miRNA Plasmid Composition for Kinase mRNA Silencing

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Solution Overview

Problem

Over-expression or mis-expression of kinases leads to homeostasis disruption and associated diseases, necessitating therapies to regulate gene expression and suppress these biomolecules.

Innovation Solution

Compositions comprising plasmids with nucleotide sequences encoding miRNA sequences that target and degrade or inactivate the mRNA of kinases, such as Bruton's tyrosine kinase, EGF, VEGF, BRAF, ALK, HER, FLT3, or PARP, to downregulate their expression and production.

Engineering Contradictions & Design Principles

VSEngineering Contradiction Analysis

1Quantity of substance

If kinases are over-expressed or mis-expressed, then biological activity is increased, but homeostasis is lost and disease occurs

Engineering Contradiction:
Improvekinase expression levelVSAvoidhomeostasis
Core Design Contradiction:
Quantity of substanceVSReliability

Solution Approach 1:

The patent extracts and utilizes miRNA sequences that naturally target and degrade kinase mRNA. By introducing these specific miRNA sequences into cells via plasmids, the invention selectively removes excess or mis-expressed kinases from the cellular proteome, thereby restoring homeostasis without affecting other biological functions.

Inventive Principle:
Principle #2Taking out (Extraction)

Solution Approach 2:

The patent employs miRNA as an intermediary molecule between the plasmid and the kinase target. The miRNA sequences act as mediators that bind to kinase mRNA and facilitate its degradation, providing a controlled and specific mechanism for suppressing kinase expression while maintaining cellular homeostasis.

Inventive Principle:
Principle #24Intermediary (Mediator)

2Reliability

If therapies are developed to suppress over-expressed kinases, then homeostasis is restored, but gene expression regulation complexity increases

Engineering Contradiction:
ImprovehomeostasisVSAvoidgene expression regulation system
Core Design Contradiction:
ReliabilityVSDevice complexity

Solution Approach 1:

The patent employs miRNA sequences that are naturally part of the cell's regulatory system. By introducing these endogenous miRNA sequences through plasmids, the invention allows the cell's own gene expression machinery to perform the suppression function, avoiding the need for complex external therapeutic agents or proteins.

Inventive Principle:
Principle #25Self-service

Solution Approach 2:

The patent changes the parameter of gene expression regulation by introducing specific miRNA sequences that alter the stability and translation of kinase mRNA. This parameter change enables precise control over kinase levels through RNA interference mechanisms, simplifying the overall therapeutic approach.

Inventive Principle:
Principle #35Parameter changes

Applied Scientific Principles

This section explains which scientific principles are used to turn an abstract innovation direction into a practical engineering solution.

Function Achieved in This Case

The compositions effectively decrease the bioavailability of target kinases, restoring homeostasis and potentially treating associated diseases by increasing endogenous production of miRNA sequences that target and silence the mRNA of these kinases.

Implementation Method 1

The sequences of miRNA may be complementary to a sequence of target messenger RNA (mRNA) that encodes for translation of a target biomolecule

Methodology Applied
Scientific EffectBase pairing:

Implementation Method 2

a backbone sequence of nucleic acids that facilitates introduction of the one or more insert sequences into one or more of a subject's cells where it is expressed and/or replicated

Methodology Applied
Scientific EffectDNA replication:

Implementation Method 3

Expression of the one or more insert sequences by one or more cells of the subject results in an increased production of the miRNA

Methodology Applied
Scientific EffectTranscription:

Data Source

PatentUS12559754B2Composition for regulating production of interfering ribonucleic acid
Publication Date: 2026.02.24 WYVERN PHARMACEUTICALS INC

AI summary

The embodiments of the present disclosure relate to decreasing the bioavailability of one or more target biomolecules by providing a composition that comprises a recombinant plasmid with one or more sequences of micro interfering ribonucleic acid (miRNA). When the recombinant plasmid interacts with a target cell, it causes the target cell to upregulate production of the miRNA, which then decreases the bioavailability of the target biomolecule. In some embodiments of the present disclosure, the target biomolecule is a kinase.