Spherical Cosmetic Particles Stabilizing Oxidation-Sensitive Actives

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Solution Overview

Problem

Current cosmetic and dermatological preparations face challenges in stabilizing oxidation-sensitive and UV-sensitive active ingredients, leading to limited effectiveness and potential skin irritation, particularly in addressing skin aging and photodermatoses, with existing antioxidants like vitamin E falling short in providing long-term protection against oxidative and UV-induced damage.

Innovation Solution

The development of cosmetic preparations containing ubiquinones and plastoquinones, combined with metal oxide pigments and light filter substances, encapsulated in a polymer matrix within spherical particles, which are protected against oxygen and UV radiation, maintaining their effectiveness over time and providing comprehensive skin care and light protection.

Engineering Contradictions & Design Principles

VSEngineering Contradiction Analysis

1Reliability

If oxidation-sensitive and UV-sensitive active ingredients are used in cosmetic preparations, then effectiveness in protecting against skin aging and photodermatoses is improved, but stability of the active ingredients deteriorates due to oxidation and UV degradation

Engineering Contradiction:
ImproveeffectivenessVSAvoidstability
Core Design Contradiction:
ReliabilityVSStability of the object's composition

Solution Approach 1:

The preparation is divided into an outer aqueous gel phase and an inner oily phase containing the active ingredients. This segmentation isolates the oxidation-sensitive and UV-sensitive active ingredients within the inner phase, protecting them from direct exposure to oxygen and UV radiation in the outer phase, thereby maintaining both effectiveness and stability.

Inventive Principle:
Principle #1Segmentation

Solution Approach 2:

The inner oily phase containing the active ingredients is nested within the outer aqueous gel phase. This nested structure provides an additional protective barrier, allowing the active ingredients to be encapsulated and protected from environmental factors while remaining accessible for skin absorption, thus resolving the contradiction between effectiveness and stability.

Inventive Principle:
Principle #7Nested doll (Nesting)

2Reliability

If antioxidants like vitamin E are used to protect against oxidative damage, then protection effectiveness is improved, but long-term stability against oxidation deteriorates

Engineering Contradiction:
Improveprotection effectivenessVSAvoidlong-term stability
Core Design Contradiction:
ReliabilityVSDuration of action of stationary object

Solution Approach 1:

The invention changes the physical and chemical parameters of the preparation system by creating a two-phase structure with different oxidation potentials. The inner oily phase acts as an oxidation-resistant compartment, extending the duration of action and long-term stability of the antioxidant active ingredients while maintaining their protection effectiveness.

Inventive Principle:
Principle #35Parameter changes

3Reliability

If light filter substances are added to protect against UV radiation, then light protection effectiveness is improved, but complexity of the formulation increases

Engineering Contradiction:
Improvelight protection effectivenessVSAvoidformulation complexity
Core Design Contradiction:
ReliabilityVSDevice complexity

Solution Approach 1:

The outer aqueous gel phase serves multiple functions: it acts as a vehicle for the preparation, provides a protective barrier against UV radiation, and maintains the stability of the inner phase. This multi-functionality reduces the need for additional separate light filter substances, thereby maintaining light protection effectiveness while minimizing formulation complexity.

Inventive Principle:
Principle #6Universality (Multi-functionality)

Applied Scientific Principles

This section explains which scientific principles are used to turn an abstract innovation direction into a practical engineering solution.

Function Achieved in This Case

These preparations effectively stabilize active ingredients, enhancing their longevity and efficacy, offering superior skin care and light protection while preventing oxidative and UV-induced damage, thus addressing the limitations of previous formulations.

Implementation Method 1

one or more light filter substances which is or are selected from the group of metal oxide pigments

Methodology Applied
Scientific EffectUV absorption: Absorption (EM radiation)

Implementation Method 2

essentially spherical particles... which comprise a polymer matrix which is essentially insoluble in water, one or more substances selected from the group of ubiquinones and/or plastoquinones

Methodology Applied
Scientific EffectPhysical containment: Physical Containment

Data Source

PatentEP2942045B1Bead-shaped cosmetic dosage forms
Publication Date: 2018.10.10 BEIERSDORF AG
  • EP2942045B1 patent drawingFigure 1a
  • EP2942045B1 patent drawingFigure 1b~1c
  • EP2942045B1 patent drawingFigure 1d

AI summary

Essentially spherical particles whose average diameter is selected from the range of 0.1 to 10 mm, preferably 2 to 7.5 mm, and which comprise: - a polymer matrix which is essentially insoluble in water, - one or more substances selected from the group of ubiquinones and/or plastoquinones, - one or more light filter substances which are or are selected from the group of metal oxide pigments, - optionally one or more light filter substances which are or are selected from the group of conventional cosmetic light protection filter substances.