IL13RA2 and BIRC5 Peptide Immunotherapy for Adrenal Cancer Recurrence

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Solution Overview

Problem

Current therapies for adrenal cancer, including surgical resection and chemotherapy, are inadequate for advanced or metastatic cases, and there is a lack of effective second-line treatments, with high recurrence rates and limited success from cancer immunotherapy.

Innovation Solution

Development of antigen-based immunotherapy targeting interleukin-13 receptor α2 (IL13RA2) and BIRC5 to stimulate an immune response against adrenal cancer, using peptides and nucleic acids to induce a cytotoxic T-lymphocyte response.

Engineering Contradictions & Design Principles

VSEngineering Contradiction Analysis

1Reliability

If surgical resection is performed for adrenal cancer, then the five-year survival rate is 50-60 percent for early-stage tumors, but the prognosis deteriorates to only 10-20 percent five-year survival when tumors have spread to nearby or distant organs

Engineering Contradiction:
Improvefive-year survival rateVSAvoidtumor metastasis
Core Design Contradiction:
ReliabilityVSObject-affected harmful factors

Solution Approach 1:

The patent applies preliminary action by administering immunotherapy treatments before tumors metastasize or progress to advanced stages. The composition stimulates the immune system in advance to recognize and attack cancer cells, preventing the deterioration from 50-60% to 10-20% five-year survival rates associated with metastatic disease

Inventive Principle:
Principle #10Preliminary action

2Adaptability or versatility

If mitotane and cytotoxic chemotherapy are used for locally advanced or metastatic adrenal cancer, then systemic treatment is provided, but no effective second-line therapies are available for patients with disease progression

Engineering Contradiction:
Improvetreatment optionsVSAvoidtreatment effectiveness
Core Design Contradiction:
Adaptability or versatilityVSReliability

Solution Approach 1:

The patent applies parameter changes by shifting from conventional cytotoxic chemotherapy to an immunotherapy approach with different mechanisms of action. The composition uses modified peptides with enhanced immunogenicity properties, changing the therapeutic parameters to overcome resistance and provide effective second-line treatment when standard therapies fail

Inventive Principle:
Principle #35Parameter changes

Solution Approach 2:

The patent applies composite materials by combining modified peptides with adjuvants in a single composition. This composite approach integrates multiple therapeutic functions - the modified peptide provides tumor-specific targeting while the adjuvant enhances immune stimulation, creating a more effective treatment than either component alone

Inventive Principle:
Principle #40Composite materials

3Ease of manufacture

If more than half of patients undergo complete surgical removal of tumors, then initial treatment is achieved, but patients are destined to have relapse often with metastases

Engineering Contradiction:
Improvesurgical resectionVSAvoidrecurrence prevention
Core Design Contradiction:
Ease of manufactureVSReliability

Solution Approach 1:

The patent applies continuity of useful action by providing ongoing immune surveillance after surgical resection. The immunotherapy composition maintains continuous immune system activation to detect and eliminate residual cancer cells, preventing relapse and metastasis that would otherwise occur in more than half of surgically treated patients

Inventive Principle:
Principle #20Continuity of useful action

4Adaptability or versatility

If cancer immunotherapy is applied to adrenal cancer, then treatment is provided, but the success rate is very limited compared to other cancer types

Engineering Contradiction:
Improveimmunotherapy applicationVSAvoidimmunotherapy success rate
Core Design Contradiction:
Adaptability or versatilityVSReliability

Solution Approach 1:

The patent applies local quality by modifying specific properties of peptides to enhance their immunogenicity for adrenal cancer treatment. The modification pattern creates localized improvements in immune recognition and activation, making the immunotherapy specifically adapted for adrenal cancer rather than using generic immunotherapy approaches

Inventive Principle:
Principle #3Local quality

Solution Approach 2:

The patent applies intermediary by using modified peptides as mediators between the immune system and adrenal cancer cells. These peptides serve as the intermediate that bridges immune recognition with tumor-specific targeting, overcoming the limited success of direct immunotherapy approaches in adrenal cancer

Inventive Principle:
Principle #24Intermediary (Mediator)

Data Source

PatentEP4045150B1Immunogenic compounds for treatment of adrenal cancer
Publication Date: 2025.11.26 ENTEROME
  • EP4045150B1 patent drawingFigure 1
  • EP4045150B1 patent drawingFigure 2
  • EP4045150B1 patent drawingFigure 3A~3B

AI summary

The present invention relates to antigen-based immunotherapy targeting interleukin 13 receptor alpha 2 (IL13RA2), BIRC5 and/or FOXM1 for treatment of adrenal cancers. In particular, the present invention provides the use of a (poly)peptide comprising an epitope of IL13RA2, BIRC5 and/or FOXM1 or a sequence variant thereof for treatment of an adrenal cancer. Moreover, the present invention also provides combinations of the (poly)peptide comprising an epitope of IL13RA2, BIRC5 and/or FOXM1 or a sequence variant thereof with (poly)peptides comprising other epitopes or sequence variants thereof for treatment of adrenal cancers.