Protective Compounds for Platelet Storage Lesion Prevention

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Solution Overview

Problem

Current methods for storing blood platelets are limited by bacterial proliferation at room temperature and cold-induced platelet storage lesions when cooled, leading to premature expiration and functional damage, necessitating the development of new compounds that can protect cells and platelets against oxidative stress and storage-related injuries.

Innovation Solution

Development of specific compounds, such as those with the structural formula (I), which protect cells and blood platelets by preventing damage from oxidative stress, cold storage lesions, and other medical indications, including ischemia and thrombotic disorders, by inhibiting cell death and maintaining platelet functionality during storage.

Engineering Contradictions & Design Principles

VSEngineering Contradiction Analysis

1Reliability

If blood platelets are stored at room temperature (20-24°C), then platelet functionality is maintained, but bacterial proliferation occurs leading to premature expiration

Engineering Contradiction:
Improveplatelet functionalityVSAvoidbacterial proliferation
Core Design Contradiction:
ReliabilityVSObject-affected harmful factors

Solution Approach 1:

The patent changes the storage temperature parameter from room temperature to refrigerated temperature (4°C), and introduces compounds that modify platelet membrane properties to prevent cold-induced damage. This parameter change allows bacterial suppression while maintaining platelet viability through chemical protection.

Inventive Principle:
Principle #35Parameter changes

Solution Approach 2:

The patent introduces compounds as intermediary substances that mediate between the cold storage environment and platelets. These compounds act as protective agents that prevent direct harmful effects of cold temperature on platelet membranes, enabling safe refrigerated storage.

Inventive Principle:
Principle #24Intermediary (Mediator)

2Object-affected harmful factors

If blood platelets are cooled to 4°C, then bacterial proliferation is prevented, but cold-induced platelet storage lesions occur causing structural and functional damage

Engineering Contradiction:
Improvebacterial proliferation preventionVSAvoidplatelet structural integrity
Core Design Contradiction:
Object-affected harmful factorsVSReliability

Solution Approach 1:

The patent applies compounds to platelets before cold storage to provide protective cushioning. These compounds are incorporated into platelet membranes in advance, creating a protective layer that cushions against cold-induced structural damage during subsequent refrigerated storage.

Inventive Principle:
Principle #11Beforehand cushioning (Prior cushioning)

Solution Approach 2:

The patent creates a composite system combining platelets with protective compounds. The compounds integrate with platelet membrane structures to form a composite material that maintains platelet integrity under cold storage conditions, preventing structural lesions while enabling bacterial suppression.

Inventive Principle:
Principle #40Composite materials

3Productivity

If storage time is extended beyond 5 days, then more platelets can be utilized, but platelet viability decreases due to storage lesions

Engineering Contradiction:
Improveplatelet utilization rateVSAvoidplatelet viability
Core Design Contradiction:
ProductivityVSReliability

Solution Approach 1:

The patent performs preliminary action by incorporating protective compounds into platelet membranes before storage. This preliminary protection enables extended storage periods while maintaining viability, allowing platelets to be stored longer than the conventional 5-day limit without significant loss of functionality.

Inventive Principle:
Principle #10Preliminary action

Applied Scientific Principles

This section explains which scientific principles are used to turn an abstract innovation direction into a practical engineering solution.

Function Achieved in This Case

The compounds effectively reduce cell death and maintain platelet functionality during storage, extending the viability and usability of blood platelets, and can be used in treating conditions related to oxidative stress and thrombotic disorders.

Implementation Method 1

oxidative stress in cells and cell damage are often related with aging and diseases related to aging

Methodology Applied
Scientific EffectOxidative stress: Oxidation

Implementation Method 2

compounds such as nitrones can be used in the treatment of ischemic stroke and as anti-cancer agents

Methodology Applied
Scientific EffectFree radical damage: Free Fall

Implementation Method 3

Platelets show cold induced platelet storage lesion (PSL) when they are cooled, even briefly to 4°C

Methodology Applied
Scientific EffectCold-induced storage lesion: Freezing

Implementation Method 4

reversible to irreversible morphological change from a discoid cell to speculated spheres with protruding filipodia, depending on the duration of exposure to temperatures less than 20°C

Methodology Applied
Scientific EffectPhase transition: Phase Change

Data Source

PatentEP3388426B1Compounds for protection of cells
Publication Date: 2023.07.05 SULFATEQ BV
  • EP3388426B1 patent drawingFigure 1
  • EP3388426B1 patent drawingFigure 2
  • EP3388426B1 patent drawingFigure 2

AI summary

This invention is related to a compound for certain uses with the structural formula (I) wherein, R1, and R2 are independently selected from the group consisting of C1-C6 alkyl and is preferably methyl, ethyl, propyl or isopropyl; R3 is selected from the group consisting of CH2NHR9, C(=O)YR10, -CH2OH