Harmful organism control composition for agricultural and horticultural use (excluding harmful organism control composition for paddy-field rice), and control method using same

Abstract

The present disclosure addresses the problem of providing: a novel harmful organism control composition for agricultural and horticultural use, which has a synergistic control effect in cultivation of plants excluding paddy-field rice; and a control method using the harmful organism control composition. The present disclosure relates to a harmful organism control composition for agricultural and horticultural use (excluding a harmful organism control composition for paddy-field rice), which comprises: (A) saccharin and / or a salt thereof; and at least one plant treatment composition selected from the group consisting of (B) an insecticidal active compound and (C) a bactericidal active compound.

Description

Agricultural and horticultural pest control compositions (excluding pest control compositions for paddy rice) and pest control methods using the same

[0001] The present disclosure relates to agricultural and horticultural pest control compositions (excluding pest control compositions for paddy rice) and pest control methods using the same.

[0002] Various pesticides have been used for the purposes of increasing agricultural crop yields, improving the quality of agricultural crops, etc. For example, in field crops, pests to be controlled include plant pathogens such as soft rot, black spot bacterial disease, and downy mildew; plant pathogens such as viruses and viroids; pests of the orders Coleoptera, Hemiptera, Diptera, Thysanoptera, and Lepidoptera; mollusks such as slugs; and nematodes such as Meloidogyne incognita. Many compositions and methods for using the same aimed at controlling these pests have been proposed (for example, Non-Patent Document 1 and Patent Document 1).

[0003] Non-Patent Document 1 describes that saccharin is effective in suppressing diseases caused by Zymoseptoria tritici in wheat. Thus, it is already known that saccharin is effective against various plant diseases. Patent Document 1 discloses a fungicide composition containing pyriophenone and at least one fungicide selected from the group consisting of bixafen, fluxapyroxad, penflufen, isopyrazam, fluopyram, ametoctrazin, fenpyrazamine, and sedaxane.

[0004] JP 2013-35823 A

[0005] Samara Mejri, Plant disease, Vol. 105, No. 4, April 2021

[0006] Repeated use of a single fungicide leads to the development of bacteria resistant to that fungicide and related fungicides. Therefore, research is being conducted to produce fungicides and fungicide compositions that are safer and more effective. The present disclosure aims to provide a novel agricultural and horticultural pest control composition that has a synergistic pest control effect in the cultivation of plants other than rice, and a control method using the same.

[0007] As a result of intensive research aimed at solving the above-mentioned problems, the present inventors have found that treatment with a composition comprising a mixture of saccharin, a salt thereof, or a mixture thereof with an insecticide or a fungicide can effectively eliminate harmful organisms in plants other than rice. The present disclosure has been completed based on this finding.

[0008] [Amendment based on Rule 91 25.04.2025] That is, the present disclosure is as follows: Item 1. An agricultural and horticultural pest control composition (excluding pest control compositions for paddy rice) containing (A) saccharin and / or a salt thereof, and at least one plant treatment composition selected from the group consisting of (B) an insecticidally active compound and (C) a fungicidal compound. Item 2. The agricultural and horticultural pest control composition (excluding pest control compositions for paddy rice) according to Item 1, wherein the agricultural and horticultural pest control composition contains the (A) saccharin and / or a salt thereof, and the (C) fungicidal compound. Item 3. The agricultural and horticultural pest control composition (excluding pest control compositions for paddy rice) according to Item 1 or 2, wherein the (C) fungicidal compound is a pesticide antibiotic. Item 4. Item 3. The agricultural and horticultural pest control composition according to Item 3 (excluding pest control compositions for paddy rice), wherein the agricultural and horticultural antibiotic comprises at least one antibiotic selected from the group consisting of chitin synthase inhibitors, enopyranuronic acid antibiotics, hexopyranosyl antibiotics, glucopyranosyl antibiotics, tetracycline antibiotics, and amphoteric macrolide antifungal antibiotics. Item 5. The agricultural and horticultural pest control composition according to Item 3 or 4 (excluding pest control compositions for paddy rice), wherein the agricultural and horticultural antibiotic is at least one compound or a salt thereof selected from the group consisting of polyoxin, kasugamycin, validamycin, streptomycin, and oxytetracycline. Item 6. The agricultural and horticultural pest control composition according to any one of Items 3 to 5 (excluding pest control compositions for paddy rice), wherein the agricultural and horticultural antibiotic is polyoxin or a salt thereof. Item 7. The (B) insecticidal compound is (b1) an acetylcholinesterase (AChE) inhibitor, (b2) a GABA-gated chloride ion channel blocker, (b3) a sodium channel modulator, (b4) a nicotinic acetylcholine receptor (nAChR) competitive modulator, (b5) a nicotinic acetylcholine receptor (nAChR) allosteric modulator - site I, (b6) a glutamate-gated chloride ion channel (GluCl) allosteric modulator, (b7) a juvenile hormone analog, (b8) other non-specific (multi-site) inhibitor, or (b9) a chordotonal organ TRPV channel modulator.(b10) mite growth inhibitors acting on CHS1, (b11) microbial insect midgut membrane disruptors, (b12) mitochondrial ATP synthase inhibitors, (b13) oxidative phosphorylation uncouplers that disrupt the proton gradient, (b14) nicotinic acetylcholine receptor (nAChR) channel blockers, (b15) chitin biosynthesis inhibitors acting on CHS1, (b16) chitin biosynthesis inhibitors (type 1), (b17) molting inhibitors (Diptera insects), (b18) ecdysone receptor agonists, (b19) octopamine receptor agonists, (b20) mitochondrial electron transport complex III inhibitors - Qo site, (b21) mitochondrial electron transport complex I inhibitors (METI), (b22) voltage-dependent sodium channel blockers, (b23) acetyl-CoA carboxylase inhibitors, (b24) mitochondrial electron transport complex IV inhibitors, (b25) mitochondrial electron transport complex II inhibitors, (b26) ryanodine receptor modulators, (b27) chordotonal organ nicotinic acid inhibitors (b28) GABA-gated chloride channel allosteric modulators, (b29) baculovirus, (b30) nicotinic acetylcholine receptor (nAChR) allosteric modulators - site II, (b31) calcium-activated potassium channel (KCa2) modulators, (b32) mitochondrial electron transport chain complex III inhibitors - Qi site, (b33) targeted suppressors via RNA interference, (b34) chordotonal organ modulators (target site unspecified), and and (b35) at least one compound selected from the group consisting of agent A with an unknown or uncertain mechanism of action, bactericidal agents (excluding BT agents) with an unknown or uncertain mechanism of action, synthetic substances, plant-derived components including extracts or unrefined oils with an unknown or uncertain mechanism of action, fungicidal agents with an unknown or uncertain mechanism of action, and physical disturbances with an unknown or uncertain mechanism of action, wherein the (C) fungicidal compound is (c1) an RNA polymerase I inhibitor, (c2) a DNA / RNA biosynthesis inhibitor, (c3) a DNA topoisomerase type II (gyrase) inhibitor, (c4) a dihydroorotate dehydrogenase inhibitor in de novo pyrimidine biosynthesis, (c5) a tubulin polymerization inhibitor, (c6) a cell division (site of action unknown) inhibitor,(c7) delocalizers of spectrin-like proteins, (c8) inhibitors of actin / myosin / fimbrin functions, (c9) inhibitors of complex I (NADH oxidoreductase), (c10) inhibitors of complex II (succinate dehydrogenase), (c11) inhibitors of complex III (ubiquinol oxidase Qo site), (c12) inhibitors of complex III (ubiquinone reductase Qi site), (c13) uncouplers of oxidative phosphorylation, (c14) inhibitors of complex III (ubiquinone reductase Qo site stigmatellin-binding subsite), (c15) inhibitors of methionine biosynthesis, (c16) inhibitors of protein biosynthesis (ribosomal translation initiation step), (c17) inhibitors of protein biosynthesis (ribosomal polypeptide elongation step), (c18) inhibitors of MAP histidine kinase (os-2, (c19) MAP / histidine kinase (os-1, Daf1) inhibitors in osmotic signal transduction, (c20) methyltransferase inhibitors in phospholipid biosynthesis, (c21) inhibitors of cellular lipid peroxidation, (c22) inhibitors of cell membrane-permeable fatty acids, (c23) inhibitors of lipid homeostasis and transport / storage, (c24) inhibitors of C14 demethylase in sterol biosynthesis, (c25) inhibitors of 3-ketoreductase in C4 demethylation in sterol biosynthesis, (c26) squalene epoxidase inhibitors in sterol biosynthesis, (c27) chitin biosynthesis enzyme inhibitors, (c28) cellulose biosynthesis enzyme inhibitors Item 8. The agricultural and horticultural pest control composition according to any one of Items 1 to 6, wherein the (B) insecticidal compound is at least one compound selected from the group consisting of (b1) an acetylcholinesterase (AChE) inhibitor, (b2) a GABA-gated chloride ion (chloride ion) channel blocker, (b3) a sodium channel modulator, (b4) a nicotinic acetylcholine receptor (nAChR) competitive modulator,(b5) nicotinic acetylcholine receptor (nAChR) allosteric modulators - site I, (b9) chordotonal organ TRPV channel modulators, (b14) nicotinic acetylcholine receptor (nAChR) channel blockers, (b16) chitin biosynthesis inhibitors (type 1), (b18) ecdysone receptor agonists, (b26) ryanodine receptor modulators, and (b33) at least one compound selected from the group consisting of oxazosulfil, benzpyrimoxane, and isocycloceram, wherein the (C) fungicidal compound is (c1) an RNA polymerase I inhibitor, (c2) a DNA / RNA biosynthesis inhibitor, (c3) a DNA topoisomerase Type II (gyrase) inhibitors, (c4) dihydroorotate dehydrogenase inhibitors in de novo pyrimidine biosynthesis, (c5) tubulin polymerization inhibitors, (c6) cell division (unknown site of action) inhibitors, (c10) complex II (succinate dehydrogenase) inhibitors, (c11) complex III (ubiquinol oxidase Qo site) inhibitors, (c12) complex III (ubiquinone reductase Qi site) inhibitors, (c16) protein biosynthesis (ribosome translation initiation step) inhibitors, (c17) protein biosynthesis (ribosome Item 8. The agricultural and horticultural pest control composition according to any one of Items 1 to 7 (excluding pest control compositions for paddy rice), which is at least one compound selected from the group consisting of (c1) a methyltransferase inhibitor in phospholipid biosynthesis, (c20) a methyltransferase inhibitor in phospholipid biosynthesis, (c24) a demethylase inhibitor at C14 position in sterol biosynthesis, (c27) a chitin biosynthesis enzyme inhibitor, (c29) a reductase inhibitor in melanin biosynthesis, (c31) a polyketamide synthase inhibitor in melanin biosynthesis, (c32) a resistance inducer in a host plant (excluding saccharin or a salt thereof), (c33) a compound with an unknown mechanism of action, (c34) a multisite contact active compound, and (c35) quinofumelin. A method for controlling pests, comprising the step of applying a composition containing (A) saccharin and / or a salt thereof and at least one plant treatment composition selected from the group consisting of (B) an insecticidal compound and (C) a fungicidal compound to pests, a habitat of pests, plants, or a cultivation carrier for plants, provided that:(excluding a method for controlling rice pests). Item 10. Use of a composition containing (A) saccharin and / or a salt thereof and at least one plant treatment composition selected from the group consisting of (B) an insecticidal compound and (C) a fungicidal compound for controlling agricultural and horticultural pests (excluding use for controlling rice pests).

[0009] According to the present disclosure, it is possible to provide a novel agricultural and horticultural pest control composition (excluding pest control compositions for paddy rice) that exhibits a remarkable synergistic plant disease control effect that cannot be predicted from the plant disease control effect obtained by using only saccharin or a salt thereof, or a mixture thereof, or by using only a plant treatment composition.

