Microbial Conversion of Rebaudioside A to D and M

Resolve Bottlenecks,
Find Innovative Solutions
Generate Solutions

Solution Overview

Problem

Current methods for producing Rebaudioside D and Rebaudioside M, which have superior taste properties compared to Rebaudioside A, are inefficient due to the rarity of these compounds in nature and the instability and cost of UDP-glucose, a necessary co-substrate for UDP-glycosyl transferases.

Innovation Solution

A method involving a host cell capable of taking up Rebaudioside A, regenerating UDP-glucose, and expressing UDP-glucosyl transferase enzymes to convert Rebaudioside A into Rebaudioside D and Rebaudioside M, using microbial species like Kluyveromyces marxianus that are safe for food use.

Engineering Contradictions & Design Principles

VSEngineering Contradiction Analysis

1Reliability

If UDP-glycosyl transferases are used to convert Rebaudioside A to Rebaudioside D and Rebaudioside M, then superior taste properties are achieved, but the process becomes inefficient due to the instability and high cost of UDP-glucose co-substrate

Engineering Contradiction:
Improvetaste propertiesVSAvoidproduction efficiency
Core Design Contradiction:
ReliabilityVSProductivity

Solution Approach 1:

The host cell is engineered to autonomously regenerate UDP-glucose from glucose-1-phosphate using engineered enzymes (phosphoglucomutase and UDP-glucose pyrophosphorylase), eliminating the need for external addition of expensive and unstable UDP-glucose. The cell's metabolic pathway is harnessed to continuously supply the required co-substrate.

Inventive Principle:
Principle #25Self-service

Solution Approach 2:

Glucose-1-phosphate serves as an intermediary substance that is stable and inexpensive to produce, which is then converted by engineered enzymes into UDP-glucose in situ. This intermediary approach bypasses the problems of directly using unstable and costly UDP-glucose.

Inventive Principle:
Principle #24Intermediary (Mediator)

2Manufacturing precision

If Rebaudioside D and Rebaudioside M are produced through natural occurrence, then high purity sweeteners are obtained, but the production is limited due to the rarity of these compounds in nature

Engineering Contradiction:
ImprovepurityVSAvoidproduction volume
Core Design Contradiction:
Manufacturing precisionVSProductivity

Solution Approach 1:

The invention extracts and utilizes only the essential genetic elements (UGT enzyme genes and UDP-glucose regeneration pathway genes) from natural sources and transfers them into a controllable host cell system. This allows production to be decoupled from natural rarity while maintaining the enzymatic specificity required for high purity product formation.

Inventive Principle:
Principle #2Taking out (Extraction)

Solution Approach 2:

The host cell's metabolic parameters are optimized through genetic engineering to favor the production of Rebaudioside D and Rebaudioside M. Expression levels of UGT enzymes and UDP-glucose regeneration enzymes are tuned to maximize conversion efficiency and product purity while maintaining cell viability.

Inventive Principle:
Principle #35Parameter changes

3Reliability

If microbial species are selected for food safety, then safe sweeteners are produced, but the ability to assimilate Rebaudioside A and regenerate UDP-glucose may be limited

Engineering Contradiction:
Improvefood safetyVSAvoidmetabolic capability
Core Design Contradiction:
ReliabilityVSAdaptability or versatility

Solution Approach 1:

The metabolic pathway is segmented into distinct functional modules: Rebaudioside A uptake system, UDP-glucose regeneration module (using phosphoglucomutase and UDP-glucose pyrophosphorylase), and glycosylation module (using UGT enzymes). Each module can be independently optimized and assembled in safe microbial hosts.

Inventive Principle:
Principle #1Segmentation

Solution Approach 2:

The host cell is engineered to perform multiple functions: taking up Rebaudioside A, regenerating UDP-glucose from glucose-1-phosphate, and catalyzing the glycosylation reactions. This multi-functionality is achieved by introducing complementary genetic pathways into a single safe microbial platform.

Inventive Principle:
Principle #6Universality (Multi-functionality)

Applied Scientific Principles

This section explains which scientific principles are used to turn an abstract innovation direction into a practical engineering solution.

Function Achieved in This Case

This method enables efficient intracellular conversion of Rebaudioside A to Rebaudioside D and Rebaudioside M, overcoming the limitations of natural availability and co-substrate stability, thereby enhancing the production of these valuable sweeteners.

Implementation Method 1

subjecting rebaudioside A to a UDP-glucosyl transferase enzyme, the UDP-glucosyl transferase enzyme is intracellularly produced by a host cell

Methodology Applied
Scientific EffectEnzyme catalysis: Enzyme

Implementation Method 2

the host cell is capable of rebaudioside A uptake from a culture medium

Methodology Applied
Scientific EffectCellular absorption: Absorption (physical)

Data Source

PatentEP3384039B1Process for producing high purity steviol glycosides
Publication Date: 2025.04.30 PURECIRCLE SDN BHD
  • EP3384039B1 patent drawingFigure 1
  • EP3384039B1 patent drawingFigure 2

AI summary

A method of producing steviol glycoside compositions and the use thereof in foods, beverages and other consumables, is described.