Combination therapy of bispecific antibodies against CEACAM5 and CD47 and bispecific antibodies against CEACAM5 and CD3
A bispecific antibody combination targeting CEACAM5 and CD47, alongside CEACAM5 and CD3, enhances tumor cell phagocytosis, addressing limitations in current cancer therapies by improving efficacy and safety for treating solid tumors.
Patent Information
- Application Number
- JP2024573315
- Authority / Receiving Office
- JP · JP
- Patent Type
- Applications
- Current Assignee / Owner
- Priority Date
- 2022-06-16
- Filing Date
- 2023-06-15
- Publication Date
- 2025-07-23
AI Technical Summary
Current cancer treatments, including immunotherapies targeting CEA and CD47, face limitations in efficacy for solid tumors, with challenges such as tumor protection mechanisms, adverse effects, and low response rates, necessitating improved strategies to enhance tumor cell killing.
A combination therapy using bispecific antibodies that target both CEACAM5 and CD47, alongside CEACAM5 and CD3, to redirect macrophages for enhanced tumor cell phagocytosis, minimizing adverse effects by optimizing binding affinities and reducing immunogenicity.
The combination therapy significantly increases tumor cell killing efficacy, particularly in low CEACAM5-expressing tumors, with reduced side effects and improved progression-free and overall survival in patients with cancers like colorectal, lung, and gastric cancer.
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Abstract
Citation Information
Patent Citations
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