Synergistic Herbicidal Composition for Weed Control

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Solution Overview

Problem

Current herbicides are inadequate in effectively controlling undesirable vegetation in agriculture, as they often require multiple applications and can lead to herbicide resistance in weeds, necessitating the development of more potent and sustainable herbicidal compositions.

Innovation Solution

A synergistic herbicidal composition combining 4-amino-3-chloro-5-fluoro-6-(4-chloro-2-fluoro-3-methoxyphenyl)pyridine-2-carboxylic acid or its agriculturally acceptable ester/salt with very long chain fatty acid (VLCFA) and fatty acid/lipid synthesis inhibiting herbicides, such as acetochlor, alachlor, and others, to enhance weed control efficacy.

Engineering Contradictions & Design Principles

VSEngineering Contradiction Analysis

1Reliability

If current herbicides are used to control undesirable vegetation, then some weed control is achieved, but multiple applications are required and herbicide resistance develops

Engineering Contradiction:
Improveweed control efficacyVSAvoidnumber of applications required
Core Design Contradiction:
ReliabilityVSLoss of time

Solution Approach 1:

The patent combines compound (I) with a VLCFA synthesis-inhibiting herbicide or fatty acid/lipid synthesis-inhibiting herbicide to create a synergistic mixture. This combination achieves superior weed control efficacy compared to individual herbicides, reducing the need for multiple applications while delaying herbicide resistance development through multi-mode-of-action.

Inventive Principle:
Principle #5Merging (Combining)

2Reliability

If current herbicides are used to control undesirable vegetation, then some weed control is achieved, but herbicide resistance in weeds develops

Engineering Contradiction:
Improveweed control efficacyVSAvoidherbicide resistance
Core Design Contradiction:
ReliabilityVSAdaptability or versatility

Solution Approach 1:

The patent combines compound (I) with a VLCFA synthesis-inhibiting herbicide or fatty acid/lipid synthesis-inhibiting herbicide to create a synergistic mixture. This combination achieves superior weed control efficacy compared to individual herbicides, reducing the need for multiple applications while delaying herbicide resistance development through multi-mode-of-action.

Inventive Principle:
Principle #5Merging (Combining)

3Reliability

If compound (I) is combined with VLCFA and fatty acid/lipid synthesis inhibiting herbicides, then herbicidal activity increases, but composition complexity increases

Engineering Contradiction:
Improveherbicidal activityVSAvoidcomposition complexity
Core Design Contradiction:
ReliabilityVSDevice complexity

Solution Approach 1:

The patent combines compound (I) with a VLCFA synthesis-inhibiting herbicide or fatty acid/lipid synthesis-inhibiting herbicide to create a synergistic mixture. This combination achieves superior weed control efficacy compared to individual herbicides, reducing the need for multiple applications while delaying herbicide resistance development through multi-mode-of-action.

Inventive Principle:
Principle #5Merging (Combining)

Data Source

PatentEP2877008B1Herbicidal compositions comprising 4-amino-3-chloro-5-fluoro-6-(4-chloro-2-fluoro-3-methoxphenyl) pyridine-2-carboxylic acid or a derivative thereof and vlcfa synthesis and fatty acid/lipid synthesis inhibiting herbicides
Publication Date: 2019.01.02 DOW AGROSCIENCES LLC
  • EP2877008B1 patent drawing
  • EP2877008B1 patent drawing
  • EP2877008B1 patent drawing

AI summary

Provided herein are synergistic herbicidal compositions containing (a) a compound of formula (I): 4-amino-3-chloro-5-fluoro-6-(4-chloro-2-fluoro-3-methoxyphenyl)pyridine-2-carboxylic acid or a derivative thereof, or an agriculturally acceptable salt or ester thereof and (b) VLCFA and fatty acid/lipid synthesis inhibiting herbicides, including but not limited to, acetochlor, alachlor, anilofos, benfuresate, cafenstrole, dimethenamid-P, fenoxasulfone, fentrazamide, indanofan, flufenacet, mefenacet, s-metolachlor, molinate, pethoxamid, pretilachlor, prosulfocarb, pyroxasulfone, thenylchlor and thiobencarb, or a salt or ester thereof, provide synergistic weed control of undesirable vegetation in direct-seeded, water-seeded and transplanted rice, cereals, wheat, barley, oats, rye, sorghum, corn or maize, sugarcane, sunflower, oilseed rape, canola, sugar beet, soybean, cotton, pineapple, pastures, grasslands, rangelands, fallow land, turf, tree and vine orchards, aquatics, plantation crops, vegetables, industrial vegetation management (IVM) or rights-of-way (ROW).