Agrohorticultural pest control composition other than the water rice pest control composition and control method using the same

Abstract

The present application provides a novel agricultural and horticultural pest control composition having synergistic control effects in the cultivation of plants other than rice, and a control method using the same. The present application relates to an agricultural and horticultural pest control composition (other than a rice pest control composition) containing (A) saccharin and / or a salt thereof, and at least one plant treatment composition selected from (B) an insecticidally active compound and (C) a fungicidally active compound.

Description

Technical Field

[0001] This invention relates to agricultural and horticultural pest control compositions other than those for rice, and methods of pest control using the same. Background Technology

[0002] In the past, various pesticides were used to increase crop yields and improve crop quality. For example, in field cultivation, pests that need to be controlled include: plant pathogens causing soft rot, bacterial black spot, and downy mildew; plant pathogens such as viruses and viroids; pests belonging to the orders Coleoptera, Hemiptera, Diptera, Thysanoptera, and Lepidoptera; mollusks such as slugs; and nematodes such as southern root-knot nematodes. To date, many compositions and methods of application for controlling these pests have been proposed (e.g., Non-Patent Literature 1 and Patent Literature 1).

[0003] Non-patent literature 1 describes the effect of saccharin in inhibiting diseases caused by Zymoseptoria tritici in wheat. Thus, it is known that saccharin is effective against various plant diseases.

[0004] Patent Document 1 discloses a fungicide composition containing benzoyl pyraclostrobin and at least one fungicide selected from bifenthiophanate-methyl, fluopyram, fluopyram, pyraclostrobin, fluopyram, pyrimethanil, fluopyram, and fluopyram.

[0005] Existing technical documents Patent documents Patent Document 1: Japanese Patent Application Publication No. 2013-35823 Non-patent literature Non-patent literature 1: Samara Mejri, Plant disease, Vol. 105, No. 4, April 2021 Summary of the Invention The technical problem that the invention aims to solve Repeated use of a single fungicide leads to the emergence of bacteria resistant to that fungicide and related fungicides. Therefore, research is underway to develop safer fungicides and fungicide compositions that offer superior efficacy.

[0006] The objective of this invention is to provide a novel agricultural and horticultural pest control composition that has a synergistic control effect in the cultivation of plants other than rice, and a method for controlling pests using the same.

[0007] Technical solutions for solving technical problems In order to solve the above-mentioned problems, the inventors conducted repeated and in-depth research and found that by treating a composition made of saccharin, its salts, or mixtures thereof with an insecticide or fungicide, harmful organisms on plants other than rice can be effectively removed. This invention is based on this insight.

[0008] That is, the present invention is as follows.

[0009] Item 1. An agricultural and horticultural pest control composition (excluding a pest control composition for rice) contains: (A) saccharin and / or its salts, and A plant treatment composition selected from at least one of (B) insecticidal active compounds and (C) fungicidal active compounds.

[0010] Item 2. The agricultural and horticultural pest control composition according to claim 1 (excluding the rice pest control composition) comprises: the (A) saccharin and / or its salt, and the (C) bactericidal active compound.

[0011] Item 3. The agricultural and horticultural pest control composition according to item 1 or 2 (excluding the pest control composition for rice), wherein the (C) bactericidal active compound is an antibiotic for pesticide use.

[0012] Item 4. According to the agricultural and horticultural pest control composition of claim 3 (excluding the pest control composition for rice), the pesticide antibiotic comprises at least one antibiotic selected from chitin synthase inhibitors, enopyranuronic acid antibiotics, hexopyranosyl antibiotics, glucopyranosyl antibiotics, tetracycline antibiotics, and amphiphilic macrolide antifungal antibiotics.

[0013] Item 5. According to item 3 or 4, the agricultural and horticultural pest control composition (excluding the rice pest control composition) wherein the pesticide antibiotic is at least one compound selected from polyoxin, kasugamycin, validamycin, streptomycin and oxytetracycline or a salt thereof.

[0014] Item 6. The agricultural and horticultural pest control composition according to any one of items 3 to 5 (except for the pest control composition for rice), wherein the pesticide antibiotic is polyoxin or a salt thereof.

[0015] Item 7. The agricultural and horticultural pest control composition according to any one of items 1 to 6 (except for the rice pest control composition), wherein the (B) insecticidal active compound is at least one compound selected from the group consisting of: (b1) Acetylcholinesterase (AChE) inhibitors, (b2) GABA-gated chloride channel blockers, (b3) Sodium channel modulators, (b4) Competitive modulators of nicotinic acetylcholine receptors (nAChR), (b5) Nicotinic acetylcholine receptor (nAChR) allosteric modulator - site I, (b6) Glutamate-gated chloride channel (GluCl) allosteric modulator, (b7) Juvenile hormone analogues, (b8) Other non-specific (multi-site) inhibitors, (b9) String tuner TRPV channel modulator, (b10) A mite growth inhibitor that acts on CHS1. (b11) Microbial-derived insect peri-feeding membrane disruptors, (b12) Inhibitor of mitochondrial ATP synthase, (b13) Oxidative phosphorylation uncoupling agents that disrupt the proton gradient. (b14) Nicotinic acetylcholine receptor (nAChR) channel blockers, (b15) Chitin biosynthesis inhibitors acting on CHS1, (b16) Chitin biosynthesis inhibitor (type 1). (b17) Eclipsis inhibitor (Diptera insects). (b18) Ecdysone (ecdysone) receptor agonist, (b19) Octopus amine receptor agonist, (b20) The Qo site, an inhibitor of mitochondrial electron transport system complex III. (b21) Inhibitor of mitochondrial electron transport system complex I (METI). (b22) Voltage-dependent sodium channel blockers, (b23) Acetyl-CoA carboxylase inhibitor, (b24) Inhibitors of mitochondrial electron transport system complex IV. (b25) Inhibitors of mitochondrial electron transport system complex II, (b26) Ryedin receptor modulator, (b27) Nicotinamide enzyme inhibitor for string instruments, (b28) GABA-gated chloride channel allosteric modulator, (b29) Baculovirus, (b30) Nicotinic acetylcholine receptor (nAChR) allosteric modulator - site II, (b31) Calcium-activated potassium channel (KCa2) regulator, (b32) Qi site, an inhibitor of mitochondrial electron transport system complex III. (b33) RNA interference-mediated target repressor, (b34) String tuning agent (target location undetermined), and (b35) Agents with unknown or uncertain mechanisms of action: A. Bacterial agents (excluding BT agents) with unknown or uncertain mechanisms of action, synthetics with unknown or uncertain mechanisms of action, plant-derived ingredients containing extracts or unrefined oils, fungal agents with unknown or uncertain mechanisms of action, and physical disturbances with unknown or uncertain mechanisms of action. The bactericidal active compound (C) is at least one compound selected from the group consisting of: (c1) RNA polymerase I inhibitor, (c2) DNA / RNA biosynthesis inhibitors, (c3) Type II DNA topoisomerase (gyrase) inhibitor, (c4) An inhibitor of dihydroorotate dehydrogenase in the de novo biosynthesis of pyrimidines. (c5) Inhibitor of microtubule polymerization, (c6) Cell division inhibitor (site of action unknown), (c7) A translocator for spectrin-like proteins. (c8) Inhibitor of actin / myosin / filamentin function. (c9) Complex I (NADH oxidoreductase) inhibitor, (C10) Complex II (succinate dehydrogenase) inhibitor, (c11) Complex III (Qo site of ubiquitin oxidase) inhibitor, (c12) Complex III (ubiquinone reductase Qi site) inhibitor, (c13) An uncoupling agent for oxidative phosphorylation. (c14) Complex III (ubiquinone reductase Qo site marker-binding subsite) inhibitor, (c15) Methionine biosynthesis inhibitor, (c16) Inhibitor of protein biosynthesis (ribosomal translation initiation), (c17) Inhibitor of protein biosynthesis (ribosomal polypeptide elongation stage), (c18) Inhibitors of MAP / histidine kinases (os-2, HOG1) in osmolar signaling. (c19) Inhibitors of MAP / histidine kinases (os-1, Daf1) in osmolarity signaling. (c20) A methyltransferase inhibitor of phospholipid biosynthesis. (c21) Inhibitor of cellular lipid peroxidation, (c22) A cell membrane permeability fatty acid inhibitor. (c23) Inhibitors of lipid homeostasis and transport / storage, (c24) An inhibitor of C14 demethylase in sterol biosynthesis. (c25) An inhibitor of 3-keto reductase in the C4 demethylation of sterol biosynthesis. (c26) Squalene cyclooxygenase inhibitor in sterol biosynthesis, (c27) Chitin biosynthesis enzyme inhibitor, (c28) Cellulose biosynthesis enzyme inhibitor, (c29) An inhibitor of reductase in melanin biosynthesis. (c30) An inhibitor of dehydrating enzymes in melanin biosynthesis. (c31) A polyketide synthase inhibitor in melanin biosynthesis. (c32) Host plant resistance inducers (excluding saccharin or its salts). (c33) Compounds with unknown mechanisms of action. (c34) Multi-point contact active compounds, and (c35) Unclassified compounds.

[0016] Item 8. The agricultural and horticultural pest control composition according to any one of items 1 to 7 (except for the rice pest control composition), wherein the (B) insecticidal active compound is at least one compound selected from the group consisting of: (b1) Acetylcholinesterase (AChE) inhibitors, (b2) GABA-gated chloride ion (chloride element ion) channel blockers, (b3) Sodium channel modulators, (b4) Competitive modulators of nicotinic acetylcholine receptors (nAChR), (b5) Nicotinic acetylcholine receptor (nAChR) allosteric modulator - site I, (b9) String tuner TRPV channel modulator, (b14) Nicotinic acetylcholine receptor (nAChR) channel blockers, (b16) Chitin biosynthesis inhibitor (type 1). (b18) Ecdysone (ecdysone) receptor agonist, (b26) Ryedin receptor modulators, and (b33) Oxazosulfyl, benzpyrimoxan and isocycloserum; The bactericidal active compound (C) is at least one compound selected from the group consisting of: (c1) RNA polymerase I inhibitor, (c2) DNA / RNA biosynthesis inhibitors, (c3) Type II DNA topoisomerase (gyrase) inhibitor, (c4) An inhibitor of dihydroorotate dehydrogenase in the de novo biosynthesis of pyrimidines. (c5) Inhibitor of microtubule polymerization, (c6) Cell division inhibitor (site of action unknown), (C10) Complex II (succinate dehydrogenase) inhibitor, (c11) Complex III (Qo site of ubiquitin oxidase) inhibitor, (c12) Complex III (ubiquinone reductase Qi site) inhibitor, (c16) Inhibitor of protein biosynthesis (ribosomal translation initiation), (c17) Inhibitor of protein biosynthesis (ribosomal polypeptide elongation stage), (c20) A methyltransferase inhibitor of phospholipid biosynthesis. (c24) An inhibitor of C14 demethylase in sterol biosynthesis. (c27) Chitin biosynthesis enzyme inhibitor, (c29) An inhibitor of reductase in melanin biosynthesis. (c31) A polyketide synthase inhibitor in melanin biosynthesis. (c32) Host plant resistance inducers (excluding saccharin or its salts). (c33) Compounds with unknown mechanisms of action. (c34) Multi-point contact active compounds, and (c35) Fluopyram.

[0017] Item 9. A method for controlling pests (excluding pest control methods for rice) includes the following steps: applying a composition to a pest, a habitat of the pest, a plant or a plant cultivation carrier, said composition containing: (A) saccharin and / or its salts, and at least one plant treatment composition selected from (B) an insecticidal active compound and (C) a fungicide active compound.

[0018] Item 10. The use of a composition in the control of pests in agriculture and horticulture (excluding the use for the control of pests in rice), wherein the composition contains: (A) saccharin and / or its salt, and at least one plant treatment composition selected from (B) an insecticidal active compound and (C) a fungicide active compound.

[0019] Invention Effects According to the present invention, a novel pest control composition for agricultural and horticultural use (excluding pest control compositions for rice) is provided, which exhibits a significant synergistic effect on plant disease control that cannot be predicted from the plant disease control effects obtained by using saccharin or its salts and mixtures alone or by using plant treatment compositions alone. Detailed Implementation

[0020] Agricultural and horticultural pest control compositions (excluding pest control compositions for rice). The agricultural and horticultural pest control composition of the present invention (excluding the pest control composition for rice) (hereinafter sometimes also referred to as "the composition of the present invention") contains: (A) Saccharin and / or its salts, and A plant treatment composition selected from at least one of (B) insecticidal active compounds and (C) fungicidal active compounds.

[0021] The agricultural and horticultural pest control composition of the present invention (excluding the pest control composition for rice) exerts excellent pest control effect in the cultivation of plants other than rice by using (A) saccharin and / or its salt in combination with at least one plant treatment composition selected from (B) insecticidal active compounds and (C) fungicidal active compounds.

[0022] (A) Saccharin and / or its salts Saccharin (1,1-dioxo-1,2-benzothiazol-3-one) is a compound represented by formula (1). Saccharin is commonly used as an artificial sweetener, but it is known to have resistance-inducing activity, and can exert a disease-inhibiting effect by inducing resistance to host plant diseases (activation of the disease control system).

[0023] [Chemistry 1] Where permitted in agriculture, the salt for saccharin can be any kind of salt. Examples of such salts include inorganic acids (e.g., hydrochlorides, sulfates, nitrates, etc.), organic acids (e.g., acetates, methanesulfonates, etc.), alkali metal salts (e.g., sodium salts, potassium salts, etc.), alkaline earth metal salts (e.g., calcium salts, etc.), quaternary ammonium salts (e.g., tetramethylammonium salts, tetraethylammonium salts, etc.), with alkali metal salts being preferred, and sodium salts being more preferred.

[0024] The application rate and concentration of the composition of the present invention can be varied according to weather conditions, application time, application location, application method, etc. The application rate of saccharin and / or its salts is usually 0.05~300 g / a, preferably 0.1~100 g / a, and more preferably 0.15~50 g / a. However, the application to crops before transplanting in plug trays, seedling pots, etc., is not limited to this.

[0025] Plant treatment compositions The compositions of the present invention comprise at least one plant treatment composition selected from (B) insecticidal active compounds and (C) fungicidal active compounds.

[0026] (B) Insecticidal compounds The agricultural and horticultural pest control compositions of the present invention (excluding rice pest control compositions) may contain known compounds that are effective against agricultural pests, without particular limitation. The insecticidal active compounds referred to herein include not only insecticides but also acaricides and nematicides. The aforementioned insecticidal active compounds may be used alone or in appropriate mixtures of two or more.

[0027] As for (B) insecticidal active compounds, there are no particular limitations. For example, compounds belonging to Groups 1 to 36 and Groups UN to UNM in the IRAC (Insecticide Resistance Action Committee) classification of action can be cited.

