Phosphazene Hydrogels with UV Cross-Linking for Biomedical Implants

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Solution Overview

Problem

Temperature-sensitive phosphazene-based polymers with chemical cross-linking are needed to improve the solidity and controlled release of drugs, as existing polymers have limitations in gel solidity and drug release profiles for applications like implant materials and artificial cartilage.

Innovation Solution

A temperature-sensitive phosphazene-based polymer with chemical cross-linking formed by UV radiation or mixing with a cross-linking agent/enzyme, allowing for sol-gel behavior and enhanced gel solidity, enabling controlled drug release and improved mechanical properties for biomedical applications.

Engineering Contradictions & Design Principles

VSEngineering Contradiction Analysis

1Reliability

If a polymer hydrogel with chemical cross-linking is prepared using conventional methods, then the gel structure is formed, but the gelation time is excessively long and physical properties are difficult to control

Engineering Contradiction:
Improvegel structure formationVSAvoidgelation time
Core Design Contradiction:
ReliabilityVSLoss of time

Solution Approach 1:

The patent changes the chemical parameters of the cross-linking system by introducing photoinitiable cross-linking groups (acrylate, methacrylate, vinyl sulfone) that can be activated by UV light. This transforms the cross-linking process from a slow thermal or enzymatic reaction to a rapid photo-induced reaction, reducing gelation time from days to minutes while maintaining controllable physical properties through parameter optimization.

Inventive Principle:
Principle #35Parameter changes

Solution Approach 2:

The patent replaces conventional thermal or enzymatic cross-linking mechanisms with photo-induced cross-linking. By substituting the activation mechanism from thermal/enzymatic to photonic, the gelation process achieves rapid and controllable network formation without the time constraints and uncontrollability of conventional methods.

Inventive Principle:
Principle #28Mechanics substitution (Replace mechanical system)

2Adaptability or versatility

If temperature-sensitive phosphazene polymer is used, then sol-gel behavior is achieved, but the gel solidity is insufficient for hydrophilic drug carrier applications

Engineering Contradiction:
Improvesol-gel behaviorVSAvoidgel solidity
Core Design Contradiction:
Adaptability or versatilityVSStrength

Solution Approach 1:

The patent merges two previously separate functionalities into a single polymer system: (1) temperature-sensitive sol-gel behavior from the phosphazene backbone with hydrophobic/hydrophilic side chains, and (2) chemical cross-linking capability from photoinitiable groups. This combination produces a hydrogel that exhibits both reversible thermal gelation and enhanced structural solidity through permanent cross-links, making it suitable for hydrophilic drug carrier applications.

Inventive Principle:
Principle #5Merging (Combining)

Solution Approach 2:

The patent creates a composite polymer structure combining phosphazene backbone, hydrophobic amino acid ester side chains, hydrophilic polyethylene glycol side chains, and photoinitiable cross-linking groups. This multi-component composite architecture provides both the temperature-sensitive sol-gel transition and the structural solidity required for biomedical applications.

Inventive Principle:
Principle #40Composite materials

3Reliability

If polyethylene glycol-based hydrogel is used for protein drug delivery, then controlled release is achieved, but the gelation process is slow and physical properties are difficult to control

Engineering Contradiction:
Improvedrug release controlVSAvoidgelation control
Core Design Contradiction:
ReliabilityVSEase of manufacture

Solution Approach 1:

The patent replaces conventional slow gelation mechanisms with photo-induced cross-linking activated by UV light. This substitution enables rapid and spatially controlled gelation, making the manufacturing process easier to control while maintaining the ability to deliver proteins and other physiological active materials through the hydrogel network.

Inventive Principle:
Principle #28Mechanics substitution (Replace mechanical system)

Applied Scientific Principles

This section explains which scientific principles are used to turn an abstract innovation direction into a practical engineering solution.

Function Achieved in This Case

The polymer exhibits improved gel solidity and controlled drug release, suitable for biomedical applications such as implant materials and artificial cartilage, with adjustable gelation temperature and biodegradability.

Implementation Method 1

A phosphazene-based polymer hydrogel with chemical cross-linkings formed by radiating ultraviolet (UV)

Methodology Applied
Scientific EffectPhotopolymerisation: Photopolymerisation

Implementation Method 2

the polymer aqueous solution maintains a liquid state at a low temperature, but it turns to a gel upon increasing temperature

Methodology Applied
Scientific EffectSol-gel transition: Gel

Implementation Method 3

Temperature-sensitive phosphazene-based polymers... show temperature sensitive polymer characteristics in which it is an aqueous solution state under a certain temperature, but it turns to a three-dimensional gel above the certain temperature

Methodology Applied
Scientific EffectThermosensitive behavior: Phase Change

Implementation Method 4

a chemical cross-linking formed by a Michael-addition-type reaction between thiol and acrylate, acrylamide, or vinyl sulfone groups

Methodology Applied
Scientific EffectMichael-addition reaction: Chemical Bonding

Data Source

PatentEP2155806B1Phosphazene hydrogels with chemical corss -link, preparation method thereof and use thereof
Publication Date: 2019.12.18 KOREA INST OF SCI & TECH
  • EP2155806B1 patent drawingFigure 1
  • EP2155806B1 patent drawingFigure 2~3
  • EP2155806B1 patent drawingFigure 4

AI summary

A phosphazene-based polymer hydrogel with a chemical cross-linkings formed by radiating ultraviolet (UV) and/or mixing with cross-linking agent and/or enzyme, a method of preparing the same, and a hydrogel forming a chemical cross-linking by radiating ultraviolet and/or mixing with a cross-linking agent and/or an enzyme; where the hydrigel shows a sol-gel behavior and has an excellent solidity by containing the phosphazene-based polymer that is capable of cross-linking at a certain concentration, are provided.