A method for the synthesis of substituted anthranilic amide compounds, intermediates and salts thereof

The method of reacting substituted isatin with a base, an amine, and an oxidizing agent addresses the inefficiencies of existing anthranilic amide synthesis methods, offering a cost-effective and environmentally friendly solution for large-scale production.

WO2025057193A1 Publication Date: 2025-03-20PI IND LTD
3 Cites 0 Cited by

Patent Information

Application Number
PCT/IN2024/051701
Authority / Receiving Office
WO · WO
Patent Type
Applications
Current Assignee / Owner
Priority Date
2023-12-19
Filing Date
2024-09-11
Publication Date
2025-03-20

AI Technical Summary

Technical Problem

Existing methods for synthesizing substituted anthranilic amide compounds are inefficient, requiring multiple steps, expensive solvents, and catalysts, making them unsuitable for large-scale commercial production.

Method used

A method involving the reaction of substituted isatin with a base, an amine, and an oxidizing agent, which simplifies the synthesis process and eliminates the need for expensive solvents and catalysts.

Benefits of technology

This method provides a cost-effective, environmentally friendly, and efficient route for producing substituted anthranilic amides, suitable for large-scale industrial production.

✦ Generated by Eureka AI based on patent content.
Patent Text Reader

Abstract

The present invention provides a method for the synthesis of compounds of formula (I), intermediates, and salts thereof, formula (I) wherein, R, R1 and n are as described in the description. The method further comprises the synthesis of anthranilic diamide compounds of formula (E), wherein the formula (E) is described in the description.
Need to check novelty before this filing date? Find Prior Art