Tau Biosensor CRISPR Screening for Genetic Modifier Detection

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Solution Overview

Problem

Current methods for identifying genetic modifiers of tau aggregation are limited in sensitivity and specificity, hindering the understanding of neurodegenerative diseases and therapeutic intervention.

Innovation Solution

A CRISPR-based screening platform is developed, utilizing FRET pairs and flow cytometry to identify genetic modifiers by culturing cells with a tau seeding agent, forming aggregates, and analyzing guide RNA abundance to determine gene disruption or activation effects on tau aggregation.

Engineering Contradictions & Design Principles

VSEngineering Contradiction Analysis

1Measurement precision

If CRISPR interference (CRISPRi) is used to knock down target genes, then gene expression is reduced, but the method lacks sensitivity and specificity in identifying genetic modifiers of tau aggregation

Engineering Contradiction:
Improveidentification accuracy of genetic modifiersVSAvoidsensitivity and specificity of screening
Core Design Contradiction:
Measurement precisionVSReliability

Solution Approach 1:

The patent introduces FRET-based biosensors as intermediaries between gene disruption and aggregation detection. The biosensors convert molecular interactions into optical signals, enabling precise measurement of tau aggregation in response to CRISPR-mediated gene disruption, thereby improving identification accuracy while maintaining screening reliability

Inventive Principle:
Principle #24Intermediary (Mediator)

Solution Approach 2:

The patent replaces traditional mechanical or chemical detection methods with optical detection using FRET (fluorescence resonance energy transfer). This substitution enables non-invasive, real-time monitoring of tau aggregation with high sensitivity and specificity, resolving the contradiction between measurement precision and screening reliability

Inventive Principle:
Principle #28Mechanics substitution (Replace mechanical system)

2Measurement precision

If FACS screening is used to detect intracellular tau aggregates, then aggregation can be detected, but the method requires cell membrane perforation which reduces cell viability and measurement accuracy

Engineering Contradiction:
Improveaggregation detection accuracyVSAvoidcell membrane damage
Core Design Contradiction:
Measurement precisionVSObject-affected harmful factors

Solution Approach 1:

The patent uses FRET-based biosensors as intermediaries that can detect tau aggregation through intact cell membranes. The optical signals generated by FRET allow aggregation detection without requiring membrane perforation, thereby eliminating cell damage while maintaining detection accuracy

Inventive Principle:
Principle #24Intermediary (Mediator)

Solution Approach 2:

The patent substitutes mechanical membrane perforation with optical detection methods. FRET-based fluorescence microscopy or flow cytometry can detect aggregation through live cells without physical disruption, replacing the harmful mechanical intervention with a non-invasive optical measurement

Inventive Principle:
Principle #28Mechanics substitution (Replace mechanical system)

3Adaptability or versatility

If genome-wide CRISPR screening is performed to identify genetic modifiers, then comprehensive gene coverage is achieved, but the complexity of the platform increases

Engineering Contradiction:
Improvegenome-wide screening capabilityVSAvoidscreening platform complexity
Core Design Contradiction:
Adaptability or versatilityVSDevice complexity

Solution Approach 1:

The patent creates a universal FRET-based biosensor platform that can be applied across genome-wide CRISPR screens. The biosensors are designed to work with various CRISPR methods (knockout, knockdown, activation) and can detect tau aggregation in multiple cell types, providing multi-functionality that simplifies the overall screening platform while maintaining genome-wide coverage capability

Inventive Principle:
Principle #6Universality (Multi-functionality)

Applied Scientific Principles

This section explains which scientific principles are used to turn an abstract innovation direction into a practical engineering solution.

Function Achieved in This Case

The platform effectively identifies genes that prevent or enhance tau aggregation, providing insights into disease progression and potential therapeutic targets.

Implementation Method 1

the first reporter and the second reporter are fluorescent proteins, wherein the first reporter and the second reporter are a fluorescence resonance energy transfer (FRET) pair

Methodology Applied
Scientific EffectFluorescence resonance energy transfer (FRET):

Implementation Method 2

the aggregation-positive population of cells and the aggregation-negative population of cells in step (e) is identified by flow cytometry

Methodology Applied
Scientific EffectFlow cytometry detection:

Data Source

PatentEP4317950B1Crispr/cas screening platform to identify genetic modifiers of tau seeding or aggregation
Publication Date: 2026.01.28 REGENERON PHARMACEUTICALS INC
  • EP4317950B1 patent drawingFigure 1~2
  • EP4317950B1 patent drawingFigure 3A
  • EP4317950B1 patent drawingFigure 3B

AI summary

Cas-protein-ready tau biosensor cells, CRISPR/Cas synergistic activation mediator (SAM)-ready tau biosensor cells, and methods of making and using such cells to screen for genetic modifiers of tau seeding or aggregation are provided. Reagents and methods for sensitizing such cells to tau seeding activity or tau aggregation or for causing tau aggregation are also provided.