Composition

By using specific plant extracts in skin care products and adjusting the proportion of ingredients, the viscosity problem when using nimethylol and cycloalanine acid is solved, achieving high moisturizing and long-lasting moisturizing effects, while improving the product usage experience.

JP7657550B2Active Publication Date: 2025-04-07KOSE CORPORATION
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Patent Information

Application Number
JP2020062386
Authority / Receiving Office
JP · JP
Patent Type
Patents
Current Assignee / Owner
Filing Date
2020-03-31
Publication Date
2025-04-07
Estimated Expiration
2040-03-31

AI Technical Summary

Technical Problem

Existing skin care products that use nimethylol and cycloalanine acid are prone to feel viscous when combined, which affects the user experience.

Method used

By adding specific plant extracts to skin care products, such as legumes, Asteraceae, Tea, Camellia, Honey, Royal Bee Honey, Sodium Disulfonate and Cordyceps extract, adjust the ingredients ratio to ensure there is no viscosity while maintaining a good moisturizing effect.

Benefits of technology

It achieves the use of high moisturizing and long-lasting moisturizing effects while avoiding the sticky feeling of skin care products, improving the product experience.

✦ Generated by Eureka AI based on patent content.

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Abstract

To provide a composition excellent in lack of stickiness and moisture retention feeling.SOLUTION: There is provided a composition which comprises the following components (A) to (C): (A) tranexamic acid or its salt, (B) niacinamide and (C) at least one cosmetic component selected from the group consisting of a leguminous plant or its extract, an Asteraceae plant or its extract, an Umbelliferae plant or its extract, a Theaceae plant or its extract, a Miscanthus plant or its extract, a Myrtaceae plant or its extract, a rutaceous plant or its extract, a buttercup plant or its extract, a labiate plant or its extract, an Osmanthus plant or its extract, a royal jelly extract, honey, sodium pyrosulfite and a cordyceps extract.SELECTED DRAWING: None
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Description

[Technical field]

[0001] The present invention relates to a composition. [Background technology]

[0002] The skin develops spots, wrinkles, sagging, pigmentation, etc. due to internal factors such as aging and stress, and external factors such as ultraviolet rays and dry air. In particular, morphological changes such as wrinkles and sagging have a large impact on the impression of the skin's appearance, so many people wish to improve them. Many drugs have been proposed to prevent and improve these wrinkles and sagging. Among these, niacinamide is known to be highly safe, and cosmetics containing it are being developed. For example, a skin anti-aging cosmetic containing nicotinamide, urea, and one or more selected from the group consisting of α-hydroxycarboxylic acid compounds having 2 to 28 carbon atoms is known (see, for example, Patent Document 1).

[0003] On the other hand, tranexamic acid is known to have an anti-inflammatory effect, and may be used for the purpose of obtaining a whitening effect. In recent years, tranexamic acid and its derivatives are known to be used as wrinkle improving agents. For example, a technique is known in which a wrinkle improving composition having a superior wrinkle improving effect is provided by using an aminocarboxylic acid derivative having a specific structure and its acid addition salt in combination with tranexamic acid and its derivatives (see, for example, Patent Document 2). [Prior art documents] [Patent documents]

[0004] [Patent Document 1] Japanese Patent Application Publication No. 10-130135 [Patent Document 2] JP 2019-206483 A Summary of the Invention [Problem to be solved by the invention]

[0005] Conventionally used niacinamide and tranexamic acid have excellent moisturizing properties, and when used in combination, a high level of moisturizing effect can be expected, but they can be less convenient to use due to stickiness, etc. Furthermore, when beauty ingredients other than niacinamide and tranexamic acid, such as plant extracts, are used in formulations, they can sometimes cause a peculiar stickiness.

[0006] Therefore, an object of the present invention is to develop a composition that has a moisturizing feel but is not sticky and has excellent usability. [Means for solving the problem]

[0007] In view of this situation, the present inventors conducted extensive research and searched for a material that maintains or further enhances the moisturizing feeling of a composition containing niacinamide and tranexamic acid and is not sticky. The inventors' research has revealed that, by using a specific beauty ingredient that has been considered to be sticky in a composition containing niacinamide and tranexamic acid, it is surprisingly possible to obtain a non-sticky composition without impairing the moisturizing feeling, and have completed the present invention.

[0008] That is, the present invention relates to the following components (A) to (C): (A) Tranexamic acid or a salt thereof (B) Niacinamide (C) At least one cosmetic ingredient selected from the group consisting of a legume plant or extract thereof, a Asteraceae plant or extract thereof, a Umbelliferae plant or extract thereof, a Theaceae plant or extract thereof, a Xanthomonas plant or extract thereof, a Myrtaceae plant or extract thereof, a Rutaceae plant or extract thereof, a Ranunculaceae plant or extract thereof, a Lamiaceae plant or extract thereof, an Oleaceae plant or extract thereof, royal jelly extract, honey, sodium metabisulfite, and Cordyceps sinensis extract. The present invention relates to a composition comprising:

[0009] The present invention also relates to the composition described above, wherein the component (C) is at least one selected from the group consisting of a plant of the genus Sophora (Fabaceae) or an extract thereof, a plant of the genus Glycyrrhiza (Fabaceae) or an extract thereof, a plant of the genus Lagodiae (Asteraceae) or an extract thereof, a plant of the genus Deutzia (Asteraceae) or an extract thereof, a plant of the genus Yarrow (Asteraceae) or an extract thereof, a plant of the genus Daucus ... Carrot (Apiaceae) or an extract thereof, a plant of the genus Camellia (Theaceae) or an extract thereof, a plant of the genus Aloe (Myrtaceae) or an extract thereof, a plant of the genus Citrus (Rutunculaceae) or an extract thereof, a plant of the genus Coptis (Ranunculaceae) or an extract thereof, a plant of the genus Rosemary (Lamiaceae) or an extract thereof, a plant of the genus Olea (Oleaceae) or an extract thereof, royal jelly extract, honey, sodium metabisulfite, and cordyceps sinensis extract.

[0010] The present invention also relates to the composition described above, wherein the component (C) is at least one selected from the group consisting of plants of the genus Sophora (Leguminosa), or extracts thereof, plants of the genus Glycyrrhiza (Leguminosa), or extracts thereof, plants of the genus Lagodiae (Asteraceae), or extracts thereof, plants of the genus Deutzia (Asteraceae), or extracts thereof, plants of the genus Yarrow (Asteraceae), or extracts thereof, plants of the genus Daucus ... Camellia (Theaceae), or extracts thereof, plants of the genus Aloe (Myrtaceae), plants of the genus Eucalyptus (Myrtaceae), plants of the genus Citrus (Rutaceae), plants of the genus Coptis (Ranunculaceae), plants of the genus Rosemary (Lamiaceae), or extracts thereof, and plants of the genus Olea (Oleaceae), or extracts thereof.

[0011] The present invention also relates to the composition described above, wherein the component (C) is at least one selected from the group consisting of royal jelly extract, honey, sodium pyrosulfite, and cordyceps sinensis extract.

[0012] The present invention also relates to the composition described above, wherein the content of the component (C) in the composition is 0.0001 to 0.01% by mass.

[0013] The present invention also relates to the composition described above, wherein the mass ratio of the component (A) to the component (B) is (A) / (B)=0.01-20.

[0014] The present invention also relates to the composition described above, wherein the mass ratio of the components (B) and (C) is (B) / (C)=10 to 10,000.