[0028] (b1) Group 1: Acetylcholinesterase (AChE) inhibitors Examples of acetylcholinesterase (AChE) inhibitors include: alanycarb, aldicarb, bendiocarb, benfuracarb, butocarboxim, butoxycarboxim, carbaryl (NAC), carbofuran, carbosulfan, ethiofencarb, fenobucarb (BPMC), formetanate, and furatin. Carbamate compounds (1A) including hiocarb, isoprocarb (MIPC), methiocarb, methomyl, metolcarb (MTMC), oxamyl, pirimicarb, propoxur (PHC), thiodicarb, thiofanox, triazamate, trimethacarb, XMC, and xylylcarb (MPMC); acephate. Azamethiphos, azinphos-ethyl, azinphos-methyl, cadusafos, chlorethoxyfos, chlorfenvinphos (CVP), chlormephos, chlorpyrifos, chlorpyrifos-methyl, coumaphos, cyanophos (CYAP), and demeton-S-methyl. Diazinon, dichlorvos (DDVP), dicrotophos, dimethoate, dimethylvinphos, disulfoton, EPN, ethion, ethoprophos, famur, fenamiphos, fenitrothion (MEP), fenthion (MPP), fosthiazate, and heptenophos.Imicafos, isofenphos, isopropyl-O-(methoxyaminothiophosphoryl)salicylate, isoxathion, malathion, mecarbam, methamidophos, methidathion (DMTP), mevinphos, monocrotophos, naled (BRP), omethoate, oxydemeton-methyl, parathion, parathion-methyl, phenthoate (PAP), phorate, p-methazophos (P-methazophos) Organophosphorus compounds (1B), including hosalone, phosmet (PMP), phosphamidon, phoxim, pirimiphos-methyl, profenofos, propetamphos, prothiofos, pyraclofos, pyridaphenthion, quinalphos, sulfotep, tebupirimfos, temephos, terbufos, tetrachlorvinphos (CVMP), thiometon, triazophos, trichlorfon (DEP), and vamidothion.

[0029] (b2) Group 2: GABA-gated chloride ion (chloride element ion) channel blockers Examples of GABA-gated chloride ion (chloride element ion) channel blockers include: cyclodiene organochlorine compounds such as chlordane and endosulfan (2A); and phenylpyrazole compounds such as ethiprole and fipronil (2B).

[0030] (b3) Group 3: Sodium channel modulators Examples of sodium channel modulators include: acrinathrin, allethrin (d-cis-trans-, d-trans-isomer), bifenthrin, bioallethrin (S-cyclopentenyl-isomer), bioresmethrin, cycloprothrin, and lambda-cyhalothrin. β -Isomer) (cyfluthrin), cyfluthrin (cyfluthrin, -isomer) λ -、 γ -Isomers (cyhalothrin), cypermethrin (cypermethrin, including...) α -、 β -、 θ -、 ζ -Isomers (cypermethrin), cyphenothrin [(1R)-trans isomer], deltamethrin, empenthrin [(EZ)-(1R)-trans isomer], esfenvalerate, etofenprox, fenpropathrin, fenvalerate, flucythrinate, flumethrin, cypermethrin τ pyrethroid compounds (3A) including fluvalinate, halfenprox, imiprothrin, kadethrin, permethrin, phenothrin ((1R)-trans isomer), prallethrin, pyrethrins, resmethrin, silafluofen, tefluthrin, tetramethrin, tetramethrin ((1R)-trans isomer), tralomethrin, and transfluthrin; DDT and methoxyDDT (3B), etc.

[0031] (b4) Group 4: Competitive modulators of nicotinic acetylcholine receptors (nAChR) As competitive regulators of nicotinic acetylcholine receptors (nAChR), examples include: neonicotinoids such as acetamiprid, clothianidin, dinotefuran, imidacloprid, nitenpyram, thiacloprid, and thiamethoxam (4A); nicotinoids such as nicotinic sulfate (4B); sulfoxide imines such as sulfoxaflor (4C); butenolates such as flupyradifurone (4D); metronidazoles such as dicloromezotiazine, fenmezoditiazine, and triflumezopyrim (4E); and pyridine subunits such as flupyrimin (4F).

[0032] (b5) Group 5: Nicotinic acetylcholine receptor (nAChR) allosteric modulators - Site I Examples of allosteric regulators of nicotinic acetylcholine receptors (nAChR) – site I include spinosomal compounds such as spintoram and spinosad.

[0033] (b6) Group 6: Allosteric regulators of glutamate-gated chloride channels (GluCl) Examples of allosteric regulators of glutamate-gated chloride channels (GluCl) include abamectin and other avermectin-like compounds, emamectin-benzoate, lepimectin, milbemectin, and other milbemectin-like compounds.

[0034] (b7) Group 7: Juvenile hormone analogs Examples of juvenile hormone analogs include: hydroprene, kinoprene, and methoprene (7A); fenoxycarb (7B); and pyriproxyfen (7C).

[0035] (b8) Group 8: Other non-specific (multi-site) inhibitors Other non-specific (multi-site) inhibitors include, for example: 1,3-dichloropropene, methyl bromide, and other halogenated alkyl compounds (8A); chloropicrin (8B); fluoride compounds such as cryolite and sulfurylfluoride (8C); borates such as borax, boric acid, disodium octaborate, sodium borate, and sodium metaborate (8D); tartaric acid (8E); methyl isothiocyanate generating agents such as dazomet, metam, and methyl isothiocyanate (8F), etc.

[0036] (b9) Group 9: String Instrument TRPV Channel Adjuster Examples of TRPV channel modulators for string instruments include pyridine diimide derivatives such as pymetrozine and pyrifluquinazon (9B); and pyropene compounds such as afidopyropen (9D).

[0037] (b10) Group 10: Mite growth inhibitors acting on CHS1 Examples of mite growth inhibitors that act on CHS1 include: clofentezine, diflovidazin, hexythiazox, etc. (10A); etoxazole (10B), etc.

[0038] (b11) Group 11: Insects of Microbial Origin Perinatal membrane Destroyer Examples of microbial insect peritrophic membrane disruptors include: Bacillus thuringiensis subsp. Israel (Bt). Bacillus thuringiensis subsp. israelensis Bacillus thuringiensis subsp. tumefaciens ( Bacillus thuringiensis subsp. Aizawai ), Bacillus thuringiensis Kustack subspecies ( Bacillus thuringiensis subsp. Kurstaki ), Bacillus thuringiensis subsp. *Tenomorphus* ( Bacillus thuringiensis subsp. tenebrionis(Proteins contained in Bt crops: Cry1Ab, Cry1Ac, Cry1Fa, Cry1A.105, Cry2Ab, Vip3A, mCry3A, Cry2Ab, Cry3Bb, Cry34Ab1 / Cry35Ab1, etc.) Bacillus thuringiensis ( Bacillus thuringiensis ) and the insecticidal proteins it produces (11A); Bacillus spheroidae ( Bacillus sphaericus (11B) etc.

[0039] (b12) Group 12: Inhibitors of mitochondrial ATP synthase Examples of mitochondrial ATP synthase inhibitors include: diafenthiuron (12A); organotin acaricides such as azocyclotin, cyhexatin, and fenbutatin oxide (12B); propargite (BPPS) (12C); and tetradifon (12D).

[0040] (b13) Group 13: Oxidative phosphorylation uncoupling agents that disrupt the proton gradient Examples of oxidative phosphorylation uncoupling agents that disrupt the proton gradient include pyrrole compounds such as chlorfenapyr; dinitrophenol compounds such as DNOC; and sulfluramid.

[0041] (b14) Group 14: Nicotinic acetylcholine receptor (nAChR) channel blockers Examples of nephrotic acetylcholine receptor (nAChR) channel blockers include bensultap, cartap hydrochloride, thiocyclam, and thiosultapsodium, which are analogues of nereistoxins.

[0042] (b15) Group 15: Chitin biosynthesis inhibitors acting on CHS1 Examples of chitin biosynthesis inhibitors that act on CHS1 include bistrifluron, chlorfluazuron, diflubenzuron, flucycloxuron, flufenoxuron, hexaflumuron, lufenuron, novaluron, noviflumuron, teflubenzuron, and triflumuron.

[0043] (b16) Group 16: Chitin biosynthesis inhibitors (type 1) Examples of chitin biosynthesis inhibitors (type 1) include buprofezin.

[0044] (b17) Group 17: Ecstasy inhibitors (Diptera) As a molting inhibitor ( Diptera Insects), for example, cyromazine, etc.

[0045] (b18) Group 18: Ecdysone (ecdysone) receptor agonists Examples of ecdysone (ecdysone) receptor agonists include diacylhydrazine compounds such as chromafenozide, halofenozide, methoxyfenozide, and tebufenozide.

[0046] (b19) Group 19: Octopus amine receptor agonists Examples of octopamine receptor agonists include amitraz.

[0047] (b20) Group 20: Inhibitors of mitochondrial electron transport system complex III - Qo site Examples of inhibitors of the mitochondrial electron transport system complex III-Qo site include: hydramethylnon (20A), acequinocyl (20B), fluacrypyrim (20C), and bifenazate (20D).

[0048] (b21) Group 21: Inhibitors of mitochondrial electron transport system complex I (METI) Examples of METI inhibitors (Mitochondrial electron transport system complex I) include: fenazaquin, fenpyroximate, pyridaben, pyrimidifen, tebufenpyrad, tolfenpyrad, etc. (21A); rotenone (21B), etc.

[0049] (b22) Group 22: Voltage-dependent sodium channel blockers Examples of voltage-dependent sodium channel blockers include oxadiazine compounds such as indoxacarb (22A) and acetamiprid compounds such as metaflumizone (22B).

[0050] (b23) Group 23: Acetyl-CoA carboxylase inhibitors Examples of acetyl-CoA carboxylase inhibitors include spirodiclofen, spiromesifen, spiropidion, spirotetramat, and other tetronic acid or tetramic acid derivatives.

[0051] (b24) Group 24: Inhibitors of mitochondrial electron transport system complex IV Examples of inhibitors of mitochondrial electron transport system complex IV include: phosphine compounds such as aluminum phosphide, calcium phosphide, phosphine, and zinc phosphide (24A); and cyanides such as hydrogen cyanide (calcium cyanide, sodium cyanide) and potassium cyanide (24B).

[0052] (b25) Group 25: Inhibitors of mitochondrial electron transport system complex II Examples of inhibitors of mitochondrial electron transport system complex II include cyenopyrafen and cyflumetofen. β - Ketone nitrile derivatives (25A); carboxylaniline compounds such as pyflubumide (25B), etc.

[0053] (b26) Group 28: Ryedin receptor modulators Examples of ryanodine receptor modulators include diamide compounds such as chlorantraniliprole, cyantraniliprole, cycloniliprole, flubendiamide, and tetrazolium.

[0054] (b27) Group 29: String tuner Examples of string tuning agents include flonicamid.

[0055] (b28) Group 30: GABA-gated chloride channel allosteric modulators Examples of GABA-gated chloride channel allosteric modulators include: broflanilide and other diamide compounds, and fluxametamide, isoxazoline compounds, and isoxazoline compounds.

[0056] (b29) Group 31: Baculoviruses Examples of baculoviruses include: codling moth (Acer palmatum) Cydia pomonella GV, false apple codling moth ( Thaumatotibia leucotreta GV and other particulate viruses (GVs); soybean cutworm ( Anticarsia gemmatalis ) MNPV, cotton bollworm ( Helicoverpa armigera Nucleopolyhedroviruses (NPVs), etc.

[0057] (b30) Group 32: Nicotinic acetylcholine receptor (nAChR) allosteric modulators - Part II Examples of allosteric regulators of nicotinic acetylcholine receptors (nAChR) at site II include GS-ω / κHXTX-Hv1a peptide.

[0058] (b31) Group 33: Calcium-activated potassium channel (KCa2) regulators Examples of calcium-activated potassium channel (KCa2) regulators include acynonapyr.

[0059] (b32) Group 34: Mitochondrial electron transport system complex III inhibitor - Qi site Examples of inhibitors of the mitochondrial electron transport system complex III, such as the Qi site, include floctoquin.

[0060] (b33) Group 35: RNA interference-mediated target inhibitors Examples of RNA interference-mediated target inhibitors include Ledprona.

[0061] (b34) Group 36: String tuning agent (target location undetermined) As a modulator of string instruments (target site not determined), examples include pyridazines such as dimpropyridazine or pyrazole carboxamides.

[0062] (b35) Group UN: Drugs with unknown or unclear mechanisms of action A Examples of agents A with unclear or unknown mechanisms of action include azadirachtin, benzoximate, benzpyrimoxan, bromopropylate, quinomethionat, dicofol, lime sulfur, mancozeb, oxazosulfyl, pyridalyl, and sulfur.

[0063] (b36) Group UNB: Bacterial agents with unknown or unclear mechanisms of action (excluding BT agents) As bacterial agents with unknown or unclear mechanisms of action (excluding BT agents), examples include Burkholderia spp. ( Burkholderia spp.), Papidiswabachian body ( Wolbachia pipientis (Zap), etc.

[0064] (b37) Group UNE: Synthetic compounds with unknown or unclear mechanisms of action, and plants containing extracts or unrefined oils. Source ingredients As a synthetic compound with an unknown or unclear mechanism of action, or a plant-derived ingredient containing extracts or unrefined oils, examples include American purslane (…). Chenopodium ambrosioides near ambrosioides Extracts of neem seeds, glycerol or propylene glycol fatty acid monoesters in neem oil, etc.

[0065] (b38) Group UNF: Fungal agents with unknown or unclear mechanisms of action As fungicides with unclear or unknown mechanisms of action, examples include *Scabies flocculationii* (Fly scale fungus). Akanthomyces muscarius ) Ve6, Beauveria bassiana strain ( Beauveria bassiana strains), Metarhizium anisopliae strains ( Metarhizium brunneum strain) F52, *Paecilomyces rosenbergii* strain ( Paecilomyces fumosoroseus Apopka strain) 97, etc.

[0066] (b39) Group UNM: Non-specific physical disturbances with unknown or unclear mechanisms of action Examples of non-specific physical disturbances with unclear or unknown mechanisms of action include diatomaceous earth and mineral oil.

[0067] In addition, well-known agricultural and horticultural pesticides can be cited as examples. These insecticidal active compounds are well-known compounds, commercially available, and therefore readily available.

[0068] In this invention, relative to 100 parts by weight of (A) saccharin and / or its salt, 0.01 to 20,000 parts by weight, preferably 0.1 to 10,000 parts by weight, and more preferably 0.5 to 1,000 parts by weight of (B) insecticidal active compound are typically added.

[0069] (C) Bactericidal active compounds The agricultural and horticultural pest control compositions of the present invention (excluding rice pest control compositions) may contain bactericidal active compounds, including compounds known to be effective against agricultural pests, without particular limitation. Here, the bactericidal active compounds include not only fungicides but also bactericides and antiviral agents. The aforementioned bactericidal active compounds may be used alone or in appropriate mixtures of two or more.