[0010] Agricultural and horticultural pest control composition (excluding pest control compositions for paddy rice) The agricultural and horticultural pest control composition of the present disclosure (excluding pest control compositions for paddy rice) (hereinafter sometimes referred to as "the composition of the present disclosure") contains (A) saccharin and / or a salt thereof, and at least one plant treatment composition selected from the group consisting of (B) an insecticidally active compound and (C) a fungicidal compound. The agricultural and horticultural pest control composition of the present disclosure (excluding pest control compositions for paddy rice) is used as a mixture combining (A) saccharin and / or a salt thereof, and at least one plant treatment composition selected from the group consisting of (B) an insecticidally active compound and (C) a fungicidal compound, and exhibits excellent pest control effects in the cultivation of plants other than paddy rice.

[0011] (A) Saccharin and / or Salts Thereof Saccharin (1,1-dioxo-1,2-benzothiazol-3-one) is a compound represented by the following formula (1): Saccharin is generally used as an artificial sweetener, but is also known to have resistance-inducing activity, and can exert a disease-suppressing effect by inducing resistance to disease in host plants (activating the disease control system).

[0012]

[0013] The saccharin salt may be any kind of salt as long as it is agriculturally acceptable. Examples of such salts include inorganic salts (e.g., hydrochloride, sulfate, nitrate, etc.), organic salts (e.g., acetate, methanesulfonate, etc.), alkali metal salts (e.g., sodium salt, potassium salt, etc.), alkaline earth metal salts (e.g., calcium salt, etc.), and quaternary ammonium salts (e.g., tetramethylammonium salt, tetraethylammonium salt, etc.), with alkali metal salts being preferred, and sodium salts being more preferred.

[0014] The application amount and application concentration of the composition of the present disclosure can be varied depending on weather conditions, application time, application location, application method, etc., but the application amount of saccharin and / or a salt thereof is usually 0.05 to 300 g / a, preferably 0.1 to 100 g / a, and more preferably 0.15 to 50 g / a, except when the composition is applied to crops in cell trays, seedling pots, etc. before planting.

[0015] Plant Treatment Composition The composition of the present disclosure comprises at least one plant treatment composition selected from the group consisting of (B) an insecticidally active compound and (C) a fungicidal compound.

[0016] (B) Insecticidally Active Compound The insecticidally active compound contained in the agricultural and horticultural pest control composition of the present disclosure (excluding the pest control composition for paddy rice) can be any compound known to have a control effect against agricultural pests, without particular limitation. The insecticidally active compound here includes not only insecticides but also miticides and nematocides. The insecticidally active compound can be formulated alone or in a suitable mixture of two or more types.

[0017] (B) The insecticidally active compound is not particularly limited, and examples thereof include compounds belonging to Groups 1 to 36 and Groups UN to UNM in the action classification by IRAC (Insecticide Resistance Action Committee).

[0018] (b1) Group 1: acetylcholinesterase (AChE) inhibitors Examples of acetylcholinesterase (AChE) inhibitors include alanycarb, aldicarb, bendiocarb, benfuracarb, butocarboxim, butoxycarboxim, carbaryl (NAC), carbofuran, carbosulfan, ethiofencarb, fenobucarb (BPMC), formetanate, furathiocarb, isoprocarb (MIPC), methiocarb, methomyl, metolcarb (MTMC), oxamyl, pirimicarb, propoxur (PHC), thiodicarb, thiofanox (thi ofanox), triazamate, trimethacarb, XMC, xylylcarb (MPMC) and other carbamate compounds (1A); acephate, azamethiphos, azinphos-ethyl, azinphos-methyl, cadusafos, chlorethoxyfos, chlorfenvinphos orfenvinphos (CVP), chlormephos (chlormephos), chlorpyrifos (chlorpyrifos), chlorpyrifos-methyl (chlorpyrifos-methyl), coumaphos (coumaphos), cyanophos (cyanophos: CYAP), demeton-S-methyl (demeton-S-methyl), diazinon (diazinon), dichlorvos (dichlorvos: DDVP), dicrotophos (dicrotophos), dimethoate (dimethoate),Dimethylvinphos, ethylthiometon (disulfoton), EPN, ethion, ethoprophos, famphur, fenamiphos, fenitrothion (MEP), fenthion (MPP), fosthiazate, heptenophos, imicyafos, isofenphos nphos), isopropyl = O- (methoxyaminothiophosphoryl) salicylate (isopropyl-O- (methoxyaminothiophosphoryl) salicylate), isoxathion (isoxathion), malathion (malathion), mecarbam (mecarbam), methamidophos (methamidophos), methidathion (methidathion: DMTP), mevinphos (mevinphos), monocrotophos (monocrotophos), naled (naled: BRP), omethoate (omethoate), oxydemeton-methyl (oxydemeton-methyl), parathion (parathion), methyl parathion (parathion-methyl), phenthoate (phenthoate: PAP), phorate (phorate), phosalone (phosalone), phosmet (phosmet: PMP), phosphamidon (phosphamidon), phoxim (phoxim), pirimiphos-methyl (pirimiphos-methyl), Profenofos (profenofos), propetamphos (propetamphos), prothiofos (prothiofos), pyraclofos (pyraclofos), pyridaphenthion (pyridaphenthion), quinalphos (quinalphos), sulfotep (sulfotep), tebupirimfos (tebupirimfos), temephos (temephos), terbufos (terbufos), tetrachlorvinphos (tetrachlorvinphos:CVMP), thiometon (thiometon),Organophosphorus compounds (1B) such as triazophos, trichlorfon (DEP), and vamidothion are included.

[0019] (b2) Group 2: GABAergic chloride ion (chloride ion) channel blockers Examples of GABAergic chloride ion (chloride ion) channel blockers include cyclic diene organic chlorine compounds (2A) such as chlordane and benzoepin (endosulfan); phenylpyrazole (fiprole) compounds (2B) such as ethiprole and fipronil.

[0020] (b3) Group 3: Sodium channel modulators Examples of sodium channel modulators include acrinathrin, allethrin (allethrin, d-cis-trans-, d-trans-isomers), bifenthrin, bioallethrin (bioallethrin, S-cyclopentenyl-isomers), bioresmethrin, cycloprothrin, cyfluthrin (cyfluthrin, β-isomers), Cyhalothrin (cyhalothrin, λ- and γ-isomers), cypermethrin (cypermethrin, α-, β-, θ-, and ζ-isomers), cyphenothrin [(1R)-trans isomer], deltamethrin, empenthrin [(EZ)-(1R)-trans isomer], esfenvalerate, etofenprox, and fenpropathrin npropathrin), fenvalerate, flucythrinate, flumethrin, fluvalinate (τ-fluvalinate), halfenprox, imiprothrin, kadethrin, permethrin, phenothrin [(1R)-trans isomer], prallethrin ), pyrethroid (pyrethrin) compounds such as pyrethrins, resmethrin, silafluofen, tefluthrin, phthalthrin (tetramethrin), tetramethrin [(1R)-trans isomer], tralomethrin, and transfluthrin (3A); DDT and methoxychlor (3B).

[0021] (b4) Group 4: Nicotinic acetylcholine receptor (nAChR) competitive modulators Examples of nicotinic acetylcholine receptor (nAChR) competitive modulators include neonicotinoid compounds (4A) such as acetamiprid, clothianidin, dinotefuran, imidacloprid, nitenpyram, thiacloprid, and thiamethoxam; nicotine sulfate (nicotine); nicotine compounds (4B) such as sulfoxaflor; sulfoximine compounds (4C) such as sulfoxaflor; butenolide compounds (4D) such as flupyradifurone; mesoionic compounds (4E) such as dichloromezotiaz, fenmezoditiaz, triflumezopyrim; and pyridylidene compounds (4F) such as flupirimine.

[0022] (b5) Group 5: Nicotinic acetylcholine receptor (nAChR) allosteric modulators - Site I Examples of nicotinic acetylcholine receptor (nAChR) allosteric modulators - Site I include spinosyn compounds such as spinetoram and spinosad.

[0023] (b6) Group 6: Glutamate-gated chloride channel (GluCl) allosteric modulators Examples of glutamate-gated chloride channel (GluCl) allosteric modulators include avermectin compounds such as abamectin, and milbemycin compounds such as emamectin benzoate, lepimectin, and milbemectin.

[0024] (b7) Group 7: Juvenile hormone mimetics Examples of juvenile hormone mimetics include juvenile hormone analogues such as hydroprene, kinoprene, methoprene (7A); fenoxycarb (7B); pyriproxyfen (7C); and the like.

[0025] (b8) Group 8: Other Nonspecific (Multi-site) Inhibitors Examples of other nonspecific (multi-site) inhibitors include alkyl halide compounds (8A) such as 1,3-dichloropropene, methyl bromide, and other alkyl halides; chloropicrin (8B); fluoride compounds (8C) such as cryolite (sodium aluminum fluoride) and sulfuryl fluoride; borax, boric acid, disodium octaborate, sodium borate, and sodium metaborate (8D); tartar emetic (8E); and methyl isothiocyanate generators (8F) such as dazomet, metam, and methyl isothiocyanate.

[0026] (b9) Group 9: Chordotonal organ TRPV channel modulators Examples of chordotonal organ TRPV channel modulators include pyridine azomethine derivatives (9B) such as pymetrozine and pyrifluquinazon; and pyropene compounds (9D) such as afidopyropen.

[0027] (b10) Group 10: Mite growth inhibitors acting on CHS1 Examples of mite growth inhibitors acting on CHS1 include clofentezine, diflovidazin, hexythiazox, etc. (10A); etoxazole (10B), etc.

[0028] (b11) Group 11: Microbial-derived insect midgut membrane disrupting agents Examples of microbial-derived insect midgut membrane disrupting agents include Bacillus thuringiensis subsp. israelensis, Bacillus thuringiensis subsp. Aizawai, Bacillus thuringiensis subsp. Kurstaki, and Bacillus thuringiensis subsp. tenebrionis (proteins contained in Bt crops: Cry1Ab, Cry1Ac, Cry1Fa, Cry1A.105, Cry2Ab, Vip3A, mCry3A, Cry2Ab, Cry3Bb, Cry34Ab1 / Cry35Ab1). thuringiensis and the insecticidal protein it produces (11A); Bacillus sphaericus (11B); and the like.

[0029] (b12) Group 12: Mitochondrial ATP synthase inhibitors Examples of mitochondrial ATP synthase inhibitors include diafenthiuron (12A); organotin acaricides such as azocyclotin, tricyclohexyltin (hexatin) hydroxide, and fenbutatin oxide (12B); propargite (BPPS) (12C); and tetradifon (12D).

[0030] (b13) Group 13: Oxidative phosphorylation uncouplers that disrupt proton gradients Examples of oxidative phosphorylation uncouplers that disrupt proton gradients include pyrrole compounds such as chlorfenapyr; dinitrophenol compounds such as DNOC; and sulfluramid.

[0031] (b14) Group 14: Nicotinic acetylcholine receptor (nAChR) channel blockers Examples of nicotinic acetylcholine receptor (nAChR) channel blockers include nereistoxin analogs such as bensultap, cartap hydrochloride, thiocyclam, and thiosultapsodium.

[0032] (b15) Group 15: Chitin Biosynthesis Inhibitors Acting on CHS1 Examples of chitin biosynthesis inhibitors acting on CHS1 include benzoylurea compounds such as bistrifluron, chlorfluazuron, diflubenzuron, flucycloxuron, flufenoxuron, hexaflumuron, lufenuron, novaluron, noviflumuron, teflubenzuron, and triflumuron.

[0033] (b16) Group 16: Chitin Biosynthesis Inhibitors (Type 1) Examples of chitin biosynthesis inhibitors (type 1) include buprofezin.

[0034] (b17) Group 17: Molting inhibitors (Diptera) Examples of molting inhibitors (Diptera) include cyromazine.

[0035] (b18) Group 18: Molting hormone (ecdysone) receptor agonists Examples of the molting hormone (ecdysone) receptor agonists include diacyl-hydrazine compounds such as chromafenozide, halofenozide, methoxyfenozide, and tebufenozide.

[0036] (b19) Group 19: Octopamine Receptor Agonists Examples of octopamine receptor agonists include amitraz.

[0037] (b20) Group 20: Mitochondrial electron transport chain complex III inhibitors-Qo site Examples of mitochondrial electron transport chain complex III inhibitors-Qo site include hydramethylnon (20A), acequinocyl (20B), fluacrypyrim (20C), bifenazate (20D), and the like.

