C-terminally Truncated Fibrillin-1 Mouse Model for NPSCL

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Solution Overview

Problem

Current transgenic non-human mammals engineered to have FBN1 mutations do not adequately reflect the symptoms of neonatal progeroid syndrome with congenital lipodystrophy (NPSCL), as they fail to accurately replicate the genetic and phenotypic characteristics of the condition.

Innovation Solution

A mouse model is developed with a mutation in the Fbn1 gene that results in a C-terminal truncation of the Fbn1 protein, leading to symptoms such as decreased body weight, decreased fat mass, increased food intake, and kyphosis, which are characteristic of NPSCL, by introducing specific mutations in the penultimate or final exon of the Fbn1 gene, disrupting the asprosin C-terminal cleavage product of pro-fibrillin-1.

Engineering Contradictions & Design Principles

VSEngineering Contradiction Analysis

1Reliability

If transgenic non-human mammals are engineered with FBN1 mutations, then the model should reflect Marfan syndrome symptoms, but the model fails to accurately represent NPSCL symptoms

Engineering Contradiction:
Improveaccuracy of disease modelVSAvoidphenotypic representation accuracy
Core Design Contradiction:
ReliabilityVSAdaptability or versatility

Solution Approach 1:

The patent applies local quality by introducing a specific mutation location (penultimate exon of Fbn1 gene) that produces a C-terminal truncated protein. This localized genetic modification creates the specific NPSCL phenotype characterized by lipodystrophy and progeroid features, rather than the Marfan syndrome phenotype. The mutation position is precisely targeted to disrupt the asprosin C-terminal cleavage product while preserving other fibrillin-1 functions, thereby achieving accurate NPSCL phenotypic representation.

Inventive Principle:
Principle #3Local quality

2Reliability

If the Fbn1 gene is mutated to produce C-terminal truncated protein, then NPSCL-like symptoms are exhibited, but the mutation disrupts the asprosin C-terminal cleavage product

Engineering Contradiction:
Improvedisease model accuracyVSAvoiddisruption of protein processing
Core Design Contradiction:
ReliabilityVSObject-generated harmful factors

Solution Approach 1:

The patent converts the harmful disruption of asprosin C-terminal cleavage into a beneficial research tool. By intentionally introducing the mutation that disrupts this cleavage process, the patent creates a model that accurately reproduces NPSCL pathology. The disruption itself becomes the mechanism for studying the disease, allowing researchers to investigate the relationship between impaired asprosin processing and NPSCL symptoms including lipodystrophy and progeroid features.

Inventive Principle:
Principle #22Blessing in disguise (Convert harm into benefit)

Data Source

PatentEP3490373B1Mice comprising mutations resulting in expression of c-truncated fibrillin-1
Publication Date: 2023.10.25 REGENERON PHARMACEUTICALS INC
  • EP3490373B1 patent drawingFigure 1~2
  • EP3490373B1 patent drawingFigure 3
  • EP3490373B1 patent drawingFigure 4~5

AI summary

Provided are non-human animals comprising a mutation in the Fbnl gene to model neonatal progeroid syndrome with congenital lipodystrophy (NPSCL). Also provided are methods of making such non-human animal models. The non-human animal models can be used for screening compounds for activity in inhibiting or reducing NPSCL or ameliorating NPSCL- like symptoms or screening compounds for activity potentially harmful in promoting or exacerbating NPSCL as well as to provide insights in to the mechanism of NPSCL and potentially new therapeutic and diagnostic targets.