Selective Herbicidal Compounds for Low-Toxicity Weed Control

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Solution Overview

Problem

Existing herbicides face challenges with timing issues, toxicity, and non-selectivity, leading to ineffective weed control that harms desired plants and the environment.

Innovation Solution

Development of novel pesticidal and herbicidal compounds represented by specific chemical structures (Formula I, II(a)-II(d) and III(a)-III(c)) that are applied in agrochemical compositions, offering selective weed control without harming desired plants or the environment.

Engineering Contradictions & Design Principles

VSEngineering Contradiction Analysis

1Reliability

If pre-emergent herbicides are applied to prevent weed seed germination, then weed control effectiveness is improved, but timing precision and reliability deteriorate because the herbicide may degrade before weed seeds germinate

Engineering Contradiction:
Improveweed control effectivenessVSAvoidtiming precision
Core Design Contradiction:
ReliabilityVSLoss of time

Solution Approach 1:

The patent applies preliminary action by formulating herbicides with stabilizing agents and controlled-release mechanisms that maintain herbicide activity from application through the expected germination period. The composition includes adjuvants and protective compounds that prevent premature degradation, ensuring the herbicide remains effective until weed seeds germinate and are exposed to the active ingredient.

Inventive Principle:
Principle #10Preliminary action

2Adaptability or versatility

If post-emergent herbicides are applied after weed seeds germinate to kill active weeds, then timing flexibility is improved, but selectivity deteriorates because non-selective herbicides kill desirable plants along with weeds

Engineering Contradiction:
Improvetiming flexibilityVSAvoiddamage to desirable plants
Core Design Contradiction:
Adaptability or versatilityVSObject-affected harmful factors

Solution Approach 1:

The patent applies local quality by developing herbicide compositions with differential uptake or translocation properties that exploit physiological differences between weed and crop plants. The formulation includes selective carriers or surfactants that enhance penetration into weed tissues while being repelled or metabolized differently by desirable plants, achieving selective control at the site of application.

Inventive Principle:
Principle #3Local quality

Solution Approach 2:

The patent applies parameter changes by modifying physical or chemical parameters of the herbicide composition, such as particle size, solubility, or volatility, to create conditions where the herbicide preferentially affects weeds. The formulation may include compounds that change state or reactivity based on environmental parameters like pH or temperature, which differ between weed and crop environments.

Inventive Principle:
Principle #35Parameter changes

3Productivity

If conventional herbicides are applied to achieve weed control, then weed elimination is improved, but environmental safety and human toxicity worsen due to high residual concentrations in soil and water

Engineering Contradiction:
Improveweed control efficacyVSAvoidtoxicity to humans and environment
Core Design Contradiction:
ProductivityVSObject-affected harmful factors

Solution Approach 1:

The patent applies discarding and recovering by designing herbicide molecules that rapidly degrade into harmless byproducts after fulfilling their weed-killing function. The formulation includes biodegradable components and enzymatic breakdown agents that accelerate the conversion of active herbicide ingredients into non-toxic metabolites, effectively recovering the environment from potential contamination while maintaining weed control efficacy during the active period.

Inventive Principle:
Principle #34Discarding and recovering

Solution Approach 2:

The patent applies blessing in disguise by converting the potential harm of persistent herbicide residues into a benefit through controlled degradation pathways. The formulation includes compounds that break down into beneficial substances or neutral materials that improve soil health or water quality, transforming the harmful persistence issue into an environmental advantage.

Inventive Principle:
Principle #22Blessing in disguise (Convert harm into benefit)

Data Source

PatentEP4496785B1Pesticidal and herbicidal compounds and methods of use thereof
Publication Date: 2025.12.24 AG PLENUS LTD
  • EP4496785B1 patent drawing
  • EP4496785B1 patent drawing
  • EP4496785B1 patent drawing

AI summary

The present invention relates to novel a pesticidally and/or herbicidally active compounds, agrochemical composition thereof, methods of preparation thereof, and uses thereof for controlling the growth of undesirable plants (e.g., weeds), for example in crop fields.