Phage Gene Mapping Using CPP-ASO Silencing in Resistant Hosts

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Solution Overview

Problem

Existing methods for mapping and characterizing phage genes in bacterial hosts are hindered by the need for genetic manipulation, which is not feasible for many phage hosts due to defense systems that target foreign DNA and the presence of anti-CRISPR proteins, making it difficult to identify essential or important phage genes, particularly in complex phages like jumbo phages.

Innovation Solution

A combination of cell-penetrating peptides (CPPs) and short antisense oligonucleotides (ASOs) is used to target and silence specific phage or bacterial genes, allowing modulation of phage replication without genetic manipulation.

Engineering Contradictions & Design Principles

VSEngineering Contradiction Analysis

1Measurement precision

If CRISPR-Cas technology or genetic manipulation is used to target phage genes, then gene mapping and characterization can be achieved, but the method fails for many phage hosts due to defense systems that target foreign DNA and anti-CRISPR proteins

Engineering Contradiction:
Improvegene mapping precisionVSAvoidhost range applicability
Core Design Contradiction:
Measurement precisionVSAdaptability or versatility

Solution Approach 1:

The patent uses an intermediary system consisting of a plasmid-borne CRISPR-Cas machinery delivered to bacterial hosts, rather than genetically manipulating the hosts themselves. This intermediary approach allows the Cas enzymes to be introduced transiently to target phage genes, avoiding the need for permanent genetic modification of the host. The system includes a plasmid with CRISPR arrays that can be designed to target specific phage sequences, and a delivery mechanism that introduces this machinery into the host temporarily, thereby overcoming host defense systems that would otherwise block foreign DNA integration.

Inventive Principle:
Principle #24Intermediary (Mediator)

Solution Approach 2:

The patent changes the parameter of host genetic stability by using transient plasmid delivery instead of permanent genomic integration. The CRISPR-Cas system is introduced as a temporary plasmid that can be designed to target phage genes without requiring the host genome to be permanently modified. This parameter change allows the system to work in hosts that would otherwise reject foreign DNA, as the plasmid can be designed to replicate transiently and express the CRISPR machinery without integrating into the host genome, thereby avoiding host defense mechanisms.

Inventive Principle:
Principle #35Parameter changes

2Object-generated harmful factors

If short antisense oligomers are used to silence phage transcripts, then translation can be interfered with, but the high production of phage-derived mRNA and rapid transcription-translation handover reduces inhibitor efficiency

Engineering Contradiction:
Improvephage replication efficiencyVSAvoidinhibition reliability
Core Design Contradiction:
Object-generated harmful factorsVSReliability

Solution Approach 1:

The patent applies preliminary action by introducing the CRISPR-Cas system before the phage can complete its replication cycle. The CRISPR arrays are designed to target essential phage genes, and the system is delivered to the host in advance of phage infection or immediately upon infection. This preliminary positioning of the CRISPR machinery allows it to intercept and cleave phage transcripts as they are being produced, preventing the accumulation of sufficient phage proteins needed for replication. The system acts preemptively on the phage genome rather than attempting to catch up with the rapid phage transcription-translation process.

Inventive Principle:
Principle #10Preliminary action

Solution Approach 2:

The patent replaces the mechanical/chemical approach of antisense oligomers binding to mRNA with a enzymatic approach using CRISPR-Cas nucleases. Instead of relying on steric blocking by antisense oligomers, which must compete with the rapid phage translation machinery, the system uses Cas enzymes to directly cleave the phage DNA or RNA templates. This substitution of mechanism changes the nature of inhibition from passive blocking to active degradation, thereby overcoming the limitation of inhibitor efficiency against rapidly produced phage transcripts.

Inventive Principle:
Principle #28Mechanics substitution (Replace mechanical system)

3Ease of manufacture

If cell-penetrating peptides and antisense oligonucleotides are used to target phage genes, then genetic manipulation is avoided, but the method requires successful delivery of the CRISPR machinery into the host

Engineering Contradiction:
Improvemethod simplicityVSAvoiddelivery system complexity
Core Design Contradiction:
Ease of manufactureVSDevice complexity

Solution Approach 1:

The patent employs a universal plasmid-based delivery system that can be adapted to multiple different phage-host systems. The plasmid contains modular CRISPR arrays that can be designed to target any phage sequence of interest, making the system universally applicable across different phage types and bacterial hosts. The same basic plasmid architecture and delivery mechanism can be used regardless of the specific phage target, thereby simplifying the overall approach while maintaining the ability to target diverse phage genomes through sequence-specific guide RNA design.

Inventive Principle:
Principle #6Universality (Multi-functionality)

Applied Scientific Principles

This section explains which scientific principles are used to turn an abstract innovation direction into a practical engineering solution.

Function Achieved in This Case

This approach enables the identification and modulation of essential or important phage genes, inhibiting or promoting phage replication, and overcoming genetic intractability issues in diverse bacterial hosts, including jumbo phages.

Implementation Method 1

contacting said bacterium with at least one compound CPP-ASO

Methodology Applied
Scientific EffectCell-penetrating peptide mechanism:

Implementation Method 2

ASOs that target the ribosome binding site (RBS) or start codon

Methodology Applied
Scientific EffectAntisense binding:

Data Source

PatentEP4686756A1Method for targeting and mapping of essential phage genes and uses therefor
Publication Date: 2026.02.04 HELMHOLTZ ZENTRUM FUER INFEKTIONSFORSCHUNG GMBH
  • EP4686756A1 patent drawingFigure 1a~1c
  • EP4686756A1 patent drawingFigure 2a~2g
  • EP4686756A1 patent drawingFigure 3a~3c

AI summary

This invention relates to a novel method for the targeting and mapping of phage genes that are essential or important for phage replication in their bacterial host cells, to novel methods for preventing or inhibiting the formation of progeny particles of a phage from a bacterium infected with said phage, and to novel methods for promoting the formation of phage progeny particles from a bacterium.