[0070] As for (C) fungicidal active compounds, there are no particular limitations. For example, in the FRAC (Fungicide Resistance Action Committee) classification of action, compounds belonging to A (nucleic acid synthesis and metabolism), B (cytoskeleton and motor proteins), C (respiration), D (amino acid and protein biosynthesis), E (signal transduction), F (lipid biosynthesis or transport / cell membrane structure or function), G (cell membrane sterol biosynthesis), H (cell wall biosynthesis), I (cell wall melanin biosynthesis), P (host plant resistance induction), M (multi-site contact active compounds), BM (biopesticides with multiple mechanisms of action: plant extracts), U (unknown mechanism of action), and unclassified compounds are preferred. Among these, the following groups are preferred: A, B, C, D, F, G, I, P, M, and U.

[0071] Group A As a group A (nucleic acid synthesis metabolism), examples include: RNA polymerase I inhibitors, adenosine deaminase, DNA / RNA biosynthesis inhibitors, type II DNA topoisomerase (gyrase) inhibitors, and dihydroorotate dehydrogenase inhibitors in the de novo biosynthesis of pyrimidines.

[0072] (c1) Group A1: RNA polymerase I inhibitor (FRAC group code 4) Examples of RNA polymerase I inhibitors include: acylalanine derivatives such as benalaxyl, benalaxyl-M, furaxyl, metalaxyl, and metalaxyl-M; oxadixyl derivatives such as oxadixyl; and butyrolactone derivatives such as ofuronide.

[0073] (c2) Group A2: Adenosine deaminase inhibitor (FRAC group code 8) Examples of adenosine deaminase inhibitors include hydroxy(2-amino)pyrimidines such as bupirimate, dimethirimol, and ethirimol.

[0074] (c3) Group A3: DNA / RNA biosynthesis inhibitors (FRAC group code 32) As inhibitors of DNA / RNA biosynthesis, examples include isoxazoles such as hymexazole and isothiazolinones such as octhilinone.

[0075] (c4) Group A4: Type II DNA topoisomerase (gyrase) inhibitor (FRAC group code 31) As a type II DNA topoisomerase ( Gyrase Inhibitors, such as carboxylic acids like oxolinic acid, are examples.

[0076] (c5) Group A5: Dihydroorotate dehydrogenase inhibitors in the de novo biosynthesis of pyrimidines (FRAC group code 52) Examples of dihydroorotate dehydrogenase inhibitors used in the de novo biosynthesis of pyrimidines include phenylpropanols such as ipflufenoquin and dihydroisoquinolines such as quinofumelin.

[0077] Group B As part of group B (cytoskeleton and motor proteins), examples include microtubule polymerization inhibitors, cell division (site of action unknown) inhibitors, spectrin-like protein translocators, actin / myosin / filamentin function inhibitors, and microtubule dynamics modulators.

[0078] (c6) Groups B1, B2, and B3: Microtubule polymerization inhibitors (FRAC group codes 1, 10, and 22) As β Microtubule polymerization inhibitors can be categorized as follows: benzimidazoles such as benomyl, carbendazim, fuberidazole, and thiabendazole; thiophanates such as thiophanate-methyl; N-phenylcarbamates such as diethofencarb; toluamides such as zoxamide; and ethylaminothiazole carbamates such as ethaboxam.

[0079] (c7) Group B4: Cell division (site of action unknown) inhibitor (FRAC group code 20) As inhibitors of cell division (with unclear sites of action), examples include phenylurea such as pencycuron.

[0080] (c8) Group B5: Spectrolin-like protein transposition agent (FRAC Group Code 43) Examples of translocators for spectroscopy-like proteins include pyridyl methylbenzamides such as fluopicolide and fluopimomide.

[0081] (c9) Group B6: Inhibitor of actin / myosin / filamentin function (FRAC group code 47) Examples of inhibitors of actin / myosin / filament protein function include: aminocyanoacrylates such as phenamacril; benzophenones such as metrafenone; and benzoylpyridines such as pyriofenone.

[0082] (c10) Group B7: Microtubule dynamics regulator (FRAC group code 53) Examples of microtubule kinetic regulators include pyridachlometyl and other pyridazine derivatives.

[0083] Group C For example, in Group C (respiration), inhibitors include: Complex I (NADH oxidoreductase) inhibitors, Complex II (succinate dehydrogenase) inhibitors, Complex III (cytochrome bc1 (ubiol oxidase) Qo site (cytb gene)) inhibitors, Complex III (ubiquinone reductase Qi site) inhibitors, oxidative phosphorylation uncoupling agents, oxidative phosphorylation, ATP synthase inhibitors, ATP transport inhibitors, and Complex III (ubiquinone reductase Qi and Qo sites, stigmatellin binding mode) inhibitors, etc.

[0084] (c11) Group C1: Complex I (NADH oxidoreductase) inhibitor (FRAC group code 39) Examples of inhibitors of complex I (NADH oxidoreductase) include: pyrimidine amines such as diflumetorim; pyrazole carboxamides such as tolfenpyrad; and quinazolines such as fenazaquin.

[0085] (c12) Group C2: Complex II (succinate dehydrogenase) inhibitor (FRAC group code 7) Examples of inhibitors of complex II (succinate dehydrogenase) include: phenylbenzamides such as benodanil, flutolanil, and mepronil; phenoxyethyl thiophenamides such as isofetamid; pyridylethyl benzamides such as fluopyram; phenylcyclobutylpyridinamides such as cyclobutrifluram; furanamides such as fenfuram; oxicarboxin and other oxothiacyclohexadiene carboxamides; thiazole carboxamides such as thifluzamide; and benzovindiflupyr and bifenthiopyr. Amines such as bixafen, fluindapyr, fluxapyroxad, furamepyr, inpyrfluxam, and isopyrazam; pyrazole-4-carboxamides such as penflufen, penthiopyrad, and sedaxane; N-cyclopropyl-N-benzylpyrazolecarboxamides such as isoflucypram; N-methoxy(phenylethyl)pyrazolecarboxamides such as pydiflumetofen; pyridinecarboxamides such as boscalid; and pyraziflumide; etc.

[0086] (c13) Group C3: Complex III (cytochrome bc1 (panthenol oxidase) Qo site (cytb gene)) inhibitor As inhibitors of Complex III (cytochrome bc1 (panthenol oxidase) Qo site (cytb gene)) (QoI fungicides (Qo inhibitors)) (FRAC group code 11), examples include: methoxyacrylates such as azoxystrobin, coumoxystrobin, enoxastrobin, flufenoxystrobin, picoxystrobin, and pyraoxystrobin; methoxyacetamides such as mandestrobin; and pyraclostrobin and pyrametostrobin. Methoxycarbamates such as chlorpyrifos (triclopyricarb); oxyiminoacetic acids such as kresoxim-methyl and trifloxystrobin; oxyiminoacetamides such as dimoxystrobin, fenaminstrobin, metominostrobin, and orysastrobin; oxazolidinones such as famoxadone; dihydrodioxazines such as fluoxastrobin; imidazolinones such as fenamidone; and benzylcarbamates such as pyribencarb.

[0087] In addition, examples of QoI bactericides (Qo inhibitors; subgroup A) (FRAC group code 11A) include tetrazolinones such as methyl tetrapyrrole.

[0088] (c14) Group C4: Complex III (ubiquinone reductase Qi site) inhibitor (FRAC group code 21) Examples of inhibitors of complex III (ubiquinone reductase Qi site) include: cyanoimidazoles such as cyazofamid; aminosulfonyl triazoles such as amisulbrom; and pyridine carboxamides such as fenpicoxamid and florylpicoxamid.

[0089] (c15) Group C5: Oxidative phosphorylation uncoupling agents (FRAC group code 29) Examples of uncoupling agents for oxidative phosphorylation include: dinitrophenyl crotonic acids such as BINAPACRIL, meptyl dinocap, and DPC; 2,6-dinitroaniline derivatives such as fluazinam; and pyrimidinone hydrazones such as ferimzone.

[0090] (c16) Group C6: Inhibitor of oxidative phosphorylation and ATP synthase (FRAC group code 30) As inhibitors of oxidative phosphorylation and ATP synthase, examples include organotin compounds such as triphenyltin (triphenyltin acetate, triphenyltin chloride, triphenyltin hydroxide), etc.

[0091] (c17) Group C7: ATP transport inhibitor (FRAC group code 38) Examples of ATP transport inhibitors include thiophene formamides such as silthiofam.

[0092] (c18) Group C8: Complex III (ubiquinone reductase Qi, Qo sites, and FRAC binding mode) inhibitor (FRAC) Group code 45) As inhibitors of complex III (ubiquinone reductase Qi, Qo sites, and marker binding mode), examples include triazolopyrimidine amines such as ametoctradin.

[0093] Group D As group D (amino acid and protein biosynthesis inhibitors), examples include: methionine biosynthesis (cgs gene) inhibitors, protein biosynthesis (ribosomal translation termination stage) inhibitors, protein biosynthesis (ribosomal translation initiation stage) inhibitors, protein biosynthesis (ribosomal polypeptide elongation stage) inhibitors, leucyl-tRNA synthesis (Leu RNA) inhibitors, etc.

[0094] (c19-1) Group D1: Methionine biosynthesis (cgs gene) inhibitor (FRAC group code 9) As inhibitors of methionine biosynthesis (cgs gene), examples include phenylamine pyrimidines such as cyprodinil, mepanipyrim, and pyrimethanil.

[0095] (c19-2) Group D2: Inhibitor of protein biosynthesis (ribosomal translation termination stage) (FRAC group code 23) Examples of inhibitors of protein biosynthesis (the termination stage of ribosomal translation) include genistein antibiotics such as blastomycin S.

[0096] (c19-3) Group D3: Inhibitor of protein biosynthesis (ribosomal translation initiation) (FRAC group code 24) Group D4: Inhibitors of protein biosynthesis (ribosomal translation initiation) (FRAC group code 25) Examples of inhibitors of protein biosynthesis (the initiation of ribosomal translation) include: hexopyranosyl antibiotics such as kasugamycin; and glucopyranosyl antibiotics such as streptomycin.

[0097] (c19-4) Group D5: Inhibitor of protein biosynthesis (ribosomal polypeptide elongation stage) (FRAC group code 41) As inhibitors of protein biosynthesis (ribosomal polypeptide elongation stage), examples include tetracycline antibiotics such as oxytetracycline.

[0098] (c19-5) Group D6: Leucyl-tRNA synthesis inhibitor (FRAC group code 54) Examples of inhibitors of leucyl-tRNA synthesis include benzoxadiborane and tavaborole.

[0099] Group E As a group E (signal transduction), examples include inhibitors of signal transduction (with unclear mechanisms of action), inhibitors of MAP / histidine kinases (os-2, HOG1) in osmolarity signal transduction, and inhibitors of MAP / histidine kinases (os-1, Daf1) in osmolarity signal transduction.

[0100] (c20) Group E1: Signal transduction (mechanism of action unknown) inhibitor (FRAC group code 13) As signal transduction inhibitors (with unclear mechanisms of action), examples include aryloxyquinolines such as quinoxyfen and quinazolinones such as proquinazid.

[0101] (c21) Group E2: MAP / histidine kinase (os-2, HOG1) inhibitors in osmolarity signal transduction (FRAC group) Code 12) As inhibitors of MAP / histidine kinases (os-2, HOG1) in osmotic signal transduction, examples include phenylpyrroles such as fenpiclonil and fludioxonil.

[0102] (c22) Group E3: MAP / histidine kinase (os-1, Daf1) inhibitors in osmolarity signal transduction (FRAC group) Code 2) As inhibitors of MAP / histidine kinases (os-1, Daf1) in osmotic signal transduction, examples include dicarboxylides such as chlozolinate, dimethachlone, iprodione, procymidone, and vinclozolin.

[0103] Group F As an F group (inhibitors of lipid biosynthesis or transport / cell membrane structure or function), examples include methyltransferase inhibitors of phospholipid biosynthesis, peroxidation inhibitors of cellular lipids, fatty acid inhibitors of cell membrane permeability, ergosterol binders, inhibitors of lipid homeostasis and transport / storage, inhibitors of interactions with cell membrane lipid components, and inhibitors of various effects on the cell membrane.

[0104] (c23) F2: Phospholipid biosynthesis methyltransferase inhibitor (FRAC group code 6) Examples of methyltransferase inhibitors for phospholipid biosynthesis include: thiophosphates such as EDDP (edifenphos), IBP (iprobenfos), and pyrazophos; and dithiopentanes such as isoprothiolane.

[0105] (c24) group F3: Inhibitor of cellular lipid peroxidation (FRAC group code 14) As inhibitors of cellular lipid peroxidation, examples include aromatic hydrocarbons such as biphenyl, chloroneb, dicloran (CNA), quintozene (PCNB), tecnazen (tetrachloronitrobenzen), and tolclofos-methyl; and 1,2,4-thiadiazoles such as etridiazole.

[0106] (c25) group F4: Cell membrane permeability fatty acid inhibitor (FRAC group code 28) Fatty acid inhibitors that impede cell membrane permeability include, for example, prothiocarb, iodocarb, propamocarb, and other carbamates.

[0107] (c26) Group F8: Ergosterol binder (FRAC group code 48) Examples of ergosterol binding agents include: natamycin (a type of phytosalicylate) and other actinomycetes such as Streptomyces natalum. Streptomyces natalensis ) or Streptomyces chatanuga ( S. chattanoogensis Amphiphilic macrolide antifungal antibiotics, etc.

[0108] (c27) Group F9: Inhibitors of lipid homeostasis and transfer / storage (FRAC group code 49) Inhibitors of lipid homeostasis and transfer / storage include, for example, piperidinyl thiazolinone, fluoxapiprolin, and other isoxazoline derivatives.

[0109] (c28) group F10: Interaction with cell membrane lipid components, inhibitors of multiple cell membrane effects (FRAC group) Code 51) Examples of inhibitors of the interaction with cell membrane lipid components and various effects on the cell membrane include peptides such as ASFBIOF01-02.

[0110] Group G As group G (inhibitors of sterol biosynthesis in the cell membrane), examples include inhibitors of C14 demethylases (erg11 / cyp51) in sterol biosynthesis, and inhibitors of Δ... 14 reductase and Δ 8 →Δ 7 Inhibitors of isomerases (erg24, erg2), inhibitors of 3-keto reductase (erg27) in C4 demethylation of sterol biosynthesis, and inhibitors of squalene cyclooxygenase (erg1) in sterol biosynthesis, etc.

