Human Antibody Production via Pre-Immunization

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Solution Overview

Problem

Current vaccine therapeutic strategies focus on antigens rather than cytokine regulation, leading to inefficiencies in addressing cytokine-related immunosuppression and inflammation, particularly in cancer and AIDS, where natural anti-cytokine antibodies with low affinity and low titers are insufficient to neutralize cytokine activity effectively.

Innovation Solution

Development of a high-yield method to produce human antibodies that neutralize the biological activity of cytokines like VEGF, IFNα, IL-4, TNFα, and TGFβ, involving immunization with stable immunogenic products comprising protein immunogene heterocomplexes and subsequent purification of polyclonal or monoclonal antibodies, Fab or F(ab)′2 fragments, and ScFv fragments.

Engineering Contradictions & Design Principles

VSEngineering Contradiction Analysis

1Reliability

If natural anti-cytokine antibodies are used, then the treatment is simple and safe, but the antibody affinity and titer are low, resulting in insufficient neutralization of cytokine activity

Engineering Contradiction:
Improveneutralization efficacyVSAvoidcomplexity of antibody production method
Core Design Contradiction:
ReliabilityVSDevice complexity

Solution Approach 1:

The patent applies preliminary action by pre-immunizing individuals with cytokines before collecting antibodies. This preliminary immunization step ensures that when blood is collected, the individuals already have high-titer, high-affinity anti-cytokine antibodies in their serum, eliminating the need for complex in vitro antibody production methods while ensuring sufficient neutralization efficacy

Inventive Principle:
Principle #10Preliminary action

Solution Approach 2:

The patent utilizes the human immune system's natural antibody production capability. By immunizing individuals and then collecting their serum, the body itself produces the required high-affinity antibodies, which are then purified through relatively simple steps. This self-service approach avoids complex recombinant DNA technology while achieving high neutralization efficacy

Inventive Principle:
Principle #25Self-service

2Manufacturing precision

If complex purification steps are implemented, then antibody purity and yield are improved, but the manufacturing process becomes more complex and time-consuming

Engineering Contradiction:
Improveantibody purityVSAvoidproduction efficiency
Core Design Contradiction:
Manufacturing precisionVSProductivity

Solution Approach 1:

The patent applies the extraction principle by directly obtaining high-affinity anti-cytokine antibodies from the serum of pre-immunized individuals. The purification process extracts the desired antibodies from serum through relatively simple steps, avoiding complex multi-stage purification protocols while maintaining high antibody purity and yield, thus preserving production efficiency

Inventive Principle:
Principle #2Taking out (Extraction)

Solution Approach 2:

The patent changes the source parameter from recombinant production to natural serum antibodies. By utilizing antibodies naturally produced in human serum after immunization, the method achieves high purity with simpler purification steps, as the antibodies are already present in high concentration and affinity, reducing the need for extensive purification

Inventive Principle:
Principle #35Parameter changes

Applied Scientific Principles

This section explains which scientific principles are used to turn an abstract innovation direction into a practical engineering solution.

Function Achieved in This Case

The method achieves high-affinity antibodies that effectively inhibit at least 50% of the maximal biological activity of target cytokines in vitro, providing a direct and efficient treatment for cytokine-mediated immunosuppression and inflammation without the need for complex purification steps.

Implementation Method 1

human antibodies that neutralize the biological activity of a human cytokine

Methodology Applied
Scientific EffectAntigen-antibody binding: Absorption (physical)

Data Source

PatentUS8679483B2High-yield method for the production of human antibodies blocking the biological activity of a human cytokine
Publication Date: 2014.03.25 NEOVACS SA

AI summary

The invention concerns a pharmaceutical composition comprising, as the active ingredient, human natural antibodies of the IgG isotype, that neutralize the activity of a human cytokine selected from VEGF, IFNα, IL-4, TNFα and TGFβ, the said neutralizing antibodies inhibiting at least 50% of the maximum biological activity induced by an amount ranging from 0.006 ng to 0.05 ng of the said cytokine in vitro.