[0015] The present invention further relates to the above-described composition, which contains a component (D) a polyhydric alcohol having 5 to 12 carbon atoms.

[0016] The present invention also relates to the composition described above, wherein the component (D) is at least one polyhydric alcohol selected from the group consisting of dipropylene glycol, tripropylene glycol, 1,2-pentanediol, 1,2-hexanediol, and 1,2-octanediol.

[0017] The present invention also relates to an external skin preparation or cosmetic composition containing the above-mentioned composition.

[0018] Furthermore, the present invention relates to an agent for reducing stickiness in a composition containing component (A) tranexamic acid or a salt thereof, and component (B) niacinamide, comprising component (C) at least one cosmetic ingredient selected from the group consisting of a legume plant or extract thereof, an Asteraceae plant or extract thereof, a Umbelliferae plant or extract thereof, a Theaceae plant or extract thereof, a Xanthomonas plant or extract thereof, a Myrtaceae plant or extract thereof, a Citrus plant or extract thereof, a Ranunculaceae plant or extract thereof, a Lamiaceae plant or extract thereof, an Oleaceae plant or extract thereof, royal jelly extract, honey, sodium metabisulfite, and Cordyceps sinensis extract.

[0019] Furthermore, the present invention relates to a method for improving stickiness in a composition containing component (A) tranexamic acid or a salt thereof, and component (B) niacinamide, using component (C) at least one cosmetic ingredient selected from the group consisting of a legume plant or extract thereof, an Asteraceae plant or extract thereof, a Umbelliferae plant or extract thereof, a Theaceae plant or extract thereof, a Xanthomonas plant or extract thereof, a Myrtaceae plant or extract thereof, a Citrus plant or extract thereof, a Ranunculaceae plant or extract thereof, a Lamiaceae plant or extract thereof, an Oleaceae plant or extract thereof, royal jelly extract, honey, sodium metabisulfite, and Cordyceps sinensis extract. Effect of the Invention

[0020] According to the present invention, it is possible to provide a composition that has a moisturizing feeling and lasts a moisturizing feeling, yet is not sticky. DETAILED DESCRIPTION OF THE PREFERRED EMBODIMENTS

[0021] The present invention will be described in detail below. In this specification, the symbol "to" means a range including the numerical values ​​before and after it.

[0022] Tranexamic acid or a salt thereof, which is the component (A) of the present invention, is a type of amino acid with the chemical name trans-4-(aminomethyl)cyclohexane-1-carboxylic acid. In the present invention, it can be used in the form of a salt, and can be a salt of an inorganic base such as a sodium salt or potassium salt, or a salt of an organic base such as triethanolamine or lysine.

[0023] The content of component (A) in the present invention is not particularly limited, but the lower limit is preferably 0.01% by mass (hereinafter simply abbreviated as "%) or more, more preferably 0.1% or more, and even more preferably 1% or more. The upper limit is preferably 10% or less, more preferably 7% or less, and even more preferably 5% or less. This range is more preferable because it provides better moisturizing feeling and non-stickiness.

[0024] Niacinamide (also known as nicotinamide), component (B) in the present invention, is also known as vitamin B3, and is a coenzyme deeply involved in various biochemical reactions in the body, such as energy metabolism and oxidation-reduction. It is said to have the effect of keeping the skin and mucous membranes normal and promoting blood flow, and it is known that a deficiency of niacinamide can cause symptoms such as "pellagra (dermatitis, gastrointestinal disorders, neurological disorders, etc.)". Niacinamide is also an ingredient that is blended into cosmetics and skin external preparations in the hope of improving the skin, since it is water-soluble; stable against heat, acid, alkali, and light; and highly safe.

[0025] The niacinamide used in the present invention may be produced by utilizing a known production method, and is also available as a raw material for foods, cosmetics, medicines, etc., or as a chemical product or reagent.

[0026] The content of component (B) in the present invention is not particularly limited, but the lower limit is preferably 0.01% or more, more preferably 0.1% or more, and even more preferably 1% or more. The upper limit is preferably 10% or less, more preferably 7% or less, and even more preferably 5% or less. This range is more preferable because it provides better moisturizing feeling and non-stickiness.

[0027] In the present invention, the composition is obtained by appropriately containing the above-mentioned components (A) and (B), but it is more preferable to specify the mass ratio of the components (A) and (B) because it is more excellent in moisturizing feeling and non-stickiness. Such mass ratio is not particularly limited, and the lower limit of the mass ratio (A) / (B) of the components (A) and (B) is preferably 0.01 or more, more preferably 0.05 or more, and even more preferably 0.1 or more. The upper limit is preferably 20 or less, more preferably 15 or less, and even more preferably 10 or less.

[0028] The component (C) in the present invention is at least one selected from the group consisting of a legume plant or its extract, a Asteraceae plant or its extract, a Umbelliferae plant or its extract, a Theaceae plant or its extract, a Xanthomonas plant or its extract, a Myrtaceae plant or its extract, a Rutaceae plant or its extract, a Ranunculaceae plant or its extract, a Lamiaceae plant or its extract, an Oleaceae plant or its extract, a royal jelly extract, honey, sodium metabisulfite, and a cordyceps sinensis extract. The details will be described below, but the plant or its extract includes the plant or its closely related species.

[0029] In the present invention, the component (C) legume plant or extract thereof is not particularly limited and can be used as long as it is a plant or extract thereof belonging to the Fabaceae family. For example, a Sophora plant or extract thereof, a Pisum plant or extract thereof, a Lupinus plant or extract thereof, a Pueraria plant or extract thereof, a Glycyrrhiza plant or extract thereof, etc. can be mentioned. Sophora plants include Sophora flavescens, etc. Pisum plants include Pisum sativum L., etc. Lupin plants include Lupinus albus, etc. Pueraria plants include Pueraria montana var. lobata, etc. Licorice plants include Glycyrrhiza glabra, etc. Among these, from the viewpoint of moisturizing feeling and non-stickiness, a Sophora plant or an extract thereof, or a Glycyrrhiza plant or an extract thereof is preferred. In particular, the use of a combination of the component (A) tranexamic acid or a salt thereof, and (B) niacinamide with an extract of Sophora flavescens (Fabaceae) and / or an extract of Glycyrrhiza glabra (Fabaceae) is more preferred, since it provides a moisturizing feeling, a sustained moisturizing feeling, and non-stickiness.

[0030] In the present invention, the component (C) Asteraceae plant or its extract can be used without any particular limitation as long as it is a plant or its extract belonging to the Asteraceae family. For example, Arnica plant or its extract, Matricaria plant or its extract, Achillea plant or its extract, Arctium plant or its extract, Calendula plant or its extract, Centaurea plant or its extract, etc. can be mentioned. Arnica unalascensis var. tschonoskyi can be mentioned as an example of Arnica plant. Matricaria plant can be mentioned as an example of Matricaria recutita. Achillea millefolium can be mentioned as an example of Achillea millefolium. Examples of plants belonging to the genus Burdock include Arctium lappa L., etc. Examples of plants belonging to the genus Calendula include Calendula officinalis, etc. Examples of plants belonging to the genus Cornflower include Centaurea cyanus, etc. Among these, from the viewpoints of moisturizing feeling and non-stickiness, plants belonging to the genus Arnica (also known as Arnica) or extracts thereof, plants belonging to the genus Matricaria or extracts thereof, and plants belonging to the genus Achillea or extracts thereof are preferred. In particular, it is more preferable to use a combination of the components (A) tranexamic acid or a salt thereof, and (B) niacinamide with one or more selected from the group consisting of an extract of Arnica unalascensis var. tschonoskyi (Asteraceae), an extract of Matricaria recutita (Asteraceae), and Achillea millefolium (Asteraceae), since this combination provides an excellent moisturizing feeling, maintains the moisturizing feeling, and is non-sticky.