[0111] (c29) Group G1: Inhibitor of C14 demethylase (erg11 / cyp51) in sterol biosynthesis (FRAC) Group code 3) Inhibitors of C14 demethylases in sterol biosynthesis include, for example: piperazines such as triforine; pyridines such as pyrifenox and pyrisoxazole; pyrimidines such as fenarimol and nuarimol; imidazoles such as imazalil, oxpoconazole, pefurazoate, prochloraz, and triflumizole; and antibiotics such as azaconazole, bitertanol, bromuconazole, cyproconazole, difenoconazole, diniconazole, epoxiconazole, etaconazole, and nitrilobenzazole. Triazoles, including fenbuconazole, fluquinconazole, flusilazole, flutriafol, hexaconazole, imibenzonazole, ipconazole, mefentrifluconazole, metconazole, miclobutanil, penconazole, propiconazole, simeconazole, tebuconazole, tetraconazole, triadimefon, triadimenol, and triticonazole; and triazolinethiophenes, including prothioconazole.

[0112] (c30) Group G2: Δ in sterol biosynthesis 14 reductase and Δ 8 →Δ 7 Inhibition of isomerases (erg24, erg2) Agent (FRAC group code 5) Δ as a component in sterol biosynthesis 14 reductase and Δ 8 →Δ 7Inhibitors of isomerases (erg24, erg2) include, for example: morpholines such as aldimorph, dodemorph, fenpropimorph, and tridemorph; piperidines such as fenpropidin and piperalin; and spiroxamines such as spiroxamine.

[0113] (c31) Group G3: Inhibitor of 3-keto reductase (erg27) in the demethylation of C4 position in sterol biosynthesis. (FRAC Group Code 17) Inhibitors of 3-keto reductase (erg27) in the demethylation of the C4 position in sterol biosynthesis include, for example, hydroxyanilines such as fenhexamid and aminopyrazolones such as fenpyrazamine.

[0114] (c32) Group G4: Inhibitor of squalene cyclooxygenase (erg1) in sterol biosynthesis (FRAC group code 18) Inhibitors of squalene epoxidase (erg1) in sterol biosynthesis include, for example, thiocarbamates such as pyributicarb; and allylamines such as naftifine and terbinafine.

[0115] Group H Examples of H-group inhibitors (cell wall biosynthesis inhibitors) include chitin synthase inhibitors and cellulose synthase inhibitors.

[0116] (c33) H4: Chitin synthase inhibitor (FRAC group code 19) Examples of chitin synthase inhibitors include peptidylpyrimidine nucleosides such as polyoxin, used as an antibiotic in pesticides. Polyoxin is produced by the actinomycete Streptomyces cocoa (…). Streptomyces cacaoi Polyoxins are antifungal (mold) antibiotics produced by [the production of polyoxins]. There are 14 types of polyoxins, with A, B, and D as the main components.

[0117] (c34) H5: Cellulose synthase inhibitor (FRAC group code 40) Examples of cinnamic acid amide inhibitors include: dimethomorph, flumorph, pyrimorph, etc.; valine amide carbamates such as benthiavalicarb, iprovalicarb, valifenalate, etc.; and mandipropamides such as mandelic acid amides.

[0118] Group I As Group I (inhibitors of melanin synthesis in the cell wall), examples include reductase inhibitors, dehydratase inhibitors, and polyketide synthase inhibitors of melanin biosynthesis.

[0119] (c35) I1: Reductase inhibitor of melanin biosynthesis (FRAC group code 16.1) Examples of reductase inhibitors that inhibit melanin biosynthesis include: isobenzofuranones such as tetrachlorophthalide; pyrroloquinolineones such as pyroquilon; and triazolobenzothiazoles such as tricyclazole.

[0120] (c36) I2: Dehydrating enzyme inhibitor of melanin biosynthesis (FRAC group code 16.2) Examples of dehydrating enzyme inhibitors used in melanin biosynthesis include: cyclopropane formamides such as carpropamid; formamides such as diclocymet; and propionamides such as fenoxanil.

[0121] (c37) Group I3: Polyketide synthase inhibitor for melanin biosynthesis (FRAC group code 16.3) Examples of polyketide synthase inhibitors used in melanin biosynthesis include trifluoroethyl carbamates such as tolprocarb.

[0122] Group P (c38) Host plant resistance inducers (excluding saccharin or its salts) Examples of P-group (host plant resistance inducers) include resistance inducers that stimulate the salicylic acid pathway, host plant resistance inducers, plant extracts that induce host plant resistance, microorganisms that induce host plant resistance, and microbial preparations. It should be noted that these host plant resistance inducers do not contain saccharin or its salts.

[0123] Group P1: Resistance inducers that stimulate the salicylic acid pathway (FRAC group code P1) Examples of benzothiadiazoles (BTH) that can stimulate the salicylic acid pathway (salicylic acid signaling) include acibenzolar-S-methyl and others.

[0124] Group P2: Host plant resistance inducer (FRAC group code P2) Examples of host plant resistance inducers (salicylic acid signaling) include benzisothiazides such as probenazole.

[0125] Group P3: Host plant resistance inducer (FRAC group code P3) Examples of host plant resistance inducers (salicylic acid signaling) include thiadinil, isothiazine, and other thiadiazole formamides.

[0126] Group P4: Host plant resistance inducer (FRAC group code P4) As host plant resistance inducers (polysaccharide elicitors, natural products), examples include laminarin and other polysaccharides.

[0127] Group P5: Plant extracts that induce host plant resistance (FRAC group code P5) Plant extracts (anthraquinone elicitors, plant extracts) that induce host plant resistance can be cited as an example: Polygonum cuspidatum ( Reynoutria sachalinensis Mixtures such as extracts, ethanol extracts (anthraquinones, resveratrol), etc.

[0128] Group P6: Microorganisms and microbial preparations that induce host plant resistance (FRAC group code P6) Microorganisms and microbial agents (microbial elicitors, microorganisms) that induce resistance in host plants can be cited as examples of Bacillus mycoides ( Bacillus mycoides ) isolate J and other bacteria of the genus Bacillus, Saccharomyces cerevisiae ( Saccharomyces cerevisiae LAS 117 strain contains cell walls and other fungi and yeasts.

[0129] Group P7: Host plant resistance inducer (FRAC group code P7) Examples of host plant resistance inducers (phosphonates) include ethyl phosphonates such as fosetyl, phosphorous acid, and their salts.

[0130] Group P8: Host plant resistance inducer (FRAC group code P8) Examples of host plant resistance inducers (salicylic acid signaling) include dichlorophenoxyacetic acid (dichlobentiazox) and other isothiazolyl methyl ethers.

[0131] (c39) Compounds with unknown mode of action (group: Unknown mode of action) (U) (FRAC group code 27) 34, 35, 36, 37, U6, U12, U13, U14, U16, U17, U18) Examples of compounds with unknown modes of action include: cyanoacetamide oximes such as cymoxanil; o-carbamoylbenzoic acids such as teclofthalam; benzotriazines such as triazine; benzenesulfonamides such as flusulfamide; pyridazinones such as diclomezine; phenylacetamides such as cyflufenamide; guanidines such as dodine; cyanomethylenethiazolidinyl oximes such as fluthianil; pyrimidinone hydrazones such as ferimzone; 4-quinolinylacetic acid such as tebufloquin; tetrazolium oximes such as picarbutrazox; and glucopyranosyl antibiotics such as validamycin.

[0132] Group M (c40) Multi-point contact active compound (M) Examples of multi-site contact active compounds (M) include inorganic compounds (electrophiles), dithiocarbamates and analogues (electrophiles), phthalimides (electrophiles), chloronitriles (phthalonitriles) (site of action unknown), biguanides (cell membrane disruptors, surfactants), triazines, quinones (anthraquinones) (electrophiles), quinoxalines (electrophiles), maleimides (electrophiles), sulfonamides, and thiocarbamates. Among these, inorganic compounds (electrophiles), chloronitriles (phthalonitriles) (site of action unknown), and biguanides (cell membrane disruptors, surfactants) are preferred as multi-site contact active compounds (M).

[0133] Inorganic compounds (electrophilic reagents) (FRAC group codes M1, M2) Examples of inorganic compounds (electrophilic reagents) include copper compounds and chalcogenides.

[0134] Examples of copper compounds include copper, DBEDC, basic copper chloride, basic copper sulfate, copper hydroxide, and copper nonylphenol sulfonate.

[0135] Examples of sulfur compounds include sulfur and lime sulfur.

[0136] Dithiocarbamates and analogues (electrophilic agents) (FRAC group code M3) Examples of dithiocarbamates and analogues (electrophilic reagents) include: amobam, ferbam, mancozeb, maneb, metiram, propineb, thiram, zinc thiazole, zineb, ziram, and other dithiocarbamates and analogues.

[0137] Phthalimides (electrophilic reagents) (FRAC group code M4) Phthalimide compounds (electrophilic reagents) include, for example, captan, captafol, and folpet.

[0138] Chloronitriles (phthalonitriles) (Method of action unknown) (FRAC group code M5) Examples of chloronitrile (phthalonitrile) compounds include chlorothalonil (TPN) and other chloronitrile (phthalonitrile) compounds.

[0139] Sulfonamides (FRAC group code M6) Examples of sulfonamides include aminosulfonic acid derivatives such as dichlofluanid and tolylfluanid.

[0140] Biguanides (cell membrane disruptors, surfactants) (FRAC group code M7) Examples of biguanides include: guazatine, iminoctadine acetate, iminoctadine albesilate (biguanidine octylamine), etc.

[0141] Triazines (FRAC group code M8) Examples of triazines include anilazine and other triazines.

[0142] Quinones (anthraquinones) (electrophilic reagents) (FRAC group code M9) Anthraquinones (electrophilic reagents) are examples of quinones such as dithianon.

[0143] Quinoxaline derivatives (electrophilic reagents) (FRAC group code M10) Examples of quinoxaline derivatives (electrophilic reagents) include quinoxaline series such as quinomethionate.

[0144] Maleimide (electrophilic reagent) (FRAC group code M11) Examples of maleimides (electrophiles) include fluoroimides and other maleimides.

[0145] Thiocarbamates (FRAC group code M12) Examples of thiocarbamates include thiocarbamates such as methasulfocarb.

[0146] BM Group (c41) Biopesticides with multiple mechanisms of action: plant extracts (BM) (FRAC group code BM1) Biopesticides with multiple mechanisms of action: Examples of plant extracts include: peptides (lectins) extracted from the cotyledons of lupin seedlings; and extracts from Philippine pectin oranges (…). Swinglea glutenosa Extracts of phenols, sesquiterpenes, triterpenes, coumarins, etc. from Melaleuca alternifolia ( Melaleuca alternifolia Extracts of tea tree oil, plant oils (mixtures), eugenol, geraniol, thymol and other terpenes, terpene alcohols and terpene phenols, etc.

[0147] As the bactericidal active compound (C), at least one compound from the group consisting of: (c1) RNA polymerase I inhibitor, (c2) DNA / RNA biosynthesis inhibitors, (c3) Type II DNA topoisomerase (gyrase) inhibitor, (c4) An inhibitor of dihydroorotate dehydrogenase in the de novo biosynthesis of pyrimidines. (c5) Inhibitor of microtubule polymerization, (c6) Cell division inhibitor (site of action unknown), (C10) Complex II (succinate dehydrogenase) inhibitor, (c11) Complex III (Qo site of ubiquitin oxidase) inhibitor, (c12) Complex III (ubiquinone reductase Qi site) inhibitor, (c16) Inhibitor of protein biosynthesis (ribosomal translation initiation), (c17) Inhibitor of protein biosynthesis (ribosomal polypeptide elongation stage), (c20) Phospholipid biosynthesis, methyltransferase inhibitor, (c24) An inhibitor of C14 demethylase in sterol biosynthesis. (c27) Chitin biosynthesis enzyme inhibitor, (c29) An inhibitor of reductase in melanin biosynthesis. (c31) A polyketide synthase inhibitor in melanin biosynthesis. (c32) Host plant resistance inducers (excluding saccharin or its salts). (c33) Compounds with unknown mechanisms of action. (c34) Multi-point contact active compounds, and (c35) Fluopyram.

[0148] Among them, the preferred bactericidal active compounds are polyoxin compounds, kasugamycin, apimycin, streptomycin, and oxytetracycline.

[0149] Polyoxin compounds are antibiotics. There are no particular limitations on the definition of a polyoxin compound; the chemical structures of major polyoxin compounds are described, for example, on page 1306 of "The Merck Index Twelfth Edition." Specifically, preferred polyoxin compounds include, for example, polyoxin itself, polyoxin salts, and polyoxin complexes.

[0150] Examples of polyoxins include polyoxin A, polyoxin B, polyoxin D, polyoxin E, polyoxin F, polyoxin G, polyoxin H, polyoxin J, polyoxin K, polyoxin L, polyoxin M, polyoxin N, and polyoxin O.

[0151] There are no particular limitations on the types of salts that can be used as polyoxins; for example, zinc salts, iron salts, titanium salts, and other metal salts can be included.

[0152] Examples of polyoxin complexes include those with polyoxin B as the main component.

[0153] Polyoxin compounds can be used alone or in combination of two or more. Sometimes, substances containing two or more polyoxins are referred to as polyoxin complexes.

[0154] It should be noted that, currently in Japan, the known active ingredients that have completed pesticide registration are polyoxin complex (a complex component mainly composed of polyoxin B) and polyoxin D zinc salt (a zinc salt mainly composed of polyoxin D).

[0155] Preferred polyoxin compounds are polyoxin complexes and polyoxin D zinc salts.

[0156] In this invention, relative to 100 parts by weight of saccharin and / or its salt (A), 0.1 to 20,000 parts by weight, preferably 1 to 10,000 parts by weight, and more preferably 5 to 5,000 parts by weight of (C) bactericidal active compound is typically added.

[0157] In addition to (A) saccharin and / or its salts, (B) insecticidal active compounds and (C) bactericidal active compounds, the compositions of the present invention may also contain appropriate auxiliary ingredients.

[0158] As an auxiliary component, anti-caking can also be achieved when manufacturing the composition of the present invention by means of additives such as talc, pyrophyllite, silica and other water-insoluble inorganic substances.

[0159] The compositions of the present invention can also be mixed or used in combination with at least one of other fungicides, insecticides, herbicides, plant growth regulators, microbial materials, mollusc control agents, and bird pest inhibitors, to a degree that does not impair the effectiveness of the compositions of the present invention. It should be noted that the aforementioned microbial materials refer to microorganisms with pest control effects (e.g., insecticidal activity, fungicidal activity, herbicidal activity, etc.) and / or microorganisms such as rhizobia and mycorrhizal fungi with plant growth regulating effects.

[0160] In addition to (A) saccharin and / or its salts, (B) an insecticidal compound, and (C) a fungicide, the compositions of the present invention may also contain metaldehyde as a molluscicide. Alternatively, the compositions of the present invention and metaldehyde may be applied simultaneously or at different times during cultivation. In this case, harmful mollusks such as golden apple snails and molluscs can be controlled.

