Phospholipid Extraction Without Chloroform or Chromatography

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Solution Overview

Problem

Existing methods for extracting and purifying phospholipids from animal brain use carcinogenic solvents like chloroform and require silica gel chromatography, resulting in contaminated products with solvent residues and protein components, and do not effectively enrich the final product in phosphatidylserine (PS).

Innovation Solution

A solvent-free extraction and purification process using acetone, methanol, and salt solutions, followed by filtration and solvent washes, to produce phospholipids with a high PS/PC ratio of 0.8-1.6, free from contaminants and solvent residues.

Engineering Contradictions & Design Principles

VSEngineering Contradiction Analysis

1Quantity of substance

If traditional extraction methods using chloroform and silica gel chromatography are employed, then phospholipids can be extracted from animal brain, but the final product is contaminated with solvent residues and protein components

Engineering Contradiction:
Improvephospholipid extraction yieldVSAvoidsolvent residues and protein contaminants
Core Design Contradiction:
Quantity of substanceVSObject-affected harmful factors

Solution Approach 1:

The invention extracts and removes harmful components (proteins, solvent residues) from the phospholipid preparation process by replacing traditional carcinogenic solvents with acetone and methanol, and eliminating silica gel chromatography in favor of selective precipitation and filtration methods that separate contaminants from the final product

Inventive Principle:
Principle #2Taking out (Extraction)

Solution Approach 2:

The invention converts the harmful effect of protein contamination into a beneficial separation process by using selective precipitation where proteins precipitate out while phospholipids remain in solution, allowing easy removal of the harmful contaminant

Inventive Principle:
Principle #22Blessing in disguise (Convert harm into benefit)

2Quantity of substance

If traditional extraction methods are used, then phospholipids can be obtained, but the final product is not enriched in phosphatidylserine (PS)

Engineering Contradiction:
Improvetotal phospholipid contentVSAvoidPS enrichment ratio
Core Design Contradiction:
Quantity of substanceVSManufacturing precision

Solution Approach 1:

The invention applies different treatment conditions to different phospholipid components during the extraction process, using selective precipitation conditions that favor the concentration and enrichment of phosphatidylserine in the final product while other phospholipids remain distributed differently

Inventive Principle:
Principle #3Local quality

Solution Approach 2:

The invention changes physical and chemical parameters (solvent composition, temperature, pH) during the extraction process to optimize for PS enrichment, adjusting conditions at different stages to selectively concentrate phosphatidylserine in the final preparation

Inventive Principle:
Principle #35Parameter changes

3Productivity

If carcinogenic solvents like chloroform are used for extraction, then phospholipids can be effectively extracted, but harmful residues remain in the final product

Engineering Contradiction:
Improveextraction efficiencyVSAvoidcarcinogenic solvent residues
Core Design Contradiction:
ProductivityVSObject-generated harmful factors

Solution Approach 1:

The invention replaces expensive and harmful carcinogenic solvents like chloroform with cheaper, non-carcinogenic alternatives such as acetone and methanol that can be completely evaporated without leaving harmful residues, sacrificing some extraction efficiency for complete product safety

Inventive Principle:
Principle #27Cheap short-living objects (Disposable)

Solution Approach 2:

The invention replaces the chemical extraction mechanism using carcinogenic solvents with a different chemical system based on acetone-methanol-water mixtures followed by evaporation and reconstitution, eliminating the harmful chemical agents while maintaining extraction capability

Inventive Principle:
Principle #28Mechanics substitution (Replace mechanical system)

4Manufacturing precision

If silica gel chromatography is used for purification, then phospholipids can be separated, but the process becomes complex and time-consuming

Engineering Contradiction:
Improvepurification qualityVSAvoidchromatography equipment and process
Core Design Contradiction:
Manufacturing precisionVSDevice complexity

Solution Approach 1:

The invention extracts and eliminates the need for complex silica gel chromatography equipment by using simple filtration and centrifugation steps that achieve comparable purification through selective precipitation and phase separation

Inventive Principle:
Principle #2Taking out (Extraction)

Solution Approach 2:

The invention creates a simplified alternative process that copies the purification function of chromatography using inexpensive filtration materials and simple centrifugation, achieving the same separation effect without complex equipment

Inventive Principle:
Principle #26Copying

Applied Scientific Principles

This section explains which scientific principles are used to turn an abstract innovation direction into a practical engineering solution.

Function Achieved in This Case

The process yields highly pure, PS-enriched phospholipids suitable for treating neuroendocrine disorders and Long-Covid symptoms by improving mental clarity and reducing fatigue, without using harmful solvents or chromatography.

Implementation Method 1

adding a mixture of solvents comprising acetone and methanol to the ground product

Methodology Applied
Scientific EffectSolvation: Solvation

Implementation Method 2

adding acetone and CaCl2 dihydrate to the subnatant of step f., stirring and settling

Methodology Applied
Scientific EffectSedimentation: Sedimentation

Implementation Method 3

adding a mixture of solvents comprising acetone and methanol to the ground product, stirring and settling

Methodology Applied
Scientific EffectPrecipitation: Precipitation

Implementation Method 4

adding water and ethanol, stirring and settling

Methodology Applied
Scientific EffectLiquid-Liquid Extraction: Liquid-Liquid Extraction

Implementation Method 5

separating the subnatant of step j., adding water and ethanol, stirring and settling; separating the subnatant of step k. by filtration through a filter with a filtration degree of 3μm, or alternatively 0.8 μm, and subsequently 0.2 μm

Methodology Applied
Scientific EffectFilter (physical): Filter (physical)

Implementation Method 6

removing the solvent under vacuum to obtain the purified phospholipids

Methodology Applied
Scientific EffectEvaporation: Evaporation

Implementation Method 7

removing the solvent under vacuum

Methodology Applied
Scientific EffectVacuum Distillation: Vacuum Distillation

Data Source

PatentEP4452277B1Industrial process for the extraction and purification of phospholipids
Publication Date: 2025.12.10 FIDIA FARM SPA

AI summary

An industrial process is described for the extraction and purification of phospholipids from animal brain, particularly pure and with a high percentage content of phosphatidylserine (PS) and phosphatidylcholine (PC), especially enriched in PS, and the use of these phospholipids in the treatment of the pathology defined as "Long-Covid".