[0031] In the present invention, the component (C) of the Apiaceae plant or its extract can be used without any particular limitation as long as it is a plant belonging to the Apiaceae family or its extract. For example, Centella plants or their extracts, Angelica plants or their extracts, Daucus plants or their extracts, etc. are included. Centella plants include Centella asiatica, etc. Angelica plants include Angelica keiskei, etc. Daucus plants include carrots (Daucus carota subsp. sativus, etc.) are included. Among these, Daucus plants or their extracts are preferred from the viewpoint of moisturizing feeling and non-stickiness. In particular, it is more preferable to use a combination of the components (A) tranexamic acid or a salt thereof, and (B) niacinamide with an extract of Daucus carota subsp. sativus of the Apiaceae family, since this combination provides excellent moisturizing sensation, lasts longer, and is non-sticky.

[0032] In the present invention, the component (C) of the Theaceae plant or its extract can be used without any particular limitation as long as it is a plant belonging to the Theaceae family or its extract. For example, the Camellia plant or its extract can be mentioned. Examples of the Camellia plant include Camellia japonica and Camellia sinensis. Among these, the Camellia plant or its extract is preferred from the viewpoint of moisturizing feeling and non-stickiness. In particular, it is more preferred to use the component (A) tranexamic acid or its salt and (B) niacinamide in combination with the extract of Camellia japonica and / or Camellia sinensis, which are both of Theaceae family, in order to provide a more excellent moisturizing feeling, its duration, and non-stickiness.

[0033] In the present invention, the component (C) Xanthorrhoeaceae plant or extract thereof can be used without any particular limitation as long as it is a plant or extract belonging to the Xanthorrhoeaceae family (also known as the Daylily family). For example, Aloe genus plants or extracts thereof, Hemerocallis genus plants or extracts thereof, etc. can be mentioned. Examples of Aloe genus plants include Aloe vera, etc. Examples of Hemerocallis genus plants include Hemerocallis fulva var. fulva, etc. Among these, Aloe genus plants or extracts thereof are preferred from the viewpoint of moisturizing feeling and non-stickiness. In particular, it is more preferred to use the component (A) tranexamic acid or its salt, and (B) niacinamide in combination with an extract of Aloe genus of Xanthorrhoeaceae, because it provides a more excellent moisturizing feeling, its duration, and non-stickiness.

[0034] In the present invention, the component (C) Myrtaceae plant or extract thereof is not particularly limited and may be any plant or extract thereof belonging to the Myrtaceae family, such as Eucalyptus plants or extracts thereof, Psidium plants or extracts thereof, and Syzygium plants or extracts thereof. Examples of Eucalyptus plants include Eucalyptus. Examples of Psidium guajava plants include Guava. Examples of Myrtaceae plants include Syzygium aromaticum. Among these, Eucalyptus plants or extracts thereof are preferred from the viewpoint of moisturizing feeling and non-stickiness. In particular, it is more preferred to use a combination of the components (A) tranexamic acid or a salt thereof and (B) niacinamide with an extract of Eucalyptus of the Myrtaceae family, since it provides a more excellent moisturizing feeling, its duration, and non-stickiness.

[0035] In the present invention, the component (C) of the citrus plant or its extract is not particularly limited and can be used as long as it is a plant belonging to the Rutaceae family or its extract. For example, Citrus plants or their extracts, Phellodendron plants or their extracts, etc. are included. Citrus plants include Citrus unshiu, Citrus junos, and Citrus limon. Phellodendron plants include Phellodendron amurense. Among these, Citrus plants or their extracts are preferred from the viewpoint of moisturizing feeling and non-stickiness. In particular, it is more preferable to use a combination of the components (A) tranexamic acid or a salt thereof, and (B) niacinamide with one or more selected from the group consisting of extracts of Citrus unshiu (Rutaceae), Citrus junos (Rutaceae), and Citrus limon (Rutaceae), since this provides an excellent moisturizing feeling, its duration, and non-stickiness.

[0036] In the present invention, the component (C) Ranunculaceae plant or extract thereof is not particularly limited as long as it is a plant belonging to the Ranunculaceae family or an extract thereof, and examples thereof include Coptis plants and extracts thereof. Examples of Coptis genus plants include Coptis japonica. Among these, Coptis genus plants or their extracts are preferred from the viewpoint of moisturizing feeling and non-stickiness. In particular, by combining the component (A) tranexamic acid or its salt and (B) niacinamide with the extract of Coptis japonica of the Ranunculaceae family, it is more preferred because it provides excellent moisturizing feeling, its duration, and non-stickiness.

[0037] In the present invention, the component (C) Lamiaceae plant or extract thereof is not particularly limited and can be used as long as it is a plant or extract thereof belonging to the Lamiaceae family. For example, Perilla plants or extracts thereof, Lavandula plants or extracts thereof, Mentha plants or extracts thereof, Salvia plants or extracts thereof, Rosmarinus plants or extracts thereof, Thymus plants or extracts thereof, etc. are included. Perilla plants include Perilla frutescens var. crispa, etc. Lavandula plants include Lavender, etc. Mentha plants include Mint, etc. Salvia plants include Sage, etc. Rosmarinus plants include Rosemary, etc. Examples of Thymus plants include Thymus L. Among these, from the viewpoint of moisturizing feeling and non-stickiness, Rosmarinus plants or their extracts are preferred. In particular, by combining the component (A) tranexamic acid or its salt and (B) niacinamide with one or more selected from the group consisting of Rosmarinus officinalis L. extract, Lavandula angustifolia, Salvia officinalis, and Thymus L., it is more preferred because it provides excellent moisturizing feeling, its duration, and non-stickiness.

[0038] In the present invention, the component (C) Oleaceae plant or extract thereof can be used without any particular limitation as long as it is a plant or extract thereof belonging to the Oleaceae family. For example, Olea plants or extracts thereof, Osmanthus plants or extracts thereof, etc. can be mentioned. Examples of Olea plants include olive (Olea europaea) and the like. Examples of Osmanthus plants include sweet osmanthus (Osmanthus fragrans var. aurantiacus) and the like. Among these, Olea plants or extracts thereof are preferred from the viewpoint of moisturizing feeling and non-stickiness. In particular, it is more preferred to use the component (A) tranexamic acid or its salt, and (B) niacinamide in combination with an extract of Olea europaea of ​​the Oleaceae family, since it provides a more excellent moisturizing feeling, its duration, and non-stickiness.

[0039] The plant in the present invention may be used as it is, but is preferably made into an extract from the viewpoint of further enhancing the effect of the present invention. The part to be extracted is not particularly limited, and flowers, leaves, stems, roots, seeds, fruits, seed coats, etc. can be used. The part to be extracted can be selected appropriately depending on the plant, and is not particularly limited. For example, the roots of a legume or its extract are preferred, the flowers of a Asteraceae plant or its extract are preferred, the roots of a Umbelliferae plant or its extract are preferred, the seeds or leaves of a Theaceae plant or its extract are preferred, the leaves or flowers of a Myrtaceae plant or its extract are preferred, the fruits or peels of a Rutaceae plant or its extract are preferred, the roots or stems of a Ranunculaceae plant or its extract are preferred, the leaves or flowers of a Lamiaceae plant or its extract are preferred, and the fruits of an Oleaceae plant or its extract are preferred.

