Uracil Compound Herbicide Selectivity Optimization

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Solution Overview

Problem

Current herbicides lack effective weed control while maintaining safety for useful plants, leading to inefficient and potentially harmful applications.

Innovation Solution

A compound represented by formula (A) is developed, formulated into a herbicidal composition with inert carriers and applied to weeds or their habitats, offering excellent weed control efficacy with low phytotoxicity to useful plants.

Engineering Contradictions & Design Principles

VSEngineering Contradiction Analysis

1Reliability

If existing herbicides are applied to control weeds, then weed control efficacy is achieved, but safety against useful plants deteriorates (high phytotoxicity)

Engineering Contradiction:
Improveweed control efficacyVSAvoidphytotoxicity to useful plants
Core Design Contradiction:
ReliabilityVSObject-affected harmful factors

Solution Approach 1:

The patent modifies the chemical structure of uracil compounds by changing parameters such as substituting hydrogen atoms with specific groups (e.g., fluorine, chlorine, methyl, ethyl groups at positions 5, 6, and 7 of the uracil ring), and adjusting the R1-R6 substituents to optimize the balance between herbicidal activity and selectivity. This structural parameter optimization enables high weed control efficacy while reducing phytotoxicity to useful plants.

Inventive Principle:
Principle #35Parameter changes

Solution Approach 2:

The herbicidal composition is segmented into multiple components: the core uracil compound (Formula A) as the active ingredient, inert carriers for delivery, and optionally adjuvants to enhance performance. This segmentation allows the active compound to be delivered selectively to weeds while inert components ensure safety and proper application characteristics.

Inventive Principle:
Principle #1Segmentation

2Productivity

If herbicidal compositions are formulated with higher concentrations of active ingredients, then weed control efficacy improves, but safety against useful plants deteriorates

Engineering Contradiction:
Improveweed control efficacyVSAvoidphytotoxicity to useful plants
Core Design Contradiction:
ProductivityVSObject-affected harmful factors

Solution Approach 1:

The patent optimizes the concentration parameters of the active ingredient within specific ranges (e.g., 0.1-1000 g AI/ha application rates, and composition formulations containing 0.1-95 wt% active ingredient) to achieve maximum weed control efficacy while maintaining safety margins for useful plants through precise parameter control.

Inventive Principle:
Principle #35Parameter changes

Data Source

PatentUS11896010B2Uracil compound and use thereof
Publication Date: 2024.02.13 SUMITOMO CHEM CO LTD
  • US11896010B2 patent drawing
  • US11896010B2 patent drawing
  • US11896010B2 patent drawing

AI summary

A compound having excellent weed control efficacy and high safety against useful plants is represented by formula (A):