Acellular Pro-inflammatory Preparations for Immune Stimulation

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Solution Overview

Problem

Current therapeutic approaches fail to effectively induce a pro-inflammatory state or immune stimulation, particularly in conditions associated with decreased or inappropriate immune responses such as cancer and infections, due to limited specificity and effectiveness of cytotoxic drugs and the inability to adequately stimulate a pro-inflammatory response.

Innovation Solution

Development of acellular pro-inflammatory preparations derived from allogeneic leukocyte populations, which are contacted under conditions to allow pro-inflammatory allo-recognition, with the resulting miRNA-enriched components being purified and formulated for administration to induce a therapeutic immune stimulation by altering the ratio of regulatory T cells to pro-inflammatory T cells.

Engineering Contradictions & Design Principles

VSEngineering Contradiction Analysis

1Quantity of substance

If chemical cytotoxic agents are used to target proliferating cells, then cancer cells are preferentially affected due to their higher mitotic rate, but the treatment lacks direct specificity towards the cancer cells

Engineering Contradiction:
Improveselectivity of cell targetingVSAvoidcomplexity of treatment approach
Core Design Contradiction:
Quantity of substanceVSEase of manufacture

Solution Approach 1:

The patent extracts and isolates specific miRNA species from allogeneic leukocytes that are responsible for inducing pro-inflammatory immune responses. These purified miRNA components are then administered therapeutically to induce immune stimulation against cancer cells, achieving targeted effect without using complex cytotoxic agents

Inventive Principle:
Principle #2Taking out (Extraction)

Solution Approach 2:

The patent uses miRNA species as intermediary molecules that mediate the immune response between the administered preparation and the cancer cells. These miRNA act as signaling molecules that trigger the patient's immune system to recognize and attack tumor cells, providing indirect but specific targeting

Inventive Principle:
Principle #24Intermediary (Mediator)

2Reliability

If clonal expansion of reactive leukocytes is induced to achieve target cell antigen-specific response, then the desired pro-inflammatory state may be stimulated, but the approach is expensive and complex

Engineering Contradiction:
Improveeffectiveness of immune stimulationVSAvoidcomplexity of treatment process
Core Design Contradiction:
ReliabilityVSDevice complexity

Solution Approach 1:

The patent uses stable, isolated miRNA species that can be produced once and stored for repeated administrations. These miRNA preparations replace complex, expensive in vivo clonal expansion protocols with simpler, more cost-effective molecular therapies that achieve similar or superior immune stimulation effects

Inventive Principle:
Principle #27Cheap short-living objects (Disposable)

Solution Approach 2:

The patent performs preliminary isolation and characterization of specific miRNA species from allogeneic leukocytes before therapeutic administration. This pre-preparation of active immune-stimulating components allows for standardized, reproducible treatments without requiring complex in vivo manipulation of entire leukocyte populations

Inventive Principle:
Principle #10Preliminary action

3Reliability

If the immune system is suppressed by regulatory T cells, then immune tolerance is maintained, but this prevents effective response to infections and cancer

Engineering Contradiction:
Improveimmune response effectivenessVSAvoidimmune suppression
Core Design Contradiction:
ReliabilityVSObject-affected harmful factors

Solution Approach 1:

The patent administers miRNA-enriched preparations that preemptively counteract the suppressive effects of regulatory T cells by inducing pro-inflammatory immune responses. The miRNA species prepare the immune system in advance to overcome Treg-mediated suppression and mount effective anti-tumor and anti-infective responses

Inventive Principle:
Principle #9Preliminary anti-action

Data Source

PatentEP3019176B1Use of acellular pro-inflammatory compositions and process for making same
Publication Date: 2020.05.06 CANADIAN BLOOD SERVICES
  • EP3019176B1 patent drawingFigure 1A~1B
  • EP3019176B1 patent drawingFigure 1C
  • EP3019176B1 patent drawingFigure 2A

AI summary

This invention relates to acellular-based therapies for decreasing the level of regulatory T cells (Treg) and/or increasing the level of pro-inflammatory T cells (Th17) to favor immune stimulation. To provide these therapeutic effects, an allogeneic leukocyte population is contacted with another leukocyte population and the acellular components produced are isolated. The leukocyte populations are contacted so as to allow pro-inflammatory allo- recognition. Acellular-based preparations and processes for achieving therapy are also provided.