TCR Antigen Identification via Combinatorial Barcoding

Resolve Bottlenecks,
Find Innovative Solutions
Generate Solutions

Solution Overview

Problem

Current methods are inefficient in identifying the specific antigen recognized by T-cell receptors, particularly for 'orphan' TCRs, which hinders the development of cancer immunotherapy and autoimmunity treatments, as they require large cell numbers and empirical testing.

Innovation Solution

A method involving combinatorial barcoding of T-cells and tumor neoantigens, where TCRα and TCRβ genes are barcoded, and their cognate antigens identified by sequencing and forming barcoded MHC-neoantigen complexes to match with TCRs, allowing for the identification of cognate antigens through shared cell-specific barcodes.

Engineering Contradictions & Design Principles

VSEngineering Contradiction Analysis

1Measurement precision

If mass spectrometry is used for antigen isolation, then unbiased antigen identification is achieved, but large cell numbers (10^7) are required

Engineering Contradiction:
Improveantigen identification accuracyVSAvoidcell number
Core Design Contradiction:
Measurement precisionVSQuantity of substance

Solution Approach 1:

The patent segments the antigen identification process into multiple steps: T-cell isolation, TCR sequencing, neoantigen prediction, and matching. This segmentation allows the use of fewer cells (10^3-10^6) by focusing on specific T-cell populations and their receptors rather than requiring large numbers for bulk analysis.

Inventive Principle:
Principle #1Segmentation

Solution Approach 2:

The patent introduces TCR sequencing and bioinformatic matching as intermediary steps between T-cell isolation and antigen identification. These intermediaries enable the identification of antigen specificity from limited T-cell samples by characterizing the TCR repertoire and matching it with predicted neoantigens.

Inventive Principle:
Principle #24Intermediary (Mediator)

2Measurement precision

If pHLA multimers are used to query T-cell specificities, then established T-cell specificities can be identified, but the method is limited to known antigens and requires empirical testing

Engineering Contradiction:
ImproveT-cell specificity identificationVSAvoidempirical testing requirements
Core Design Contradiction:
Measurement precisionVSDevice complexity

Solution Approach 1:

The patent performs preliminary bioinformatic analysis to predict neoantigens from tumor sequencing data before experimental validation. This preliminary action identifies candidate antigens in silico, reducing the need for extensive empirical testing with pHLA multimers and enabling the study of previously unknown tumor antigens.

Inventive Principle:
Principle #10Preliminary action

Solution Approach 2:

The patent replaces the mechanical/physical approach of pHLA multimer binding assays with a bioinformatic approach: sequencing TCRs, predicting neoantigens from tumor genomes, and using computational algorithms to match TCRs with their cognate antigens. This substitution eliminates the need for empirical testing with known antigens.

Inventive Principle:
Principle #28Mechanics substitution (Replace mechanical system)

3Measurement precision

If combinatorial barcoding is implemented, then TCR-antigen matching precision is improved, but the process complexity increases

Engineering Contradiction:
ImproveTCR-antigen matching accuracyVSAvoidbarcoding process complexity
Core Design Contradiction:
Measurement precisionVSDevice complexity

Solution Approach 1:

The patent uses combinatorial barcoding to create molecular copies of TCR sequences and neoantigen sequences with unique identifier tags. These barcoded copies allow high-throughput tracking and matching of TCR-antigen pairs through sequencing, achieving precise matching while automating the process to manage the complexity.

Inventive Principle:
Principle #26Copying

Data Source

PatentEP3807636B1A system for identification of antigens recognized by t cell receptors expressed on tumor infiltrating lymphocytes
Publication Date: 2024.01.31 F HOFFMANN LA ROCHE & CO AG
  • EP3807636B1 patent drawingFigure 1
  • EP3807636B1 patent drawingFigure 2
  • EP3807636B1 patent drawingFigure 2

AI summary

The invention is a method of identifying a cognate antigen for a T-cell receptor using neoantigens from a patient's tumor cells combined with the patient's T-cells and using cell sorting, genome sequencing, expressing TCR genes, presenting tumor neoantigens on MHC complex and uniquely barcoding the T-cells where TCR recognition occurs to tag all components of the TCR recognition complex.