Triple Epitope Tag Sequences for Antibody Fragment Detection

Resolve Bottlenecks,
Find Innovative Solutions
Generate Solutions

Solution Overview

Problem

Existing epitope tag combinations are often inaccessible due to protein secondary and tertiary structures, and can alter protein expression and stability in display systems, limiting detection, capture, and purification of antibody fragments like single chain antibodies and Fab fragments.

Innovation Solution

A novel triple tag sequence comprising a 6X histidine tag, a c-myc tag positioned between the 6X histidine and V5 tag, which remains accessible for antibody binding, allowing for efficient detection, capture, and purification of proteins of interest without affecting their expression or display in libraries.

Engineering Contradictions & Design Principles

VSEngineering Contradiction Analysis

1Reliability

If epitope tags are inserted into proteins for detection and purification, then detection and purification capability is improved, but tag accessibility is reduced due to protein secondary and tertiary structures

Engineering Contradiction:
Improvedetection and purification capabilityVSAvoidtag accessibility
Core Design Contradiction:
ReliabilityVSDifficulty of detecting and measuring

Solution Approach 1:

The invention divides the tagging function into multiple separate epitope tags (V5, c-myc, 6X histidine) positioned at different locations on the protein. This segmentation ensures that at least one tag remains accessible for detection and purification even if others are buried in protein structure, resolving the contradiction between detection capability and tag accessibility.

Inventive Principle:
Principle #1Segmentation

2Reliability

If multiple epitope tags are added to proteins for enhanced detection, then detection capability is improved, but protein expression and stability are altered

Engineering Contradiction:
Improvedetection capabilityVSAvoidprotein expression and stability
Core Design Contradiction:
ReliabilityVSStability of the object's composition

Solution Approach 1:

The invention applies different types of epitope tags (V5, c-myc, 6X histidine) with distinct properties at different positions on the protein. Each tag has been selected for its specific binding characteristics and minimal interference with protein folding and stability, allowing enhanced detection capability while maintaining protein expression and stability.

Inventive Principle:
Principle #3Local quality

3Productivity

If antibody fragments like scFv and Fab are captured using Fc region reagents, then capture efficiency is improved, but capture is precluded for fragments lacking Fc domains

Engineering Contradiction:
Improvecapture efficiencyVSAvoidcapture applicability to different antibody fragments
Core Design Contradiction:
ProductivityVSAdaptability or versatility

Solution Approach 1:

The invention creates a universal tagging system that can be applied to all antibody fragments regardless of their class or presence of Fc domains. The multiple epitope tags (V5, c-myc, 6X histidine) provide universal capture handles that work with scFv, Fab, and other fragments lacking Fc regions, greatly expanding the versatility of capture methods while maintaining efficiency.

Inventive Principle:
Principle #6Universality (Multi-functionality)

4Reliability

If Fab fragments are captured using anti-Fab antibodies, then capture capability is improved, but antigen binding is interfered with

Engineering Contradiction:
Improvecapture capabilityVSAvoidinterference with antigen binding
Core Design Contradiction:
ReliabilityVSObject-generated harmful factors

Solution Approach 1:

The invention extracts the capture function from the antibody-antigen binding site by using separate epitope tags (V5, c-myc, 6X histidine) that are distinct from the antigen-binding Fab region. This allows capture of Fab fragments using anti-tag antibodies without interfering with the intact antigen-binding capability of the Fab region.

Inventive Principle:
Principle #2Taking out (Extraction)

Data Source

PatentEP2344686B1Novel triple tag sequences and methods of use thereof
Publication Date: 2014.03.05 XOMA TECHNOLOGY LTD(US)
  • EP2344686B1 patent drawingFigure 1
  • EP2344686B1 patent drawingFigure 2
  • EP2344686B1 patent drawingFigure 3

AI summary

The present disclosure relates to novel triple tag sequences that may comprise a 6X histidine tag, a c-myc tag and a V5 tag. The present disclosure also provides polynucleotides, proteins, vectors and host cells that comprise the triple tag sequence of the present disclosure, including libraries of such polynucleotides, proteins, vectors and host cells. The novel triple tag sequences of the present disclosure may be used in phage display vectors and phage libraries and in methods for detection, screening, capture, purification, quantitation, and/or recovery of proteins of interest to which they are linked. Proteins of interest include antibodies such as single chain antibodies, single chain antibodies, and Fab fragments of antibodies or peptides such as non-antibody peptides.