Aminoquinolinones useful as CD38 inhibitors

Aminoquinolinones are developed to inhibit CD38, addressing the need for treating metabolic and other disorders by increasing cellular NAD levels, effectively managing conditions like obesity and diabetes.

WO2026143049A1PCT designated stage Publication Date: 2026-07-02NEOLAIA INC
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Patent Information

Application Number
PCT/US2025/060994
Authority / Receiving Office
WO · WO
Patent Type
Applications
Current Assignee / Owner
Priority Date
2025-07-15
Filing Date
2025-12-22
Publication Date
2026-07-02

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Abstract

The present invention relates to compounds that have activity as cluster of differentiation 38 (CD38) inhibitors, compositions of such compounds, and methods using such compounds for preventing or treating diseases and disorders such as, for example, diseases and disorders of metabolism.
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