SNP-Based Statin Response Prediction and Cardiovascular Risk Assessment

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Solution Overview

Problem

Current methods lack effective genetic markers to predict individual responsiveness to statins and identify those at risk for cardiovascular diseases such as coronary heart disease and stroke, leading to inadequate treatment and prevention strategies.

Innovation Solution

Identification of specific single nucleotide polymorphisms (SNPs) associated with variability in response to statins, which can be used to develop diagnostic and prognostic reagents and therapeutic agents for predicting individual responses to statin treatment and assessing cardiovascular disease risk.

Engineering Contradictions & Design Principles

VSEngineering Contradiction Analysis

1Measurement precision

If current methods are used for cardiovascular disease treatment and prevention, then general population approaches are applied, but individual responsiveness to statins cannot be predicted and treatment efficacy is insufficient

Engineering Contradiction:
Improveprediction accuracy of individual statin responseVSAvoidtreatment effectiveness
Core Design Contradiction:
Measurement precisionVSReliability

Solution Approach 1:

The invention segments the population into distinct genetic subgroups based on SNP profiles (e.g., CYP3A5*3 polymorphisms). By dividing the homogeneous treatment approach into heterogeneous genetically-defined groups, the patent enables precision medicine strategies where treatment decisions are tailored to individual genetic characteristics, thereby improving both measurement precision of response prediction and reliability of treatment outcomes

Inventive Principle:
Principle #1Segmentation

Solution Approach 2:

The invention changes the parameter used for treatment selection from general clinical factors to specific genetic parameters (SNP genotypes). By identifying and measuring specific genetic polymorphisms such as CYP3A5*3, the patent transforms the approach from empirical treatment to genetically-informed treatment, enhancing the ability to predict individual statin response and improve treatment effectiveness

Inventive Principle:
Principle #35Parameter changes

2Adaptability or versatility

If genetic markers are not used, then treatment decisions are made without genetic information, but personalized treatment approaches cannot be implemented

Engineering Contradiction:
Improvepersonalization of treatment approachVSAvoidgenetic information about individual risk and response
Core Design Contradiction:
Adaptability or versatilityVSLoss of information

Solution Approach 1:

The invention performs preliminary genetic testing to identify SNP profiles (such as CYP3A5*3 polymorphisms) before making treatment decisions. By obtaining genetic information in advance, the patent enables clinicians to adapt treatment approaches based on individual genetic characteristics, preventing the loss of valuable predictive information and allowing personalized medicine strategies to be implemented from the outset

Inventive Principle:
Principle #10Preliminary action

Solution Approach 2:

The invention introduces genetic markers (SNPs) as intermediary variables that mediate between statin treatment and clinical outcomes. These genetic markers serve as informative intermediaries that carry information about individual susceptibility and response, enabling the translation of genetic variation into actionable treatment decisions without directly measuring the complex biological pathways involved

Inventive Principle:
Principle #24Intermediary (Mediator)

3Reliability

If specific SNPs are identified for statin response prediction, then personalized treatment can be achieved, but additional diagnostic testing and genetic analysis are required

Engineering Contradiction:
Improveaccuracy of treatment response predictionVSAvoiddiagnostic testing requirements
Core Design Contradiction:
ReliabilityVSDevice complexity

Solution Approach 1:

The invention extracts and focuses on specific, high-value genetic markers (such as CYP3A5*3 polymorphisms) that have been shown to be strongly associated with statin response. By selecting and isolating these key SNPs rather than analyzing the entire genome or numerous low-value markers, the patent achieves reliable prediction of treatment response while minimizing diagnostic complexity and testing requirements

Inventive Principle:
Principle #2Taking out (Extraction)

Solution Approach 2:

The invention identifies SNPs that serve multiple functions: they predict statin response, indicate cardiovascular disease risk, and guide treatment selection. By finding genetic markers with multiple clinical applications, the patent reduces the need for separate diagnostic tests for different purposes, thereby improving prediction reliability without proportionally increasing diagnostic complexity

Inventive Principle:
Principle #6Universality (Multi-functionality)

Data Source

PatentUS11827937B2Genetic polymorphisms associated with statin response and cardiovascular diseases, methods of detection and uses thereof
Publication Date: 2023.11.28 CELERA CORP

AI summary

The present invention provides compositions and methods based on genetic polymorphisms that are associated with response to statin treatment, particularly for reducing the risk of cardiovascular disease, especially coronary heart disease (such as myocardial infarction) and stroke. For example, the present invention relates to nucleic acid molecules containing the polymorphisms, variant proteins encoded by these nucleic acid molecules, reagents and kits for detecting the polymorphic nucleic acid molecules and variant proteins, and methods of using the nucleic acid molecules and proteins as well as methods of using reagents and kits for their detection.