Protease Variants With Targeted Substitutions for Cleaning Activity

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Solution Overview

Problem

There is a need for engineered proteases with enhanced proteolytic and cleaning activities suitable for specific conditions and uses.

Innovation Solution

Development of protease variants with specific amino acid substitutions, such as S078N-G097A-G128S-Y217Q, that exhibit improved proteolytic and cleaning activities compared to the BPN' protease, along with methods for producing and using these variants in compositions for cleaning applications.

Engineering Contradictions & Design Principles

VSEngineering Contradiction Analysis

1Productivity

If protease variants with specific amino acid substitutions (S078N-G097A-G128S-Y217Q) are developed, then proteolytic activity and cleaning activity are enhanced, but protein structure complexity increases

Engineering Contradiction:
Improveproteolytic activityVSAvoidprotein structure complexity
Core Design Contradiction:
ProductivityVSDevice complexity

Solution Approach 1:

The patent applies parameter changes by modifying specific amino acid residues (S078N, G097A, G128S, Y217Q) in the protease sequence to enhance proteolytic and cleaning activities. This targeted substitution approach optimizes enzyme performance while maintaining structural feasibility through controlled parameter modification.

Inventive Principle:
Principle #35Parameter changes

Solution Approach 2:

The invention implements local quality by introducing specific amino acid substitutions at particular positions (78, 97, 128, 217) within the protease sequence. These localized modifications enhance specific functional properties (proteolytic activity, cleaning activity) without altering the entire protein structure, thereby resolving the contradiction between enhanced functionality and structural complexity.

Inventive Principle:
Principle #3Local quality

2Productivity

If protease variants with specific amino acid substitutions (S078N-G097A-G128S-Y217Q) are developed, then cleaning activity is enhanced, but manufacturing complexity increases

Engineering Contradiction:
Improvecleaning activityVSAvoidmanufacturing complexity
Core Design Contradiction:
ProductivityVSEase of manufacture

Solution Approach 1:

The patent modifies specific amino acid parameters (S078N, G097A, G128S, Y217Q) to enhance cleaning activity. These targeted changes allow for improved performance while maintaining relatively simple manufacturing processes through site-directed mutagenesis and standard recombinant expression techniques.

Inventive Principle:
Principle #35Parameter changes

Solution Approach 2:

By applying localized amino acid substitutions at specific positions rather than global sequence modification, the invention achieves enhanced cleaning activity with minimal impact on manufacturing complexity. The local quality approach enables precise functional optimization using established protein engineering methods.

Inventive Principle:
Principle #3Local quality

3Productivity

If multiple amino acid substitutions are introduced to enhance proteolytic activity, then enzyme performance improves, but sequence identity to original BPN' protease decreases

Engineering Contradiction:
Improveproteolytic activityVSAvoidsequence identity
Core Design Contradiction:
ProductivityVSManufacturing precision

Solution Approach 1:

The patent introduces specific amino acid substitutions (S078N, G097A, G128S, Y217Q) to enhance proteolytic activity while maintaining at least 80% sequence identity to BPN' protease. This controlled parameter modification approach optimizes enzyme performance within acceptable sequence deviation limits.

Inventive Principle:
Principle #35Parameter changes

Solution Approach 2:

The invention applies local quality by limiting modifications to specific amino acid positions (78, 97, 128, 217) while preserving the majority of the original BPN' sequence. This localized approach enhances proteolytic activity while maintaining sufficient sequence identity for structural integrity and manufacturability.

Inventive Principle:
Principle #3Local quality

Applied Scientific Principles

This section explains which scientific principles are used to turn an abstract innovation direction into a practical engineering solution.

Function Achieved in This Case

The protease variants demonstrate enhanced proteolytic and cleaning activities, making them suitable for various industrial and personal care applications, including cleaning compositions and methods.

Implementation Method 1

the variant has enhanced proteolytic activity and/or cleaning activity compared to the proteolytic activity and/or cleaning activity of the BPN' protease

Methodology Applied
Scientific EffectProteolysis: Hydrolysis

Data Source

PatentEP3599279B1Compositions and methods comprising protease variants
Publication Date: 2026.02.18 DANISCO US INC
  • EP3599279B1 patent drawingFigure 1
  • EP3599279B1 patent drawingFigure 2
  • EP3599279B1 patent drawingFigure 3

AI summary

The present invention provides protease variants, compositions comprising protease variants, and methods of using such protease variants and compositions.