Silencing Oligonucleotide for Padlock Probe Specificity

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Solution Overview

Problem

Current methods for removing unhybridized padlock probes in nucleic acid detection assays are inefficient, particularly in homogenous solutions, and can lead to mis-priming and reduced specificity and sensitivity due to the presence of free padlock probes.

Innovation Solution

The use of a silencing oligonucleotide that hybridizes to the ends of padlock probes, preventing them from participating in further reactions by creating a gap that keeps the ends apart, ensuring the probes are functionally inactivated unless a correct template is present, allowing for RCA to be initiated only after the silencing oligonucleotide is present.

Engineering Contradictions & Design Principles

VSEngineering Contradiction Analysis

1Reliability

If free padlock probes are removed by washing or enzymatic digestion, then mis-priming is reduced, but the method requires additional steps (washing, solid phase, or enzyme inactivation) that reduce ease of operation

Engineering Contradiction:
ImprovespecificityVSAvoidease of operation
Core Design Contradiction:
ReliabilityVSEase of operation

Solution Approach 1:

A silencing oligonucleotide is introduced as an intermediary substance that hybridizes to free padlock probes to prevent mis-priming. This mediator allows the system to achieve high specificity without requiring washing steps, solid phases, or enzyme inactivation, thereby maintaining ease of operation while improving reliability

Inventive Principle:
Principle #24Intermediary (Mediator)

Solution Approach 2:

The harmful function of free padlock probes (mis-priming) is extracted and neutralized by the silencing oligonucleotide, which specifically binds to and silences unligated probes. This separates the problematic free probes from the functional ligated probes without requiring physical removal steps

Inventive Principle:
Principle #2Taking out (Extraction)

2Reliability

If exonuclease is used to digest free padlock probes, then specificity is improved, but the method requires additional expense and enzyme inactivation steps

Engineering Contradiction:
ImprovespecificityVSAvoidcomplexity
Core Design Contradiction:
ReliabilityVSDevice complexity

Solution Approach 1:

The silencing oligonucleotide serves as a simple, inexpensive, single-use reagent that replaces expensive enzymes like exonuclease. It performs the function of selectively silencing free probes without requiring enzyme inactivation steps, reducing both cost and procedural complexity

Inventive Principle:
Principle #27Cheap short-living objects (Disposable)

Solution Approach 2:

The biochemical mechanism of enzymatic digestion by exonuclease is replaced with a simpler hybridization-based silencing mechanism. The silencing oligonucleotide uses base-pairing to neutralize free probes instead of requiring enzymatic activity, eliminating the need for enzyme addition and inactivation steps

Inventive Principle:
Principle #28Mechanics substitution (Replace mechanical system)

Applied Scientific Principles

This section explains which scientific principles are used to turn an abstract innovation direction into a practical engineering solution.

Function Achieved in This Case

This approach enhances the specificity and sensitivity of nucleic acid detection assays by preventing non-specific reactions and improving signal detection, particularly in homogenous formats, without the need for additional enzymatic steps or solid phases.

Implementation Method 1

a silencing oligonucleotide which comprises first and second silencing regions which are complementary to the target-binding regions at the ends of the padlock probe

Methodology Applied
Scientific EffectHybridization:

Implementation Method 2

RCA is commonly used for such amplification, and is typically used in conjunction with padlock probes. RCA utilises a strand displacement polymerase enzyme, and requires a circular amplification template

Methodology Applied
Scientific EffectRolling circle amplification:

Implementation Method 3

the ends of the probe may be ligated together to circularise the probe

Methodology Applied
Scientific EffectLigation:

Data Source

PatentEP4590852B1Method of detection of a target nucleic acid sequence
Publication Date: 2026.04.22 READILY AB
  • EP4590852B1 patent drawingFigure 1
  • EP4590852B1 patent drawingFigure 2A~2C
  • EP4590852B1 patent drawingFigure 3

AI summary

The present invention provides a method for detecting a target nucleic acid molecule in a sample, using padlock probes and rolling circle amplification. The method herein provides a new way of removing free padlock probes which have failed to hybridise to their target, or to be ligated, and involves the use of a "silencing" oligonucleotide to "block" such unbound, or unligated, padlock probes.