[0161] Other mollusc control agents include bis(tributyltin)oxide, allicin, bromoacetamide, cloethocarb, copper sulfate, fentin, ferric phosphate (III), methiocarb, niclosamide, pentachlorophenol, sodium pentachlorophenoxide, tazimcarb, thiacloprid, thiodicarb, tralopyril, trifenmorph, trimethacarb, cartap, and bensultap.

[0162] In addition to (A) saccharin and / or its salts, (B) an insecticidal compound, and (C) a fungicide, the compositions of the present invention may also contain anthraquinone as a bird repellent. Alternatively, the compositions of the present invention and anthraquinone may be applied simultaneously or at different times during cultivation. In this case, bird-induced damage in the cultivation of plants other than rice can be suppressed.

[0163] Other bird pest control agents include chloralose, copper oxychloride, diazinon, guazatine, methiocarb, thiram, trimethacarb, ziram, and zinc oxide.

[0164] In addition to (A) saccharin and / or its salts, (B) an insecticidal active compound and (C) a fungicide active compound, the compositions of the present invention may also contain herbicides and / or phytotoxicity reducers. Alternatively, the compositions of the present invention may be applied simultaneously or at different times during cultivation. In this case, weeds in the cultivation of plants other than rice can be controlled.

[0165] Examples of herbicide-damage mitigators include AD-67, BAS-145138, benoxacor, cloquintocet-mexyl, cyometrinil, 2,4-D, DKA-24, dichlormid, daimuron, fenchlorim, fenchlorazole-ethyl, flurazole, fluxofenim, furilazole, isoxadifen-ethyl, mefenpyr-diethyl, MG-191, naphthalenecarboxylic anhydride, oxabetrinil, PPG-1292, and R-29148.

[0166] Method for manufacturing agricultural and horticultural pest control compositions In the composition of the present invention, no other ingredients may be added, only (A) saccharin and / or its salt, (B) insecticidal active compound and (C) bactericidal active compound. Generally, solid carriers, liquid carriers and gaseous carriers (propellants) can be mixed, and surfactants and other formulation adjuvants can be added as needed. According to the usual formulation method, it can be made into oil, emulsion, wettable powder, suspension, granules, powder, aerosol, smoke agent and so on for use.

[0167] In these formulations, the combined amount of (A) saccharin and / or its salt, (B) insecticidal active compound and / or (C) fungicide active compound as active ingredients may typically be 0.01 to 95% by weight, preferably 0.05 to 80% by weight, more preferably 0.1 to 70% by weight.

[0168] Solid carriers used in formulation include, for example, clays (kaolin clay, diatomaceous earth, synthetic hydrated silica, bentonite, fubasami clay, acid clay, etc.), talc, ceramics, other inorganic minerals (celite, quartz, sulfur, activated carbon, calcium carbonate, hydrated silica, etc.), and chemical fertilizers (ammonium sulfate, ammonium phosphate, ammonium nitrate, urea, ammonium chloride, etc.) in the form of fine powders or granules.

[0169] Examples of liquid carriers include water, alcohols (methanol, ethanol, etc.), ketones (acetone, methyl ethyl ketone, etc.), aromatic hydrocarbons (benzene, toluene, xylene, ethylbenzene, methylnaphthalene, etc.), aliphatic hydrocarbons (hexane, cyclohexane, kerosene, light oil, etc.), esters (ethyl acetate, butyl acetate, etc.), nitriles (acetonitrile, isobutyronitrile, etc.), ethers (diisopropyl ether, dioxane, etc.), amides (N,N-dimethylformamide, N,N-dimethylacetamide, etc.), halogenated hydrocarbons (dichloromethane, trichloroethane, carbon tetrachloride, etc.), dimethyl sulfoxide, soybean oil, cottonseed oil, and other vegetable oils.

[0170] Examples of gaseous carriers include butane, LPG (liquefied petroleum gas), dimethyl ether, and carbon dioxide.

[0171] Examples of surfactants include: alkyl sulfates, alkyl sulfonates, alkyl aryl sulfonates, alkyl aryl ethers and their polyoxyethylene compounds, polyethylene glycol ethers, polyol esters, sugar alcohol derivatives, etc.

[0172] Examples of pharmaceutical adjuvants include fixatives, dispersants, and stabilizers.

[0173] Examples of fixatives or dispersants include casein, gelatin, polysaccharides (starch, gum arabic, cellulose derivatives, alginic acid, etc.), lignin derivatives, bentonite, sugars, and synthetic water-soluble polymers (polyvinyl alcohol, polyvinylpyrrolidone, polyacrylic acid, etc.). Examples of stabilizers include PAP (isopropyl phosphate), BHT (2,6-di-tert-butyl-4-methylphenol), BHA (a mixture of 2-tert-butyl-4-methoxyphenol and 3-tert-butyl-4-methoxyphenol), vegetable oils, mineral oils, fatty acids, or their esters.

[0174] The composition of this invention can be used directly or diluted with water or other solvents. Alternatively, it can be used in combination with other insecticides, fungicides, herbicides, plant growth regulators, synergists, soil conditioners, animal feeds, etc., or used simultaneously without mixing.

[0175] When the composition of the present invention contains both components (A) and (B), or components (A) and (C), the total amount thereof is typically 0.01 to 95% by mass, preferably 0.05 to 80% by mass, and more preferably 0.1 to 50% by mass.

[0176] When combined with the above three components (A), (B) and (C), the total amount of components (A) to (C) can typically be 0.01 to 95% by mass, preferably 0.05 to 80% by mass, and more preferably 0.1 to 70% by mass.

[0177] The dosage of the composition of the present invention is per 1a (100m 2 The amount is typically 0.05g to 600g, preferably 0.1g to 200g, and more preferably 0.5g to 100g.

[0178] When the synergistic insecticide composition of the present invention in the form of emulsion, wettable powder, suspension, liquid, etc., is diluted with water, the application concentration is usually 0.1~300000ppm, preferably 1~30000ppm, and more preferably 10~8000ppm.

[0179] At this time, the application concentration of component (A) is typically 0.05 to 150,000 ppm, preferably 0.5 to 10,000 ppm, and more preferably 5 to 4,000 ppm. The application concentration of component (B) is typically 0.05 to 150,000 ppm, preferably 0.5 to 10,000 ppm, and more preferably 5 to 4,000 ppm. The application concentration of component (C) is typically 0.05 to 150,000 ppm, preferably 0.5 to 10,000 ppm, and more preferably 5 to 4,000 ppm.

[0180] For example, in conventional spraying, the application concentration of the composition of the present invention is typically 0.1 to 10,000 ppm, preferably 1 to 5,000 ppm, and more preferably 10 to 1,000 ppm. In the case of infusion, the application concentration of the composition of the present invention is generally 1 to 300,000 ppm, preferably 10 to 30,000 ppm, and more preferably 100 to 8,000 ppm.

[0181] In addition, granules, powders, etc., can be applied directly as a formulation without any dilution with water.

[0182] The dosage and concentration of these substances vary depending on the type of formulation, application time, application location, application method, type of pest, and degree of damage. They can be increased or decreased and are not limited to the above ranges.

[0183] Examples of pests that can be controlled by the composition of the present invention include insects, mites, nematodes, mollusks, and plant pathogens such as filamentous fungi, bacteria, and viruses.

[0184] Insects, mites, nematodes, mollusks, etc., that can be controlled by the composition of the present invention, specifically the following types can be mentioned.

[0185] insect Hemiptera ( Hemiptera Grey planthopper ( Laodelphax striatellus Brown planthopper ( Nilaparvata lugens White-backed planthopper ( Sogatella furcifera ), corn flower winged planthopper ( The pilgrim maid ), Gubei planthopper ( Javesella pellucida ), sugarcane flat-horned planthopper ( Perkinsiella saccharicida ), rice stalk planthopper ( Tagosodes oryzicolus Planthoppers (family Planthopperidae) Delphicidae ); Black-tailed leafhopper ( Nephotettix cincticeps ), two-spotted black-tailed leafhopper ( Nephotettix virescens ), two-spotted black-tailed leafhoppers ( Black-spotted Nephotettix ), electric leafhopper ( Dorsal Recilia ), small green leafhopper ( Grandson's Empoasca ), potato leafhopper ( Bean sprouts ), corn leafhopper ( Maiden's scythe ), large white leafhopper ( Ghostly hood Cicadidae (etc.) Leafhoppers ); Sugarcane cicada ( Mahanarva walled Sugarcane root grasshopper ( Mahanarva fringed ) and other cicadas ( Cercopidae beet aphid ( Bean aphid ), soybean aphid ( Wisteria aphids ), cotton aphids ( Aphis gossypii Apple aphids Apple aphid ), Spiraea aphid ( Aphis spiraecola ), Peach aphid ( Myzus peaches ), Prunus shorttail aphid ( Brachycaudus helichrysi ), cabbage aphid ( Brassica oleracea ), plantain roundtail aphid ( Dysaphis plantain Radish aphid ( Lipaphis erysimi), potato aphid ( Euphorbia macrosiphum ), potato tube aphid ( Aulacorthumsolani ), lettuce aphids ( Nasovia blackcurrant ), cereal constrictor aphid ( Rhopalosiphum padi ), corn aphids ( Rhopalosiphum maidis ), Citrus aphid ( Toxoptera citricida ), Peach Pink Aphid ( Hyalopterus plumi ), sugarcane aphid ( Melanophis sugar ), Black-bellied Four-veined Aphid ( Tetraneura nigriabdominalis Sugarcane aphid ( Ceratovacuum woolen clothes Apple woolly aphid ( Eriosoma woolly Aphids (and other aphids) Aphids ); grape phylloxera ( Daktulosphaira vitifoliae ), American pecan phylloxera ( Phylloxera devastating ), pecan leaf phylloxera ( Notable phylloxera ), South American pecan leaf phylloxera ( Phylloxera russelliana ) and other rhizophora (family Aphididae) Phylloxera ); Hemlock ball aphid ( Adelges hemlock ), fir ball aphid ( Adelges piceus ) and fir ball aphid ( Aphrastasia pectinata ) and other aphids ( Adelgids ); Rice black bug ( Scotinophara dirty ), Malayan rice black bug ( Scotinophara coarctata ), Black-bearded rice green bug ( Nezara antennata ), Northern Two-Star Bug ( Eysarcoris aureus ), Japanese two-star bug ( Eysarcoris lewisi ), Guang Erxing bug ( Eysarcoris ventralis ), pseudo-two-star bug ( Eysarcoris annamita ), tea-winged bug ( Haliomorpha haly ), rice green bug ( Green-leaved nezara ), brown bug ( Euschistus the hero ), Red-banded bug ( Piezodorus guild of guilds ), rice bug ( The fighting bull ), Green-bellied bug ( Dichelops melacanthus ) and other bugs ( Pentatomidae ); brown soil bug ( Chestnut-colored Scaptocoris ) and other soil bugs ( Cydniidae ); Spotted bee periwinkle ( Footsteps ), Chinese rice bug ( Leptocorisa chinensis ), Large Rice Bug ( Leptocorisa sharp Spider bugs (Arachnidae) Alydidae ); Rice spiny-edged bug ( Cletus the Punctualist ), Australian leaf-footed bug ( Leptoglossus southern ) etc. family ( Coreidae ); Sugarcane stink bug ( Caverelius saccharivore ), gourd bug ( Togo half-winged ), wheat bug ( Blissus leucopterus ) Equal-length bugs ( Lygaeidae ); Red-bearded blind bug ( Trigonotylus celestialis ), Red-striped filamentous mirid bug ( Red-bellied scaly-headed ), Two-spined narrow-skinned bug ( Stenodema calcarata ), American mirid bug ( Lygus lineolaris Miridae ( ) Miridae Greenhouse whiteflies ( Trialeurodes vaporariorum ), whitefly ( Bemisia tabaci citrus whiteflies ( Dialeurodes lemons ), black thorn whitefly ( Aleurocanthus spiniferus ), tea black thorn whitefly ( Aleurocanthus camellias ), tea whitefly ( Pealius Euryae Whitefly family ( ) Aleyrodidae ); Tea long-rooted round gecko ( Abgralaspis cyanophyllus ), Red round scale ( Aonidiella aurantii ), pear-shaped gecko ( Diaspidiotus destructive ), Mulberry Scale ( Pseudoulacaspis pentagona ), arrowhead scale ( Unaspis yanensis ), Orange Arrowhead Scale ( Lemon peel ) and other families such as the scale insect family ( Diaspididae ); Red wax scale ( Red wax moth ) and other species of scale insects ( Coccidae ); Blowing cotton-shelled gecko ( Icerya purchasi ), Silver-haired cottony mealybug ( Seychelles ice cream ) etc., Shuojie Science ( Margarididae Lycoris radiata and mealybug ( Nightshade ), Hibiscus mealybug ( Phenacococcus sunflower ), Japanese mealybug ( Planococcus kraunhiae ), Comstock mealybug ( Pseudococci comstock Orange-skinned beetle ( Planococcus citri Pseudococcus Calceolaria ), long-tailed mealybug ( Pseudococcus longispinus ), rice mealybug ( I am holding a brevet. ) and other mealybugs ( Pseudococcidae ); citrus psyllid ( Citrus diaphorine ), African citrus psyllid ( Trioza erythraea ), pear psyllid ( Cacopsylla pyrisuga ), Chinese pear psyllid ( Cacopsylla chinensis ), potato psyllid ( Bactericera cockerelli ), pear psyllid ( Cacopsylla pyricola Psyllidaceae ( Psyllididae ); Sycamore lace bug ( Corythucha ciliata ), Chrysanthemum-winged lace bug ( Corythucha marmorata ), pear-crowned lace bug ( Stephanitis nashi ), Cuckoo lace bug ( Stephanitis pyrioides ) and other lace bugs ( Tingidae Temperate bedbugs ( Bed bug Bedbugs (family Cladosporidae) Bedbugs ); and giant cicadas ( Quesada the giant Cicadas (and other cicada species) Cicadas ).

