Spray Dried Myrosinase Ascorbate Mixture for Isothiocyanate Production

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Solution Overview

Problem

The conversion of glucosinolates to isothiocyanates, such as sulforaphane, is inefficient due to the presence of epithiospecifier protein (ESP) which competes with the desired reaction pathway, resulting in reduced yield and purity of sulforaphane production.

Innovation Solution

A spray dried myrosinase/ascorbate mixture is created by heating a source of myrosinase with ascorbate to a temperature of about 40°C or higher, deactivating ESP and improving the stability and activity of myrosinase, which is then mixed with glucosinolates in water at a pH of 5 to 6.5 to enhance the conversion to sulforaphane.

Engineering Contradictions & Design Principles

VSEngineering Contradiction Analysis

1Productivity

If myrosinase is used to convert glucosinolates to isothiocyanates, then the chemoprotective effect is achieved, but the yield and purity are reduced due to competing reaction pathways catalyzed by ESP

Engineering Contradiction:
Improveyield of isothiocyanatesVSAvoidcompeting reaction products
Core Design Contradiction:
ProductivityVSObject-generated harmful factors

Solution Approach 1:

The patent removes the harmful ESP component from the reaction system by separating it from the myrosinase source (broccoli seeds) through controlled extraction and purification processes, allowing myrosinase to act without competing reaction pathways

Inventive Principle:
Principle #2Taking out (Extraction)

Solution Approach 2:

The patent creates optimal local conditions for myrosinase activity by controlling pH (using citrate buffer at pH 5.0), temperature (37°C water bath), and substrate concentration, while the competing ESP remains inactive under these specific conditions

Inventive Principle:
Principle #3Local quality

2Ease of operation

If plant material containing both myrosinase and glucosinolates is used, then the conversion can occur, but the presence of ESP reduces the efficiency and consistency of isothiocyanate production

Engineering Contradiction:
Improvesimplicity of processVSAvoidrate of conversion
Core Design Contradiction:
Ease of operationVSProductivity

Solution Approach 1:

The patent separates the myrosinase enzyme source from the glucosinolate substrate, processing broccoli seeds to extract and purify myrosinase independently, then combining it with glucoraphanin in controlled conditions to eliminate ESP interference

Inventive Principle:
Principle #1Segmentation

Solution Approach 2:

The patent performs preliminary extraction and purification of myrosinase from broccoli seeds before the conversion reaction, removing ESP and other interfering components in advance to ensure efficient and consistent isothiocyanate production

Inventive Principle:
Principle #10Preliminary action

Applied Scientific Principles

This section explains which scientific principles are used to turn an abstract innovation direction into a practical engineering solution.

Function Achieved in This Case

The process results in a more stable and active myrosinase/ascorbate mixture that increases the yield and rate of sulforaphane production, providing a consistent and potent chemoprotective agent.

Implementation Method 1

Myrosinase catalyzes the conversion of glucosinolates to isothiocyanates

Methodology Applied
Scientific EffectEnzyme catalysis: Enzyme

Implementation Method 2

Glucosinolates may be converted to isothiocyanates through the use of myrosinase enzymes

Methodology Applied
Scientific EffectHydrolysis: Hydrolysis

Implementation Method 3

heating the mixture in a solvent to a temperature of about 104° F. (about 40° C.) or higher, and spray drying the myrosinase/ascorbate mixture

Methodology Applied
Scientific EffectThermal deactivation: Heating

Implementation Method 4

spray drying the myrosinase/ascorbate mixture

Methodology Applied
Scientific EffectSpray drying: Evaporation

Data Source

PatentUS10925934B2Spray dried myrosinase and use to produce isothiocynates
Publication Date: 2021.02.23 CAUDILL SEED

AI summary

A spray dried myrosinase/ascorbate mixture is formed from the steps comprising: providing a source of myrosinase, adding ascorbate to the source of myrosinase, heating the source of myrosinase to a temperature of about 104° F. (about 40° C.) or higher, and spray drying the myrosinase/ascorbate mixture. The spray dried myrosinase/ascorbate mixture may be used to prepare isothiocyanates. The spray dried myrosinase/ascorbate mixture may also be mixed with glucoraphanin and used in an activated tablet or capsule.