[0038] (b21) Group 21: Mitochondrial Electron Transport Complex I Inhibitors (METI) Examples of mitochondrial electron transport complex I inhibitors (METI) include METI agents (21A) such as fenazaquin, fenpyroximate, pyridaben, pyrimidifen, tebufenpyrad, and tolfenpyrad; and derris (rotenone) (21B).

[0039] (b22) Group 22: Voltage-dependent sodium channel blockers Examples of voltage-dependent sodium channel blockers include oxadiazine compounds (22A) such as indoxacarb; semicarbazone compounds (22B) such as metaflumizone; and the like.

[0040] (b23) Group 23: Acetyl-CoA Carboxylase Inhibitors Examples of the acetyl-CoA carboxylase inhibitors include tetronic acid or tetramic acid derivatives such as spirodiclofen, spiromesifen, spiropidione, and spirotetramat.

[0041] (b24) Group 24: Mitochondrial Electron Transport Complex IV Inhibitors Examples of mitochondrial electron transport complex IV inhibitors include phosphine compounds (24A) such as aluminum phosphide, calcium phosphide, hydrogen phosphide, and zinc phosphide; and cyanides (24B) such as hydrocyanic acid (calcium cyanide, sodium cyanide), potassium cyanide, and the like.

[0042] (b25) Group 25: Mitochondrial Electron Transport Complex II Inhibitors Examples of mitochondrial electron transport complex II inhibitors include β-ketonitrile derivatives (25A) such as cyenopyrafen and cyflumetofen; carboxanilide compounds (25B) such as pyflubumide; and the like.

[0043] (b26) Group 28: Ryanodine Receptor Modulators Examples of ryanodine receptor modulators include diamide compounds such as chlorantraniliprole, cyantraniliprole, cycloniliprole, flubendiamide, and tetraniliprole.

[0044] (b27) Group 29: Chordotonal organ modulators Examples of chordotonal organ modulators include flonicamid.

[0045] (b28) Group 30: GABA-gated chloride ion channel allosteric modulators Examples of the GABA-gated chloride ion channel allosteric modulators include metadiamide compounds such as broflanilide, and isoxazoline compounds such as fluxametamide and isocycloseram.

[0046] (b29) Group 31: Baculoviruses Examples of baculoviruses include granulosis viruses (GVs) such as codling moth Cydia pomonella GV and false codling moth Thaumatotibia leucotreta GV, and polyhedrosis viruses (NPVs) such as velvet bean caterpillar Anticarsia gemmatalis MNPV and cotton bollworm Helicoverpa armigera NPV.

[0047] (b30) Group 32: Nicotinic acetylcholine receptor (nAChR) allosteric modulators - site II Examples of nicotinic acetylcholine receptor (nAChR) allosteric modulators - site II include GS-omega / kappa HXTX-Hv1a peptide.

[0048] (b31) Group 33: Calcium-activated potassium channel (KCa2) modulators Examples of calcium-activated potassium channel (KCa2) modulators include acinonapyr.

[0049] (b32) Group 34: Mitochondrial electron transport complex III inhibitors-Qi site Examples of mitochondrial electron transport complex III inhibitors-Qi site include flometoquin.

[0050] (b33) Group 35: Targeted Inhibitors Mediated by RNA Interference Examples of targeted inhibitors mediating RNA interference include Ledprona.

[0051] (b34) Group 36: Chordotonal organ modulators (unspecified target site) Examples of chordotonal organ modulators (unspecified target site) include pyridazines or pyrazole carboxamides such as dimpropyridaz.

[0052] (b35) Group UN: Agent A with an unknown or unclear mechanism of action Examples of Agent A with an unknown or unclear mechanism of action include azadirachtin, benzoximate, benzpyrimoxan, bromopropylate, quinomethionat, dicofol, lime sulfur mixture, manzeb, oxazosulfyl, pyridalyl, sulfur, etc. (b36) Group UNB: Bacterial agents with an unknown or unclear mechanism of action (excluding BT agents) Examples of bacterial agents with an unknown or unclear mechanism of action (excluding BT agents) include Burkholderia spp, Wolbachia pipientis (Zap), etc. (b37) Group UNE: Plant-derived ingredients including synthetic compounds, extracts, or unrefined oils with an unknown or unclear mechanism of action. Examples of plant-derived ingredients including synthetic compounds, extracts, or unrefined oils with an unknown or unclear mechanism of action include Chenopodium ambrosioides near ambrosioides, (American ant-weed) extract, and fatty acid monoesters of glycerin or propanediol in neem oil. (b38) Group UNF: Antifungal agents with an unknown or unclear mechanism of action. Examples of antifungal agents with an unknown or unclear mechanism of action include Akanthomyces muscarius Ve6, Beauveria bassiana strains, Metarhizium brunneum strain F52, and Paecilomyces fumosoroseus Apopka strain 97. (b39) Group UNM: Nonspecific physical perturbations with an unknown or unclear mechanism of action. Examples of nonspecific physical perturbations with an unknown or unclear mechanism of action include diatomaceous earth and mineral oil.

[0053] Other examples include known agricultural and horticultural insecticides. These insecticidal compounds are known compounds and are commercially available, so they are easily available.

[0054] In the present disclosure, (B) an insecticidal active compound is typically blended in an amount of 0.01 to 20,000 parts by mass, preferably 0.1 to 10,000 parts by mass, more preferably 0.5 to 1,000 parts by mass per 100 parts by mass of (A) saccharin and / or its salt.

[0055] (C) Fungicidal Compounds The fungicidal compounds contained in the agricultural and horticultural pest control compositions of the present disclosure (excluding pest control compositions for paddy rice) can be any known compounds that have a control effect on agricultural pests, without particular limitation. The fungicidal compounds herein include not only fungicides but also bactericides and virucides. The fungicidal compounds can be used alone or in combination of two or more.

[0056] (C) The fungicidal compound is not particularly limited, and examples thereof include compounds classified as A (nucleic acid synthesis metabolism), B (cytoskeleton and motor protein), C (respiration), D (amino acid and protein biosynthesis), E (signal transduction), F (lipid biosynthesis or transport / cell membrane structure or function), G (cell membrane sterol biosynthesis), H (cell wall biosynthesis), I (cell wall melanin biosynthesis), P (host plant resistance induction), M (multi-site contact active compound), BM (biopesticide with multiple mechanisms of action: plant extract), U (mechanism of action unknown), and unclassified. Among these, the following A group, B group, C group, D group, F group, G group, I group, P group, M group, and U group are preferred.

[0057] Group A Group A (nucleic acid synthesis metabolism) includes, for example, RNA polymerase I inhibitors, adenosine deaminase, DNA / RNA biosynthesis inhibitors, DNA topoisomerase type II (gyrase) inhibitors, and dihydroorotate dehydrogenase inhibitors in de novo pyrimidine biosynthesis.

[0058] (c1) Group A1: RNA polymerase I inhibitors (FRAC group code 4) Examples of RNA polymerase I inhibitors include acylalanines such as benalaxyl, benalaxyl-M, furalaxyl, metalaxyl, and metalaxyl-M; oxazolidinones such as oxadixyl; and butyrolactones such as ofurace.

[0059] (c2) Group A2: Adenosine deaminase inhibitors (FRAC group code 8) Examples of adenosine deaminase inhibitors include hydroxy(2-amino-)pyrimidines such as bupirimate, dimethirimol, and ethirimol.

[0060] (c3) Group A3: DNA / RNA biosynthesis inhibitors (FRAC group code 32) Examples of DNA / RNA biosynthesis inhibitors include isoxazoles such as hydroxyisoxazole (hymexazole), and isothiazolones such as octhilinone.

[0061] (c4) Group A4: DNA topoisomerase type II (gyrase) inhibitors (FRAC group code 31) Examples of DNA topoisomerase type II (gyrase) inhibitors include carboxylic acids such as oxolinic acid. (c5) Group A5: Dihydroorotate dehydrogenase inhibitors in de novo pyrimidine biosynthesis (FRAC group code 52) Examples of dihydroorotate dehydrogenase inhibitors in de novo pyrimidine biosynthesis include phenylpropanols such as ipflufenoquine, and dihydroisoquinolines such as quinofumelin.

[0062] Group B Group B (cytoskeleton and motor proteins) includes, for example, tubulin polymerization inhibitors, cell division (unknown site of action) inhibitors, delocalizing agents of spectrin-like proteins, inhibitors of actin / myosin / fimbrin function, and tubulin dynamics modulators.

[0063] (c6) Group B1, B2, B3: Tubulin polymerization inhibitors (FRAC group codes 1, 10, 22) Examples of β-tubulin polymerization inhibitors include benzimidazoles such as benomyl, carbendazim, fuberidazole, and thiabendazole; thiophanates such as thiophanate and thiophanate-methyl; N-phenylcarbamates such as diethofencarb; toluamides such as zoxamide; and ethylaminothiazolecarboxamides such as ethaboxam.

[0064] (c7) Group B4: Cell division (unknown site of action) inhibitors (FRAC group code 20) Examples of cell division (unknown site of action) inhibitors include phenylureas such as pencycuron.

[0065] (c8) Group B5: Delocalizing Agents for Spectrin-Like Proteins (FRAC Group Code 43) Examples of the delocalizing agents for spectrin-like proteins include pyridinylmethylbenzamides such as fluopicolide and fluopimomide.

[0066] (c9) Group B6: Inhibitors of actin / myosin / fimbrin function (FRAC group code 47) Examples of inhibitors of actin / myosin / fimbrin function include aminocyanoacrylates such as phenamacril; benzophenones such as metrafenone; benzoylpyridines such as pyriophenone; and the like.

[0067] (c10) Group B7: Tubulin Dynamics Modulators (FRAC Group Code 53) Examples of the tubulin dynamics modulators include pyridazines such as pyridachlometyl.

[0068] Group C Examples of Group C (respiration) inhibitors include complex I (NADH oxidoreductase) inhibitors, complex II (succinate dehydrogenase) inhibitors, complex III (cytochrome bc1 (ubiquinol oxidase) Qo site (cytb gene)) inhibitors, complex III (ubiquinone reductase Qi site) inhibitors, uncouplers of oxidative phosphorylation, inhibitors of oxidative phosphorylation and ATP synthase, ATP transport inhibitors, and complex III (ubiquinone reductase Q1, Qo site, stigmatellin binding mode) inhibitors.

[0069] (c11) Group C1: Complex I (NADH oxidoreductase) inhibitors (FRAC group code 39) Examples of complex I (NADH oxidoreductase) inhibitors include pyrimidinamines such as diflumetorim; pyrazolecarboxamides such as tolfenpyrad; quinazolines such as fenazaquin; and the like.

[0070] (c12) Group C2: Complex II (succinate dehydrogenase) inhibitors (FRAC group code 7) Examples of complex II (succinate dehydrogenase) inhibitors include phenylbenzamides such as benodanil, flutolanil, mepronil, etc.; phenyloxoethylthiophenamides such as isofetamide, etc.; pyridinylethylbenzamides such as fluopyram, etc.; phenylcyclobutylpyridine amides such as cyclobutrifluram, etc.; furancarboxamides such as fenfuram, etc.; oxathiincarboxamides such as carboxin, oxycarboxin, etc.; thiazolecarboxamides such as thifluzamide, etc.; benzovindiflupyr, Examples of the antipyretic agent include pyrazole-4-carboxamides such as bixafen, fluindapyr, fluxapyroxad, furametpyr, inpirfluxam, isopyrazam, penflufen, penthiopyrad, and sedaxane; N-cyclopropyl-N-benzylpyrazolecarboxamides such as isoflucypram; N-methoxy(phenylethyl)pyrazolecarboxamides such as pydiflumetofen; pyridinecarboxamides such as boscalid; and pyrazinecarboxamides such as pyraziflumide.