[0040] The plant extracting solvent in the present invention is not particularly limited, and may be selected from one or more of water, organic solvents, etc. Also, carbon dioxide or water in a supercritical state may be used.

[0041] As the organic solvent, for example, one or more selected from alcohols; ketones such as acetone; ethers such as ethyl ether; esters such as ethyl acetate; and hydrocarbons such as hexane and benzene can be used.

[0042] Examples of the alcohols include lower monohydric alcohols (e.g., methanol, ethanol, etc.); liquid polyhydric alcohols (e.g., 1,3-butylene glycol, propylene glycol, glycerin, etc.). The alcohols are preferably monohydric alcohols and dihydric alcohols, and the number of carbon atoms of the alcohols is preferably about 1 to 5.

[0043] Of the above-mentioned extraction solvents, water and / or alcohols (preferably having 1 to 4 carbon atoms) are preferred. As the above-mentioned alcohols, one or more selected from methanol, ethanol, propylene glycol and 1,3-butylene glycol are preferred. Among these extraction solvents, more preferred are a mixture of one or more selected from water, ethanol and 1,3-butylene glycol, more preferred are water, ethanol, 1,3-butylene glycol, an ethanol-water mixed solution, a 1,3-butylene glycol-water mixed solution, and even more preferred is a 1,3-butylene glycol-water mixed solution. In the case of an alcohol aqueous solution, the alcohol concentration (V / V) is preferably 0 to 100% by volume, more preferably 20 to 80% by volume.

[0044] The royal jelly extract (C) of the present invention is a jelly-like substance obtained by mixing secretions from the hypopharyngeal gland and mandibular gland of worker honeybees. Royal jelly extract is known to have effects such as nutritional tonic, anti-aging, and growth promotion.

[0045] Honey is made by honeybees sucking nectar from the flowers of plants, decomposing it with enzymes secreted from the salivary glands, and concentrating it. Nectar for honey can be selected from various plants, such as plum, mandarin orange, cherry blossom, manuka, etc. The honey in the present invention is not particularly limited, but manuka honey is preferred from the viewpoint of moisturizing feeling.

[0046] Sodium metabisulfite can also be produced by the dehydration of sodium bisulfite or by the addition of sulfur dioxide to sodium sulfite. Sodium metabisulfite has reducing properties and is used as a food bleach and as an antioxidant in wine.

[0047] In addition, Cordyceps sinensis extract is an extract of the fruiting body of Cordyceps sinensis, which parasitizes the larvae of insects such as those of the Pterygota moth family, forms a sclerotium inside the body, and is formed on the body surface of the host insect or its larvae in the summer.

[0048] The content of component (C) in the present invention is not particularly limited, but the lower limit, calculated as solid content, is preferably 0.0001% or more, more preferably 0.0005% or more, and even more preferably 0.001% or more. The upper limit is preferably 0.01% or less, more preferably 0.007% or less, and even more preferably 0.005% or less. This range is more preferable because it provides better moisturizing feeling and non-stickiness.

[0049] In the present invention, the composition is obtained by appropriately containing the components (B) and (C), but it is more preferable to specify the mass ratio of the components (B) and (C) because it is more excellent in moisturizing feeling and non-stickiness. Such mass ratio is not particularly limited, and the lower limit of the mass ratio (B) / (C) of the components (B) and (C) is preferably 10 or more, more preferably 50 or more, and even more preferably 100 or more. The upper limit is preferably 10,000 or less, more preferably 5,000 or less, and even more preferably 1,000 or less.

[0050] In the present invention, the composition is obtained by appropriately containing the components (A) and (C), but it is more preferable to specify the mass ratio of the components (A) and (C) because it is more excellent in moisturizing feeling and non-stickiness. Such mass ratio is not particularly limited, and the lower limit of the mass ratio (A) / (C) of the components (A) and (C) is preferably 10 or more, more preferably 50 or more, and even more preferably 100 or more. The upper limit is preferably 10,000 or less, more preferably 5,000 or less, and even more preferably 2,000 or less.

[0051] In the present invention, the composition is obtained by appropriately containing the above-mentioned components (A), (B) and (C), but it is preferable to specify the mass ratio of the components (A), (B) and (C) because a higher effect can be expected. Such mass ratio is not particularly limited, and the lower limit of the total amount of components (A) and (B) and the mass ratio of component (C) [(A)+(B)] / (C) is preferably 100 or more, more preferably 500 or more, and even more preferably 1000 or more. The upper limit is preferably 12000 or less, more preferably 10000 or less, and even more preferably 5000 or less. This range is more preferable because it provides better moisturizing feeling and non-stickiness.

[0052] The present invention may further contain a polyhydric alcohol having 5 to 12 carbon atoms as component (D). The polyhydric alcohol of component (D) in the present invention is not particularly limited as long as it has 5 to 12 carbon atoms, and the lower limit of the carbon number is preferably 5 or more, preferably 6 or more, and more preferably 7 or more. The upper limit of the carbon number is preferably 12 or less, preferably 10 or less, and more preferably 9 or less. This range is more preferable because it provides better moisturizing feeling and non-stickiness. Examples of such polyhydric alcohols include dipropylene glycol, tripropylene glycol, diglycerin, 1,2-pentanediol, 1,2-hexanediol, 1,2-octanediol, and 1,2-decanediol, and one or more of these may be used in combination. Among these, at least one selected from the group consisting of dipropylene glycol, tripropylene glycol, 1,2-pentanediol, 1,2-hexanediol, and 1,2-octanediol is preferred, at least one selected from the group consisting of dipropylene glycol, tripropylene glycol, and 1,2-pentanediol is more preferred, and dipropylene glycol and / or tripropylene glycol is even more preferred.

[0053] The content of component (D) in the present invention is not particularly limited, but the lower limit is preferably 0.1% or more, more preferably 1% or more, and even more preferably 3% or more.The upper limit is preferably 50% or less, more preferably 30% or less, and even more preferably 15% or less.This range is more preferable because it provides better moisturizing feeling and non-stickiness.

[0054] The present invention may further contain an aqueous component other than component (D) as component (E). The aqueous component other than component (D) means water or a mixture of a component soluble in water and water. For example, lower alcohols such as ethyl alcohol and isopropyl alcohol can be mentioned. The content of the aqueous component in the present invention is not particularly limited, and the lower limit is preferably 10% or more, more preferably 30% or more, and even more preferably 50% or more. The upper limit is preferably 90% or less, more preferably 80% or less, and even more preferably 70% or less. This range is more preferable because it provides excellent moisturizing feeling and its duration, and is not sticky.

