Vitamin D Detection Using Carbamate Derivatives and Specific Binding

Resolve Bottlenecks,
Find Innovative Solutions
Generate Solutions

Solution Overview

Problem

Current methods for determining vitamin D levels in biological samples lack accuracy and sensitivity, particularly in distinguishing between vitamin D and its analogs and metabolites, which is crucial for diagnosing related disorders.

Innovation Solution

A method involving specific binding members and compounds that form complexes with vitamin D, allowing for the measurement of vitamin D levels through signal-producing systems, including antibodies and chemiluminescent particles, to accurately quantify vitamin D in samples.

Engineering Contradictions & Design Principles

VSEngineering Contradiction Analysis

1Measurement precision

If conventional methods are used for determining vitamin D levels, then the determination can be performed with standard procedures, but the accuracy and sensitivity are insufficient for distinguishing between vitamin D and its analogs and metabolites

Engineering Contradiction:
Improveaccuracy and sensitivity of vitamin D level determinationVSAvoidcomplexity of binding members and compounds
Core Design Contradiction:
Measurement precisionVSDevice complexity

Solution Approach 1:

The patent introduces specific binding members (antibodies) and specially designed compounds as intermediaries to enable accurate detection of vitamin D. These binding members specifically recognize and bind to vitamin D and its analogs, allowing differentiation between similar molecules. The compounds contain specific structural features (substituents at positions 22 and 23) that enhance binding specificity, serving as mediators between the sample and detection system.

Inventive Principle:
Principle #24Intermediary (Mediator)

2Measurement precision

If specific binding members and specialized compounds are used to improve detection accuracy, then sensitivity and precision increase, but the device and method complexity increases

Engineering Contradiction:
Improvesensitivity of vitamin D detectionVSAvoidcomplexity of assay procedure
Core Design Contradiction:
Measurement precisionVSDifficulty of detecting and measuring

Solution Approach 1:

The patent employs compounds that are pre-designed with specific structural characteristics (substituents at positions 22 and 23 of the steroid nucleus) to enhance binding affinity and specificity before the actual detection process. This preliminary structural optimization ensures that when the binding members are introduced, they can immediately and specifically recognize the target molecules, reducing the need for complex procedural steps during detection.

Inventive Principle:
Principle #10Preliminary action

3Measurement precision

If conventional detection methods are used, then the procedure is simpler, but the ability to distinguish between vitamin D, analogs, and metabolites is insufficient for accurate diagnosis

Engineering Contradiction:
Improveability to distinguish vitamin D from analogs and metabolitesVSAvoidamount of reagents and binding members required
Core Design Contradiction:
Measurement precisionVSQuantity of substance

Solution Approach 1:

The patent applies local quality by introducing specific substituents at particular positions (22 and 23) of the steroid nucleus in the detection compounds. These localized structural modifications create specific binding pockets that recognize unique features of vitamin D and its analogs, enabling differentiation based on local molecular characteristics rather than requiring overall structural matching. This allows specific detection of target molecules even in complex biological samples containing multiple similar compounds.

Inventive Principle:
Principle #3Local quality

Applied Scientific Principles

This section explains which scientific principles are used to turn an abstract innovation direction into a practical engineering solution.

Function Achieved in This Case

This approach provides a sensitive and accurate means to determine the presence and amount of vitamin D, enabling better diagnosis and management of related disorders by enhancing the precision of vitamin D level assessments.

Implementation Method 1

a specific binding member for vitamin D... The combination is subjected to conditions for binding of the compound to the specific binding member to form a complex

Methodology Applied
Scientific EffectSpecific binding:

Implementation Method 2

signal-producing systems, including antibodies and chemiluminescent particles

Methodology Applied
Scientific EffectChemiluminescence: Chemiluminescence

Data Source

PatentEP2926143B1Compositions and methods for detecting vitamin d
Publication Date: 2019.03.27 SIEMENS HEALTHCARE DIAGNOSTICS INC
  • EP2926143B1 patent drawingFigure 1
  • EP2926143B1 patent drawingFigure 2
  • EP2926143B1 patent drawing

AI summary

Compounds include carbamate derivatives of vitamin D including vitamin D3 and vitamin D2. The compounds are useful in methods and kits for determining the presence and/or total amount of vitamin D, including vitamin D analogs and metabolites thereof, in a sample suspected of containing the same.