Oral Retention Composition Using Shellac-Coated Functional Substances

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Solution Overview

Problem

Functional substances in oral compositions are easily washed away by saliva and exudates, and retention-enhancing substances often interact with functional substances, reducing their effectiveness, especially when acidic polysaccharides are used with basic or polyphenolic substances.

Innovation Solution

An oral retention composition comprising shellac or zein-coated functional substances mixed with acidic polysaccharides, such as carrageenan, hyaluronic acid, or xanthan gum, to enhance retention time in the oral cavity without significantly impairing the retention-imparting function of the acidic polysaccharides.

Engineering Contradictions & Design Principles

VSEngineering Contradiction Analysis

1Duration of action of moving object

If retention-enhancing substances are added to improve functional substance retention in the oral cavity, then retention time is extended, but the functional substances interact with retention-enhancing substances, greatly reducing or eliminating their effects

Engineering Contradiction:
Improveretention time of functional substanceVSAvoideffectiveness of functional substance
Core Design Contradiction:
Duration of action of moving objectVSReliability

Solution Approach 1:

The invention divides the functional substance into coated particles, where each particle is individually coated with a protective layer. This segmentation prevents interaction between the functional substance and acidic polysaccharides while maintaining retention enhancement, thereby preserving both retention time and effectiveness

Inventive Principle:
Principle #1Segmentation

Solution Approach 2:

The invention introduces an intermediary coating layer (such as shellac, zein, or other protective coatings) between the functional substance and acidic polysaccharides. This intermediary prevents direct interaction that would otherwise reduce effectiveness, while still allowing the acidic polysaccharides to provide retention enhancement

Inventive Principle:
Principle #24Intermediary (Mediator)

2Duration of action of moving object

If acidic polysaccharides are used as retention-enhancing substances, then viscosity is increased to improve retention, but when functional substances are basic substances or polyphenols, the retention-enhancing action is greatly reduced

Engineering Contradiction:
Improveretention time of functional substanceVSAvoidcompatibility with basic substances and polyphenols
Core Design Contradiction:
Duration of action of moving objectVSAdaptability or versatility

Solution Approach 1:

By coating basic substances and polyphenols as separate particles before mixing with acidic polysaccharides, the invention prevents direct chemical interaction that would reduce viscosity. Each coated particle maintains its integrity while the acidic polysaccharides provide retention enhancement through viscosity increase

Inventive Principle:
Principle #1Segmentation

Solution Approach 2:

The coating layer acts as an intermediary barrier that prevents direct interaction between basic substances/polyphenols and acidic polysaccharides. This allows the acidic polysaccharides to maintain their viscosity-imparting properties while still providing retention enhancement for the functional substances

Inventive Principle:
Principle #24Intermediary (Mediator)

Applied Scientific Principles

This section explains which scientific principles are used to turn an abstract innovation direction into a practical engineering solution.

Function Achieved in This Case

The composition effectively prolongs the retention of functional substances in the oral cavity, suppressing the decrease in viscosity of acidic polysaccharides and maintaining their antimicrobial and biofilm inhibition activities, thereby extending the duration of their effects.

Implementation Method 1

the functional substance coated with the at least one compound selected from the group consisting of shellac and zein

Methodology Applied
Scientific EffectCoating: Coatings

Implementation Method 2

the retention-enhancing action (e.g., viscosity-imparting) of the acidic polysaccharide

Methodology Applied
Scientific EffectViscosity-imparting:

Implementation Method 3

the decrease in the viscosity of the acidic polysaccharide caused by the functional substance can be suppressed

Methodology Applied
Scientific EffectViscosity stabilization:

Data Source

PatentUS20230276836A1Oral retention composition
Publication Date: 2023.09.07 BIZEN CHEM
  • US20230276836A1 patent drawing
  • US20230276836A1 patent drawing

AI summary

An object of the present invention is to provide an oral retention composition in which a decrease in the viscosity of an acidic polysaccharide due to a functional substance is suppressed even when the functional substance is basic. The present invention relates to an oral retention composition comprising at least one compound selected from the group consisting of shellac and zein, a functional substance, and an acidic polysaccharide, the functional substance coated with the at least one compound selected from the group consisting of shellac and zein being mixed with the acidic polysaccharide.