tRNA-Enhanced Lipofection for Mammalian Gene Transfer

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Solution Overview

Problem

Current gene transfer methods to mammalian cells, such as the lipofection method, face inefficiencies compared to virus vector methods, and existing methods do not effectively utilize tRNA for enhancing gene transfer efficiency.

Innovation Solution

Combining tRNA with a lipofection reagent, specifically using yeast-derived, calf liver-derived, wheat germ-derived, or E. coli-derived tRNA, at concentrations ranging from 3 to 50 µg/mL, along with polyethylene glycol of molecular weights between 2,000 to 6,000, to improve gene transfer efficiency in mammalian cells.

Engineering Contradictions & Design Principles

VSEngineering Contradiction Analysis

1Ease of operation

If the lipofection method is used for gene transfer to mammalian cells, then the method is simple and versatile, but the gene transfer efficiency is inferior to virus vector methods

Engineering Contradiction:
ImprovesimplicityVSAvoidgene transfer efficiency
Core Design Contradiction:
Ease of operationVSProductivity

Solution Approach 1:

The patent changes the chemical parameters of the lipofection system by introducing tRNA as a co-transfectant agent. This parameter change transforms the lipofection method from a simple but inefficient process to an enhanced system that achieves virus-vector-like efficiency while maintaining operational simplicity. The tRNA component modifies the interaction between liposome and DNA, improving uptake efficiency without complicating the basic procedure.

Inventive Principle:
Principle #35Parameter changes

Solution Approach 2:

The patent creates a composite transfection system combining lipofection reagents with tRNA. This composite approach merges the simplicity of lipofection with the high efficiency of virus vector methods. The tRNA acts as an auxiliary agent that enhances the liposome-DNA complex interaction, creating a synergistic effect that achieves both ease of operation and high productivity.

Inventive Principle:
Principle #40Composite materials

2Productivity

If virus vector methods are used for gene transfer, then gene transfer efficiency is high, but the process is time-consuming and requires specialized facilities and personnel

Engineering Contradiction:
Improvegene transfer efficiencyVSAvoidtime for virus production
Core Design Contradiction:
ProductivityVSLoss of time

Solution Approach 1:

The patent extracts the essential function of virus vectors (high efficiency gene transfer) while removing the time-consuming and complex components (virus production, specialized facilities, skilled personnel). By using tRNA-enhanced lipofection, the method achieves virus-like efficiency without requiring virus cultivation time or specialized containment facilities, thus separating the beneficial outcome from the cumbersome process.

Inventive Principle:
Principle #2Taking out (Extraction)

Solution Approach 2:

The patent replaces complex, time-consuming virus vector systems with a simpler, faster lipofection-based system using tRNA. This approach uses readily available reagents and cells, eliminating the need for expensive virus production infrastructure and specialized personnel, while achieving comparable or superior gene transfer efficiency in a fraction of the time.

Inventive Principle:
Principle #27Cheap short-living objects (Disposable)

3Productivity

If tRNA is added to lipofection solution, then gene transfer efficiency is significantly improved, but the complexity of the procedure increases

Engineering Contradiction:
Improvegene transfer efficiencyVSAvoidprocedure complexity
Core Design Contradiction:
ProductivityVSDevice complexity

Solution Approach 1:

The patent merges tRNA with the lipofection reagent in a single combined solution, treating the enhancement agent as an integral part of the transfection system. This merging approach simplifies the procedure by eliminating separate addition steps and ensuring proper mixing, while maintaining the efficiency boost. The tRNA is incorporated into the liposome-DNA complex formation process itself, rather than being added as a separate subsequent step.

Inventive Principle:
Principle #5Merging (Combining)

Applied Scientific Principles

This section explains which scientific principles are used to turn an abstract innovation direction into a practical engineering solution.

Function Achieved in This Case

This combination significantly enhances gene transfer efficiency, as demonstrated by up to 58-fold increases in luciferase activity assays, indicating effective gene incorporation into mammalian cells.

Implementation Method 1

The lipofection method is a method which involves forming a liposome-DNA complex by the electric interaction between a lipid bilayer membrane vesicle consisting of a positively charged lipid or the like (liposome) and DNA to be transferred and incorporating the complex into host cells by phagocytosis or membrane fusion.

Methodology Applied
Scientific EffectLipofection:

Implementation Method 2

forming a liposome-DNA complex by the electric interaction between a lipid bilayer membrane vesicle consisting of a positively charged lipid or the like (liposome) and DNA to be transferred

Methodology Applied
Scientific EffectElectric interaction: Electrostatics

Data Source

PatentEP2548958B1Agent for improving gene transfer efficiency to mammalian cells
Publication Date: 2017.11.22 YAMAGUCHI UNIV
  • EP2548958B1 patent drawingFigure 1
  • EP2548958B1 patent drawingFigure 2
  • EP2548958B1 patent drawingFigure 3

AI summary

Provided is an efficiency improving agent for gene transfer to mammalian cells, a method for improving efficiency of gene transfer to mammalian cells, and a method for transforming mammalian cells. The method is characterized in that tRNA is used in combination with a lipofection reagent. Preferably, the agent may be used so that the tRNA concentration in a lipofection solution falls within the range of 3 to 50 µg/mL, and the concentration in a culture is approximately 1/10. More preferably, tRNA and PEG may be used in combination with a lipofection reagent. According to the present invention, gene transfer to mammalian cells with high efficiency can be achieved.