[0055] In particular, among the aqueous components, a compound containing one or more structural units selected from the group consisting of polyoxyethylene units (hereinafter sometimes abbreviated as EO units), polypropylene units (hereinafter sometimes abbreviated as PO units), and polyoxybutylene units (hereinafter sometimes abbreviated as BO units) is more preferable because it provides a more excellent moisturizing feeling. Such a compound is an ether in which EO units, PO units, and BO units are randomly or block-copolymerized with alcohol. The number of carbon atoms in the alcohol is not particularly limited, but a carbon number of 1 to 3 is preferred. In addition, the alcohol is not particularly limited, but may be any monohydric to trihydric alcohol, more preferably a trihydric alcohol, and even more preferably glycerin. For example, polyoxypropylene butyl ether (3PO), polyoxyethylene polyoxypropylene butyl ether (10EO) (7PO), polyoxyethylene polyoxypropylene dimethyl ether (14EO) (7PO), polyoxybutylene polyoxyethylene polyoxypropylene glyceryl ether (3BO) (8EO) (5PO), etc. can be mentioned. In the present invention, the content of the compound that comprises one or more structural units selected from the group consisting of EO unit, PO unit, and BO unit is not particularly limited, but the lower limit is preferably 0.001% or more, more preferably 0.005% or more, and even more preferably 0.01% or more.The upper limit is preferably 5% or less, more preferably 3% or less, and even more preferably 1% or less.This range is more preferable because it is more excellent in the sustained moisturizing feeling.

[0056] The present invention may further contain a component (F) film-forming agent. The film-forming agent in the present invention is a substance that forms a film when applied. The film-forming agent in the present invention has the effect of keeping the components (A) and (B) in place for a long time, thereby further enhancing the duration of the moisturizing feeling. Such a film-forming agent is not particularly limited, and various types can be used.

[0057] Examples of the film-forming agent include water-soluble film-forming agents, emulsion polymer-type film-forming agents, and oil-based film-forming agents. More specifically, examples of the water-soluble film-forming agent include polyvinylpyrrolidone and polyvinyl alcohol. Examples of the emulsion polymer-type film-forming agent include copolymers having alkyl acrylate, ethylenic polymer, and vinylpyrrolidone or vinyl alcohol as monomer units. Examples of the film-forming agent include (acrylates / VP) copolymer, (styrene / VP) copolymer, (ethylene / VA) copolymer, (acrylates / VA) copolymer, and (VP / VA) copolymer. Examples of the oil-based film-forming agent include silicone-based resins such as trimethylsiloxysilicate, polymethylsilsesquioxane, and acrylic-modified silicone, rosin-modified phenolic resin, and rosin acid-based resins such as rosin ester. Among these, water-soluble film-forming agents are preferred from the viewpoint of sustained moisturizing feeling.

[0058] In addition to the above-mentioned components, the composition of the present invention may contain optional components within the range that does not impair the effects of the present invention, such as powders, water-soluble polymers, colorants, preservatives, antibacterial agents, UV absorbers, fragrances, antioxidants, pH adjusters, chelating agents, cosmetic ingredients other than the components (A) to (C), etc.

[0059] The method for producing the composition of the present invention is not particularly limited as long as it is a known mixing method, and may be, for example, dispersion mixing, solubilization, high-pressure emulsification, or the like.

[0060] According to the present invention, a composition containing component (A) tranexamic acid or a salt thereof and component (B) niacinamide is provided by containing component (C) at least one cosmetic ingredient selected from the group consisting of a legume plant or an extract thereof, a Asteraceae plant or an extract thereof, a Umbelliferae plant or an extract thereof, a Theaceae plant or an extract thereof, a Xanthomonas plant or an extract thereof, a Myrtaceae plant or an extract thereof, a Citrus plant or an extract thereof, a Ranunculaceae plant or an extract thereof, a Labiatae plant or an extract thereof, an Oleaceae plant or an extract thereof, a royal jelly extract, honey, sodium metabisulfite, and a Cordyceps sinensis extract, which are at least one cosmetic ingredient selected from the group consisting of a Fabaceae plant or an extract thereof, a Ranunculaceae plant or an extract thereof, a Labiatae plant or an extract thereof, an Oleaceae plant or an extract thereof, a royal jelly extract, honey, sodium metabisulfite, and a Cordyceps sinensis extract. The preferred components and contents of components (A) to (C) of the stickiness reducing agent of the present invention, the mass ratios of components (A) to (C), and the like are the same as those of the above composition.

[0061] In addition, the present invention provides a method for improving stickiness of a composition containing component (A) tranexamic acid or a salt thereof and component (B) niacinamide, by containing component (C) at least one cosmetic ingredient selected from the group consisting of a legume plant or an extract thereof, an Asteraceae plant or an extract thereof, a Umbelliferae plant or an extract thereof, a Theaceae plant or an extract thereof, a Xanthomonas plant or an extract thereof, a Myrtaceae plant or an extract thereof, a Citrus plant or an extract thereof, a Ranunculaceae plant or an extract thereof, a Labiatae plant or an extract thereof, an Oleaceae plant or an extract thereof, a royal jelly extract, honey, sodium metabisulfite, and a Cordyceps sinensis extract. The preferred components and contents of components (A) to (C) in the method for improving stickiness of the present invention, and the mass ratios of components (A) to (C) are the same as those of the above composition.

[0062] The formulation of the composition of the present invention is not particularly limited, and any of the formulations such as aqueous solution, oil-in-water type, water-in-oil type, and powder can be used for washing, with aqueous solution and oil-in-water type being preferred. The properties are also not particularly limited, and the composition can be in various formulations such as liquid, gel, paste, cream, and solid.

[0063] The composition of the present invention can be used, for example, as a cosmetic, an external skin preparation, a medicine, a food, and the like.

[0064] The composition of the present invention can be applied as cosmetics. For example, skin care cosmetics such as lotion, milky lotion, cream, eye cream, beauty essence, massage agent, pack agent, hand cream, body milk, body cream, hair styling agent, sunscreen cosmetic, hair cosmetics such as shampoo, rinse, hair cream, cleansing cosmetics such as body soap, hand soap, face wash, cleansing agent, makeup cosmetics such as lipstick, powder foundation, liquid foundation, cream foundation, concealer, face powder, makeup base, blusher, eye shadow, mascara, eyeliner, eyebrow, etc., and the method of use thereof can be a method using hands, cotton, puff, etc., a method of applying to nonwoven fabric, etc., a method of spraying from a spray container, etc.

[0065] The composition of the present invention can also be used as a skin external preparation. Examples of the composition include external liquid preparations, external gel preparations, cream preparations, ointments, liniments, lotions, poultices, plasters, sprays, aerosols, etc. The method of use can be the same as that of the above-mentioned cosmetics.

[0066] The composition of the present invention can also be used as a food. For example, it can be used as a nutritional supplement, a health supplement, a functional health food, a food for specified health uses, a supplement, etc. More specifically, Examples include candy, yogurt, soup, fruit juice, vegetable juice, soft drinks, etc. EXAMPLES

[0067] The present invention will be described in more detail below by way of examples, but the present invention is not limited to these in any way. Example 1 (Products 1 to 14 of the present invention) and Comparative Example (Comparative Products 1 to 4): Cosmetic Compositions The compositions shown in Table 1 were prepared by the manufacturing method described below, and evaluated and judged according to the evaluation methods and judgment criteria described below, and the results are also shown in Table 1. The extracts and fruit juices listed in this example table refer to values ​​converted into solid content concentrations.

[0068] [Table 1]

[0069] (Manufacturing method) A: Mix and dissolve ingredients (1) to (12) uniformly. B: Add ingredients (13) to (14) and mix evenly. C: The mixture was filled into a container to obtain a cosmetic composition.

