A piperonyl-quinone conjugate having insecticidal activity and its preparation method and application

By synthesizing piperine-morrhagic ketone compound, the problems of insufficient activity and high cost of single compounds have been solved, achieving high-efficiency insecticidal activity and stability, making it suitable for large-scale agricultural applications.

CN122404306APending Publication Date: 2026-07-17YIBIN SOUTHWEST JIAOTONG UNIV RES INST
View PDF 0 Cites 0 Cited by

Patent Information

Authority / Receiving Office
CN · China
Patent Type
Applications(China)
Current Assignee / Owner
YIBIN SOUTHWEST JIAOTONG UNIV RES INST
Filing Date
2026-04-28
Publication Date
2026-07-17

AI Technical Summary

Technical Problem

Existing plant-derived pesticides contain single active compounds with insufficient insecticidal activity, high costs, and poor stability of compound formulations, making it difficult to meet the needs of large-scale agricultural production.

Method used

By synthesizing piperine-morrhagic ketone composites, piperine and morrhagic ketone molecules are covalently linked using specific chemical reaction steps to form piperine-morrhagic ketone composites with insecticidal activity.

Benefits of technology

It significantly improves insecticidal activity and cytotoxicity against lepidopteran insects, reduces production costs, is suitable for industrial production, and the compound exhibits greater insecticidal and stomach poison activity than the single compound at the same concentration.

✦ Generated by Eureka AI based on patent content.

Smart Images

  • Figure CN122404306A_ABST
    Figure CN122404306A_ABST
Patent Text Reader

Abstract

本发明公开了一种具有杀虫活性的胡椒碱‑梣酮拼合物及其制备方法和应用,涉及医药化学技术领域。该胡椒碱‑梣酮拼合物由胡椒碱与梣酮通过酯基和肟酯基进行拼合。本发明还提供了胡椒碱‑梣酮拼合物的制备方法和应用。本发明提供的胡椒碱‑梣酮拼合物对鳞翅目昆虫表现出显著的杀虫活性及细胞毒性,可应用于天然植物源杀虫剂的开发,在制备新型环境友好型农药领域展现出潜在应用价值,有效解决了单一天然产物活性不足以及作用谱窄的问题。
Need to check novelty before this filing date? Find Prior Art