Recombinant Sclerotium Rolfsii Lectin for Targeted Inflammation Control

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Solution Overview

Problem

Current treatments for inflammatory diseases are costly, have significant side effects, and lack specificity, necessitating a more effective and economical biologic option.

Innovation Solution

Utilization of a recombinant lectin derived from Sclerotium rolfsii with an amino acid sequence of SEQ ID NO: 2, which inhibits inflammatory cytokine secretion, reduces C-reactive protein levels, and stimulates ALP activity and collagen levels, administered via various routes to treat and prevent inflammation.

Engineering Contradictions & Design Principles

VSEngineering Contradiction Analysis

1Reliability

If conventional medications (NSAIDs, DMARDs, biologics, corticosteroids) are used to treat inflammatory diseases, then inflammation can be reduced, but cost increases and side effects occur

Engineering Contradiction:
Improveanti-inflammatory efficacyVSAvoidside effects and cost
Core Design Contradiction:
ReliabilityVSObject-affected harmful factors

Solution Approach 1:

The patent employs a recombinant lectin protein derived from Sclerotium rolfsii, which is a cost-effective alternative to expensive biologics. The lectin is produced through recombinant DNA technology in host cells, enabling scalable production at lower cost while maintaining therapeutic efficacy with fewer side effects

Inventive Principle:
Principle #27Cheap short-living objects (Disposable)

Solution Approach 2:

The patent modifies the amino acid sequence of the Sclerotium rolfsii lectin (SEQ ID NO: 2) to enhance its anti-inflammatory properties. Specific amino acid changes were introduced to improve binding affinity and functional activity, allowing optimization of therapeutic parameters without increasing cost

Inventive Principle:
Principle #35Parameter changes

2Manufacturing precision

If biologics are used to treat inflammatory diseases, then specificity and efficacy improve, but cost and availability worsen

Engineering Contradiction:
Improvespecificity of actionVSAvoidproduction scalability and cost
Core Design Contradiction:
Manufacturing precisionVSEase of manufacture

Solution Approach 1:

The patent creates a recombinant copy of the Sclerotium rolfsii lectin protein using DNA cloning techniques. The gene encoding the lectin is inserted into host cells (such as E. coli or yeast) that replicate and produce the protein, enabling large-scale manufacturing while maintaining the specific anti-inflammatory properties of the original lectin

Inventive Principle:
Principle #26Copying

Solution Approach 2:

The recombinant lectin protein serves multiple functions: it binds to specific carbohydrate structures on cell surfaces, activates immune cells, and modulates inflammatory responses. This multi-functionality allows a single protein to address various aspects of inflammatory disease pathology, reducing the need for multiple specialized drugs

Inventive Principle:
Principle #6Universality (Multi-functionality)

Data Source

PatentEP3849586B1Sclerotium rolfsii lectin for treatment of inflammatory diseases
Publication Date: 2026.03.11 UNICHEM LAB LTD
  • EP3849586B1 patent drawingFigure 1~2
  • EP3849586B1 patent drawingFigure 3~4
  • EP3849586B1 patent drawing

AI summary

The present invention relates to a lectin for use in the treatment, reduction in progression and curing of inflammation in a subject in need thereof. Pharmaceutical compositions comprising said lectin are also described. The lectin may comprise an amino acid sequence having sequence of SEQ ID NO: 1 or at least 60% homology to SEQ ID NO: 1.