[0070] (Evaluation items) B. Moisturizing feeling B. Sustained moisturizing effect C. Non-stickiness

[0071] (Evaluation method) Six expert panelists (women in their 30s to 50s) were selected who were trained in the sensory evaluation of cosmetics and able to evaluate them according to certain standards. They were asked to apply each sample to the area around their cheeks, and after blending it in, they were asked to evaluate (a) whether they felt moisturizing (answer "good" if they felt moisturizing, and "bad" if they did not), (b) whether the moisturizing sensation continued even after several hours had passed (answer "good" if they felt moisturizing three hours after application, and "bad" if they did not), and (c) whether they felt sticky (answer "good" if they felt sticky, and "bad" if they did not). They reported the results and judged them according to the following criteria.

[0072] (Evaluation based on certain criteria) Six expert panel members undergo sensory evaluation of cosmetics. In order to confirm that the evaluation can be performed according to a consistent standard, the following three types of samples were prepared, and 5g of each sample was applied to the skin (forearm) of the expert panel members, and the degree of stickiness and moisturizing sensation was checked.

[0073] (Confirmation sample) Sample A: Glycerin Sample B: 20% glycerin aqueous solution Sample C: Purified water

[0074] After applying the three samples, the expert panel judged each sample's lack of stickiness and moisturizing sensation as good or bad. In the present invention, the condition of the panel is that the panel can answer sample a or sample b as good for moisturizing sensation, and sample b or sample c as good for lack of stickiness. Furthermore, the condition of the expert panel, who has been trained in sensory evaluation of cosmetics, is that the panel can answer only sample b as good for moisturizing sensation and lack of stickiness.

[0075] (Judgment criteria) (Judgment): (Evaluation) A: 5 or more people answered that it would be good B: 3 to 4 people are best C: 1 to 2 people are better D: Everyone answered that it was bad.

[0076] As is clear from the results in Table 1, the Examples (Products 1 to 14 of the present invention) were superior to the Comparative Examples in terms of moisturizing feeling, sustained moisturizing feeling, and non-stickiness. On the other hand, Comparative Product 1, which does not contain Component (A), and Comparative Product 2, which does not contain Component (B), did not provide satisfactory quality in terms of moisturizing feeling and sustained moisturizing feeling, and Comparative Product 3, which does not contain Component (C), and Comparative Product 4, in which Component (C) was replaced with another plant extract, did not provide satisfactory quality in terms of non-stickiness.

[0077] Example 2 Oil-in-water emulsion cream Ingredients (%) 1.1,3-Butylene glycol 12 2. Glycerin 5 3. Remaining purified water 4. Niacinamide 4 5. Tranexamic acid 0.4 6. Licorice extract 0.1 7. Sodium N-stearoyl-N-methyl taurate 0.5 8. PEG-40 Stearate 1 9. Heavy Liquid Isoparaffin 3 10. Dimethylpolysiloxane (25℃ kinematic viscosity 10CS) 1 11. Ceramide 2 0.1 12. Ethyl oleate 0.01 13. DL-α-tocopherol acetate 0.01 14. Cetostearyl alcohol 2 15. Behenyl Alcohol 1 16. Pentylene glycol 0.1 17. Acrylic acid / alkyl methacrylate copolymer 0.15 18. Gellan gum 0.1 19. Sodium hydroxide 2% solution 0.2 20. Fragrance (Citrus) 0.1 (Manufacturing method) A: Dissolve and mix ingredients 1 to 6 uniformly at 70°C. B: Components 7 to 16 are dissolved and mixed uniformly at 80°C. C: Add B to A and emulsify at 70℃. D: Ingredients 17 to 20 were added to C and mixed, then cooled to 40°C to obtain an oil-in-water emulsion cream. (evaluation) The oil-in-water emulsion cream of Example 2 was excellent in all respects: moisturizing feeling, sustained moisturizing feeling, and non-stickiness.

[0078] Example 3 Water-in-oil liquid foundation Ingredients (%) 1. Spherical polyethylene (average particle size 5 μm) 5 2. Spherical silica (average particle size 5 μm) 1.5 3. Fine particle titanium dioxide *1 8 4. Fine particle zinc oxide *2 5 5. Isododecane 15 6. Hydrogenated polyisobutene 3 7. Ethylhexyl methoxycinnamate 5 8. Bis-ethylhexyloxyphenol Methoxyphenyltriazine 1 9. Diisopropyl Sebacate 3 10. Cetyl ethylhexanoate 2 11. Lauryl PEG-9 Polydimethylsiloxyethyl dimethicone※9 3 12. Remaining purified water 13. Niacinamide 7 14. Tranexamic acid 2 15. Ethanol 3 16. Tripropylene glycol 2 17.1,3-Butylene glycol 2 18. Methylenebisbenzotriazolyltetramethylbutylphenol 2 19. Honey 0.01 20. Eucalyptus extract 0.01 21. Carrot extract 0.01 22. Rosemary extract 0.01 23. Hydrolyzed collagen 0.001 24. Ceramide NG 0.005 25. Stearyl hectorite 0.3 26. Dimethylstearylammonium Hectorite 0.2 27. Coloring agent ※3 2 28.2% lecithin-treated talc 4 29. Glyceryl Tribehenate 2 30. Propylene glycol dicaprate 8 31. Glyceryl tri-2-ethylhexanoate 6 *1: 2% isopropyl triisostearate titanium treatment *2: 3% methylhydrogenpolysiloxane treatment *3: 2% triethoxycaprylylsilane-treated pigment-grade titanium dioxide 1.2%, 2% stearoyl glutamate disodium-treated red iron oxide 0.2%, 1% lauroyl lysine 0.4% yellow iron oxide, 0.1% black iron oxide, 0.05% ferric ferrite, 0.05% titanium mica mixture (Manufacturing method) A: Dissolve and mix ingredients 29 to 31 uniformly at 70°C. B: Add ingredients 25 to 28 to A and mix uniformly using a roll mill. C: Add B to A and mix evenly. D: Add ingredients 1 to 11 to C and mix evenly. E: Mix ingredients 12 to 24 uniformly at room temperature. F: E was added to C and emulsified to obtain a water-in-oil liquid foundation. (evaluation) The water-in-oil liquid foundation of Example 3 was excellent in all respects: moisturizing feeling, sustained moisturizing feeling, and non-stickiness.

[0079] Example 4: Powder eye shadow Ingredients (%) 1. Spherical cellulose (average particle size 12 μm) 2 2. Spherical hollow silica (average particle size 5 μm) 1.5 3.Synthetic phlogopite 8 4. Zinc oxide (hexagonal plate shape, average particle size 0.3 μm) 3 5.2% Amodimethicone-treated mica remaining 6. Amino-modified silicone-treated talc *4 20 7. Glass powder ※5 13 8. Aluminum powder ※6 8 9. Red iron oxide coated titanium mica ※7 12 10. (PET / Methacrylate) Laminate 5 11. Cetyl ethylhexanoate 3 12. Diisostearyl malate 8 13. Sorbitan sesquistearate 0.5 14. Hydrogenated polyisobutene 2 15. Microcrystalline wax 1 16. Tripropylene glycol 0.2 17. Polyoxybutylene Polyoxyethylene Polyoxypropylene glyceryl ether (3BO)(8EO)(5PO) 0.3 18.Purified water 3 19. Niacinamide 1 20. Tranexamic acid 5 21. Sodium pyrosulfite 0.01 22. Aloe extract 0.01 23. Sophora Extract 0.001 24. Ascorbic acid 0.1 25. Polyethylene glycol 0.1 26. Alkyl acrylate / methacrylic acid copolymer 0.2 27. Glycerin 3 28. Quaternium-18 Hectorite 0.4 29. Phenoxyethanol 0.2 30. Chlorphenesin 0.3 *4: SE-TA-EX (manufactured by Miyoshi Chemicals) *5: Metashine MC2080PS (manufactured by Nippon Sheet Glass Co., Ltd.) *6: COSMICOLOR CE. TECLA GR (manufactured by Toyo Aluminum Co., Ltd.) *7: GEMTONE TAN OPAL G305 (manufactured by BASF) (Manufacturing method) A: Mix ingredients 16 to 30 evenly. B: Heat ingredients 11 to 15 to 90°C and dissolve uniformly. C: Mix ingredients 1 to 10 evenly. D: Add B to C and mix uniformly at room temperature. E: Add A to D at room temperature and mix to obtain a cosmetic composition. F: 60 parts by mass of 30% ethanol water is added to 100 parts by mass of the cosmetic composition to form a slurry. G:E was filled into a resin dish and compressed using a porous press head while removing the 30% ethanol water to obtain a solid powder eye shadow. (evaluation) The solid powder eye shadow of Example 4 was excellent in all respects: moisturizing feeling, sustained moisturizing feeling, and non-stickiness.

