TDP-43 Transgenic Mouse Model for FTLD-U Pathogenesis

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Solution Overview

Problem

The causative role of TDP-43 in the pathogenesis of frontotemporal lobar degeneration with ubiquitin-positive inclusions (FTLD-U) remains undefined, and existing models do not adequately address the molecular and cellular properties of TDP-43 in neurodegenerative diseases.

Innovation Solution

A transgenic mouse model with increased expression of TDP-43 in the hippocampus and cortex, but not the cerebellum and spinal cord, using a CaMKIIα promoter, which mimics the phenotypic characteristics of FTLD-U, including impaired learning and motor functions, and exhibits TDP-43 protein inclusion bodies.

Engineering Contradictions & Design Principles

VSEngineering Contradiction Analysis

1Reliability

If TDP-43 is overexpressed in the central nervous system using a Thy-1 promoter, then neuronal aggregates containing ubiquitinated TDP-43 are formed, but the model also causes degeneration of motor neurons and nonmotor cortical neurons, leading to spastic quadriplegia and FTLD-like symptoms

Engineering Contradiction:
Improvemodel reliability for studying TDP-43 pathogenesisVSAvoidneuronal degeneration and spastic quadriplegia
Core Design Contradiction:
ReliabilityVSObject-affected harmful factors

Solution Approach 1:

The patent uses the CaMKIIα promoter to achieve region-specific overexpression of TDP-43 in forebrain neurons (cortex and hippocampus) while avoiding expression in spinal cord and cerebellum. This local quality approach allows the model to study FTLD-U pathology without causing the widespread neuronal degeneration and spastic quadriplegia seen in Thy-1 promoter models, thereby reducing harmful effects while maintaining model reliability for forebrain-specific pathogenesis studies

Inventive Principle:
Principle #3Local quality

2Manufacturing precision

If TDP-43 is overexpressed to form cytoplasmic inclusion bodies, then the model mimics FTLD-U pathological features, but the causative role of TDP-43 in FTLD-U pathogenesis remains undefined

Engineering Contradiction:
Improvepathological feature accuracyVSAvoidcausative role definition
Core Design Contradiction:
Manufacturing precisionVSReliability

Solution Approach 1:

The patent segments the expression pattern of TDP-43 to match the regional distribution observed in FTLD-U patients (forebrain-specific expression in cortex and hippocampus). This segmentation allows the model to accurately reproduce FTLD-U pathological features including cytoplasmic inclusion bodies and TDP-43 depleted nuclei in forebrain regions, while avoiding expression in spinal cord and cerebellum, thereby providing a more reliable model for defining the causative role of TDP-43 in FTLD-U specifically

Inventive Principle:
Principle #1Segmentation

3Adaptability or versatility

If a transgenic model is created to study TDP-43 in FTLD-U, then valuable tools for mechanistic analysis are provided, but existing models do not adequately address the molecular and cellular properties of TDP-43 in neurodegenerative diseases

Engineering Contradiction:
Improvemodel utility for therapeutic developmentVSAvoidmolecular and cellular property representation
Core Design Contradiction:
Adaptability or versatilityVSReliability

Solution Approach 1:

The patent changes the expression parameters of TDP-43 by using the CaMKIIα promoter to achieve forebrain-specific overexpression (2-3 fold increase) in cortex and hippocampus, matching the molecular and cellular properties observed in FTLD-U patients. This parameter change approach provides a reliable model that accurately represents TDP-43 pathology in the most affected brain regions, enabling versatile applications in mechanistic analysis and therapeutic development while maintaining fidelity to human disease characteristics

Inventive Principle:
Principle #35Parameter changes

Data Source

PatentEP2258857B1TDP-43 transgenic mouse model for frontotemporal lobar degeneration with ubiquitin-positive inclusions (FTLD-U)
Publication Date: 2015.04.29 ACAD SINICA
  • EP2258857B1 patent drawingFigure 1A~1E
  • EP2258857B1 patent drawingFigure 2A~2F
  • EP2258857B1 patent drawingFigure 3A~3B

AI summary

Non-human animal models for frontotemporal lobar degeneration with ubiquitin-positive inclusions (FTLD-U) are disclosed. The invention relates to a transgenic mouse whose genome comprises a transgene operably linked to a neuronal specific promoter effective for an increased expression of the transgene in the brain of the mouse, in which the transgene comprises a nucleotide sequence encoding TAR DNA-binding protein 43 (TDP-43). The transgenic mouse exhibits reduced or impaired learning and memory capacity, and may further exhibits progressively impaired or reduced motor functions. Methods of using such animal models are also disclosed.