Synthetic GPL Peptides for Specific Mycobacterium avium paratuberculosis Detection

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Solution Overview

Problem

Current diagnostic tests for Mycobacterium avium subsp. paratuberculosis (Map) infections face challenges due to cross-reacting antibodies from related mycobacteria, leading to non-specific reactions and the need for costly and time-consuming pre-absorption steps, and existing antigens used in skin tests and gamma-interferon assays produce false positives in young animals.

Innovation Solution

The use of synthetic peptides, such as DPhe-NMeVal-Ile-Phe-Ala-OMe and its derivatives, which mimic the lipopeptide Para-LP-01, for in vitro detection and quantification of specific anti-Map antibodies and T-cell immune responses, allowing for more specific and efficient diagnosis.

Engineering Contradictions & Design Principles

VSEngineering Contradiction Analysis

1Measurement precision

If crude fractions of mycobacteria are used as antigens in ELISA, then the detection sensitivity is improved, but false-positive reactions occur due to cross-reacting antibodies from related bacteria

Engineering Contradiction:
Improvedetection sensitivityVSAvoidspecificity
Core Design Contradiction:
Measurement precisionVSReliability

Solution Approach 1:

The patent segments the crude mycobacterial fraction into specific peptide components (GPL peptides with sequences like D-Phe-D-Allo-Thr-D-Ala-L-Alaninol) that are unique to Map. This segmentation allows the diagnostic test to target only Map-specific antigens rather than using whole crude extracts, thereby maintaining sensitivity while eliminating cross-reactivity with other mycobacteria.

Inventive Principle:
Principle #1Segmentation

Solution Approach 2:

The patent applies local quality by identifying and utilizing specific structural features of Map's GPL peptides (such as the particular amino acid sequence and lipid composition) that distinguish Map from other mycobacteria. By focusing on these localized unique characteristics rather than general mycobacterial components, the test achieves high specificity while maintaining detection sensitivity.

Inventive Principle:
Principle #3Local quality

2Reliability

If pre-absorption with crude fractions from M. phlei is performed to reduce cross-reacting antibodies, then the specificity of ELISA is improved, but the procedure becomes expensive and time-consuming

Engineering Contradiction:
ImprovespecificityVSAvoiddiagnostic procedure time
Core Design Contradiction:
ReliabilityVSLoss of time

Solution Approach 1:

The patent extracts and uses only the essential Map-specific GPL peptide antigens directly in the ELISA assay, eliminating the need for pre-absorption steps with M. phlei. By taking out only the necessary diagnostic components (Map-specific peptides) and removing unnecessary procedural steps (pre-absorption), the patent achieves high specificity while significantly reducing both time and cost.

Inventive Principle:
Principle #2Taking out (Extraction)

Solution Approach 2:

The patent performs preliminary identification and characterization of Map-specific GPL peptide sequences and structures, allowing these purified peptides to be used directly as antigens without requiring subsequent pre-absorption steps. This preliminary characterization enables the elimination of time-consuming pre-absorption procedures while maintaining diagnostic specificity.

Inventive Principle:
Principle #10Preliminary action

3Measurement precision

If avian or Johnin PPD antigens are used in skin tests and gamma-interferon assays, then the detection of T-cell-mediated immune response is improved, but non-specific reactions occur in young animals

Engineering Contradiction:
Improveimmune response detectionVSAvoidspecificity in young animals
Core Design Contradiction:
Measurement precisionVSReliability

Solution Approach 1:

The patent segments the conventional PPD antigen into specific Map-derived GPL peptides (such as the tetrapeptide or pentapeptide sequences). This segmentation allows the immune assay to detect T-cell responses specific to Map infection rather than general mycobacterial exposure, thereby eliminating non-specific reactions in young animals while maintaining detection sensitivity for Map-specific immunity.

Inventive Principle:
Principle #1Segmentation

Solution Approach 2:

The patent changes the antigenic parameter from conventional PPD (a mixture of mycobacterial proteins) to specific Map-derived GPL peptides with defined sequences and lipid compositions. This parameter change ensures that the antigen specifically recognizes Map-specific T-cell responses, eliminating cross-reactivity with other mycobacteria in young animals while maintaining the ability to detect Map-induced immunity.

Inventive Principle:
Principle #35Parameter changes

Data Source

PatentEP3406261B1Synthetic antigenic peptides and lipopeptides derived from mycobacterium avium subsp. paratuberculosis
Publication Date: 2024.08.21 INST PASTEUR
  • EP3406261B1 patent drawingFigure 1A~1B
  • EP3406261B1 patent drawingFigure 2
  • EP3406261B1 patent drawingFigure 3

AI summary

The invention relates to synthetic pentapeptides and lipopentapeptides and to their use for the diagnosis and treatment of diseases resulting from infections by Mycobacterium avium subsp. paratuberculosis .