[0186] Lepidoptera ( Lepidoptera ): Borer borer ( Chilo suppressalis ), Black-headed moth ( Kilo polychrome ), rice stem borer ( Scirpophaga innotata ), rice stem borer ( Scirpophaga incertulas ), South American white borer ( White ruffe ), rice leaf roller ( Cnaphalocrocis medinalis ), broad-striped rice leaf roller ( Marasmia patnalis ), Rice leaf roller ( Marasmia minor ), cotton leaf borer ( Notarch derogated Asian corn borer ( Furnacian oyster ), European corn borer ( Clouded oyster ), vegetable moth ( Hellula undalis Grape leafminer ( Herpetogramma melancholy Bluegrass moth ( Pediatrics little fox ), rice three-spotted stem borer ( Nymphula depunctalis ), sugarcane borer ( Diatraea saccharalis ) and other herbaceous moths ( Crambidae ); South American corn seedling borer ( Elasmopalpus lignosellus Indian meal borer ( Plodia interpunct Pyralidae ( Pyralidae ); Spodoptera litura ( Spodoptera litura ), beet armyworm ( Spodoptera small ), armyworms ( Separate myths ), cabbage moth ( Brassica napus ), giant borer ( Bringing sesame seeds ), Grey-winged Noctuid Moth ( Spodoptera mauritia ), rice stem borer ( Orange blossom Fall armyworm ( Spodoptera frugiperda African fall armyworm ( Spodoptera exempta ), small cutworm ( Agrotis ipsilon Black-spotted Silver-striped Noctuid Moth ( Black-lettered autographs Golden-spotted moth ( Plus flakes ), soybean silver-striped noctuid moth ( Including Chrysodeixis ), genus *Pseudococcus* ( Trichoplusia spp.), tobacco bud moth ( Heliothis virescens ) and other moths of the genus *Cypripedium* Heliothis spp.), cotton bollworm ( Helicoverpa armor-bearer ), grain moth ( Helicoverpa zea ) etc. of the genus *Bulbus* ( Helicoverpa spp.), Bean moth ( Anticarsia gemmatalis ), cotton leafminer moth ( Alabama clay ), Hops vine borer ( Hydraecia monstrous Noctuidae (etc.) Noctuidae );cabbage butterfly( Pieris turnips Pieridae (and other families) Pieridae ); Pear fruit moth ( Grapholite pest ), Li Xiaoshi Xin Chong ( Grapholita dimorpha ), soybean pod borer ( Leguminous glycine ), Bean leafroller ( Matsumuraeses azukivora ), Cotton brown leafroller ( Adoxophyes orange banded ), tea leafroller ( Adoxophyes honmai ), tea long-haired moth ( Magnanimous people ), Apricot Yellow Roller ( Archips fuscocupreanus Apple codling moth ( Cydia pomonella Sugarcane borer ( Tetramoera schistose ), bean shoot leafroller ( Epinotia aporema ), Citrus fruit borer ( Ecdytolopha aurantiana ) and other members of the family Lepidoptera ( Tortricidae Tea moth (); Caloptilia theivora ), Golden-striped fine moth ( Phyllonorycter small ring ) and other moths (family Scleroderidae) Gracillariidae ); Peach fruit moth ( Carposina sasakii Fruit borers (family: ) Carposinidae Coffee leafminer ( Leucoptera coffeella Peach leafminer ( Lyonetia clerkella ), Silver Leafminer ( Lyonetia prunifoliella ) and other moths ( Lionetiidae ); Gypsy moth ( Lymantria uneven ) and other tussock moths ( Lymantria spp.), tea tussock moth ( Euproctis pseudoconspersa ) and other species of yellow moth ( Euproctis spp.) and other tussock moths ( Lymantriidae Diamondback moth (); Plutella xylostella) and other members of the Prunella vulgaris family ( Plutellidae ); Peach bark moth ( Anarsia lineatella ), sweet potato moth ( Helcystogramma three-ringed ), pink bollworm ( Pectinophora gossypiella ), potato tuber moth ( Phthorimaea lid Tomato leafminer ( Absolutely safe ) and other moths (family Agromycetes) Gelechiidae ); American white moth ( Hyphantria wedge ) and other moths (family Lithopodidae) Arctiidae ); large sugarcane borer ( Telchin lich ) and other butterfly moths ( Castniidae ); small wood-boring moth ( Islander's Cossus Wood-boring moths ( ) and other wood-boring moths ( Cossidae ); Great bridge-building insect ( Ascot moon Geometridae (etc.) Geometridae ); Green tussock moth ( Nice parasites ) and other Limacodidae ( Slugidae ); persimmon calyx worm ( Stathmopoda masinissa ) and other moths (family Lepidoptera) Stathmopodidae ); Ghostface hawkmoth ( Acherontia lachesis ) and other sphingomycetes ( Sphingidae Kiwifruit clearwing moth ( Wild Nokona Clearwing moths ( ) and other clearwing moths ( Sesiidae Straight-striped rice skipper ( Parnara guttata ) and other butterfly families ( Hesperiidae ).

[0187] Thysanoptera ( Thysanoptera ): Western flower thrips ( Frankliniella occidentalis Palm thrips ( Palm thrips ), Tea yellow thrips ( Scirtothrips dorsalis ), onion thrips ( Tobacco thrips ), flower thrips ( Frankliniella intonsa ), rice thrips ( Stenchaetothrips biformis ), thrips ( American thrips Thrips (and other thrips families) Thripidae Rice thrips ( Haplothrips aculeatus Thripsidae (etc.) Phlaeothripidae ).

[0188] Diptera ( Diptera Seed fly ( Delia's flat ), onion fly ( Ancient Delia Spinach leafminer ( Pegomya cunicularis ) and other families such as the flower fly family ( Anthomyiidae Beet fly ( ); beet leaf fly ( Myopaeform tetanus ) and other leafhoppers ( Ulidiidae ); Japanese rice miner ( Agromyza rice beetle ), American serpentine leafminer ( Liriomyza sativa ), trifoliate leafminer ( Liriomyza trifolii ), Pea miner ( Chromatomyia horticola ) and other leafminer family ( Agromyzidae Rice straw flies ( Chlorops oryzae ) and other stem flies ( Chloropidae ); melon fly ( Bactrocera squash ), the orange fruit fly ( Bactrocera dorsalis Broadband fruit fly ( Bactrocera latifrons Olive fruit fly ( Bactrocera oleae Queensland fruit fly ( Bactrocera tryoni Mediterranean fruit fly ( ) Ceratitis capitata Apple fruit fly ( Rhagoletis pomonella ), Japanese cherry fruit fly ( Rhacochlaena Japanese Fruit flies (Fungidae) Tephritidae Rice leafminer ( ); Hydrellia griseola ), Philippine hairy-eyed water fly ( Philippine Hydrellia ), rice stalk hairy water fly ( Hydrellia sasakii ) and other water flies ( Ephrydidae ); Spotted-winged fruit fly ( Drosophila suzukii Drosophila (Fructus Drosophila) Drosophila ); East Asian flea fly ( Megaselia spiracle ) and other fleas (Flea family ( Phoridae ); white-spotted moth fly ( Clogmia albipunctata ) and other mothflies ( Psychodidae ); *Heterophthalmos fasciatus* ( Bradysia difformis ) and other fungiidae ( Sciaridae Black forest gall midge ( ); Black forest gall midge ( Mayetiola destructor ), Asian rice gall midge ( Oryzae Gallidae (etc.) Cecidomyiidae ); Big-eyed Exophthalmos ( Diopsis macrophthalmus ) and other families such as Exophthalmosidae ( Diopsidae ); Rice mosquito ( Aino pepper ), common mosquito ( Onion ), European giant mosquito ( Marsh sedge Mosquito family ( ) etc. Tipulidae ); Culex pipiens pallens ( Pale pipiens mosquito Aedes aegypti ( Aedes aegypti ), Aedes albopictus ( The white-painted house Anopheles sinensis ( Anopheles hyracanus sinensis Culex pipiens quinquefolius ( ) Five-banded mosquito ), harassing Culex mosquitoes ( The annoying pipiens mosquito Forskal Mosquitoes ( ) and other mosquitoes Mosquitoes ); Black Spotted Fly ( Proximum from Yezo ), decorative short-necked beetle ( Ornamental ant ) and other species of gnats ( Simidae Trigonella foetida ( ) Horsefly triangle ) and other horseflies ( Horsefly ); housefly ( Housefly ), stable fly ( Stall fly Flies (Fly family) Fly family )wait.

[0189] Coleoptera ( Beetles Western corn rootworm ( Diabrotica virgifera virgifera Southern corn rootworm ( Diabrotica undecimpuncatata Howard ), Northern corn rootworm ( Diabrotica barbers Mexican corn rootworm ( Diabrotica virgifera zeae ), spotted cucumber leaf beetle ( Diabrotica belted ), Cucurbitaceae beetles ( Speciiform Diabrotica ), bean leaf beetle ( Cerotoma trifurcata ), Black-horned mud beetle ( Oulema melanopus ), Huang Shougua ( Aulacophora femoralis ), Yellow-striped flea beetle ( Phyllotreta striped ), Cabbage flea beetle ( Phyllotreta crucifera ), Western Black Jump Armor ( Phyllotreta pusilla ), cabbage stem flea beetle ( Psylliodes chrysocephalus ), Hubu Jump Armor ( Psylliodes punctulata ), potato beetle ( Leptinotarsa ​​ten-lineata Rice leaf beetle ( Rice weevil ), grape leaf beetle ( Collapse brown ), corn flea beetle ( Chaetocnema pulicaria ), sweet potato flea beetle ( Chaetocnema confinans ), Potato flea beetle ( Cucumber ), rice iron beetle ( Dicladispa armigera Southern corn leaf beetle ( Myochrous denticollis ), sweet potato and tortoise shell ( Laccoptera quadrimamaculata ), tobacco flea beetle ( Hairy-billed ibis Chrysophagaceae ( ) etc. Chrysomelidae ); Corn-seed chestnut brown ground beetle ( Stenolophus I lied. ), corn seed beetle ( Clivina impressifrons ) etc., Argonautidae ( Carabidae ); Bronze Elegant Golden Tortoise ( Copper anomaly ), Bean beetle ( Anomaly red-copper ), Little Bronze Tortoise ( White-haired anomaly ), Japanese beetle ( Japanese popillia ), Huang Changli Golden Turtle ( Heptophylla picea ), European Golden Beetle ( Rhizotrogus majalis ), Black-spotted Golden Beetle ( Humpbacked Tomarus ), genus *Hemiberlesia lataniae* ( Holotrichia spp.), June beetle ( Phyllophaga hairy ) etc. ( ) genus of golden beetles Phyllophagus spp.), Argentine rhinoceros beetle ( Diloboderus abderus Argentine small scabbard (etc.) Diloboderusspp.) and other scarab beetles ( Scarabaeidae Coffee Elephant ( Araecerus coffeae ), Sweet Potato Elephant ( Cylas anteater West Indian sweet potato weevil ( Euscepes postfasciatus ), alfalfa leaf weevil ( Backyard ), corn weevil ( Sitophilus zeamais ), rice weevil ( Echinocnemus squameus ), Rice water weevil ( Lissorhoptrus rice-loving Palm weevil ( Rhabdoscelus lineatocollis ), Cotton Boll Weevil ( Anthonom big ), lawn weevil ( Sphenophorus hunted s), Southern Corn Weevil ( Callosus sphenophorus ), soybean stem weevil ( Sternechus subscriptus Sugarcane weevil ( Sphenophorus levis ), Gray gourd weevil ( Gray skeptic ), Brown gourd weevil ( Skeptic in uniform ), Brazilian bean weevil ( Zabrotes underdressed ), Pine pit pruning beetle ( Tomicus piniperda Coffee berry borer ( Hypotheneum hampi Moss's spiny elephant ( Aracanthus mourei ) etc., genus *Echinochloa* Arachnanthus spp.), cotton root weevil ( Eutinobothrus brasiliensis Elephant family ( ) Weevils ); Red grain beetle ( Tribolium chestnut ), miscellaneous grain thief ( Tribolium confusa ) and other tenebrionid A family ( Tenebrionidae ); Ladybug with twenty-eight spots ( Epilachna vigintioctopunctata Ladybugs ( ) and other ladybugs ( Ladybirds Bamboo powder beetle ( Lyctus brown ) Equal longhorn beetles ( Bostrychidae Spider beetles ( ); Spider family ( Ptiniidae ); Longhorn beetle ( Anoplophora Malaysian ), Freund's naked-horned longhorn beetle ( Almond fryanus Longhorn beetles ( ) Beetles ); Okinawa sugarcane shell ( Melanotus okinawaensis ), fine chest nail ( Brown-bellied woodpecker ), horn comb, claws, nails ( Melanotan ambassador ), genus *Spinythoracis* ( Anchast spp.), *Broad-chested Talonoptera* ( Conoderus spp.), genus *Cypripedium* ( Ctenicera spp.), genus *Tectus* ( ... Limonius spp.), genus Aeolus ( Aeolus spp.) and other family of cladocerans ( Elateridae ); Paederus fuscipes ) and other rove beetles ( Staphylinidae ).

[0190] Orthoptera ( Orthoptera Locusts Migratory locust ), Moroccan locust ( Dociostaurus Moroccan ), Australian locust plague Chortoicetes terminifera ), red locust ( Nomads seven-banded ), brown locust ( Leopard locust Tree locusts ( Anacridium melanorhodon ), Italian locust ( Calliptamus italicum ), American migratory locust ( Melanoplus differentialis ), double-banded black locust ( Melanoplus bivittatus ), migratory black locusts ( Melanoplus sanguineus ), Red-legged Black Locust ( Melanoplus red thigh ), clearwing locust ( Transparent tube Desert locusts Schistocerca gregarious ), Yellow-winged locust ( Gastromargus musician ), spiky locust ( Austracris guttulus ), small-winged rice locust ( Oxya yezoensis ), Japanese rice locust (Oxya japonica), Indian yellow-spined locust ( Short-tailed batangas ) and other Acrididae ( Grasshoppers Oriental mole cricket ( Gryllotalpa orientalis Mole crickets (family Mole cricket family) Gryllotalpidae ); house cricket ( Domestic catfish ), Yellow-faced oil gourd ( Teleogryllus emma ) and other cricket families ( Gryllids Mormon Grasshopper ( Anabrus simplex ) etc. katydids ( Tettigoniidae ).

[0191] Hymenoptera ( Hymenoptera Turnip leaf bee ( Athalia roses ), Japanese Sawfly ( Athaliah Japanese ) and other leaf bee families ( Tenthredinidae Fire ants ( ) Nightshade spp.), Barcher leaf ants ( Atta capiguara Ants (e.g., ants) Ants )wait.

[0192] Blattales ( Cockroach German cockroach ( German cockroach ) and other Blattodea families ( Blattellidae Black-breasted cockroach ( ); Periplaneta fuliginosa American cockroach ( Periplaneta americana Brown-spotted cockroach ( Periplaneta brunnea Oriental cockroach ()Blatta orientalis Blattodea (family Blattodea) Blattidae ); North African termites ( Reticulitermes speratus ), Formosan subterranean termite ( Coptotermes formosanus ), small jacaranda termites ( Incisitermes minor ), truncated sand termites ( Cryptotermes domesticus ), black-winged subterranean termites ( Odontotermes formosanus Hengchun new termites ( Neotermes koshunensis ), Satsuma tree termites ( Glyptotermes satsumensis ), Nakajima tree termites ( Glyptotermes nakajimai ), black tree termites ( Glyptotermes fuscus ), forest termites ( Hodotermopsis sjostedti ), Guangzhou subterranean termite ( Coptotermes guangzhouensis Amami subterranean termites ( Reticulitermes amamianus ), Miyamoto termites ( Reticulitermes miyatakei ), close the door to release termites ( Reticulitermes kanmonensis ), Takasago termites ( Nasutitermes takasagoensis ), Nitobe near-twisted termites ( Pericapritermes nitobei ), Taiwan Wicked Termites ( Sinocapritermes mushae ), sand-dwelling termites ( Cornitermes cumulans Termites (family Termitidae) Termitidae ).