[0071] (c13) Group C3: Complex III (cytochrome bc1 (ubiquinol oxidase) Qo site (cytb gene)) inhibitors Complex III (cytochrome bc1 (ubiquinol oxidase) Qo site (cytb gene)) inhibitors (QoI fungicides (Qo inhibitors)) (FRAC group code 11) include, for example, methoxyacrylates such as azoxystrobin, cumoxystrobin, enoxastrobin, flufenoxystrobin, picoxystrobin, and pyraoxystrobin; methoxyacetamides such as mandestrobin; pyraclostrobin, pyrametostrobin, and triclopyricarb. Examples of QoI fungicides (Qo inhibitors; subgroup A) (FRAC group code 11A) include tetrazolinones such as methyltetrapyrrole, methyltetrapyrrole, and the like.

[0072] (c14) Group C4: Complex III (ubiquinone reductase Qi site) inhibitors (FRAC group code 21) Examples of complex III (ubiquinone reductase Qi site) inhibitors include cyanoimidazoles such as cyazofamid; sulfamoyltriazoles such as amisulbrom; picolinamides such as fenpicoxamid and florylpicoxamid.

[0073] (c15) Group C5: Uncouplers of Oxidative Phosphorylation (FRAC Group Code 29) Examples of uncouplers of oxidative phosphorylation include dinitrophenylcrotonates such as binapacryl, meptyl dinocap, and DPC (dinocap); 2,6-dinitroanilines such as fluazinam; and pyrimidinone hydrazones such as ferimzone.

[0074] (c16) Group C6: Inhibitors of oxidative phosphorylation and ATP synthase (FRAC group code 30) Examples of inhibitors of oxidative phosphorylation and ATP synthase include triphenyltin compounds such as organotins (triphenyltin acetate, triphenyltin chloride, triphenyltin hydroxide).

[0075] (c17) Group C7: ATP transport inhibitors (FRAC group code 38) Examples of ATP transport inhibitors include thiophenecarboxamides such as silthiofam.

[0076] (c18) Group C8: Complex III (ubiquinone reductase Q1, Qo site, stigmatellin binding mode) inhibitors (FRAC group code 45) Examples of complex III (ubiquinone reductase Q1, Qo site, stigmatellin binding mode) inhibitors include triazolopyrimidylamines such as ametoctradin.

[0077] [Correction based on Rule 91 25.04.2025] Group D Group D (amino acid and protein biosynthesis inhibitors) includes, for example, methionine biosynthesis (cgs gene) inhibitors, protein biosynthesis (ribosome translation termination step) inhibitors, protein biosynthesis (ribosome translation initiation step) inhibitors, protein biosynthesis (ribosome polypeptide elongation step) inhibitors, leucyl-tRNA synthesis (LeuRNA) inhibitors, etc.

[0078] (c19-1) Group D1: Methionine biosynthesis (cgs gene) inhibitors (FRAC group code 9) Examples of methionine biosynthesis (cgs gene) inhibitors include anilinopyrimidines such as cyprodinil, mepanipyrim, and pyrimethanil.

[0079] [Correction based on Rule 91 25.04.2025] (c19-2) Group D2: Protein biosynthesis (ribosomal translation termination) inhibitors (FRAC group code 23) Examples of protein biosynthesis (ribosomal translation termination) inhibitors include enopyranuronic acid antibiotics such as Blasticidin S.

[0080] [Correction based on Rule 91 25.04.2025] (c19-3) Group D3: Protein biosynthesis (ribosomal translation initiation stage) inhibitors (FRAC group code 24), Group D4: Protein biosynthesis (ribosomal translation initiation stage) inhibitors (FRAC group code 25) Examples of protein biosynthesis (ribosomal translation initiation stage) inhibitors include hexopyranosyl antibiotics such as kasugamycin; glucopyranosyl antibiotics such as streptomycin; etc.

[0081] [Correction based on Rule 91 25.04.2025] (c19-4) Group D5: Inhibitors of protein biosynthesis (ribosomal polypeptide elongation stage) (FRAC Group Code 41) Examples of inhibitors of protein biosynthesis (ribosomal polypeptide elongation stage) include tetracycline antibiotics such as oxytetracycline.

[0082] (c19-5) Group D6: Leucyl-tRNA synthase (LeuRNA) inhibitors (FRAC group code 54) Examples of leucyl-tRNA synthase (LeuRNA) inhibitors include benzoxanboroles such as tavaborole.

[0083] Group E Examples of Group E (signal transduction) include signal transduction (mechanism of action unknown) inhibitors, MAP / histidine kinase (os-2, HOG1) inhibitors in osmotic signal transduction, and MAP / histidine kinase (os-1, Daf1) inhibitors in osmotic signal transduction.

[0084] (c20) Group E1: Signal Transduction (Mechanism of Action Unknown) Inhibitors (FRAC Group Code 13) Examples of signal transduction (mechanism of action unknown) inhibitors include allyloxyquinolines such as quinoxyfen; quinazolinones such as proquinazid; and the like.

[0085] (c21) Group E2: MAP / histidine kinase (os-2, HOG1) inhibitors in osmotic signal transduction (FRAC group code 12) Examples of MAP / histidine kinase (os-2, HOG1) inhibitors in osmotic signal transduction include phenylpyrroles such as fenpiclonil and fludioxonil.

[0086] (c22) Group E3: MAP / histidine kinase (os-1, Daf1) inhibitors in osmotic signal transduction (FRAC group code 2) Examples of MAP / histidine kinase (os-1, Daf1) inhibitors in osmotic signal transduction include dicarboximides such as chlozolinate, dimethachlone, iprodione, procymidone, and vinclozolin.

[0087] Group F Group F (inhibitors of lipid biosynthesis or transport / cell membrane structure or function) include, for example, methyltransferase inhibitors of phospholipid biosynthesis, inhibitors of cellular lipid peroxidation, inhibitors of cell membrane permeable fatty acids, ergosterol binders, inhibitors of lipid homeostasis and transfer / storage, inhibitors of interactions with cell membrane lipid fractions, inhibitors of multiple actions on cell membranes, etc.

[0088] (c23) Group F2: phospholipid biosynthesis methyltransferase inhibitors (FRAC group code 6) Examples of phospholipid biosynthesis methyltransferase inhibitors include phosphorothiolates such as EDDP (edifenphos), IBP (iprobenfos), and pyrazophos; and dithiolanes such as isoprothiolane.

[0089] (c24) Group F3: Cellular lipid peroxidation inhibitors (FRAC group code 14) Examples of cellular lipid peroxidation inhibitors include aromatic hydrocarbons such as biphenyl, chloroneb, CNA (dicloran), PCNB (quintozene), tecnazen, and tolclofos-methyl; and 1,2,4-thiadiazoles such as eclomezole (etridiazole).

[0090] (c25) Group F4: Cell membrane-permeable fatty acid inhibitors (FRAC group code 28) Examples of the cell membrane-permeable fatty acid inhibitors include carbamates such as prothiocarb, iodocarb, propamocarb, and propamocarb.

[0091] (c26) Group F8: Ergosterol Binders (FRAC Group Code 48) Examples of ergosterol binders include amphoteric macrolide antifungal antibiotics such as natamycin (pimaricin) produced by actinomycetes Streptomyces natalensis or S. chattanoogensis.

[0092] (c27) Group F9: Inhibitors of lipid homeostasis and transfer / storage (FRAC group code 49) Examples of inhibitors of lipid homeostasis and transfer / storage include piperidinylthiazole isoxazolines such as oxathiapiprolin and fluoxapiprolin.

[0093] (c28) Group F10: Inhibitors of interaction with cell membrane lipid fractions and multiple actions on cell membranes (FRAC group code 51) Examples of inhibitors of interaction with cell membrane lipid fractions and multiple actions on cell membranes include polypeptides such as ASFBIOF01-02.

[0094] G Group G Group (cell membrane sterol biosynthesis inhibitors) include, for example, inhibitors of the C14 demethylase (erg11 / cyp51) in sterol biosynthesis, Δ １４ Reductase and Δ ８ →Δ ７ Examples of inhibitors include inhibitors of isomerase (erg24, erg2), inhibitors of 3-ketoreductase (erg27) in C4 demethylation in sterol biosynthesis, and inhibitors of squalene epoxidase (erg1) in the sterol biosynthesis system.

[0095] (c29) Group G1: Inhibitors of C14 demethylase (erg11 / cyp51) in sterol biosynthesis (FRAC group code 3) Examples of inhibitors of C14 demethylase in sterol biosynthesis include piperazines such as triforine; pyridines such as pyrifenox and pyrisoxazole; pyrimidines such as fenarimol and nuarimol; imidazoles such as imazalil, oxypoconazole, pefurazoate, prochloraz, and triflumizole; triazoles such as nbuconazole, fluquinconazole, flusilazole, flutriafol, hexaconazole, imibenconazole, ipconazole, mefentrifluconazole, metconazole, myclobutanil, penconazole, propiconazole, simeconazole, tebuconazole, tetraconazole, triadimefon, triadimenol, and triticonazole; and triazolinethiones such as prothioconazole.

[0096] (c30) Group G2: Δ in sterol biosynthesis １４ Reductase and Δ ８ →Δ ７ Inhibitors of isomerases (erg24, erg2) (FRAC group code 5) Δ in sterol biosynthesis １４ Reductase and Δ ８ →Δ ７ Examples of inhibitors of isomerases (erg24, erg2) include morpholines such as aldimorph, dodemorph, fenpropimorph, and tridemorph; piperidines such as fenpropidin and piperalin; and spiroketalamines such as spiroxamine.

[0097] (c31) Group G3: 3-ketoreductase (erg27) inhibitors in demethylation at the C4 position of sterol biosynthesis (FRAC group code 17) Examples of 3-ketoreductase (erg27) inhibitors in demethylation at the C4 position of sterol biosynthesis include hydroxyanilides such as fenhexamid; aminopyrazolinones such as fenpyrazamine; and the like.

[0098] (c32) Group G4: Inhibitors of squalene epoxidase (erg1) in sterol biosynthesis (FRAC group code 18) Examples of inhibitors of squalene epoxidase (erg1) in sterol biosynthesis include thiocarbamates such as pyributicarb; and allylamines such as naftifine and terbinafine.

[0099] Group H Examples of group H (cell wall biosynthesis inhibitors) include chitin synthase inhibitors and cellulose synthase inhibitors.

[0100] (c33) Group H4: Chitin synthase inhibitors (FRAC group code 19) Examples of chitin synthase inhibitors include peptidylpyrimidine nucleosides such as polyoxins, which are agricultural antibiotics. Polyoxins are antifungal antibiotics produced by the actinomycete Streptomyces cacaoi. There are 14 types of polyoxins, with the main components being A, B, and D.

[0101] (c34) Group H5: Cellulose synthase inhibitors (FRAC group code 40) Examples of cellulose synthase inhibitors include cinnamic acid amides such as dimethomorph, flumorph, pyrimorph, etc.; valinamide carbamates such as benthiavalicarb, iprovalicarb, valifenalate, etc.; mandelic acid amides such as mandipropamide, etc.

[0102] Group I Group I (cell wall melanin synthesis inhibitors) include, for example, reductase inhibitors of melanin biosynthesis, dehydratase inhibitors of melanin biosynthesis, and polyketide synthase inhibitors of melanin biosynthesis.

[0103] (c35) Group I1: Reductase inhibitors of melanin biosynthesis (FRAC group code 16.1) Examples of reductase inhibitors of melanin biosynthesis include isobenzofuranones such as fthalide; pyrroloquinolinones such as pyroquilon; triazolobenzothiazoles such as tricyclazole; and the like.

[0104] (c36) Group I2: Dehydratase inhibitors of melanin biosynthesis (FRAC group code 16.2) Examples of dehydratase inhibitors of melanin biosynthesis include cyclopropanecarboxamides such as carpropamid; carboxamides such as diclocymet; propionamides such as fenoxanil; and the like.

[0105] (c37) Group I3: Polyketide synthase inhibitors in melanin biosynthesis (FRAC group code 16.3) Examples of polyketide synthase inhibitors in melanin biosynthesis include trifluoroethylcarbamates such as tolprocarb.

[0106] Group P (c38) Host plant resistance inducers (excluding saccharin and its salts) Group P (host plant resistance inducers) include, for example, resistance inducers that stimulate the salicylic acid pathway, host plant resistance inducers, plant extracts that induce resistance in host plants, microorganisms and microbial preparations that induce resistance in host plants, etc. Note that saccharin and its salts are not included in the host plant resistance inducers.

