Pyridine-Based Herbicidal Compounds for Improved Weed Control

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Solution Overview

Problem

Existing herbicides, such as those disclosed in WO 2002/42275 and U.S. Pat. No. 6,010,980, do not effectively address the need for herbicidally active compounds with improved efficacy against undesirable plant growth in crops.

Innovation Solution

Development of novel herbicidal compounds of formula (I) with specific substituent combinations, including various alkyl, haloalkyl, alkoxy, and heteroatom-containing groups, which exhibit enhanced herbicidal activity.

Engineering Contradictions & Design Principles

VSEngineering Contradiction Analysis

1Reliability

If existing herbicides (WO 2002/42275 and U.S. Pat. No. 6,010,980) are used, then herbicidal activity is achieved, but efficacy against undesirable plant growth is insufficient

Engineering Contradiction:
Improveherbicidal activityVSAvoidefficacy against undesirable plant growth
Core Design Contradiction:
ReliabilityVSProductivity

Solution Approach 1:

The patent applies parameter changes by systematically varying the substituent groups R1-R19 on the pyridine core structure, exploring different combinations of alkyl, haloalkyl, alkoxy, and heteroatom-containing groups to optimize herbicidal efficacy while maintaining reliable herbicidal activity

Inventive Principle:
Principle #35Parameter changes

Solution Approach 2:

The invention creates composite molecular structures by combining the pyridine core with diverse substituent groups (alkyl, haloalkyl, alkoxy, heteroatom-containing groups) to generate compounds with enhanced and versatile herbicidal properties that overcome the limitations of existing single-structure herbicides

Inventive Principle:
Principle #40Composite materials

Data Source

PatentUS20250212879A1Herbicidal compounds
Publication Date: 2025.07.03 SYNGENTA CROP PROTECITON AG
  • US20250212879A1 patent drawing
  • US20250212879A1 patent drawing
  • US20250212879A1 patent drawing

AI summary

Compounds of the formula (I) wherein the substituents are as defined in claim 1, useful as a pesticides, especially as herbicides.