[0080] Example 5 Oily solid lip balm Ingredients (%) 1. Polyethylene 3 2. Microcrystalline wax 2 3. Fischer-Tropsch wax 5 4. Polybutene 6 5. Hydrogenated polyisobutene 3 6. Bis-diglyceryl polyacyladipate-2 4 7. Vaseline (melting point 58°C) 20 8. Dilinoleic acid di(phytosteryl / isostearyl) / Cetyl / Stearyl / Behenyl) 8 9. Dihydrogenated rosin dimer dilinoleyl 3 10. Diisostearyl malate 4 11. Polyglyceryl-2 Diisostearate 6 12. Polyglyceryl-2 triisostearate remaining 13. Polyglyceryl-10 Decaisostearate 2 14. Polyglyceryl-10 Pentaisostearate 1 15. Tranexamic acid 0.1 16. Niacinamide 2 17. Tripropylene glycol 2 18. Dipropylene glycol 1 19. Yarrow Extract 0.001 20. Cinnamon Water 1 21. Red No. 218 0.01 22. Red No. 223 0.03 23. Yellow No. 5 0.05 twenty four. (Manufacturing method) A: Heat ingredients 1 to 14 to 110°C and dissolve uniformly. B: Add ingredients 15 to 24 to A and mix uniformly at room temperature. C: B is heated to 90°C, filled into a stick container from the front, and cooled to -5°C. D: C was returned to room temperature to obtain an oily solid lip balm. (evaluation) The oil-based solid lip cream of Example 5 was excellent in all respects: moisturizing feeling, sustained moisturizing feeling, and non-stickiness.

[0081] Example 6 Ointment Ingredients (%) 1. Tranexamic acid 8 2. Niacinamide 0.8 3. Orange juice 0.001 4. Polyethylene glycol (average molecular weight 400) 1 5. Remaining purified water 6.1,3-Butylene glycol 3 7. Glycerin 4 8. Ethanol 8 9. Stearic acid 2 10. Stearyl alcohol 0.3 11. Behenyl alcohol 0.2 12. Vaseline 40 13. Lanolin 5 14. Fragrance (Citrus) 0.001 (Manufacturing method) A: Dissolve ingredients 1 to 8 uniformly at room temperature. B: Heat ingredients 9 to 14 to 60°C and mix uniformly. C: Add A to B at 80°C and emulsify. D: C was brought to room temperature and filled into a jar to obtain an ointment. (evaluation) The ointment of Example 6 was excellent in all respects: moisturizing feeling, sustained moisturizing feeling, and non-stickiness.

Claims

1. The following components (A) to (D'): (A) Tranexamic acid or a salt thereof (B) Niacinamide (C) at least one cosmetic ingredient selected from the group consisting of a plant of the genus Sophora of the family Fabaceae or an extract thereof, a plant of the genus Glycyrrhiza of the family Fabaceae or an extract thereof, a plant of the genus Achillea of ​​the family Asteraceae or an extract thereof, a plant of the genus Daucus of the family Apiaceae or an extract thereof, a plant of the genus Camellia of the family Theaceae or an extract thereof, a plant of the genus Aloe of the family Xanthomoniaceae or an extract thereof, a plant of the genus Eucalyptus of the family Myrtaceae or an extract thereof, a plant of the genus Citrus of the family Rutaceae or an extract thereof, and a plant of the genus Rosemary of the family Lamiaceae or an extract thereof (D') A skin preparation or cosmetic composition containing a polyhydric alcohol having 7 to 12 carbon atoms.

2. 2. The skin topical preparation or cosmetic according to claim 1, wherein a content mass ratio of the component (A) to the component (B) is (A) / (B) = 0.05 to 15, and a content mass ratio of the total amount of the component (A) and the component (B) to the component (C), [(A) + (B)] / (C), is 100 to 10,000.

3. The following components (A) to (C): (A) Tranexamic acid or a salt thereof (B) Niacinamide (C) at least one cosmetic ingredient selected from the group consisting of a plant of the genus Sophora of the family Fabaceae or an extract thereof, a plant of the genus Glycyrrhiza of the family Fabaceae or an extract thereof, a plant of the genus Achillea of ​​the family Asteraceae or an extract thereof, a plant of the genus Daucus of the family Apiaceae or an extract thereof, a plant of the genus Camellia of the family Theaceae or an extract thereof, a plant of the genus Aloe of the family Xanthomoniaceae or an extract thereof, a plant of the genus Eucalyptus of the family Myrtaceae or an extract thereof, a plant of the genus Citrus of the family Rutaceae or an extract thereof, and a plant of the genus Rosemary of the family Lamiaceae or an extract thereof A skin external preparation or cosmetic comprising: A skin external preparation or cosmetic composition (excluding a lotion having the following formulation (1) and excluding a milky lotion having the following formulation (2)) in which the content mass ratio of the component (A) to the component (B) is (A) / (B)=0.05 to 15, and the content mass ratio of the total amount of the component (A) and the component (B) to the component (C), [(A)+(B)] / (C), is 100 to 10,000. 【Table 1】 【Table 2】

4. The following components (A) to (C): (A) Tranexamic acid or a salt thereof (B) Niacinamide (C) at least one cosmetic ingredient selected from the group consisting of a plant of the genus Sophora of the family Fabaceae or an extract thereof, a plant of the genus Glycyrrhiza of the family Fabaceae or an extract thereof, a plant of the genus Achillea of ​​the family Asteraceae or an extract thereof, a plant of the genus Camellia of the family Theaceae or an extract thereof, a plant of the genus Aloe of the family Xanthomoniaceae or an extract thereof, a plant of the genus Eucalyptus of the family Myrtaceae or an extract thereof, and a plant of the genus Citrus of the family Rutaceae or an extract thereof A skin external preparation or cosmetic comprising: A skin external preparation or cosmetic, wherein the content mass ratio of the component (A) to the component (B) is (A) / (B)=0.05 to 15, and the content mass ratio of the total amount of the component (A) and the component (B) to the component (C), [(A)+(B)] / (C), is 100 to 10,000.

5. The skin external preparation or cosmetic preparation according to claim 3 or 4, further comprising component (D) a polyhydric alcohol having 5 to 12 carbon atoms.

