Variant Cry1B Polypeptides for Broad-Spectrum Pest Control

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Solution Overview

Problem

Existing genetically engineered crops provide resistance to only a narrow range of economically important insect pests, necessitating the development of new Bacillus thuringiensis (Bt) toxins with improved insecticidal activity against insects from the orders Lepidoptera and Coleoptera, and biopesticides with broader activity against various insect pests.

Innovation Solution

Development of variant Cry1B polypeptides with enhanced insecticidal activity against corn earworm and fall armyworm, encoded by recombinant nucleic acids, which are expressed in transgenic plants to control Lepidopteran pests.

Engineering Contradictions & Design Principles

VSEngineering Contradiction Analysis

1Adaptability or versatility

If genetically engineered crops produce pesticidal proteins from Bacillus, then insect resistance is enhanced, but the spectrum of pest control remains narrow

Engineering Contradiction:
Improvespectrum of pest controlVSAvoidcomplexity of developing new toxin variants
Core Design Contradiction:
Adaptability or versatilityVSDevice complexity

Solution Approach 1:

The patent applies parameter changes by systematically mutating specific amino acid residues in the Cry1B polypeptide sequence to alter its insecticidal properties. Multiple variants are created with different amino acid substitutions at positions known to affect toxin activity, thereby expanding the spectrum of pest control while maintaining a relatively simple development framework based on structured mutagenesis

Inventive Principle:
Principle #35Parameter changes

Solution Approach 2:

The patent achieves universality by developing a single Cry1B polypeptide variant system that can control multiple pest species across different orders (Lepidoptera and Coleoptera). The engineered variants maintain core functionality while gaining broader applicability, allowing one toxin system to serve multiple pest control functions

Inventive Principle:
Principle #6Universality (Multi-functionality)

2Reliability

If broad-spectrum chemical insecticides are used, then pest control effectiveness is high, but environmental hazards increase

Engineering Contradiction:
Improvepest control effectivenessVSAvoidenvironmental hazards
Core Design Contradiction:
ReliabilityVSObject-affected harmful factors

Solution Approach 1:

The patent replaces chemical insecticide systems with a biological control system based on genetically engineered Bacillus thuringiensis-derived polypeptides. These biopesticides maintain high pest control effectiveness through targeted action on insect gut receptors while eliminating the environmental hazards associated with broad-spectrum chemical insecticides, as they are highly specific to certain insect orders

Inventive Principle:
Principle #28Mechanics substitution (Replace mechanical system)

Solution Approach 2:

The patent modifies the biological parameters of the pesticidal proteins by engineering amino acid variations that enhance both effectiveness and environmental safety. The engineered variants achieve improved binding affinity to insect gut receptors for higher effectiveness while maintaining biodegradability and species-specificity for reduced environmental harm

Inventive Principle:
Principle #35Parameter changes

Data Source

PatentEP3442994B1Insecticidal polypeptides having improved activity spectrum and uses thereof
Publication Date: 2025.10.29 PIONEER HI BREED INTERNATIONAL INC
  • EP3442994B1 patent drawingFigure 1A
  • EP3442994B1 patent drawingFigure 1B
  • EP3442994B1 patent drawingFigure 1C

AI summary

The disclosure provides nucleic acids, and variants and fragments thereof, derived from strains of Bacillus thuringiensis encoding variant polypeptides having increased pesticidal activity against insect pests, including Lepidoptera and Coleopteran. Particular embodiments of the disclosure provide isolated nucleic acids encoding pesticidal proteins, pesticidal compositions, DNA constructs, and transformed microorganisms and plants comprising a nucleic acid of the embodiments. These compositions find use in methods for controlling pests, especially plant pests.