[0107] Group P1: Plant resistance inducers that stimulate the salicylic acid pathway (FRAC group code P1) Plant resistance inducers that stimulate the salicylic acid pathway (salicylic acid signaling) include, for example, benzothiadiazoles (BTHs) such as acibenzolar-S-methyl.

[0108] Group P2: Host plant resistance inducers (FRAC group code P2) Examples of host plant resistance inducers (salicylic acid signaling) include benzisothiazoles such as probenazole. Group P3: Host plant resistance inducers (FRAC group code P3) Examples of host plant resistance inducers (salicylic acid signaling) include thiadiazolecarboxamides such as thiadinil and isothianiil.

[0109] Group P4: Resistance inducers in host plants (FRAC group code P4) Examples of resistance inducers in host plants (polysaccharide elicitors, natural products) include polysaccharides such as laminarin. Group P5: Plant extracts that induce resistance in host plants (FRAC group code P5) Examples of plant extracts (anthraquinone elicitors, plant extracts) that induce resistance in host plants include mixtures such as giant knotweed extract, ethanol extracts (anthraquinones, resveratrol), etc. Group P6: Microorganisms and microbial preparations that induce resistance in host plants (FRAC group code P6) Examples of microorganisms and microbial preparations (microbial elicitors, microorganisms) that induce resistance in host plants include bacteria from the genus Bacillus, such as Bacillus mycoides isolate J, and fungi from the genus Saccharomyces, such as the cell wall of Saccharomyces cerevisiae strain LAS117.

[0110] Group P7: Host plant resistance inducers (FRAC group code P7) Examples of host plant resistance inducers (phosphonates) include ethyl phosphonates such as fosetyl, phosphorous acid and salts, etc. Group P8: Host plant resistance inducers (FRAC group code P8) Examples of host plant resistance inducers (salicylic acid signaling) include isothiazolyl methyl ethers such as dichlobentiazox, etc.

[0111] (c39) Compounds with unknown mode of action (Group: Unknown mode of action) (U) (FRAC group codes 27, 34, 35, 36, 37, U6, U12, U13, U14, U16, U17, U18) Compounds with unknown mode of action (Group: Unknown mode of action) Examples of antibiotics with a specific action include cyanoacetamide oximes such as cymoxanil; phthalamic acids such as teclofthalam; benzotriazines such as triazoxide; benzenesulfonamides such as flusulfamide; pyridazinones such as diclomezine; phenylacetamides such as cyflufenamide; guanidines such as dodine; cyanomethylenethiazolidines such as fluthianil; pyrimidinone hydrazones such as ferimzone; 4-quinolylacetic acids such as tebufloquin; tetrazolyl oximes such as picarbutrazox; and glucopyranosyl antibiotics such as validamycin.

[0112] M Group (c40) Multisite Contact-Active Compounds (M) Examples of multisite contact-active compounds (M) include inorganic compounds (electrophiles), dithiocarbamate compounds and analogs (electrophiles), phthalimides (electrophiles), chloronitriles (phthalonitriles) (site of action unknown), bisguanidines (cell membrane disruptors, surfactants), triazines, quinones (anthraquinones) (electrophiles), quinoxalines (electrophiles), maleimides (electrophiles), sulfamides, thiocarbamates, etc. Preferred multisite contact-active compounds (M) are inorganic compounds (electrophiles), chloronitriles (phthalonitriles) (site of action unknown), and bisguanidines (cell membrane disruptors, surfactants).

[0113] Inorganic Compounds (Electrophiles) (FRAC Group Codes M1 and M2) Examples of inorganic compounds (electrophiles) include copper compounds and sulfur-based compounds. Examples of copper compounds include copper, DBEDC, basic copper chloride, basic copper sulfate, copper hydroxide, and copper nonylphenol sulfonate. Examples of sulfur-based compounds include sulfur and lime sulfur.

[0114] Dithiocarbamates and Analogues (Electrophiles) (FRAC Group Code M3) Examples of dithiocarbamates and analogues (electrophiles) include dithiocarbamates and analogues such as amobam, ferbam, mancozeb, maneb, metiram, propineb, thiuram, zinc thiazole, zineb, and ziram.

[0115] Phthalimides (Electrophiles) (FRAC Group Code M4) Examples of phthalimide compounds (electrophiles) include phthalimides such as captan, captafol, and folpet.

[0116] Chloronitriles (phthalonitriles) (site of action unknown) (FRAC group code M5) Examples of chloronitrile (phthalonitrile) compounds include chloronitriles (phthalonitriles) such as chlorothalonil (TPN).

[0117] Sulfamides (FRAC Group Code M6) Examples of sulfamides include sulfamine-based sulfamides (dichlofluanid), tolylfluanid, and the like.

[0118] Bisguanidines (cell membrane disruptors, surfactants) (FRAC group code M7) Examples of bisguanidines include guazatine, iminoctadine acetate, iminoctadine albesilate (iminoctadine), etc. Triazines (FRAC group code M8) Examples of triazines include anilazine, etc.

[0119] Quinones (anthraquinones) (electrophiles) (FRAC group code M9) Examples of quinones (anthraquinones) (electrophiles) include quinones (anthraquinones) such as dithianon.

[0120] Quinoxalines (electrophiles) (FRAC group code M10) Examples of quinoxalines (electrophiles) include quinoxalines such as quinoxaline-based (quinomethionate) compounds.

[0121] Maleimides (electrophiles) (FRAC group code M11) Examples of maleimides (electrophiles) include maleimides such as fluoroimide. Thiocarbamates (FRAC group code M12) Examples of thiocarbamates include thiocarbamates such as methasulfocarb.

[0122] BM Group (c41) Biological pesticides with multiple modes of action: plant extracts (BM) (FRAC group code BM1) Biological pesticides with multiple modes of action: plant extracts include polypeptides (lectins) such as extracts from cotyledons of lupin seedlings; phenols, sesquiterpenes, triterpenoids, coumarins, etc. such as extracts from Swinglea glutunosa; extracts of Melaleuca alternifolia (tea tree oil), vegetable oils (mixtures), terpene hydrocarbons such as eugenol, geraniol, thymol, terpene alcohols, and terpene phenols.

[0123] [Amendment under Rule 91 25.04.2025] (C) Preferred fungicidal compounds include (c1) RNA polymerase I inhibitors, (c2) DNA / RNA biosynthesis inhibitors, (c3) DNA topoisomerase type II (gyrase) inhibitors, (c4) dihydroorotate dehydrogenase inhibitors in de novo pyrimidine biosynthesis, (c5) tubulin polymerization inhibitors, (c6) cell division (site of action unknown) inhibitors, (c10) complex II (succinate dehydrogenase) inhibitors, (c11) complex III (ubiquinol oxidase Qo site) inhibitors, (c12) complex III (ubiquinone reductase Qi site) inhibitors, (c16) protein biosynthesis (ribosome translation initiation step) inhibitors, (c17) protein biosynthesis (ribosome (c20) inhibitors of phospholipid biosynthesis, methyltransferase, (c24) inhibitors of demethylase at C14 position in sterol biosynthesis, (c27) inhibitors of chitin biosynthesis enzyme, (c29) inhibitors of reductase in melanin biosynthesis, (c31) inhibitors of polyketamide synthase in melanin biosynthesis, (c32) resistance inducers in host plants (excluding saccharin or a salt thereof), (c33) compounds with an unknown mechanism of action, (c34) multisite contact active compounds, and (c35) at least one compound selected from the group consisting of quinofumelin.

[0124] Among these, preferred fungicidal compounds are polyoxin compounds, kasugamycin, validamycin, streptomycin, and oxytetracycline. Polyoxin compounds are antibiotics, and the polyoxin compounds are not particularly limited. The chemical structures of major polyoxin compounds are described, for example, in "THE MERCK INDEX TWELFTH EDITION," page 1306. Specific preferred polyoxin compounds include polyoxin, polyoxin salts, polyoxin complexes, and the like. Examples of polyoxins include polyoxin A, polyoxin B, polyoxin D, polyoxin E, polyoxin F, polyoxin G, polyoxin H, polyoxin J, polyoxin K, polyoxin L, polyoxin M, polyoxin N, and polyoxin O. The type of polyoxin salt is not particularly limited, and examples include metal salts such as zinc salts, iron salts, and titanium salts. Examples of polyoxin complexes include complex components mainly composed of polyoxin B. A single polyoxin compound may be used alone, or two or more may be selected and used in combination. Here, a compound containing two or more polyoxins is sometimes referred to as a polyoxin complex. Currently, in Japan, two active ingredients are known to be registered as pesticides: a polyoxin complex (a complex component mainly composed of polyoxin B) and polyoxin D zinc salt (a zinc salt mainly composed of polyoxin D). Preferred polyoxin compounds are the polyoxin complex and polyoxin D zinc salt.

[0125] In the present disclosure, (C) the fungicidal active compound is typically blended in an amount of 0.1 to 20,000 parts by mass, preferably 1 to 10,000 parts by mass, more preferably 5 to 5,000 parts by mass per 100 parts by mass of (A) saccharin and / or its salt.

[0126] The composition of the present disclosure may contain appropriate auxiliary components in addition to (A) saccharin and / or a salt thereof, (B) an insecticidal compound, and (C) a fungicidal compound. By adding, as the auxiliary component, an auxiliary agent such as a water-insoluble inorganic substance, e.g., talc, rosestone, or silica, it is possible to prevent the composition of the present disclosure from caking during production.

[0127] The composition of the present disclosure can also be mixed or used in combination with at least one optional component selected from the group consisting of other fungicides, insecticides, herbicides, plant growth regulators, microbial materials, mollusk control agents, and bird pest control agents, to the extent that the effects of the composition of the present disclosure are not impaired. The microbial materials are microorganisms that have a pest control effect (e.g., insecticidal activity, fungicidal activity, herbicidal activity, etc.) and / or a plant growth regulating effect such as rhizobia and mycorrhizal fungi.

[0128] The composition of the present disclosure may contain metaldehyde, a molluscicide, in addition to (A) saccharin and / or its salt, (B) an insecticidal compound, and (C) a fungicidal compound. Alternatively, the composition of the present disclosure and metaldehyde can be applied simultaneously or at different times during the cultivation period. In this case, harmful mollusks such as apple snails and lymnaea can be controlled. Other mollusk control agents include bis(tributyltin)oxide, allicin, bromoacetamide, cloethocarb, copper sulfate, fentin, ferric phosphate, methiocarb, niclosamide, pentachlorophenol, sodium pentachlorophenoxide, tazimcarb, thiacloprid, thiodicarb, tralopyril, trifenmorph, trimethacarb, cartap, and bensultap.

[0129] The composition of the present disclosure may contain anthraquinone, a bird repellent, in addition to (A) saccharin and / or its salt, (B) an insecticidal compound, and (C) a fungicidal compound. Alternatively, the composition of the present disclosure and anthraquinone can be applied simultaneously or at different times during the cultivation period. In this case, bird damage to cultivated plants other than paddy rice can be suppressed. Other bird pest control agents include chloralose, basic copper chloride (copperoxychloride), diazinon, guazatine, methiocarb, thiram, trimethacarb, ziram, zinc oxide, etc.

[0130] The composition of the present disclosure may contain a herbicide and / or a safener in addition to (A) saccharin and / or a salt thereof, (B) an insecticidally active compound, and (C) a fungicidal compound. Alternatively, the composition of the present disclosure and the herbicide and / or safener can be applied simultaneously or at different times during the cultivation period. In this case, weeds can be controlled in the cultivation of plants other than paddy rice. Examples of safeners include AD-67, BAS-145138, benoxacor, cloquintocet-mexyl, cyometrinil, 2,4-D, DKA-24, dichlormid, dymron, fenclorim, fenchlorazole-ethyl, flurazole, fluxofenim, furilazole, isoxadifen-ethyl, mefenpyr-diethyl, MG-191, naphthalic anhydride, oxabetrinil, PPG-1292, and R-29148.