[0193] mites Mites ( Acari Two-spotted spider mite ( Tetranychus urticae ), Tetranychus kamizawa ( Tetranychus kanzawai ), Tetranychus edodes ( Tetranychus evansi ), Citrus red claw mite ( Panonychus citri Apple parsnip ( Panonychus ulmi ), genus *M.* Oligonychus Tetranychids (spp.) and other spider mites ( Tetranychidae ); Citrus rust mite ( Aculops pelekassi ), Ryukyu citrus rust mite ( Phyllocoptruta citri ), tomato rust mite ( Aculops lycopersici ), tea orange gall mite ( Calacarus carinatus Tea gall mite ( Acaphylla theavagrans ), pear rust gall mite ( Eriophyes chibaensis ), Apple rust mite ( Aculus schlechtendali ), persimmon gall mite ( Aceria diospyri ), wheat gall mite ( Aceria tosichella ), Perilla gall mite ( Shevtchenkella sp.) and other gallomites (spe.) Eriophyidae ); tea yellow mite ( Polyphagotarsonemus latus ) and other Tardiidae (Tarsonemidae ); Purple-red short-haired mite ( Brevipalpus phoenicis ) and other fine-toothed mites ( Tenuipalpidae ); Takkarya ( Tuckerellidae ); Longhorn Haemaphysalis ( Haemaphysalis longicornis ), brown haematopoiet ( ), Taiwan tick ( Haemaphysalis flava American dog ticks ( ) Dermacentor taiwanensis Dermacentor variabilis ), oval hard tick ( Ixodes ovatus ), whole furrow hard tick ( Ixodes persulcatus ), shoulder tick ( Ixodes scapularis ), American flower tick ( Amblyomma americanum ), tiny ticks ( Boophilus microplus ), Blood-red fan-head tick ( Rhipicephalus sanguineus ) and other hard ticks (family Ixodidae) Ixodidae ); Tyrophagus putrificans ( Tyrophagus putrescentiae ), Tyrophagus-like mites ( Tyrophagus similis ) and other acarids ( Acaridae ); dust mites ( Dermatophagoides farinae House dust mites ( Dermatophagoides pteronyssinus ) and other dust mite families ( Pyroglyphidae ); Common carnivorous mites ( Cheyletus eruditus ), Malacca carnivorous mite ( Cheyletus malaccensis Southern carnivorous mite ( Cheyletus moorei ), Canis chelicerata ( Cheyletiella yasguri Carnivorous mites ( ) and other carnivorous mites Cheyletidae ); Canine ear mites ( Otodectes cynotis ), human scabies mite ( Sarcoptes scabiei Sarcoptes (family Sarcoptidae) Sarcoptidae ); canine demodicosis ( Demodex canis Demodex family ( ) Demodicidae ); Trichodermatidae ( Listrophoridae ); Avian mites ( Haplochthoniidae ); Burke's avian spiny mite ( Ornithonyssus bacoti ), forest birds tussock mites ( Ornithonyssus sylviarum ) and other giant spiny mites ( Macronyssidae Chicken skin mites (); Dermanyssus gallinae ) and other dermatophytes ( Dermanyssidae ); Red chigger mite ( Leptotrombidium akamushi ) and other mites (family Chrystomidae) Trombiculidae )wait.

[0194] Nematodes Nematodes ( Nematoda Rice stem nematode ( Aphelenchoides besseyi ) and other families of slippery blades ( Aphelenchoididae ); coffee short-bodied nematode ( Pratylenchus coffeae ), short-tailed short-bodied nematode ( Pratylenchus brachyurus Neglecting the short-bodied nematode ( Pratylenchus neglectus), similar perforating nematodes ( Radopholus similis ) and other short-body subjects ( Pratylenchidae Javan root-knot nematode ( Meloidogyne javanica Southern root-knot nematode ( Meloidogyne incognita ), Northern root-knot nematodes ( Meloidogyne hapla ), soybean cyst nematode ( Heterodera glycines ), potato nematode ( Globodera rostochiensis ), potato white nematode ( Globodera pallida ) and other heterodermataceae ( Heteroderidae ); Nematode nematode ( Rotylenchulus reniformis ) and other linking disciplines ( Hoplolaimidae ); Strawberry bud nematode ( Nothotylenchus acris ), bulb nematode ( Ditylenchus dipsaci ) etc. Gramineae Anguinidae ); Citrus semi-piercing nematode ( Tylenchulus semipenetrans Semi-puncture department () Tylenchulidae ); Standard nematode ( Xiphinema index ) and length needle family ( Longidoridae ); Nematodae ( Trichodoridae ); Pine wood nematode ( Bursaphelenchus xylophilus Parasitic Scalyflies ( ) and other families of parasites Parasitaphelenchidae )wait.

[0195] soft animals Gastropoda ( Gastropods Reticulated slug ( Margined slug ), yellow slug ( Yellow slug Slugidae ( Slugs ); Two-lined slug ( Meghimatium bilineatum ) and other slime slugs ( Philomycidae ); Golden apple snail ( Pomacea canaliculata ) and other families such as the bottlenose family ( Amphillidae ); Small cone snail ( Austropeplea small bottle Examples include the Lymnaeidae family.

[0196] Specifically, the following plant diseases originating from plant pathogens that can be prevented and controlled by the compositions of the present invention can be listed as examples. The scientific names of the plant pathogens causing each disease are indicated in parentheses.

[0197] plant disease Wheat diseases: powdery mildew ( Erysiphe grass Fusarium head blight ( Fusarium gramineae , F. oatmeal , F. culms , Snowdrop ), rust ( Puccinia striiformis , P. grass , P. confidita Red snow rot ( Micronectriella nivale ), sclerotinia nivalis disease ( Typhula sp.), loose smut ( Wheat blight ), smut disease ( Tilletia caries ), eye wrinkles ( Pseudocercosporella herpotrichoides Leaf blight ( Mycosphaerella graminicola ), glumpy disease ( Stagonospora nodorum ), macular degeneration ( Pyrenophora tritici-repentis )wait.

[0198] Barley diseases: Powdery mildew ( Erysiphe grass Fusarium head blight ( Fusarium gramineae , F. oatmeal , F. culms , Snowdrop ), rust ( Puccinia striiformis , P. grass , Barley gram Loose smut ( Naked scald ), cloud pattern disease ( Naked scald ), reticulate disease ( Pyrenophora teres ), spotted disease ( Cochliobolus sativus ), leaf spot disease ( Pyrenophora grass ), by Rhizoctonia spp. ( Rhizoctonia Seedling blight caused by fungi ( ) Rhizoctonia solani )wait.

[0199] Corn diseases: smut ( May burning ), Sesame leaf blight ( Snail heterostrophe Leopard disease () Gloeocercospora sorghi Southern rust ( Puccinia polysora Gray leaf spot ( Cercospora zeae-maydis Damping-off disease caused by Rhizoctonia spp. Rhizoctonia solani )wait.

[0200] Citrus diseases: Black spot disease ( Citrus diaportha ), scabies ( Elsinoe fawcetti ), Penicillium ( Penicillium digitatum , P. italicum Phytophthora ( Phytophthora parasitic , Phytophthora citrophthora )wait.

[0201] Apple diseases: Brown rot ( Evil's necklace ), rot disease ( Valsae ceratosperma ),powdery mildew( Podosphaera leucotricha ), leaf spot disease ( Podosphaera leucotricha ), black star disease ( Ventura unequal ),anthrax( Colletotrichum acutatum ), epidemic ( Phytophthora cactorum )wait.

[0202] Pear diseases: Black spot ( Venturia nashicola , V. pear ), black spot disease ( Alternaria alternate J Japanese pear pathotype ), red star disease ( Gymnosporangium haraeanum ), epidemic ( Phytophthora cactorum )wait.

[0203] Peach diseases: Brown rot ( Monilinia fructifera ), black star disease ( Cladosporium carpophilous ), stem spot rot ( Phomopsis sp.) etc.

[0204] Grape diseases: Black rot ( Elsinore ampelina ),anthrax( Glomerella cingulata ),powdery mildew( The hook-killer ), rust ( Phakopsora ampelopsidis ), black rot ( Guignard Bidwell's Downy mildew ( Plasmopara viticola )wait.

[0205] Diseases of persimmons: Anthracnose ( Gloeosporium kaki ), leaf disease ( Cercospora kaki , Mycosphaerella nawae )wait.

[0206] Diseases of melons: Anthracnose ( Colletotrichum lagenarium ),powdery mildew( Spheroid sooty ), vine blight ( Mycosphaerella melonis ), wilt disease ( Fusarium oxysporum Downy mildew ( Pseudoperonospora cubensis ), epidemic ( Phytophthora sp.), seedling blight ( Pythium sp.) etc.

[0207] Tomato diseases: ring rot ( Alternaria solani Leaf mold ( Cladosporium fulvum ), epidemic ( Phytophthora infestans ).

[0208] Eggplant diseases: Brown spot ( Phomopsis vexans ),powdery mildew( Erysiphe cichoracea )wait.

[0209] Diseases of cruciferous vegetables: Black spot ( Alternaria japonica ), vitiligo ( Cercosporella cabbages ), root nodule disease ( Brassica spp. Downy mildew ( Downy mildew), bacterial black spot disease ( Pseudomonas syringae pv. maculicola and Pseudomonas cannabina pv.alisalensis ), soft rot ( Pectobacterium carotovora subsp. carrot-eating )wait.

[0210] Diseases of scallions: Rust ( Garlic powder Downy mildew ( Downy mildew ), soft rot ( Pectobacterium carotovora subsp. carrot-eating )wait.

[0211] Soybean diseases: Purple spot disease ( Cercospora kikuchii ), black spot disease ( Elsinore wisteria Black spot disease ( Diaporthe phaseolorum var. soy Brown stripe disease Septoria wisteria ), spotted disease ( Cercospora soybean ), rust ( Phakopsora pachyrhizi ), stem blight ( Phytophthora sojae Damping-off disease caused by Rhizoctonia solani ( Rhizoctonia solani Brown ring spot disease ( Corynespora cashew nut ), sclerotinia stem rot Sclerotinia sclerotiorum )wait.

[0212] Diseases of green beans: Anthracnose ( Colletotrichum lindemuthianum )wait.

[0213] Peanut diseases: Black spot ( Cercospora personata Brown spot disease ( Cercospora peanut White silk disease ( Sclerotium rolfsii )wait.

[0214] Pea diseases: powdery mildew ( Erysiphe pea )wait.

[0215] Potato diseases: Early blight ( Alternaria solani ), epidemic ( Phytophthora infestans Red rot ( Phytophthora erythroseptica ), powdery scab ( Spongospora subterranean f. sp. underground )wait.

[0216] Strawberry diseases: powdery mildew ( Sphaerotheca humuli ),anthrax( Glomerella cingulata )wait.

[0217] Tea diseases: Net cake disease ( Reticulated exobasidium ), white star disease ( Elsinoe leucospila ), ring spot disease ( Pestalotiopsis sp.), anthrax ( Colletotrichum theae-sinensis )wait.

[0218] Tobacco diseases: Red spot disease ( Alternaria longipes ),powdery mildew( Erysipelas chicory ),anthrax( Colletotrichum tabacum Downy mildew ( Tobacco powdery mildew ), epidemic ( Phytophthora nicotianae )wait.

[0219] Rapeseed diseases: Sclerotinia stem rot ( Sclerotinia sclerotiorum Damping-off disease caused by Rhizoctonia spp. Rhizoctonia solani )wait.

[0220] Diseases of cotton: Damping-off caused by Rhizoctonia solani (…) Rhizoctonia solani ), white mold ( Mycosphaerella areola ), by Rhizosphere mold ( Thielaviopsis Black root rot caused by fungi ( ) Thielaviopsis basicola )wait.

[0221] Coffee diseases: Rust ( Hemileia the destroyer )wait.

[0222] Sugarcane diseases: Rust ( Puccinia melanocephala , Puccinia kuehnii ),smut( The scytamine-like plant )wait.

[0223] Sunflower diseases: Rust ( Puccinia helianthus )wait.

[0224] Diseases of sugar beets: Brown spot ( Cercospora beticola Leaf rot ( Thanatephorus cucumber ), root rot ( Cucumber beetle ), black root disease ( Aphanomyces cochlioides )wait.

[0225] Rose diseases: Black spot ( Diplocarpon rosae ),powdery mildew( Sphaerotheca pannosa Downy mildew ( Downy mildew )wait.

[0226] Diseases of chrysanthemums and Asteraceae vegetables: Downy mildew ( Bremia lettuce Brown spot disease ( Septoria chrysanthemums-indicia White rust ( Puccinia horiana )wait.

[0227] Diseases of various plants: Diseases caused by Pythium fungi ( Pythium aphanidermatum , P. Debarian , P. graminicola , P. irregulare , P. ultimum ), gray mold ( Botrytis cinerea ), sclerotinia stem rot Sclerotinia sclerotiorum )wait.

[0228] Radish diseases: Black spot disease Alternaria brassicicola )wait.

[0229] Lawn diseases: Coin spot ( Sclerotinia homoeocarpa Brown spot disease and large spot disease ( Rhizoctonia solani )wait.

[0230] Banana diseases: Leaf spot ( Mycosphaerella fijiensis , Mycosphaerella musicola )wait.

[0231] Sunflower diseases: Downy mildew ( Plasmopara halstedii )wait.

[0232] By Aspergillus ( Aspergillus ), Penicillium ( Penicillium Fusarium ( ) Fusarium ), Gibberellins ( Gibberella Trichoderma ( ) Trichoderma ), Rhizophora genus ( Thielaviopsis Rhizopus ( ) Rhizopus Mucor ( ) Mucor ), genus *Fougella* Corticium ), Phytophthora spp. Phoma ), Rhizoctonia spp. ( Rhizoctonia ) and Chlorodiclofenac ( Diplodia Various seed diseases or diseases in the early stages of plant growth caused by fungi, etc.

[0233] In addition, by controlling harmful insects belonging to the order Hemiptera, the composition of the present invention can also protect crops from viral diseases mediated by these insects, such as tomato yellow leaf curl virus, cucumber mosaic virus and turnip mosaic virus, beet western yellows virus and cauliflower mosaic virus.

[0234] Application method As for the application methods of the compositions of the present invention, for example, in the case of granules, planting hole treatment at the time of planting and root treatment of plants can be cited, and in the case of liquid formulations, immersion treatment, pre-planting irrigation treatment, root irrigation treatment of plants, soil irrigation treatment, foliar spraying, and aerial spraying can be cited.

