Plant Extract Composition for Metabolic Disorder Treatment

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Solution Overview

Problem

Current treatments for type 2 diabetes, particularly those involving metformin and other antidiabetic agents, come with significant contraindications and adverse effects, making it challenging to manage the condition effectively and safely, especially in patients with renal insufficiency, and often require multiple medications that can increase cardiovascular risk and mortality.

Innovation Solution

A composition comprising a mixture of extracts from Chrysanthellum indicum, Cynara scolymus, Vaccinium myrtillus, and Piper (including piperine), which acts synergistically to improve carbohydrate and lipid metabolism, reducing blood sugar levels, improving insulin sensitivity, and addressing cardiovascular risk factors with fewer side effects.

Engineering Contradictions & Design Principles

VSEngineering Contradiction Analysis

1Reliability

If metformin and other antidiabetic agents are used to treat type 2 diabetes, then blood sugar levels are reduced and insulin sensitivity is improved, but contraindications and adverse effects increase, especially in patients with renal insufficiency

Engineering Contradiction:
Improveeffectiveness of diabetes treatmentVSAvoidcontraindications and adverse effects
Core Design Contradiction:
ReliabilityVSObject-affected harmful factors

Solution Approach 1:

The patent uses plant extracts (Chrysanthellum indicum, Cynara scolymus, Vaccinium myrtillus, and Piper) as natural, short-acting alternatives to long-term pharmaceutical interventions. These extracts provide therapeutic effects without the cumulative toxicity and renal accumulation issues associated with metformin, allowing patients to receive treatment even with compromised kidney function.

Inventive Principle:
Principle #27Cheap short-living objects (Disposable)

Solution Approach 2:

The plant extracts serve as intermediaries that bridge the gap between lifestyle modifications and strong pharmaceutical interventions. They provide a middle-ground therapeutic approach that is gentler than metformin but more effective than diet alone, reducing the need for aggressive pharmacological treatment and its associated side effects.

Inventive Principle:
Principle #24Intermediary (Mediator)

2Reliability

If multiple antidiabetic agents are combined to manage type 2 diabetes and cardiovascular risk factors, then metabolic control is improved, but the risk of serious side reactions and mortality increases

Engineering Contradiction:
Improvemetabolic controlVSAvoidside reactions and mortality risk
Core Design Contradiction:
ReliabilityVSObject-generated harmful factors

Solution Approach 1:

The patent combines multiple plant extracts with complementary mechanisms of action into a single formulation. This synergistic combination addresses multiple metabolic pathways (carbohydrate metabolism, lipid metabolism, insulin sensitivity) simultaneously, replacing the need for multiple separate pharmaceutical agents and their associated interaction risks.

Inventive Principle:
Principle #5Merging (Combining)

Solution Approach 2:

The invention creates a composite therapeutic formulation integrating four different plant extracts, each contributing unique bioactive compounds. This composite approach provides multi-target therapy with a single product, reducing the complexity of polypharmacy and minimizing drug-drug interactions while maintaining comprehensive metabolic control.

Inventive Principle:
Principle #40Composite materials

3Productivity

If traditional antidiabetic treatments are initiated quickly to manage type 2 diabetes, then metabolic parameters are controlled, but the complexity of managing contraindications and adverse effects increases

Engineering Contradiction:
Improvespeed of treatment initiationVSAvoidcomplexity of treatment management
Core Design Contradiction:
ProductivityVSDevice complexity

Solution Approach 1:

The patent extracts the therapeutic benefits from complex pharmaceutical regimens and consolidates them into a single plant-based formulation. This extraction process removes the need to manage multiple separate medications, their contraindications, and their interactions, simplifying treatment while maintaining effectiveness.

Inventive Principle:
Principle #2Taking out (Extraction)

Data Source

PatentEP3533454B1Composition comprising a mixture of plant extracts or a mixture of molecules contained in said plants and use to act on the carbohydrate and/or lipid metabolism
Publication Date: 2022.04.20 VALBIOTIS
  • EP3533454B1 patent drawingFigure 1~2
  • EP3533454B1 patent drawingFigure 3~4
  • EP3533454B1 patent drawingFigure 5~6

AI summary

The object of the invention is a composition comprising at least one mixture of molecules obtained from at least: - Chrysanthellum indicum, and - Cynara scolymus, and - Vaccinium myrtillus, said mixture of molecules also comprising piperine. This composition is particularly useful as a nutritional or health product for preventing and/or combating disorders of carbohydrate and/or lipid metabolism in humans or animals.