Rumen-Resistant Microgranules for Controlled Post-Ruminal Release

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Solution Overview

Problem

Existing compositions for delivering physiologically active substances to ruminants suffer from poor stability during feedstuff production, inadequate ruminal protection, and low post-ruminal digestibility, leading to insufficient bioavailability of these substances.

Innovation Solution

A rumen-resistant microgranule composition with a core containing active substances and a matrix, coated with multiple layers to protect against ruminal degradation, featuring disintegrant agents for controlled release in the abomasum and small intestine, enhancing bioavailability.

Engineering Contradictions & Design Principles

VSEngineering Contradiction Analysis

1Reliability

If active substances are mixed with feedstuff in conventional formulations, then they are administered orally to animals, but they undergo enzymatic chemical degradation in the rumen and during processing, resulting in poor preservation stability and low bioavailability

Engineering Contradiction:
Improvestability of active substancesVSAvoiddegradation of active substances
Core Design Contradiction:
ReliabilityVSLoss of substance

Solution Approach 1:

The formulation is segmented into distinct functional components: active substances (5-50% w/w), protective agents (50-95% w/w), and optional binders or fillers. This segmentation allows the active substances to be physically separated from the feed matrix, protecting them from ruminal degradation while maintaining stability during processing and storage.

Inventive Principle:
Principle #1Segmentation

Solution Approach 2:

Protective agents serve as intermediaries between the active substances and the ruminal environment. These agents (fats, oils, waxes, proteins, or their derivatives) form a protective barrier that prevents enzymatic degradation in the rumen while allowing controlled release in the lower digestive tract, thus resolving the contradiction between protection and bioavailability.

Inventive Principle:
Principle #24Intermediary (Mediator)

2Reliability

If protective coatings are applied to protect active substances from ruminal degradation, then rumen bypass is improved, but post-ruminal digestibility and bioavailability are reduced

Engineering Contradiction:
Improverumen protectionVSAvoidreduced post-ruminal digestibility
Core Design Contradiction:
ReliabilityVSLoss of substance

Solution Approach 1:

The protective agents are selected and formulated with specific physical and chemical parameters: melting points above ruminal temperature (38-42°C) to maintain protection, but below colonic temperature (35-37°C) to allow release. Fats and oils with melting points of 35-45°C, waxes with melting points of 40-60°C, and proteins with appropriate solubility characteristics are used to achieve the desired parameter balance for both protection and release.

Inventive Principle:
Principle #35Parameter changes

Solution Approach 2:

The formulation uses composite protective systems combining multiple agents (fats, oils, waxes, proteins, or their derivatives) with complementary properties. This composite approach provides synergistic protection during ruminal passage while ensuring adequate release in the lower digestive tract, resolving the contradiction between protection and digestibility.

Inventive Principle:
Principle #40Composite materials

3Productivity

If active substances are concentrated in the formulation, then higher zootechnical performance can be achieved, but they become more susceptible to degradation during mixing, packaging, storage, and compaction

Engineering Contradiction:
Improvezootechnical performanceVSAvoiddegradation during processing
Core Design Contradiction:
ProductivityVSLoss of substance

Solution Approach 1:

The active substances are extracted from the conventional feed matrix and formulated as a separate concentrated composition with protective agents. This extraction allows higher concentrations of active substances (5-50% w/w) to be incorporated while the protective agents shield them from degradation during mixing, packaging, storage, and compaction operations.

Inventive Principle:
Principle #2Taking out (Extraction)

Solution Approach 2:

Protective agents (fats, oils, waxes, proteins, or their derivatives) are incorporated beforehand to cushion and protect the active substances from mechanical stress, heat, and moisture during processing and storage. This prior cushioning prevents degradation before the substances are exposed to harmful conditions, enabling higher concentrations to be used safely.

Inventive Principle:
Principle #11Beforehand cushioning (Prior cushioning)

Applied Scientific Principles

This section explains which scientific principles are used to turn an abstract innovation direction into a practical engineering solution.

Function Achieved in This Case

The composition achieves improved ruminal bypass and post-ruminal digestibility, resulting in higher total bioavailability of active substances, maintaining chemical and physical stability during processing and administration.

Implementation Method 1

The microgranules comprise at least two coating layers, in which the first coating layer consists of a substance or mixture of substances having hydrophobic properties

Methodology Applied
Scientific EffectHydrophobic barrier: Hydrophobe

Implementation Method 2

The core comprises one or more physiologically active substances and a matrix, in which at least one disintegrant agent is included

Methodology Applied
Scientific EffectDisintegration:

Data Source

PatentEP3585362B1Composition for controlled release of physiologically active substances and process for its preparation
Publication Date: 2026.04.01 BALCHEM ITALIA SRL

AI summary

The present invention relates to a rumen-resistant composition in the form of microgranules, a process for its production and a feedstuff containing such composition.