Stabilized Calcium Phosphate with Pendant Polymerizable Groups

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Solution Overview

Problem

Existing calcium phosphate materials used in dental and biomedical applications face challenges such as instability in acidic conditions, limited mechanical strength, and poor compatibility with monomers, which restricts their use in load-bearing applications and restorative dentistry.

Innovation Solution

A method of forming stabilized calcium phosphate by reacting a calcium salt with an organic phosphate having a polymerizable methacrylate or vinyl group, such as bis[2-(methacryloyloxy)ethyl] phosphate, and an inorganic phosphate source, resulting in a calcium phosphate with pendant polymerizable groups that enhances stability and bioactivity, allowing integration with resin systems and improved mechanical properties.

Engineering Contradictions & Design Principles

VSEngineering Contradiction Analysis

1Reliability

If amorphous calcium phosphate is used in dental restorative materials, then it can release calcium and phosphate ions for remineralization, but it turns into hydroxyapatite when in contact with water, losing its stability

Engineering Contradiction:
ImprovestabilityVSAvoidchemical integrity
Core Design Contradiction:
ReliabilityVSStability of the object's composition

Solution Approach 1:

The patent creates a composite material consisting of calcium phosphate particles dispersed in a polymer matrix. The polymer component provides structural stability and prevents premature transformation of the amorphous calcium phosphate into hydroxyapatite, while still allowing controlled ion release for dental remineralization applications

Inventive Principle:
Principle #40Composite materials

Solution Approach 2:

The patent modifies the physical and chemical parameters of the calcium phosphate by controlling particle size, surface area, and dispersion characteristics within the polymer matrix. These parameter changes enhance stability while maintaining bioactivity and ion release capabilities

Inventive Principle:
Principle #35Parameter changes

2Stability of the object's composition

If crystalline hydroxyapatite is produced by high temperature sintering, then it achieves high crystallinity and structural stability, but it has limited solubility and reduced resorbability

Engineering Contradiction:
ImprovecrystallinityVSAvoidsolubility
Core Design Contradiction:
Stability of the object's compositionVSReliability

Solution Approach 1:

The patent produces calcium phosphate particles with controlled crystallinity through wet chemical methods rather than high-temperature sintering. By controlling parameters such as pH, temperature, and reaction time during synthesis, the patent achieves a balance between crystalline structure and solubility, enabling both stability and resorbability for biomedical applications

Inventive Principle:
Principle #35Parameter changes

Solution Approach 2:

The patent creates particles with heterogeneous internal structure, where the core maintains crystalline order for stability while the surface retains higher solubility characteristics. This local quality variation allows simultaneous achievement of structural integrity and controlled resorption in the body

Inventive Principle:
Principle #3Local quality

3Reliability

If calcium phosphate materials are used in load-bearing applications, then they provide good tissue compatibility, but they have limited mechanical strength

Engineering Contradiction:
Improvetissue compatibilityVSAvoidmechanical strength
Core Design Contradiction:
ReliabilityVSStrength

Solution Approach 1:

The patent develops composite materials combining calcium phosphate particles with polymer matrices or other reinforcing phases. This composite structure provides both the biocompatibility of calcium phosphate and enhanced mechanical strength from the polymer or reinforcement, making the material suitable for load-bearing biomedical applications

Inventive Principle:
Principle #40Composite materials

Solution Approach 2:

The patent creates porous calcium phosphate structures with controlled pore size and distribution. The porous architecture reduces overall density and can improve mechanical properties through optimized load distribution, while maintaining high surface area for bone ingrowth and tissue compatibility

Inventive Principle:
Principle #31Porous materials

Applied Scientific Principles

This section explains which scientific principles are used to turn an abstract innovation direction into a practical engineering solution.

Function Achieved in This Case

The stabilized calcium phosphate exhibits higher stability, mechanical strength, and bioactivity, enabling effective use in polymerizable resin systems, bioactive fillers for dental restoratives, and bone substitutes, with enhanced ion release and bone growth promotion.

Implementation Method 1

reacting a calcium salt with an organic phosphate having a polymerizable methacrylate or vinyl group

Methodology Applied
Scientific EffectChemical Bonding: Chemical Bonding

Implementation Method 2

organic phosphate having a polymerizable methacrylate or vinyl group

Methodology Applied
Scientific EffectPhotopolymerisation: Photopolymerisation

Data Source

PatentEP3265046B1Stabilized calcium phosphate and methods of forming same
Publication Date: 2024.09.04 MODERN IDEAS LLC
  • EP3265046B1 patent drawingFigure 1
  • EP3265046B1 patent drawingFigure 2
  • EP3265046B1 patent drawingFigure 3

AI summary

A method of forming a stabilized calcium phosphate moiety for use in dental or biomedical applications includes providing a solution or dispersion including a calcium salt and reacting an organic phosphate having a polymerizable methacrylate or vinyl group with the solution or dispersion in order to form the calcium phosphate moiety having at least one pendant polymerizable group and at least one organic functional group, which may be the same group. A polymerizable composite system having a stabilized calcium phosphate formed according to the method is also provided.