CRISPR-Cas Guide RNA Architecture for Scalable Genome Editing

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Solution Overview

Problem

Current genome editing technologies, such as designer zinc fingers and TALEs, are not scalable, easy to set up, or affordable for targeting multiple positions within the eukaryotic genome, limiting their applicability in advanced biological and medical applications.

Innovation Solution

The development of a CRISPR-Cas system using engineered guide RNA molecules, such as chimeric single guide RNA (sgRNA) and dual guide RNA (dgRNA), which can be programmed to target specific DNA sequences without requiring customized proteins, enabling efficient genome editing by forming a CRISPR-Cas complex that can manipulate target nucleic acids in prokaryotic and eukaryotic cells.

Engineering Contradictions & Design Principles

VSEngineering Contradiction Analysis

1Manufacturing precision

If customized proteins are used for genome targeting (e.g., designer zinc fingers, TALEs), then targeting specificity is achieved, but device complexity and manufacturing cost increase significantly

Engineering Contradiction:
Improvetargeting specificityVSAvoidsystem complexity
Core Design Contradiction:
Manufacturing precisionVSDevice complexity

Solution Approach 1:

The patent uses RNA copies (guide RNA) to replace complex protein-based targeting systems. Instead of designing custom proteins for each target, a simple RNA sequence complementary to the target DNA serves as the targeting element, dramatically simplifying the system while maintaining specificity

Inventive Principle:
Principle #26Copying

Solution Approach 2:

The Cas9 enzyme serves as a universal platform that can target any genomic location by simply changing the guide RNA sequence. This single protein performs multiple targeting functions without requiring customization, reducing device complexity while maintaining versatility

Inventive Principle:
Principle #6Universality (Multi-functionality)

2Manufacturing precision

If customized proteins are used for each target position, then targeting precision is maintained, but productivity and scalability decrease

Engineering Contradiction:
Improvetargeting precisionVSAvoidscalability
Core Design Contradiction:
Manufacturing precisionVSProductivity

Solution Approach 1:

RNA sequences can be rapidly copied and modified through standard molecular biology techniques. Multiple guide RNAs can be designed and synthesized quickly to target different genomic positions, enabling high-throughput genome-wide studies without the time-consuming protein engineering required by previous methods

Inventive Principle:
Principle #26Copying

Solution Approach 2:

The patent changes the fundamental parameter from protein sequence design to RNA sequence design. This allows researchers to use simple nucleotide sequence changes rather than complex protein engineering, dramatically increasing productivity and enabling simultaneous targeting of multiple genes

Inventive Principle:
Principle #35Parameter changes

3Adaptability or versatility

If complex protein systems are used for genome editing, then functional capability is achieved, but ease of operation and setup become difficult

Engineering Contradiction:
Improvefunctional capabilityVSAvoidease of setup
Core Design Contradiction:
Adaptability or versatilityVSEase of operation

Solution Approach 1:

The guide RNA acts as a simple informational copy that directs the Cas9 enzyme to target sequences. This RNA-based addressing system is much easier to design and implement than protein-based systems, allowing researchers with basic molecular biology skills to perform genome editing without specialized protein engineering expertise

Inventive Principle:
Principle #26Copying

Solution Approach 2:

The guide RNA serves as an intermediary between the researcher's intent and the Cas9 enzyme's action. By designing a simple RNA sequence complementary to the target, researchers can program the complex Cas9 enzyme without directly manipulating it, greatly simplifying the operational process

Inventive Principle:
Principle #24Intermediary (Mediator)

Applied Scientific Principles

This section explains which scientific principles are used to turn an abstract innovation direction into a practical engineering solution.

Function Achieved in This Case

This approach simplifies genome editing methodologies, enhances targeting specificity, and accelerates the cataloging and mapping of genetic factors associated with various biological functions and diseases, providing a robust and scalable solution for genome engineering.

Implementation Method 1

a guide sequence capable of hybridizing to a target sequence in a genomic locus of interest

Methodology Applied
Scientific EffectHybridization:

Data Source

PatentEP4219699A1Engineering of systems, methods and optimized guide compositions with new architectures for sequence manipulation
Publication Date: 2023.08.02 THE BROAD INST INC
  • EP4219699A1 patent drawingFigure 1
  • EP4219699A1 patent drawingFigure 2
  • EP4219699A1 patent drawingFigure 3A

AI summary

The invention provides for systems, methods, and compositions for altering expression of target gene sequences and related gene products. Provided are structural information on the Cas protein of the CRISPR-Cas system, use of this information in generating modified components of the CRISPR complex, vectors and vector systems which encode one or more components or modified components of a CRISPR complex, as well as methods for the design and use of such vectors and components. Also provided are methods of directing CRISPR complex formation in eukaryotic cells and methods for utilizing the CRISPR-Cas system. In particular the present invention comprehends optimized functional CRISPR-Cas enzyme systems. In particular the present invention comprehends engineered new guide architectures to be used in optimized CRISPR-Cas enzyme systems.