Antigen-Specific T Cell Generation via Allogeneic MHC Co-Transfection

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Solution Overview

Problem

Current adoptive cell therapies for treating solid tumors face challenges such as the slow activation and expansion of specific T cells, risk of graft-versus-host disease, and inefficacy in rapidly progressing tumors due to limitations in generating T cells with high functional avidity that can recognize tumor-specific MHC-peptide ligands without attacking normal tissues.

Innovation Solution

The method involves co-transfecting dendritic cells with RNA encoding allogeneic MHC molecules and tumor-associated antigens to prime peripheral blood lymphocytes, allowing for the selection and expansion of antigen-specific CD4+ and CD8+ T cells with high affinity TCRs, which can be used to treat solid tumors without the risk of graft-versus-host disease.

Engineering Contradictions & Design Principles

VSEngineering Contradiction Analysis

1Productivity

If unselected lymphocyte populations are transferred in donor lymphocyte infusions, then the elimination of malignant cells can occur, but the activation and expansion of specific T cells takes several months up to a year

Engineering Contradiction:
Improvetumor cell elimination rateVSAvoidT cell activation time
Core Design Contradiction:
ProductivityVSLoss of time

Solution Approach 1:

The patent applies preliminary action by pre-activating and expanding tumor-specific T cells ex vivo before transfer to the patient. T cells are stimulated with antigen-presenting cells and cytokines in culture to generate large numbers of activated, tumor-specific effector cells that can immediately attack tumor cells upon infusion, eliminating the months-long in vivo activation period required by conventional DLI approaches.

Inventive Principle:
Principle #10Preliminary action

2Productivity

If unselected lymphocyte populations are transferred to speed up immune response, then T cells can be expanded faster, but the risk of graft-versus-host disease increases

Engineering Contradiction:
Improveimmune response speedVSAvoidgraft-versus-host disease risk
Core Design Contradiction:
ProductivityVSObject-affected harmful factors

Solution Approach 1:

The patent applies the extraction principle by isolating and selecting only the tumor-specific T cell subset from the total lymphocyte population through antigen-specific stimulation and expansion. This enriches the transferred cell product for cytotoxic T cells with defined tumor reactivity while removing or minimizing regulatory T cells and other lymphocyte subsets that could mediate graft-versus-host disease, thereby achieving rapid antitumor immunity with reduced toxicity.

Inventive Principle:
Principle #2Taking out (Extraction)

3Productivity

If T cells with high affinity TCRs are generated to effectively target tumor cells, then tumor eradication is more effective, but the risk of attacking normal tissues increases

Engineering Contradiction:
Improvetumor eradication effectivenessVSAvoidnormal tissue attack
Core Design Contradiction:
ProductivityVSObject-affected harmful factors

Solution Approach 1:

The patent applies local quality by generating T cell populations with heterogeneous TCR affinities rather than uniformly high-affinity clones. The antigen-specific expansion process naturally selects for cells with appropriate affinity ranges, and the polyclonal nature of the product ensures diverse target recognition. This allows effective tumor cell killing while reducing the risk of autoimmunity compared to highly purified single clones with extremely high affinity.

Inventive Principle:
Principle #3Local quality

Solution Approach 2:

The patent applies partial action by transferring a polyclonal population of antigen-specific T cells rather than maximizing the frequency of the single most effective clone. This approach achieves sufficient antitumor activity through the combined effect of multiple T cell clones with different specificities and affinities, while maintaining safety through the dilution effect and presence of regulatory cells within the polyclonal mixture.

Inventive Principle:
Principle #16Partial or excessive action

4Object-affected harmful factors

If stem cell transplantation is performed to establish tolerance before T cell transfer, then graft-versus-host disease is reduced, but the treatment time and complexity increase

Engineering Contradiction:
Improvegraft-versus-host diseaseVSAvoidtreatment protocol complexity
Core Design Contradiction:
Object-affected harmful factorsVSDevice complexity

Solution Approach 1:

The patent applies the intermediary principle by using antigen-specific T cell expansion as a bridge between bone marrow transplantation and tumor therapy. The method generates tumor-specific effector cells ex vivo that can be transferred after standard bone marrow recovery, serving as an intermediary step that provides targeted antitumor immunity without requiring complex protocols to induce tolerance. The antigen-specific nature of the cells inherently limits their reactivity to host tissues.

Inventive Principle:
Principle #24Intermediary (Mediator)

Data Source

PatentEP2327763B1Generation of antigen specific T cells
Publication Date: 2018.03.14 HELMHOLTZ ZENT MUENCHEN DEUT FORSCHUNGSZENTRUM FUER GESUNDHEIT & UMWELT (GMBH)
  • EP2327763B1 patent drawingFigure 1
  • EP2327763B1 patent drawingFigure 2
  • EP2327763B1 patent drawingFigure 3a

AI summary

The present invention is directed to a method of generating antigen specific T cells. Furthermore, the invention is directed to antigen specific T cells, isolated transgenic TCR's, pharmaceutical compositions containing same and their use in adoptive cell therapy. This invention in particular pertains to the use of cells co-expressing allogeneic MHC molecules and antigens to induce peptide-specific T cells from non-selected allogeneic T cell repertoires.