Pyridone Herbicidal Derivatives for Selective Weed Control

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Solution Overview

Problem

Existing herbicides do not effectively address the need for selective and efficient weed control in agricultural and horticultural settings, particularly in crops of useful plants.

Innovation Solution

Development of novel pyridone derivatives with specific structural features, such as C1-C6alkyl, C1-C6alkoxy, C2-C6alkenyl, C2-C6alkynyl, C1-C6alkoxyC1-C6alkyl, or C3-C6cycloalkyl substituents, which exhibit herbicidal activity when applied as active ingredients in agrochemical compositions.

Engineering Contradictions & Design Principles

VSEngineering Contradiction Analysis

1Reliability

If existing herbicides are used, then weed control is achieved, but the herbicidal activity is insufficient for selective and efficient weed control in agricultural and horticultural settings

Engineering Contradiction:
Improveherbicidal activityVSAvoidselective weed control
Core Design Contradiction:
ReliabilityVSAdaptability or versatility

Solution Approach 1:

The patent applies parameter changes by systematically modifying the chemical structure of pyridone derivatives through varying substituents at different positions (R1-R6 groups including alkyl, alkoxy, alkenyl, alkynyl, cycloalkyl groups). These structural parameter changes result in compounds with enhanced herbicidal activity and improved selectivity for weed control in agricultural and horticultural settings, directly resolving the contradiction between sufficient herbicidal activity and selective control capability

Inventive Principle:
Principle #35Parameter changes

Data Source

PatentUS20260013501A1Herbicidal derivatives
Publication Date: 2026.01.15 SYNGENTA CROP PROTECITON AG
  • US20260013501A1 patent drawing
  • US20260013501A1 patent drawing
  • US20260013501A1 patent drawing

AI summary

Compounds of Formula (I) wherein the substituents are as defined in claim 1. The invention further relates to herbicidal compositions which comprise a compound of Formula (I) and to the use of compounds of Formula (I) for controlling weeds, in particular in crops of useful plants.