[0235] The composition of the present invention prepared in this way can control the growth of unwanted plants relative to the useful plants by acting simultaneously or separately on the useful plants, or on the site where the useful plants are to grow, or on the site where they are growing. Furthermore, the aforementioned useful plants include field crops, horticultural crops, lawns, fruit trees, and non-agricultural land, etc.

[0236] The application amount and concentration of the composition of the present invention can be varied in a wide range depending on weather conditions, application period, application location, application method, etc. However, the application amount of components (A) to (C) contained in the composition of the present invention is usually about 0.05 to 600 g / a in total, preferably 0.1 to 200 g / a, and more preferably 0.5 to 100 g / a.

[0237] Example The present invention will be described in more detail below through examples, but the technical scope of the present invention is not limited to these examples.

[0238] Examples of formulations are shown below. It should be noted that "parts" refers to "parts by weight". However, the formulations described are not limited to those shown and can vary widely.

[0239] Formulation Example 1 (Emulsion) Dissolve 10 parts of each of the compositions of the present invention in 45 parts of Solvesso 150 and 35 parts of N-methylpyrrolidone, add 10 parts of emulsifier (trade name: Sorpol 3005X, manufactured by Toho Chemical Co., Ltd.), and stir to obtain 10% emulsions of each.

[0240] Formulation Example 2 (Wettable Powder) Add 20 parts of each of the compositions of the present invention to a mixture of 2 parts sodium dodecyl sulfate, 4 parts sodium lignosulfonate, 20 parts synthetic hydrous silica micro powder and 54 parts clay, and mix with a juice mixer to obtain a 20% wettable powder.

[0241] Formulation Example 3 (Granules) To each of the 5 parts of the composition of the present invention, add 2 parts of sodium dodecylbenzenesulfonate, 10 parts of bentonite, and 83 parts of clay, and mix thoroughly. Add an appropriate amount of water, stir further, granulate using a granulator, and dry in an air-conditioned environment to obtain 5% granules.

[0242] Formulation Example 4 (Powder) Dissolve one part of each of the compositions of the present invention in an appropriate amount of acetone, add five parts of synthetic aqueous silica micro powder, 0.3 parts of isopropyl phosphate (PAP) and 93.7 parts of clay, mix with a juice mixer, evaporate to remove acetone, and obtain a 1% powder.

[0243] Formulation Example 5 (Suspension) Mix 20 parts of each of the compositions of the present invention with 20 parts of water containing 3 parts of polyoxyethylene tristyrene phenyl ether phosphate triethanolamine and 0.2 parts of Rhodorsil 426R, wet pulverize using a sand mill, and then mix with 60 parts of water containing 8 parts of propylene glycol and 0.32 parts of xanthan gum to obtain a 20% aqueous suspension.

[0244] Formulation Example 6 (Liquid) Mix 10 parts of each of the compositions of the present invention, 5 parts of polyoxyethylene dehydrated sorbitol monostearate, 5 parts of propylene glycol and 70 parts of water to obtain 10% liquid solutions of each.

[0245] For specific combinations of particularly preferred compositions, the effects are confirmed through biological testing.

[0246] Biological Experiment Example 1: Preventive Effect For Chinese cabbage seedlings grown in 6.5cm plastic pots, spray with a solution containing compounds (A) and (C) shown in Table 1 (with 5000 times diluted Kumitene (registered trademark)) and air dry. Approximately 24 hours after spraying, spray inoculate with a suspension of cruciferous bacterial black spot fungus (containing 500 ppm Tween-20aq.) and manage in a humidified room set at 25°C. After 6 days, count the number of lesions and calculate the control value using the following formula. This experiment was conducted with 5 plants per plot and 1 replicate.

[0247] Control value = (1 - (average number of lesions in the treated area / average number of lesions in the untreated area)) × 100 The results are shown in Table 1.

[0248] [Table 1] To demonstrate the degree of synergistic effect, the "expected value of prevention and control" is calculated using the Colby method according to the following formula. A synergistic effect is considered to occur when the prevention and control value is greater than the "expected value of prevention and control".

[0249] Expected value = X + Y - XY / 100 X: Prevention value in area A (single-use zone) Y: Prevention value in C single-use zone result As a result, the plant pest control composition containing compounds (A) and (C) showed a synergistic effect on bacterial black spot disease of Chinese cabbage when applied to the target plant.

[0250] Biological Experiment Example 2: Therapeutic Effect For Chinese cabbage seedlings grown in 6.5cm plastic pots, a suspension of cruciferous bacterial black spot fungus (containing 500ppm Tween-20aq.) was sprayed and managed in a humidified room at 25°C for 1 day. Approximately 24 hours after inoculation, a solution containing compounds (A) and (C) shown in Table 2 (with 5000 times diluted Kumitene (registered trademark)) was sprayed and returned to the humidified room. After 6 days, the number of lesions was counted, and the control value was calculated using the following formula. This experiment was conducted with 5 plants per plot and 1 replicate.

[0251] Control value = (1 - (average number of lesions in the treated area / average number of lesions in the untreated area)) × 100 The results are shown in Table 2.

[0252] [Table 2] result As a result, the plant pest control composition containing compounds (A) and (C) showed a synergistic effect on bacterial black spot disease of Chinese cabbage when applied to the target plant.

[0253] Biological Experiment Example 3: Preventive Effect For cabbage seedlings grown in 6.5cm plastic pots, a solution containing compounds (A) and (C) shown in Table 3 (with 3300 times diluted Kumitene (registered trademark)) was sprayed. Approximately 24 hours after spraying, mycelial discs were prepared from a plate medium pre-cultured with sclerotium tumefaciens and inoculated onto the leaves. The plants were then managed in a humidified room set at 20°C. After 3 days, the diameter of the lesions was measured, and the control value was calculated using the following formula. This experiment was conducted with 5 plants per plot and 1 replicate.

[0254] Control value = (1 - (diameter of lesions in the treated area / diameter of lesions in the untreated area)) × 100 The results are shown in Table 3.

[0255] [Table 3] result As a result, the plant pest control composition containing compounds (A) and (C) showed a synergistic effect on cabbage sclerotinia stem rot when applied to the target plant.

[0256] This application claims priority based on Japanese Patent Application No. 2023-185781, filed on October 30, 2023. Japanese Patent Application No. 2023-185781 is incorporated herein by reference.

Claims

1. An agricultural and horticultural pest control composition, excluding rice pest control compositions, characterized in that, contain: (A) Saccharin and / or its salts, and A plant treatment composition selected from at least one of (B) insecticidal active compounds and (C) fungicidal active compounds.

2. The agricultural and horticultural pest control composition other than the rice pest control composition according to claim 1, wherein, The agricultural and horticultural pest control composition comprises (A) saccharin and / or its salt, and (C) a bactericidal active compound.

3. The agricultural and horticultural pest control composition other than the rice pest control composition according to claim 2, wherein, The bactericidal active compound (C) is an antibiotic for pesticide use.

4. The agricultural and horticultural pest control composition other than the rice pest control composition according to claim 3, wherein, The pesticide antibiotics comprise at least one antibiotic selected from chitin synthase inhibitors, enylpyranoside antibiotics, hexopyranosyl antibiotics, glucopyranosyl antibiotics, tetracycline antibiotics, and amphiphilic macrolide antifungal antibiotics.

5. The agricultural and horticultural pest control composition other than the water-removing rice pest control composition according to claim 4, wherein The antibiotic used in pesticides is at least one compound selected from polyoxin, kasugamycin, apigenin, streptomycin, and oxytetracycline, or a salt thereof.

6. The agricultural and horticultural pest control composition other than the water-removing rice pest control composition according to claim 5, wherein The antibiotic used in pesticides is polyoxin or its salt.

7. An agricultural and horticultural pest control composition other than the water-removing rice pest control composition according to claim 1, wherein The insecticidal active compound (B) is at least one compound selected from (b1) to (b35) below: (b1) Acetylcholinesterase (AChE) inhibitors, (b2) GABA-gated chloride channel blockers, (b3) Sodium channel modulators, (b4) Competitive modulators of nicotinic acetylcholine receptors (nAChR), (b5) Nicotinic acetylcholine receptor (nAChR) allosteric modulator - site I, (b6) Glutamate-gated chloride channel (GluCl) allosteric modulator, (b7) Juvenile hormone analogues, (b8) Other non-specific (multi-site) inhibitors, (b9) String tuner TRPV channel modulator, (b10) A mite growth inhibitor that acts on CHS1. (b11) Microbial-derived insect peri-feeding membrane disruptors, (b12) Inhibitor of mitochondrial ATP synthase, (b13) Oxidative phosphorylation uncoupling agents that disrupt the proton gradient. (b14) Nicotinic acetylcholine receptor (nAChR) channel blockers, (b15) Chitin biosynthesis inhibitors acting on CHS1, (b16) Chitin biosynthesis inhibitor (type 1). (b17) Eclipsis inhibitor (Diptera insects). (b18) Ecdysone (ecdysone) receptor agonist, (b19) Octopus amine receptor agonist, (b20) The Qo site, an inhibitor of mitochondrial electron transport system complex III. (b21) Inhibitor of mitochondrial electron transport system complex I (METI). (b22) Voltage-dependent sodium channel blockers, (b23) Acetyl-CoA carboxylase inhibitor, (b24) Inhibitors of mitochondrial electron transport system complex IV. (b25) Inhibitors of mitochondrial electron transport system complex II, (b26) Ryedin receptor modulator, (b27) Nicotinamide enzyme inhibitor for string instruments, (b28) GABA-gated chloride channel allosteric modulator, (b29) Baculovirus, (b30) Nicotinic acetylcholine receptor (nAChR) allosteric modulator - site II, (b31) Calcium-activated potassium channel (KCa2) regulator, (b32) Qi site, an inhibitor of mitochondrial electron transport system complex III. (b33) RNA interference-mediated target repressor, (b34) String tuning agent (target location undetermined), and (b35) Agents with unknown or uncertain mechanisms of action: A. Bacterial agents with unknown or uncertain mechanisms of action other than BT agents, synthetic agents with unknown or uncertain mechanisms of action, plant-derived ingredients containing extracts or unrefined oils, fungal agents with unknown or uncertain mechanisms of action, and physical disturbances with unknown or uncertain mechanisms of action. The bactericidal active compound (C) is at least one compound selected from (c1) to (c35): (c1) RNA polymerase I inhibitor, (c2) DNA / RNA biosynthesis inhibitors, (c3) Type II DNA topoisomerase (gyrase) inhibitor, (c4) An inhibitor of dihydroorotate dehydrogenase in the de novo biosynthesis of pyrimidines. (c5) Inhibitor of microtubule polymerization, (c6) Cell division inhibitor (site of action unknown), (c7) A translocator for spectrin-like proteins. (c8) Inhibitor of actin / myosin / filamentin function. (c9) Complex I (NADH oxidoreductase) inhibitor, (C10) Complex II (succinate dehydrogenase) inhibitor, (c11) Complex III (Qo site of ubiquitin oxidase) inhibitor, (c12) Complex III (ubiquinone reductase Qi site) inhibitor, (c13) An uncoupling agent for oxidative phosphorylation. (c14) Complex III (ubiquinone reductase Qo site marker-binding subsite) inhibitor, (c15) Methionine biosynthesis inhibitor, (c16) Inhibitor of protein biosynthesis (ribosomal translation initiation), (c17) Inhibitor of protein biosynthesis (ribosomal polypeptide elongation stage), (c18) Inhibitors of MAP / histidine kinases (os-2, HOG1) in osmolar signaling. (c19) Inhibitors of MAP / histidine kinases (os-1, Daf1) in osmolarity signaling. (c20) A methyltransferase inhibitor of phospholipid biosynthesis. (c21) An inhibitor of cellular lipid peroxidation. (c22) A cell membrane permeability fatty acid inhibitor. (c23) Inhibitors of lipid homeostasis and transport / storage, (c24) An inhibitor of C14 demethylase in sterol biosynthesis. (c25) An inhibitor of 3-keto reductase in the C4 demethylation of sterol biosynthesis. (c26) Squalene cyclooxygenase inhibitor in sterol biosynthesis, (c27) Chitin biosynthesis enzyme inhibitor, (c28) Cellulose biosynthesis enzyme inhibitor, (c29) An inhibitor of reductase in melanin biosynthesis. (c30) An inhibitor of dehydrating enzymes in melanin biosynthesis. (c31) A polyketide synthase inhibitor in melanin biosynthesis. (c32) Host plant resistance inducers other than saccharin or its salts. (c33) Compounds with unknown mechanisms of action. (c34) Multi-point contact active compounds, and (c35) Unclassified compounds.

8. An agricultural and horticultural pest control composition other than the water-removing rice pest control composition according to claim 1, wherein The insecticidal active compound (B) is at least one compound selected from the group consisting of: (b1) Acetylcholinesterase (AChE) inhibitors, (b2) GABA-gated chloride ion (chloride element ion) channel blockers, (b3) Sodium channel modulators, (b4) Competitive modulators of nicotinic acetylcholine receptors (nAChR), (b5) Nicotinic acetylcholine receptor (nAChR) allosteric modulator - site I, (b9) String tuner TRPV channel modulator, (b14) Nicotinic acetylcholine receptor (nAChR) channel blockers, (b16) Chitin biosynthesis inhibitor (type 1). (b18) Ecdysone (ecdysone) receptor agonist, (b26) Ryedin receptor modulators, and (b33) Oxazolidinone, pyrimethanil and isoxazolidinamide; The bactericidal active compound (C) is at least one compound selected from the group consisting of: (c1) RNA polymerase I inhibitor, (c2) DNA / RNA biosynthesis inhibitors, (c3) Type II DNA topoisomerase (gyrase) inhibitor, (c4) An inhibitor of dihydroorotate dehydrogenase in the de novo biosynthesis of pyrimidines. (c5) Inhibitor of microtubule polymerization, (c6) Cell division inhibitor (site of action unknown), (C10) Complex II (succinate dehydrogenase) inhibitor, (c11) Complex III (Qo site of ubiquitin oxidase) inhibitor, (c12) Complex III (ubiquinone reductase Qi site) inhibitor, (c16) Inhibitor of protein biosynthesis (ribosomal translation initiation), (c17) Inhibitor of protein biosynthesis (ribosomal polypeptide elongation stage), (c20) A methyltransferase inhibitor of phospholipid biosynthesis. (c24) An inhibitor of C14 demethylase in sterol biosynthesis. (c27) Chitin biosynthesis enzyme inhibitor, (c29) An inhibitor of reductase in melanin biosynthesis. (c31) A polyketide synthase inhibitor in melanin biosynthesis. (c32) Host plant resistance inducers other than saccharin or its salts. (c33) Compounds with unknown mechanisms of action. (c34) Multi-point contact active compounds, and (c35) Fluopyram.

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