6. The skin topical preparation or cosmetic preparation according to any one of claims 1, 2 and 5, wherein the component (D') or the component (D) is at least one polyhydric alcohol selected from the group consisting of tripropylene glycol and 1,2-octanediol.

7. The skin topical preparation or cosmetic according to any one of claims 1 to 6, wherein the content of the component (C) in the skin topical preparation or cosmetic is 0.0001 to 0.01 mass%.

8. The skin topical preparation or cosmetic according to any one of claims 1 to 7, wherein the mass ratio of the component (B) to the component (C) is (B) / (C) = 10 to 10,000.

9. The skin topical preparation or cosmetic according to any one of claims 1 to 8, wherein the mass ratio of the component (A) to the component (C) is (A) / (C) = 10 to 10,000.

10. A skin topical preparation or cosmetic composition described in any one of claims 1 to 9, further comprising, as component (E), an aqueous component excluding components (D) and (D').

11. A skin topical preparation or cosmetic preparation described in any one of claims 1 to 10, further containing component (F) a film-forming agent.

12. 2. A skin topical preparation or cosmetic composition comprising component (A) tranexamic acid or a salt thereof, component (B) niacinamide, and component (D') a polyhydric alcohol having 7 to 12 carbon atoms, comprising component (C) an agent for reducing stickiness by at least one cosmetic ingredient selected from the group consisting of a plant of the genus Sophora of the family Fabaceae or an extract thereof, a plant of the genus Glycyrrhiza of the family Fabaceae or an extract thereof, a plant of the genus Achillea of ​​the family Asteraceae or an extract thereof, a plant of the genus Daucus of the family Apiaceae or an extract thereof, a plant of the genus Camellia of the family Theaceae or an extract thereof, a plant of the genus Aloe of the family Xanthomoniaceae or an extract thereof, a plant of the genus Eucalyptus of the family Myrtaceae or an extract thereof, a plant of the genus Citrus of the family Rutaceae or an extract thereof, and a plant of the genus Rosemary of the family Lamiaceae or an extract thereof.

13. A method for improving stickiness in a skin topical preparation or cosmetic composition containing component (A) tranexamic acid or a salt thereof, component (B) niacinamide, and component (D') a polyhydric alcohol having 7 to 12 carbon atoms, using component (C) at least one cosmetic ingredient selected from the group consisting of a plant of the genus Sophora of the Leguminosae family or an extract thereof, a plant of the genus Glycyrrhiza of the Leguminosae family or an extract thereof, a plant of the genus Achillea of ​​the Asteraceae family or an extract thereof, a plant of the genus Daucus of the Umbelliferae family or an extract thereof, a plant of the genus Camellia of the Theaceae family or an extract thereof, a plant of the genus Aloe of the Xanthomoniaceae family or an extract thereof, a plant of the genus Eucalyptus of the Myrtaceae family or an extract thereof, a plant of the genus Citrus of the Rutaceae family or an extract thereof, and a plant of the genus Rosemary of the Lamiaceae family or an extract thereof.

14. In a skin topical preparation or cosmetic composition containing component (A) tranexamic acid or a salt thereof, and component (B) niacinamide, component (C) is a plant of the genus Sophora or an extract thereof of the genus Licorice of the genus Fabaceae or an extract thereof, a plant of the genus Achillea of ​​the genus Asteraceae or an extract thereof, a plant of the genus Daucus of the genus Daucus of the genus Camellia of the genus Theaceae or an extract thereof, a plant of the genus Aloe of the genus Xanthomoniaceae or an extract thereof, a plant of the genus Eucalyptus of the genus Myrtaceae or an extract thereof, a plant of the genus Citrus of the genus Rutaceae or an extract thereof, and a plant of the genus Mannonia of the genus Lamiaceae or an extract thereof A stickiness improving agent containing at least one or more cosmetic ingredients selected from the group consisting of plants of the genus Wax or extracts thereof, wherein the mass ratio of the components (A) and (B) is (A) / (B)=0.05 to 15, and component (C) is used so that the mass ratio of the total amount of the components (A) and (B) to the component (C), [(A)+(B)] / (C), is 100 to 10,000 (however, excluding a lotion having the following formulation (1) and excluding a milky lotion having the following formulation (2)). 【Table 3】 【Table 4】

15. In a skin topical preparation or cosmetic composition containing component (A) tranexamic acid or a salt thereof, and component (B) niacinamide, component (C) is a plant of the genus Sophora or an extract thereof of a plant of the genus Glycyrrhiza of the family Fabaceae, a plant of the genus Achillea or an extract thereof of a plant of the genus Yarrow of the family Asteraceae, a plant of the genus Daucus of the family Apiaceae or an extract thereof, a plant of the genus Camellia of the family Theaceae or an extract thereof, a plant of the genus Aloe of the family Xanthomoniaceae or an extract thereof, a plant of the genus Eucalyptus of the family Myrtaceae or an extract thereof, a plant of the genus Citrus of the family Rutaceae or an extract thereof, and a plant of Roseola of the family Lamiaceae A method for improving stickiness using at least one or more cosmetic ingredients selected from the group consisting of plants of the genus Corbicula or extracts thereof, the method using component (C) such that the content mass ratio of component (A) to component (B) is (A) / (B)=0.05 to 15, and the content mass ratio of the total amount of component (A) and component (B) to component (C), [(A)+(B)] / (C), is 100 to 10,000 (however, excluding lotions formulated as in the following formulation (1) and excluding emulsions formulated as in the following formulation (2)). 【Table 5】 【Table 6】

16. A stickiness-improving agent for a skin topical preparation or cosmetic preparation containing component (A) tranexamic acid or a salt thereof, and component (B) niacinamide, comprising component (C) at least one or more cosmetic ingredients selected from the group consisting of a plant of the genus Sophora of the family Fabaceae or an extract thereof, a plant of the genus Glycyrrhiza of the family Fabaceae or an extract thereof, a plant of the genus Achillea of ​​the family Asteraceae or an extract thereof, a plant of the genus Camellia of the family Theaceae or an extract thereof, a plant of the genus Aloe of the family Xanthomoniaceae or an extract thereof, a plant of the genus Eucalyptus of the family Myrtaceae or an extract thereof, and a plant of the genus Citrus of the family Rutaceae or an extract thereof, wherein the mass ratio of said component (A) to said component (B) is (A) / (B) = 0.05 to 15, and component (C) is used such that the mass ratio of the total amount of said component (A) and said component (B) to said component (C), [(A) + (B)] / (C), is 100 to 10,000.

17. A method for improving stickiness in a skin topical preparation or cosmetic preparation containing component (A) tranexamic acid or a salt thereof, and component (B) niacinamide, using component (C) at least one or more cosmetic ingredients selected from the group consisting of a plant of the genus Sophora of the family Fabaceae or an extract thereof, a plant of the genus Glycyrrhiza of the family Fabaceae or an extract thereof, a plant of the genus Achillea of ​​the family Asteraceae or an extract thereof, a plant of the genus Camellia of the family Theaceae or an extract thereof, a plant of the genus Aloe of the family Xanthomoniaceae or an extract thereof, a plant of the genus Eucalyptus of the family Myrtaceae or an extract thereof, and a plant of the genus Citrus of the family Rutaceae or an extract thereof, wherein the mass ratio of the content of component (A) to the content of component (B) is (A) / (B) = 0.05 to 15, and component (C) is used such that the mass ratio of the content of the total amount of component (A) and component (B) to component (C), [(A) + (B)] / (C), is 100 to 10,000.

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