Topical Formulations for STD Prevention via Film-Forming Excipients

Resolve Bottlenecks,
Find Innovative Solutions
Generate Solutions

Solution Overview

Problem

Current topical formulations for preventing sexually transmitted diseases (STDs) often cause irritation and are not effective in providing a physical barrier against pathogen transmission, especially when used in conjunction with condoms.

Innovation Solution

The development of non-irritating topical protective formulations that utilize a combination of film-forming excipients, including skin protectants like zinc oxide, glycerin, lanolin, and silicone derivatives, to create a persistent hydrophobic barrier on the skin, inhibiting the penetration of pathogens.

Engineering Contradictions & Design Principles

VSEngineering Contradiction Analysis

1Reliability

If chemical actives such as nonoxynol-9 are used in topical formulations to reduce STD transmission, then the rate of STD transmission is reduced, but local irritation, inflammation, and ulcerations are induced which may favor STD transmission

Engineering Contradiction:
ImproveSTD transmission preventionVSAvoidlocal irritation and inflammation
Core Design Contradiction:
ReliabilityVSObject-affected harmful factors

Solution Approach 1:

The patent removes harmful chemical actives (nonoxynol-9, benzalkonium chloride, povidone-iodine) from the formulation while retaining the protective barrier function through film-forming excipients alone, thereby eliminating irritation while maintaining STD prevention capability

Inventive Principle:
Principle #2Taking out (Extraction)

Solution Approach 2:

The patent converts the previously harmful approach of using chemical microbicides into a beneficial physical barrier approach using only film-forming excipients, where the barrier property itself becomes the protective mechanism without chemical irritation

Inventive Principle:
Principle #22Blessing in disguise (Convert harm into benefit)

2Reliability

If chemical microbicides are used to provide protection against STDs, then STD transmission is reduced, but the formulations cause skin irritation and ulcerations

Engineering Contradiction:
Improveprotection against STDsVSAvoidskin irritation and ulcerations
Core Design Contradiction:
ReliabilityVSObject-generated harmful factors

Solution Approach 1:

The patent extracts and removes all chemical microbicide components from the formulation, relying solely on the physical barrier properties of film-forming excipients to provide protection, thereby eliminating the source of skin irritation and ulcerations

Inventive Principle:
Principle #2Taking out (Extraction)

Solution Approach 2:

The patent uses film-forming excipients as an intermediary physical barrier between the pathogen and the skin, replacing the need for chemical microbicides and eliminating their harmful side effects while maintaining protective function

Inventive Principle:
Principle #24Intermediary (Mediator)

3Reliability

If prior art formulations are used, then chemical active ingredients are present, but none provide a physical barrier to pathogen permeation without causing irritation

Engineering Contradiction:
Improvepathogen transmission inhibitionVSAvoidskin irritation
Core Design Contradiction:
ReliabilityVSObject-affected harmful factors

Solution Approach 1:

The patent employs film-forming excipients that create a flexible physical barrier film on the skin surface, providing a non-irritating yet effective shield against pathogen permeation, contrasting with prior art that relied on chemical actives without such physical barrier properties

Inventive Principle:
Principle #30Flexible shells and thin films

Applied Scientific Principles

This section explains which scientific principles are used to turn an abstract innovation direction into a practical engineering solution.

Function Achieved in This Case

These formulations effectively prevent the transmission of STDs by forming a durable, non-irritating physical barrier on the skin, providing enhanced protection against viral, bacterial, and fungal pathogens, even when used in combination with condoms.

Implementation Method 1

The products of the present invention are persistent in that they form a film or barrier on healthy or even damaged skin... This forms a physical hydrophobic layer, which resides on the skin surface (including mucosal membranes) and provides a barrier, which would inhibit penetration of liquids, and pathogens

Methodology Applied
Scientific EffectHydrophobic barrier formation: Hydrophobe

Implementation Method 2

They liquefy and spread over the skin as a result of exposure to body heat. This forms a physical hydrophobic layer, which resides on the skin surface (including mucosal membranes) and provides a barrier, which would inhibit penetration of liquids, and pathogens

Methodology Applied
Scientific EffectPhysical containment: Physical Containment

Data Source

PatentEP2644193B1Topical formulations for the prevention of sexually transmitted disease and methods of producing the same
Publication Date: 2014.10.08 CLJI IP COMPANY LLC

AI summary

The present invention is directed towards various topical protective formulations, which may be used as an adjunct in preventing the spread of a broad range of sexually transmitted diseases. The product is intended to be used as a topical lotion, cream, emulsion, or the like. The film forming excipients and active ingredients in the following formulations have demonstrated unique skin protective barrier properties with enhanced persistence that inhibits transmission of sexually transmitted diseases.