Mutant Phi29 DNA Polymerase Thermostability and Processivity

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Solution Overview

Problem

The existing bacteriophage phi29 DNA polymerase has limitations due to its relatively low thermostability, which restricts its application in DNA amplification techniques, particularly with high G/C content DNA and at elevated temperatures, leading to slower reaction kinetics and increased formation of non-specific products.

Innovation Solution

Mutations such as E221K, M8R, V51A, M97T, G197D, K209E, E239G, Q497P, K512E, and F526L are introduced into the phi29 DNA polymerase to enhance its thermostability, processivity, and fidelity, allowing for more efficient DNA amplification at higher temperatures.

Engineering Contradictions & Design Principles

VSEngineering Contradiction Analysis

1Productivity

If phi29 DNA polymerase is used at elevated temperatures to improve reaction kinetics, then DNA amplification efficiency increases, but the enzyme's thermostability is insufficient leading to reduced enzyme stability

Engineering Contradiction:
ImproveDNA amplification efficiencyVSAvoidenzyme stability
Core Design Contradiction:
ProductivityVSReliability

Solution Approach 1:

The patent applies parameter changes by modifying amino acid residues at specific positions (e.g., E221K, M8R, V51A, M97T, G197D, K209E, E239G, Q497P, K512E, F526L) to alter the enzyme's physical-chemical properties. These mutations increase thermostability while preserving catalytic activity, enabling the enzyme to function effectively at elevated temperatures up to 40°C and beyond, thus resolving the contradiction between reaction kinetics and enzyme stability

Inventive Principle:
Principle #35Parameter changes

2Adaptability or versatility

If phi29 DNA polymerase is used for DNA amplification with high G/C content, then amplification of difficult templates is achieved, but non-specific product formation increases due to low reaction temperature

Engineering Contradiction:
Improveability to amplify high G/C content DNAVSAvoidspecificity of amplification
Core Design Contradiction:
Adaptability or versatilityVSManufacturing precision

Solution Approach 1:

The mutated phi29 DNA polymerase exhibits enhanced thermostability that enables reactions at elevated temperatures (up to 40°C and higher). This temperature increase improves the specificity of DNA amplification by reducing non-specific product formation, while the enzyme's modified structure maintains its ability to handle high G/C content templates effectively

Inventive Principle:
Principle #35Parameter changes

3Reliability

If wild-type phi29 DNA polymerase is used at 30°C optimal temperature, then enzyme stability is maintained, but reaction kinetics are slower

Engineering Contradiction:
Improveenzyme stabilityVSAvoidreaction kinetics
Core Design Contradiction:
ReliabilityVSSpeed

Solution Approach 1:

The patent introduces multiple amino acid mutations that collectively enhance the enzyme's thermostability parameters. This allows the enzyme to maintain stability at higher temperatures where reaction kinetics are inherently faster, thus resolving the trade-off between stability at low temperature and speed at high temperature

Inventive Principle:
Principle #35Parameter changes

4Manufacturing precision

If phi29 DNA polymerase is used for whole genome amplification, then complete genome coverage is achieved, but amplification bias occurs due to processivity limitations

Engineering Contradiction:
Improvegenome coverage completenessVSAvoidamplification speed and efficiency
Core Design Contradiction:
Manufacturing precisionVSProductivity

Solution Approach 1:

The mutations in phi29 DNA polymerase enhance processivity by improving the enzyme's ability to remain bound to DNA during synthesis. This increased processivity reduces amplification bias and improves genome coverage completeness while simultaneously enhancing overall amplification efficiency and speed

Inventive Principle:
Principle #35Parameter changes

Data Source

PatentEP3093347B1DNA polymerase mutants having increased thermostability and processivity
Publication Date: 2019.08.07 THERMO FISHER SCI BALTICS UAB
  • EP3093347B1 patent drawingFigure 1
  • EP3093347B1 patent drawingFigure 2
  • EP3093347B1 patent drawingFigure 2

AI summary

Mutants of bacteriophage phi29 DNA polymerase with increased protein stability and increased half-life, compared to wild type DNA polymerase. The disclosed mutants are more stable in reaction mixtures with or without DNA. The inventive phi29 DNA polymerase mutants generate more amplification product. The inventive phi29 DNA polymerase mutants amplify genomic DNA with less bias compared to wild type DNA polymerase. Selected mutations increase the affinity of polymerase for DNA template.