[0131] Method for manufacturing agricultural and horticultural pest control compositions The composition of the present disclosure need only contain (A) saccharin and / or a salt thereof, (B) an insecticidal compound, and (C) a fungicidal compound without adding any other ingredients. However, it is usually preferable to mix a solid carrier, a liquid carrier, or a gaseous carrier (propellant), add a surfactant or other formulation adjuvants as needed, and formulate the composition into an oil solution, emulsion, wettable powder, flowable agent, granules, dust, aerosol, fog, or the like according to a conventional formulation method for use.

[0132] These formulations contain the active ingredients (A) saccharin and / or a salt thereof, (B) an insecticidal compound, and / or (C) a fungicidal compound in a total amount of usually 0.01 to 95% by weight, preferably 0.05 to 80% by weight, and more preferably 0.1 to 70% by weight.

[0133] Examples of solid carriers used in formulation include fine powders or granules of clays (kaolin clay, diatomaceous earth, synthetic hydrous silicon oxide, bentonite, fubasami clay, acid clay, etc.), talcs, ceramics, other inorganic minerals (celite, quartz, sulfur, activated carbon, calcium carbonate, hydrated silica, etc.), and chemical fertilizers (ammonium sulfate, ammonium phosphate, ammonium nitrate, urea, ammonium chloride, etc.).

[0134] Examples of liquid carriers include water, alcohols (methanol, ethanol, etc.), ketones (acetone, methyl ethyl ketone, etc.), aromatic hydrocarbons (benzene, toluene, xylene, ethylbenzene, methylnaphthalene, etc.), aliphatic hydrocarbons (hexane, cyclohexane, kerosene, diesel, etc.), esters (ethyl acetate, butyl acetate, etc.), nitriles (acetonitrile, isobutyronitrile, etc.), ethers (diisopropyl ether, dioxane, etc.), acid amides (N,N-dimethylformamide, N,N-dimethylacetamide, etc.), halogenated hydrocarbons (dichloromethane, trichloroethane, carbon tetrachloride, etc.), dimethyl sulfoxide, soybean oil, cottonseed oil, and other vegetable oils.

[0135] Examples of gaseous carriers include butane gas, LPG (liquefied petroleum gas), dimethyl ether, and carbon dioxide gas.

[0136] Examples of surfactants include alkyl sulfates, alkyl sulfonates, alkylaryl sulfonates, alkylaryl ethers and their polyoxyethylenated products, polyethylene glycol ethers, polyhydric alcohol esters, and sugar alcohol derivatives.

[0137] Examples of formulation adjuvants include adhesives, dispersants, stabilizers, and the like.

[0138] Examples of fixing agents or dispersing agents include casein, gelatin, polysaccharides (starch powder, gum arabic, cellulose derivatives, alginic acid, etc.), lignin derivatives, bentonite, sugars, and synthetic water-soluble polymers (polyvinyl alcohol, polyvinylpyrrolidone, polyacrylic acids, etc.). Examples of stabilizers include PAP (acid isopropyl phosphate), BHT (2,6-di-tert-butyl-4-methylphenol), BHA (a mixture of 2-tert-butyl-4-methoxyphenol and 3-tert-butyl-4-methoxyphenol), vegetable oil, mineral oil, fatty acid, or an ester thereof.

[0139] The composition of the present disclosure may be used as is or after diluting with water, etc. It may also be used with or without mixing with other insecticides, fungicides, herbicides, plant growth regulators, synergists, soil conditioners, animal feed, etc.

[0140] When the composition of the present disclosure contains two components, component (A) and component (B), or component (A) and component (C), the total amount thereof can be generally 0.01 to 95% by mass, preferably 0.05 to 80% by mass, and more preferably 0.1 to 50% by mass. When the composition of the present disclosure contains three components, component (A), component (B), and component (C), the total amount of components (A), (B), and (C) can be generally 0.01 to 95% by mass, preferably 0.05 to 80% by mass, and more preferably 0.1 to 70% by mass.

[0141] The application amount of the composition of the present disclosure is usually 1 a (100 m ２ The application concentration of the synergistic insecticide composition of the present disclosure, in the form of an emulsifiable concentrate, wettable powder, flowable formulation, liquid formulation, or the like, is usually 0.05 g to 600 g, preferably 0.1 to 200 g, and more preferably 0.5 to 100 g, per 1000 gram of water. When the synergistic insecticide composition of the present disclosure, in the form of an emulsifiable concentrate, wettable powder, flowable formulation, liquid formulation, or the like, is diluted with water and used, the application concentration is usually 0.1 to 300,000 ppm, preferably 1 to 30,000 ppm, and more preferably 10 to 8,000 ppm. In this case, the application concentration of the component (A) is usually 0.05 to 150,000 ppm, preferably 0.5 to 10,000 ppm, and more preferably 5 to 4,000 ppm. The application concentration of the component (B) is usually 0.05 to 150,000 ppm, preferably 0.5 to 10,000 ppm, and more preferably 5 to 4,000 ppm. The application concentration of the component (C) is usually 0.05 to 150,000 ppm, preferably 0.5 to 10,000 ppm, and more preferably 5 to 4,000 ppm. For example, in the case of normal spray application, the application concentration of the composition of the present disclosure is usually 0.1 to 10,000 ppm, preferably 1 to 5,000 ppm, and more preferably 10 to 1,000 ppm. In the case of drenching, the application concentration of the composition of the present disclosure is usually 1 to 300,000 ppm, preferably 10 to 30,000 ppm, and more preferably 100 to 8,000 ppm. Granules, dusts, and the like are applied as formulated without any dilution with water.

[0142] These application amounts and application concentrations vary depending on the type of formulation, application time, application location, application method, type of pest, degree of damage, and other conditions, and can be increased or decreased without being limited to the above ranges.

[0143] Examples of pests that can be controlled by the composition of the present disclosure include pests such as insects, mites, nematodes, and mollusks; and plant pathogens such as mold, bacteria, and viruses.

[0144] Specific examples of insects, mites, nematodes, mollusks, and the like that can be controlled by the composition of the present disclosure include the following.

[0145] Insects Hemiptera: Small brown planthopper (Laodelphax striatellus), Brown planthopper (Nilaparvata lugens), White-backed planthopper (Sogatella furcifera), Corn planthopper (Peregrinus maidis), Yellow leafhopper (Javesella pellucida), Black horned planthopper (Perkinsiella saccharicida), Tagosodes orizicolus and other Delphacidae; Green rice leafhopper (Nephotettix cincticeps), Taiwanese green rice leafhopper (Nephotettix virescens), Black-striped green rice leafhopper (Nephotettix nigropictus), Lightning leafhopper (Recilia dorsalis), Tea green leafhopper (Empoasca onukii), Potato leafhopper (Empoasca fabae), corn leafhopper (Dalbulus maidis), white leafhopper (Cofana spectra), etc., Cicadellidae; Cercopidae, such as Mahanarva posticata and Mahanarva fimbriolata;Black bean aphid (Aphis fabae), soybean aphid (Aphis glycines), cotton aphid (Aphis gossypii), European apple aphid (Aphis pomi), willow aphid (Aphis spiraecola), green peach aphid (Myzus persicae), strawberry aphid (Brachycaudus helichrysi), radish aphid (Brevicoryne brassicae), rosy apple aphid (Dysaphis plantaginea), false radish aphid (Lipaphis erysimi), tulip aphid (Macrosiphum euphorbiae), potato aphid (Aulacorthum solani), lettuce aphid (Nasonovia ribisnigri), wheat neck aphid (Rhopalosiphum padi), corn aphid (Rhopalosiphum maidis), citrus aphid (Toxoptera citricida), peach butterbur aphid (Hyalopterus pruni), barnyard millet aphid (Melanaphis sacchari), Japanese black aphid (Tetraneura nigriabdominalis), citrus cotton aphid (Ceratovacuna lanigera), apple aphid (Eriosoma lanigerum), etc.; phylloxeridae, such as grape aphid (Daktulosphaira vitifoliae), pecan phylloxera (Phylloxera devastatrix), pecan leaf phylloxera (Phylloxera notabilis), and southern pecan leaf phylloxera (Phylloxera russellae); Adelgidae, such as Adelges tsugae, Adelges piceae, and Aphrastasia pectinatae;Pentatomidae, such as the black rice bug (Scotinophara lurida), Malayan rice black bug (Scotinophara coarctata), green stink bug (Nezara antennata), thorny spotted bug (Eysarcoris aeneus), large thorny spotted bug (Eysarcoris lewisi), white spotted bug (Eysarcoris ventralis), purple spotted bug (Eysarcoris annamita), brown marmorated stink bug (Halyomorpha halys), southern green stink bug (Nezara viridula), brown stink bug (Euschistus heros), red banded stink bug (Piezodorus guildinii), Oebalus pugnax, and Dichelops melacanthus; Burrower brown Cydnidae, such as the narrow-leaved stink bug (Scaptocoris castanea); Alydidae, such as the narrow-leaved stink bug (Riptortus pedestris), the spider stink bug (Leptocorisa chinensis), and the narrow-leaved stink bug (Leptocorisa acuta); Coreidae, such as the narrow-leaved stink bug (Cletus punctiger) and the foot-striped stink bug (Leptoglossus australis); Caverelius saccharivorus, the rice-winged long-horn bug (Togo hemipterus), and the American long-horned stink bug (Blissus Lygaeidae, such as Trigonotylus caelestialium, Stenotus rubrovittatus, Stenodema calcarata, and Lygus lineolaris; Miridae, such as Trigonotylus caelestialium, Stenotus rubrovittatus, Stenodema calcarata, and Lygus lineolaris;Whiteflies (Aleyrodidae) such as the greenhouse whitefly (Trialeurodes vaporariorum), the tobacco whitefly (Bemisia tabaci), the citrus whitefly (Dialeurodes citri), the citrus spine whitefly (Aleurocanthus spiniferus), the tea spine whitefly (Aleurocanthus camelliae), and the Japanese oak cotton whitefly (Pealius euryae); the palm scale (Abgrallaspis cyanophylli), the red scale (Aonidiella aurantii), the pear scale (Diaspidiotus perniciosus), the white mulberry scale (Pseudaulacaspis pentagona), the Yanon scale (Unaspis yanonensis), and the false Yanon scale (Unaspis Diaspididae such as Ceroplastes rubens; Coccidae such as Ceroplastes rubens; Margarodidae such as Icerya purchasi and Icerya seychellarum; Phenacoccus solani, Phenacoccus solenopsis, Planococcus kraunhiae, Pseudococcus comstocki, Planococcus citri, Pseudococcus calceolariae, Pseudococcus longispinus), tuttlemea bug (Brevennia rehi), and other mealybugs (Pseudococcidae);Psyllidae family such as the citrus psyllid (Diaphorina citri), the citrus psyllid (Trioza erytreae), the pear psyllid (Cacopsylla pyrisuga), the Chinese pear psyllid (Cacopsylla chinensis), the potato psyllid (Bactericera cockerelli), and the pear psylla (Cacopsylla pyricola); Tingidae family such as the plane tree earworm (Corythucha ciliata), the goldenrod earworm (Corythucha marmorata), the pear earworm (Stephanitis nashi), and the azalea earworm (Stephanitis pyrioides); Cimicidae family such as the bedbug (Cimex lectularius), and the cicada family such as the giant cicada (Quesada gigas). ;

