Paraquat Emulsion Composition for Stable Multi-Herbicide Formulations

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Solution Overview

Problem

Formulating paraquat with other herbicides like butafenacil and S-metolachlor is challenging due to paraquat's high ionic strength, leading to formulation complications and surfactant incompatibility, and existing emulsifier systems fail to create stable emulsions.

Innovation Solution

A stable emulsion is achieved using an emulsifier package comprising a polyvinylalcohol-acetate copolymer, sorbitan ester surfactant, and polymeric ethoxylated sorbitan ester, which dissolves paraquat and maintains stability even with additional pesticidal active ingredients.

Engineering Contradictions & Design Principles

VSEngineering Contradiction Analysis

1Adaptability or versatility

If paraquat is formulated with additional herbicides using conventional emulsifier systems, then the formulation complexity increases, but the emulsion stability deteriorates due to surfactant incompatibility caused by paraquat's high ionic strength

Engineering Contradiction:
Improveformulation compatibilityVSAvoidemulsion stability
Core Design Contradiction:
Adaptability or versatilityVSStability of the object's composition

Solution Approach 1:

The patent employs a composite emulsifier system comprising multiple components (polyvinyl alcohol, sorbitan esters, and ethoxylated sorbitan esters) that work synergistically to stabilize the emulsion. This composite approach allows the formulation to accommodate paraquat's high ionic strength while maintaining emulsion stability and enabling the inclusion of additional herbicides like butafenacil and S-metolachlor

Inventive Principle:
Principle #40Composite materials

Solution Approach 2:

The polyvinyl alcohol acts as an intermediary substance that mediates between the charged paraquat molecules and the oil phase containing additional herbicides. This intermediary component facilitates compatibility among ingredients that would otherwise be incompatible due to electrostatic repulsion and surfactant interference

Inventive Principle:
Principle #24Intermediary (Mediator)

2Device complexity

If polyvinyl alcohol is used as an emulsifier with highly charged active ingredients like glyphosate and gluphosinate, then the formulation simplicity is maintained, but the polyvinyl alcohol precipitates out of solution

Engineering Contradiction:
Improveformulation simplicityVSAvoidpolyvinyl alcohol solubility
Core Design Contradiction:
Device complexityVSStability of the object's composition

Solution Approach 1:

The patent modifies the chemical parameters of the emulsifier system by selecting specific types of sorbitan esters and ethoxylated sorbitan esters that are compatible with polyvinyl alcohol in the presence of paraquat. This parameter optimization allows polyvinyl alcohol to remain soluble and functional with highly charged active ingredients, preventing precipitation while maintaining formulation simplicity

Inventive Principle:
Principle #35Parameter changes

3Reliability

If a stable emulsion is achieved with paraquat and additional herbicides, then the pesticidal efficacy is enhanced, but the formulation development time increases due to surfactant compatibility challenges

Engineering Contradiction:
Improvepesticidal efficacyVSAvoidformulation development time
Core Design Contradiction:
ReliabilityVSLoss of time

Solution Approach 1:

The patent applies preliminary action by pre-selecting and optimizing the emulsifier package composition before final formulation development. The identified combination of polyvinyl alcohol, sorbitan esters, and ethoxylated sorbitan esters is pre-tested for compatibility with paraquat and additional herbicides, establishing a reliable base formulation that reduces subsequent development time and accelerates product deployment

Inventive Principle:
Principle #10Preliminary action

Data Source

PatentEP3883383B1Paraquat formulation
Publication Date: 2025.07.16 SYNGENTA CROP PROTECITON AG

AI summary

The present invention relates to pesticidal emulsions comprising an aqueous continuous phase comprising paraquat and at least one polyvinylalcohol or polyvinylalcohol derivative; a dispersed oil phase; a pesticidal active ingredient; and at least two polymeric surfactants selected from a sorbitan ester and an ethoxylated sorbitan ester. It also relates to the use of a pesticidal emulsion to control undesired vegetation.