Small-molecule compound as well as synthesis method and application thereof

By developing a new type of small molecule compound, using specific structural formulas and synthesis methods, we have solved the problem of existing drugs being unable to effectively treat androgenic alopecia, achieved the effect of promoting hair growth and improving the hair growth cycle, and are suitable for many patients. treatment of diseases.

CN104193699AActive Publication Date: 2014-12-10TECHNODERMA MEDICINES
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Patent Information

Application Number
CN201410398184.1
Authority / Receiving Office
CN · China
Patent Type
Applications(China)
Current Assignee / Owner
Filing Date
2014-08-14
Publication Date
2014-12-10
Estimated Expiration
2034-08-14

AI Technical Summary

Technical Problem

Existing drugs for the treatment of alopecia cannot effectively solve the problem of androgenic alopecia, and there is insufficient research on the diversity and diversification of drugs for regulating hair growth, making them unable to meet the needs of modern people.

Method used

A new type of small molecule compound was developed to promote hair growth through a specific structural formula and synthesis method. The specific steps include using 4-methoxyphenol and 1,2,3-trichloro-5-nitrobenzene as The initial raw materials undergo a series of reactions to generate N1-(3,5-dichloro-4-(3-(substituted benzyl)-4-hydroxyphenoxy)phenyl)-N2-oxalylhydroxylamine compounds, which are used for Treating androgenetic alopecia.

Benefits of technology

This small molecule compound significantly changes the hair growth cycle and promotes hair growth in mouse hair growth tests, has no toxic side effects, slows body weight changes, and has obvious hair growth effects. It is suitable for the treatment of androgenetic alopecia and other diseases such as osteoporosis. disease, obesity, etc.

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Abstract

The invention provides a small-molecule compound which is characterized by being shown in a structure formula which is as shown in the specification. Various concentration dosages of the small-molecule compound are capable of remarkably changing the hair growth period and promoting the hair growth; the small-molecule compound shows a remarkable hair growth promotion effect; and moreover, the body weight change of mice in each group is very slow, which means that the tested compound does not cause weight loss of the animals.
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