Recombinant Virion Arrays for Membrane Protein Profiling

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Solution Overview

Problem

Current methods for studying membrane proteins, especially those with multi-pass transmembrane domains, are limited by the need for embedding in a membrane and require posttranslational modifications, making high-throughput profiling challenging, and there is a need for cost-effective and time-efficient production of high-quality antibodies for these proteins.

Innovation Solution

The development of recombinant herpesviridae virion arrays with heterologous membrane-bound proteins that retain native conformations, allowing for the detection of binding events and the production of specific antibodies through a high-throughput platform.

Engineering Contradictions & Design Principles

VSEngineering Contradiction Analysis

1Productivity

If membrane proteins are purified using biochemical methods with detergents, then the proteins can be isolated, but the throughput is limited and subsequent manipulation becomes difficult

Engineering Contradiction:
ImprovethroughputVSAvoiddifficulty of manipulation
Core Design Contradiction:
ProductivityVSEase of manufacture

Solution Approach 1:

The patent uses detergents as intermediaries to solubilize membrane proteins during purification while maintaining their native conformations. The detergent micelles act as mediators between the hydrophobic membrane proteins and the aqueous environment, enabling high-throughput purification without denaturation. This resolves the contradiction by allowing both high throughput and ease of manipulation through the intermediary detergent system.

Inventive Principle:
Principle #24Intermediary (Mediator)

Solution Approach 2:

The patent changes physical parameters by using specific detergent concentrations and buffer conditions to maintain membrane proteins in soluble, active states during purification. By optimizing detergent type, concentration, and pH parameters, the method achieves high throughput purification while keeping proteins manipulable and active, thus resolving the contradiction between productivity and ease of manufacture.

Inventive Principle:
Principle #35Parameter changes

2Reliability

If membrane proteins are embedded in membranes to maintain native conformation, then the proteins retain their native conformations and interactions, but high-throughput profiling becomes challenging

Engineering Contradiction:
Improvenative conformation retentionVSAvoidthroughput
Core Design Contradiction:
ReliabilityVSProductivity

Solution Approach 1:

The patent employs detergents as intermediaries that replace the native membrane environment, allowing membrane proteins to maintain their native conformations and interactions in a soluble state. This intermediary system enables high-throughput profiling by eliminating the need for actual membrane embedding while preserving protein functionality and native structures.

Inventive Principle:
Principle #24Intermediary (Mediator)

Solution Approach 2:

The patent creates a simplified copy or surrogate of the native membrane environment using detergent micelles. Instead of requiring actual biological membranes, the detergent-based system replicates the essential properties needed for maintaining native protein conformations, enabling high-throughput experiments without the complexity of true membrane systems.

Inventive Principle:
Principle #26Copying

3Measurement precision

If antibodies are produced through traditional methods, then specific antibodies to membrane proteins can be obtained, but the process is costly and time-consuming

Engineering Contradiction:
Improveantibody specificityVSAvoidproduction time
Core Design Contradiction:
Measurement precisionVSLoss of time

Solution Approach 1:

The patent uses the membrane protein arrays to screen and select antibodies automatically, allowing the system to identify specific antibodies without extensive manual testing. The high-throughput array format enables the antibodies to be self-sorted based on their binding specificity to different membrane proteins, dramatically reducing both time and cost while maintaining high specificity.

Inventive Principle:
Principle #25Self-service

Solution Approach 2:

The patent changes the screening parameters by using high-throughput array formats that can simultaneously test thousands of antibody-protein interactions. This parameter change from sequential to parallel screening reduces production time and cost while maintaining or improving antibody specificity through comprehensive screening capabilities.

Inventive Principle:
Principle #35Parameter changes

Data Source

PatentEP3011061B1Virion display array for profiling functions and interactions of human membrane proteins
Publication Date: 2021.12.29 JOHNS HOPKINS UNIVERSITY
  • EP3011061B1 patent drawingFigure 1a
  • EP3011061B1 patent drawingFigure 1b
  • EP3011061B1 patent drawingFigure 1c

AI summary

Provided herein are recombinant virion arrays comprising human membrane bound proteins that retain their native conformations and/or interactions, recombinant HSV-1 virions, and methods of use including high-content, high-throughput assays for screening for ligands and/or drugs that bind human membrane bound proteins, diagnostic assays, proteomic assays, and biosensor assays. Also provided are recombinant HSV-1 virions comprising an envelope comprising a plurality of heterologous membrane bound proteins that retain their native conformations and/or interactions as well as recombinant HSV-1 bacterial artificial chromosome (BAC) clones encoding heterologous membrane polypeptides.