Saccharide-Coated Solid-Phase Carrier for Specific Capture

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Solution Overview

Problem

Existing solid-phase carriers for capturing target substances face challenges with high nonspecific adsorption of biological substances, which complicates the detection and purification of specific proteins, peptides, nucleic acids, and cells, and can reduce the activity of bound ligands.

Innovation Solution

A solid-phase carrier with a saccharide-coated base material and a linker of 5-100 atoms having a reactive functional group for binding ligands, designed to minimize nonspecific adsorption and maintain ligand activity, is developed. This carrier is produced by chemically binding a saccharide to a linker molecule and then to a base material, such as magnetic particles, creating a surface suitable for specific interactions.

Engineering Contradictions & Design Principles

VSEngineering Contradiction Analysis

1Reliability

If conventional affinity resins are used for capturing target substances, then the capture capability is achieved, but nonspecific adsorption of biological substances occurs which complicates detection and purification

Engineering Contradiction:
Improvespecific capture capabilityVSAvoidnonsspecific adsorption
Core Design Contradiction:
ReliabilityVSObject-generated harmful factors

Solution Approach 1:

The patent introduces a spacer arm as an intermediary component between the solid-phase carrier and the ligand. This spacer arm mediates the interaction by providing physical separation that prevents nonspecific adsorption of biological substances onto the carrier surface, while still allowing the ligand to maintain its specific binding capability to the target substance.

Inventive Principle:
Principle #24Intermediary (Mediator)

Solution Approach 2:

The patent applies different functional properties to different parts of the carrier structure. The solid-phase carrier surface is designed to be non-adsorptive (low nonspecific binding), while the ligand-bound region maintains high specific binding affinity. This spatial differentiation of functional qualities resolves the contradiction between specific capture and nonspecific adsorption.

Inventive Principle:
Principle #3Local quality

2Reliability

If conventional solid-phase carriers are used, then target substance capture is possible, but the activity of bound ligands is reduced

Engineering Contradiction:
Improvetarget capture functionVSAvoidligand activity
Core Design Contradiction:
ReliabilityVSLoss of substance

Solution Approach 1:

The spacer arm serves as a protective intermediary that separates the ligand from the solid-phase carrier surface. This separation prevents the carrier surface from interacting with and potentially deactivating the ligand, thereby maintaining ligand activity while still enabling target capture function.

Inventive Principle:
Principle #24Intermediary (Mediator)

Solution Approach 2:

The patent extends the ligand-carrying structure into the third dimension by using a spacer arm that protrudes from the carrier surface. This dimensional extension places the ligand in a different spatial zone away from the carrier surface, reducing unwanted interactions and preserving ligand activity.

Inventive Principle:
Principle #17Another dimension (Dimensionality change)

Applied Scientific Principles

This section explains which scientific principles are used to turn an abstract innovation direction into a practical engineering solution.

Function Achieved in This Case

The solution significantly reduces nonspecific adsorption of biological substances, allowing for efficient capture and maintaining the activity of bound ligands, thereby enhancing the detection and purification of target substances.

Implementation Method 1

The presence of a nonspecific intermolecular interaction that prevents the selection and purification of a desired molecule based on a specific intermolecular interaction has raised a problem

Methodology Applied
Scientific EffectNonspecific adsorption: Adsorption

Implementation Method 2

a linker of 5 to 100 atoms having a reactive functional group for binding a ligand that specifically binds to a target substance, in which the saccharide is chemically bound to the linker

Methodology Applied
Scientific EffectChemical bonding: Chemical Bonding

Implementation Method 3

an attempt to capture a molecule that exhibits a specific interaction with a particular molecule using a technique based on intermolecular interactions

Methodology Applied
Scientific EffectSpecific intermolecular interaction: Adsorption

Data Source

PatentEP3109637B1Method for capturing target substance, solid-phase carrier for capturing target substance, and method for producing solid-phase carrier
Publication Date: 2019.08.14 JSR CORPORATION
  • EP3109637B1 patent drawingFigure 1
  • EP3109637B1 patent drawingFigure 2
  • EP3109637B1 patent drawing

AI summary

To provide a solid-phase carrier that has extremely low nonspecific adsorption of biological substances such as proteins, peptides, nucleic acids and cells, and is capable of maintaining the activity of bound ligands at a high level; and a method for capturing a target substance using the solid-phase carrier. A method for capturing a target substance, including: a step for preparing a solid-phase carrier for capturing a target substance, the carrier having a base material, at least a portion of the surface thereof being formed oforcoatedwitha saccharide, and having a linker of 5-100 atoms having a reactive functional group for binding a ligand that specifically binds to the target substance, wherein the saccharide is chemically bound to the linker; a step for binding the ligand to the solid-phase carrier to obtain a solid-phase carrier having a ligand bound thereto; and a step for bringing the solid-phase carrier having the ligand bound thereto into contact with a sample containing the target substance that specifically binds to the ligand.