[0146] Lepidoptera: Rice stem borer (Chilo suppressalis), Darkheaded stem borer (Chilo polychrysus), White stem borer (Scirpophaga innotata), White stem borer (Scirpophaga incertulas), Rupela albina, Rice leaf borer (Cnaphalocrocis medinalis), Marasmia patnalis, Rice casino borer (Marasmia exigua), Cotton borer (Notarcha derogata), European corn borer (Ostrinia furnacalis), European corn borer (Ostrinia nubilalis), Hellula undalis, Black rice borer (Herpetogramma luctuosale), Grass moth (Pediasia teterrellus), Rice case worm (Nymphula depunctalis), Sugarcane Crambidae, such as the borer (Diatraea saccharalis); Pyralidae, such as the corn moth (Elasmopalpus lignosellus) and the Indian meal moth (Plodia interpunctella);Spodoptera litura, Spodoptera exigua, Mythimna separata, Mamestra brassicae, Sesamia inferens, Spodoptera mauritia, Naranga aenescens, Spodoptera frugiperda, Spodoptera exempta, Agrotis ipsilon, Autographa nigrisigna, Plusia festucae, Chrysodeixis includens, Trichoplusia spp., Heliothis virescens, and other Heliothis species Helicoverpa spp., such as the cotton bollworm (Helicoverpa armigera) and the American tobacco budworm (Helicoverpa zea), Noctuidae, such as the velvetbean caterpillar (Anticarsia gemmatalis), the cotton leafworm (Alabama argillacea), and the hop vine borer (Hydraecia immanis); Pieridae, such as the cabbage white butterfly (Pieris rapae);Tortricidae such as the pear fruit moth (Grapholita molesta), the plum fruit moth (Grapholita dimorpha), the bean fruit moth (Leguminivora glycinivorella), the adzuki bean pea moth (Matsumuraeses azukivora), the apple tortrix moth (Adoxophyes orana fasciata), the tea tortrix moth (Adoxophyes honmai), the tea tortrix moth (Homona magnanima), the green tea tortrix moth (Archips fuscocupreanus), the codling moth (Cydia pomonella), the citrus fruit borer (Tetramoera schistaceana), the bean shoot borer (Epinotia aporema), and the citrus fruit borer (Ecdytolopha aurantiana); Gracilariae (Gracillariidae) such as Carposina ringoniella; Carposinidae (Carposinidae) such as Carposina sasakii; Lyonetiidae (Lyonetiidae) such as Coffee Leaf miner (Leucoptera coffeella), Peach leafminer (Lyonetia clerkella), and Silver leafminer (Lyonetia prunifoliella); Lymantriidae (Lymantria spp.) such as Lymantria dispar (Lymantria dispar), Euproctis spp. such as Euproctis pseudoconspersa (Euproctis pseudoconspersa); Plutellidae (Plutellidae) such as Plutella xylostella (Plutella xylostella);Gelechiidae, such as the peach leaf moth (Anarsia lineatella), the potato leaf moth (Helcystogramma triannulella), the red cotton moth (Pectinophora gossypiella), the potato tuber moth (Pthorimaea operculella), and Tuta absoluta; Arctiidae, such as the American fall webworm (Hyphantria cunea); Castniidae, such as the giant sugarcane borer (Telchin licus); Cossidae, such as the small sugarcane moth (Cossus insularis); Geometridae, such as the arthropod geometridae (Ascotis selenaria); Parasa Limacodidae such as Stathmopoda lepida; Stathmopodidae such as Stathmopoda masinissa; Sphingidae such as Acherontia lachesis; Sesiidae such as Nokona feralis; Hesperiidae such as Parnara guttata.

[0147] Thysanoptera: Thripidae such as western flower thrips (Frankliniella occidentalis), southern green thrips (Thrips palmi), green tea thrips (Scirtothrips dorsalis), onion thrips (Thrips tabaci), plain leaf thrips (Frankliniella intonsa), rice thrips (Stenchaetothrips biformis), and white-streaked thrips (Echinothrips americanus); Phlaeothripidae such as rice thrips (Haplothrips aculeatus).

[0148] Diptera: Anthomyiidae such as Delia platura, Delia antiqua, and Pegomya cunicularia; Ulidiidae such as Tetanops myopaeformis; Agromyzidae such as Agromyza oryzae, Liriomyza sativae, Liriomyza trifolii, and Chromatomyia horticola; Chloropidae such as Chlorops oryzae; Bactrocera cucurbitae, Bactrocera citri dorsalis), Bactrocera latifrons, Bactrocera oleae, Bactrocera tryoni, Ceratitis capitata, Rhagoletis pomonella, Rhacochlaena japonica, and other Tephritidae; Hydrellia griseola, Hydrellia philippina, Hydrellia sasakii, and other Ephydridae; Drosophilidae, Drosophila suzukii, and other Drosophila suzukii; Megaselia Phoridae, such as the Japanese bush fly (Clogmia spiracularis); Psychodidae, such as the Japanese bush fly (Clogmia albipunctata); Sciaridae, such as the Japanese bush fly (Bradysia difformis);Cecidomyiidae, such as the Hessian fly (Mayetioladestructor) and the rice rot gall midge (Orseolia oryzae); Diopsidae, such as Diopsis macrophthalma; Tipulidae, such as the Japanese crane fly (Tipula aino), the common crane fly (Tipula oleracea), and the European crane fly (Tipula paludosa); Culex pipiens pallens, Aedes aegypti, Aedes albopicutus, Anopheles hyracanus sinesis, Culex quinquefasciatus, and Culex pipiens molestus Culicidae such as Prosimulium yezoensis and Simulium ornatum, Tabanidae such as Tabanus trigonus, Musca domestica, Muscina stabulans, Muscidae, etc.;

[0149] Coleoptera: Western corn rootworm (Diabrotica virgifera virgifera), Southern corn rootworm (Diabrotica undecimpunctata howardi), Northern corn rootworm (Diabrotica barberi), Mexican corn rootworm (Diabroticavirgifera zeae), Banded cucumber beetle (Diabrotica balteata), Cucurbit beetle (Diabrotica speciosa), Bean leaf beetle (Cerotoma trifurcata), Red-necked leaf beetle (Oulema melanopus), Cucurbit leaf beetle (Aulacophora femoralis), Striped flea beetle (Phyllotreta striolata), Cabbage flea beetle (Phyllotreta cruciferae), Western black flea beetle (Phyllotreta pusilla), Cabbage stem flea beetle (Psylliodes Chrysomelidae, such as the hop flea beetle (Psylliodes punctulata), Colorado potato beetle (Leptinotarsa ​​decemlineata), rice leaf beetle (Oulema oryzae), grape colaspis (Colaspis brunnea), corn flare beetle (Chaetocnema pulicaria), sweet potato stag beetle (Chaetocnema confinis), potato flare beetle (Epitrix cucumeris), rice spur beetle (Dicladispa armigera), southern corn leaf beetle (Myochrous denticollis), four-legged tortoise beetle (Laccoptera quadrimaculata), and tobacco flea beetle (Epitrix hirtipennis);Carabidae, such as the seedcorn beetle (Stenolophus lecontei) and the slender seedcorn beetle (Clivina impressifrons); Scarabaeidae, such as the cuprea beetle (Anomala cuprea), the dwarf beetle (Anomala rufocuprea), the green beetle (Anomala albopilosa), the Japanese beetle (Popillia japonica), the long-legged beetle (Heptophylla picea), the European chafer (Rhizotrogus majalis), the black-legged beetle (Tomarus gibbosus), the genus Holotrichia (Holotrichia spp.), and the June beetle (Phyllophaga crinita); Scarabaeidae, such as the genus Diloboderus (Diloboderus spp.), and the like;Boll weevil (Araecerus coffeae), sweet potato weevil (Cylas formicarius), potato weevil (Euscepes postfasciatus), alfalfa weevil (Hypera postica), maize weevil (Sitophilus zeamais), rice weevil (Echinocnemus squameus), rice water weevil (Lissorhoptrus oryzophilus), white-spotted weevil (Rhabdoscelus lineatocollis), boll weevil (Anthonomus grandis), grass banded weevil (Sphenophorus venatus), Southern corn billbug (Sphenophorus callosus), soybean stalk weevil (Sternechus subsignatus), sugarcane weevil (Sphenophorus levis), rust gourd weevil (Scepticus griseus), brown gourd weevil (Scepticus uniformis), Brazilian bean weevil (Zabrotes subfasciatus), pine bark beetle (Tomicus piniperda), coffee berry borer (Hypothenemushampei), Aracanthus spp. such as Aracanthus mourei, cotton root borer (Eutinobothrus brasiliensis), etc. Curculionidae; Tenebrionidae; Tribolium castaneum; Tribolium confusum; Coccinellidae; Lyctus Bostrychidae, such as Bostrychidae brunneus; Ptinidae;Cerambycidae, such as the spotted longhorn beetle (Anoplophora malasiaca) and Migdolus fryanus; Elateridae, such as the Okinawan wireworm beetle (Melanotus okinawensis), the brown-headed wireworm beetle (Agriotes fuscicollis), the comb beetle (Melanotus legatus), the Anchastus spp., the Conoderus spp., the Ctenicera spp., the Limonius spp., and the Aeolus spp.; Staphylinidae, such as the blue-leaf rove beetle (Paederus fuscipes).

[0150] Orthoptera: Migratory locust (Locusta migratoria), Moroccan locust (Dociostaurus maroccanus), Australian locust (Chortoicetes terminifera), Red locust (Nomadacris septemfasciata), Brown locust (Locustana pardalina), Tree locust (Anacridium melanorhodon), Italian locust (Calliptamus italicus), Differential grasshopper (Melanoplus differentialis), Two-striped grasshopper (Melanoplus bivittatus), Migratory grasshopper (Melanoplus sanguinipes), Red-legged grasshopper (Melanoplus femurrubrum), Clearwinged grasshopper (Camnula pellucida), Desert locust (Schistocerca gregaria), Yellow-winged locust (Gastrimargus The grasshoppers (Acrididae) include the Japanese grasshopper (Oxya musicus), the spur-throated locust (Austracris guttulosa), the oriental grasshopper (Oxya yezoensis), the long-winged grasshopper (Oxya japonica), and the Taiwan ground locust (Patanga succincta); the grasshoppers (Gryllotalpidae) include the European house cricket (Acheta domestica) and the field cricket (Teleogryllus emma); and the grasshoppers (Tettigoniidae) include the Mormon cricket (Anabrus simplex).

[0151] Hymenoptera: Tenthredinidae such as Athalia rosae and Athalia japonica; Formicidae such as Solenopsis spp. and Brown leaf-cutting ant Atta capiguara.

[0152] Order Blattodea: Family Blattellidae such as the German cockroach (Blattella germanica); Family Blattidae such as the American cockroach (Periplaneta fuliginosa), the American cockroach (Periplaneta americana), the brown cockroach (Periplaneta brunnea), and the Asian cockroach (Blatta orientalis); Family Reticulitermes speratus, Formosan termite (Coptotermes formosanus), American dry wood termite (Incisitermes minor), Formosan termite (Cryptotermes domesticus), Formosan termite (Odontotermes formosanus), Japanese termite (Neotermes koshunensis), Satsuma termite (Glyptotermes satsumensis), and Nakajima termite (Glyptotermes Termites of the termite family (Termitidae), such as the Japanese termite (Glyptotermes fuscus), the Japanese formosan termite (Hodotermopsis sjostedti), the Formosan termite (Coptotermes guangzhouensis), the Amami termite (Reticulitermes amamianus), the Miyatake termite (Reticulitermes miyatakei), the Formosan termite (Reticulitermes kanmonensis), the Takasago termite (Nasutitermes takasagoensis), the Sinocapritermes nitobei, the Musha termite (Sinocapritermes mushae), and the Cornitermes cumulans.

[0153] Mites (Acari): Tetranychidae, such as Tetranychus urticae, Tetranychus kanzawai, Tetranychus evansi, Panonychus citri, Panonychus ulmi, and Oligonychus spp.; Aculops pelekassi, Phyllocoptruta citri, Aculops lycopersici, Calacarus carinatus, Acaphylla theavagrans, Eriophyes chibaensis, Aculus schlechtendali, and Aceria diospyri), Aceria tosichella, Shevtchenkella sp. and other Eriophyidae mites; Tarsonemidae mites such as Polyphagotarsonemuslatus; Tenuipalpidae mites such as Brevipalpus phoenicis; Tuckerellidae mites; Haemaphysalis longicornis, Haemaphysalis flava, Dermacentor taiwanensis, Dermacentor variabilis, Ixodes ovatus, Ixodes persulcatus, Ixodes scapularis, Amblyomma Ixodidae, such as Rhipicephalus americanum, Boophilus microplus, and Rhipicephalus sanguineus;Acaridae, such as Tyrophagus putrescentiae and Tyrophagus similis; Pyroglyphidae, such as Dermatophagoides farinae and Dermatophagoides pteronyssinus; Cheyletidae, such as Cheyletus eruditus, Cheyletus malaccensis, Cheyletus moorei, and Cheyletiella yasguri; Sarcoptidae, such as Otodectes cynotis and Sarcoptes scabiei; Demodex Demodicidae such as Ornithonyssus canis; Listrophoridae; Haplochthoniidae; Macronyssidae such as Ornithonyssus bacoti and Ornithonyssus sylviarum; Dermanyssidae such as Dermanyssus gallinae; Trombiculidae such as Leptotrombidium akamushi;

[0154] Nematodes Nematodes (Nematoda): Aphelenchoididae such as the rice root-lesion nematode (Aphelenchoides besseyi); Pratylenchidae such as the southern root-lesion nematode (Pratylenchus coffeae), Pratylenchus brachyurus, the wheat root-lesion nematode (Pratylenchus neglectus), and Radopholus similis; Java root-knot nematode (Meloidogyne javanica), sweet potato root-knot nematode (Meloidogyne incognita), northern root-knot nematode (Meloidogyne hapla), soybean cyst nematode (Heterodera glycines), potato cyst nematode (Globodera rostochiensis), potato white cyst nematode (Globodera Heteroderidae such as Rotylenchulus reniformis; Hoplolaimidae such as Rotylenchulus reniformis; Anguinidae such as Nothotylenchus acris and Ditylenchus dipsaci; Tylenchulidae such as Tylenchulus semipenetrans; Longidoridae such as Xiphinema index; Trichodoridae; Parasitaphelenchidae such as Bursaphelenchus xylophilus.

[0155] Mollusk Gastropoda: Limacidae family such as Limax marginatus and Limax flavus; Philomycidae family such as Meghimatium bilineatum; Ampullariidae family such as Pomacea canaliculata; Lymnaeidae family such as Austropeplea ollula; etc.

[0156] Specific examples of plant diseases caused by plant pathogenic fungi that can be controlled by the composition of the present disclosure include the following. The scientific names of the plant pathogenic fungi that cause each disease are shown in parentheses. Plant diseases (plant pathogens) Wheat diseases: powdery mildew (Erysiphe graminis), head blight (Fusarium graminearum, F. avenacerum, F. culmorum, Microdochium nivale), rust (Puccinia striiformis, P. graminis, P. recondita), pink snow blight (Micronectriella nivale), snow blight sclerotinia (Typhula sp.), naked smut (Ustilago tritici), cattail smut (Tilletia caries), eyespot (Pseudocercosporella herpotrichoides), leaf blight (Mycosphaerella graminicola), leaf spot blight (Stagonospora nodorum), yellow spot (Pyrenophora tritici-repentis), etc. Barley diseases: powdery mildew (Erysiphe graminis), head blight (Fusarium graminearum, F. avenacerum, F. culmorum, Microdochium nivale), rust (Puccinia striiformis, P. graminis, P. hordei), naked smut (Ustilago nuda), scald (Ustilago nuda), net blotch (Pyrenophora teres), leaf spot (Cochliobolus sativus), leaf spot (Pyrenophora graminea), seedling damping-off caused by Rhizoctonia genus fungi (Rhizoctonia solani), etc. Corn diseases: ear smut (Ustilago maydis), whole leaf blight (Cochliobolus heterostrophus), hail blotch (Gloeocercospora sorghi), southern rust (Puccinia polysora), gray leaf spot (Cercospora zeae-maydis), seedling damping-off caused by Rhizoctonia solani, etc.

[0157] Citrus diseases: black spot (Diaporthe citri), common scab (Elsinoe fawcetti), fruit rot (Penicillium digitatum, P. italicum), phytophthora (Phytophthora parasitica, Phytophthora citrophthora), etc. Apple diseases: monilinia (Monilinia mali), canker (Valsa ceratosperma), powdery mildew (Podosphaera leucotricha), leaf spot (Podosphaera leucotricha), black spot (Venturia inaequalis), anthracnose (Colletotrichum acutatum), late blight (Phytophtora cactorum), etc. Pear diseases: black spot (Venturia nashicola, V. pirina), black spot (Alternaria alternata Japanese pear pathotype), red spot (Gymnosporangium haraeanum), late blight (Phytophtora cactorum), etc. Peach diseases: brown spot (Monilinia fructicola), black spot (Cladosporium carpophilum), Phomopsis rot (Phomopsis sp.), etc. Grape diseases: black rot (Elsinoe ampelina), late rot (Glomerella cingulata), powdery mildew (Uncinula necator), rust (Phakopsora ampelopsidis), black rot (Guignardia bidwellii), downy mildew (Plasmopara viticola), etc. Persimmon diseases: Anthracnose (Gloeosporium kaki), leaf spot (Cercospora kaki, Mycosphaerella nawae), etc.Cucurbit diseases: Anthracnose (Colletotrichum lagenarium), powdery mildew (Sphaerotheca fuliginea), vine blight (Mycosphaerella melonis), vine wilt (Fusarium oxysporum), downy mildew (Pseudoperonospora cubensis), late blight (Phytophthora sp.), seedling damping-off (Pythium sp.), etc. Tomato diseases: Ring spot (Alternaria solani), leaf mold (Cladosporium fulvum), late blight (Phytophthora infestans). Eggplant diseases: Brown spot (Phomopsis vexans), powdery mildew (Erysiphe cichoracearum), etc. Diseases of cruciferous vegetables: black spot (Alternaria japonica), white spot (Cercosporella brassicae), clubroot (Plasmodiophora brassicae), downy mildew (Peronospora parasitica), bacterial black spot (Pseudomonas syringae pv. maculicola and Pseudomonas cannabina pv. alisalensis), soft rot (Pectobacterium carotovora subsp. carotovora), etc. Diseases of leeks: rust (Puccinia allii), downy mildew (Peronospora destructor), soft rot (Pectobacterium carotovora subsp. carotovora), etc.

[0158] Soybean diseases: purple spot (Cercospora kikuchii), black rot (Elsinoe glycines), black spot (Diaporthe phaseolorum var. sojae), brown spot (Septoria glycines), leaf spot (Cercospora sojina), rust (Phakopsora pachyrhizi), stem rot (Phytophthora sojae), seedling damping-off caused by Rhizoctonia solani, brown ring spot (Corynespora cassiicola), sclerotinia sclerotiorum, etc.; kidney bean diseases: anthracnose (Colletotrichum lindemuthianum), etc.; peanut diseases: black spot (Cercospora personata), brown spot (Cercospora arachidicola), southern blight (Sclerotium rolfsii), etc. Pea diseases: powdery mildew (Erysiphe pisi), etc. Potato diseases: summer blight (Alternaria solani), late blight (Phytophthora infestans), scarlet rot (Phytophthora erythroseptica), powdery scab (Spongospora subterranean f.sp. subterranea), etc. Strawberry diseases: powdery mildew (Sphaerotheca humuli), anthracnose (Glomerella cingulata), etc. Tea diseases: net blight (Exobasidium reticulatum), white spot (Elsinoe leucospila), ring spot (Pestalotiopsis sp.), anthracnose (Colletotrichum theae-sinensis), etc. Tobacco diseases: red star (Alternaria longipes), powdery mildew (Erysiphe cichoracearum), anthracnose (Colletotrichum tabacum), downy mildew (Peronospora tabacina), late blight (Phytophthora nicotianae), etc.Rapeseed diseases: Sclerotinia sclerotiorum, seedling damping-off caused by Rhizoctonia solani, etc. Cotton diseases: Seedling damping-off caused by Rhizoctonia solani, white mold (Mycosphaerella areola), black root rot caused by Thielaviopsis basicola, etc. Coffee diseases: Rust (Hemileia vastatrix), etc. Sugarcane diseases: Rust (Puccinia melanocephela, Puccinia kuehnii), smut (Ustilago scitaminea), etc. Sunflower diseases: Rust (Puccinia helianthi), etc. Sugar beet diseases: brown spot (Cercospora beticola), leaf rot (Thanatephorus cucumeris), root rot (Thanatephorus cucumeris), black root rot (Aphanomyces cochlioides), etc. Rose diseases: black scab (Diplocarpon rosae), powdery mildew (Sphaerotheca pannosa), downy mildew (Peronospora sparsa), etc. Chrysanthemum and Asteraceae vegetable diseases: downy mildew (Bremia lactucae), brown spot (Septoria chrysanthemi-indici), white rust (Puccinia horiana), etc. Diseases of various plants: diseases caused by Pythium fungi (Pythium aphanidermatum, P. debarianum, P. graminicola, P. irregulare, P. ultimum), gray mold (Botrytis cinerea), sclerotinia sclerotiorum, etc. Diseases of radish: black spot (Alternaria brassicicola), etc. Diseases of turfgrass: dollar spot (Sclerotinia homoeocarpa), brown patch, and large patch (Rhizoctonia solani), etc.Banana diseases: Sigatoka disease (Mycosphaerella fijiensis, Mycosphaerella musicola), etc. Sunflower diseases: downy mildew (Plasmopara halstedii), etc. Seed diseases or diseases in the early stages of growth of various plants caused by fungi of the genera Aspergillus, Penicillium, Fusarium, Gibberella, Tricoderma, Thielaviopsis, Rhizopus, Mucor, Corticium, Phoma, Rhizoctonia, and Diplodia, etc.

[0159] Furthermore, the composition of the present disclosure can control harmful insects belonging to the order Hemiptera, and thereby protect crops from viral diseases transmitted by these insects, such as Tomato yellow leaf curl virus, Cucumber mosaic virus and Turnip mosaic virus, Beet western yellows virus, and Cauliflower mosaic virus.

[0160] Application Methods of the composition of the present disclosure include, for example, planting hole treatment at planting time and base treatment for granules, and immersion treatment, pre-planting irrigation treatment, base irrigation treatment, soil irrigation treatment, foliar spray, aerial spray, etc. for liquid formulations. The composition of the present disclosure prepared in this manner can be applied simultaneously or in divided doses to useful plants or to the area where useful plants are intended to grow or are growing, thereby controlling the growth of undesirable plants relative to useful plants. Note that the above-mentioned useful plants include field crops, horticultural crops, turf, fruit trees, non-agricultural land, etc.

[0161] The application amount and application concentration of the composition of the present disclosure can vary over a wide range depending on weather conditions, application time, application location, application method, etc., but the application amount of components (A) to (C) contained in the composition of the present disclosure is usually about 0.05 to 600 g / a in total, preferably 0.1 to 200 g / a, and more preferably 0.5 to 100 g / a.

[0162] The present disclosure will be explained in more detail below using examples, but the technical scope of the present disclosure is not limited to these examples.

[0163] Formulation examples are shown below. Note that "parts" means "parts by mass." However, the formulations are not limited to those shown and can be varied widely.

[0164] Formulation Example 1 (Emulsion) 10 parts of each of the compositions of the present disclosure were dissolved in 45 parts of Solvesso 150 and 35 parts of N-methylpyrrolidone, and 10 parts of an emulsifier (trade name: Sorpol 3005X, manufactured by Toho Chemical Industry Co., Ltd.) were added thereto, followed by stirring and mixing to obtain 10% emulsions of each composition.

[0165] Formulation Example 2 (wettable powder) 20 parts of each of the compositions of the present disclosure were added to a mixture of 2 parts of sodium lauryl sulfate, 4 parts of sodium lignin sulfonate, 20 parts of synthetic hydrous silicon oxide fine powder, and 54 parts of clay, and the mixture was stirred and mixed in a juice mixer to obtain a 20% wettable powder.

[0166] Formulation Example 3 (Granules) 2 parts of sodium dodecylbenzenesulfonate, 10 parts of bentonite, and 83 parts of clay were added to 5 parts of each composition of the present disclosure and thoroughly mixed. The required amount of water was added, and the mixture was further stirred. The mixture was granulated in a granulator and air-dried to obtain 5% granules.

[0167] Formulation Example 4 (Dust) One part of each of the compositions of the present disclosure is dissolved in an appropriate amount of acetone, and to this is added 5 parts of synthetic hydrous silicon oxide fine powder, 0.3 parts of acid isopropyl phosphate (PAP), and 93.7 parts of clay. The mixture is stirred and mixed in a juice mixer, and the acetone is evaporated off to obtain a 1% dust.

[0168] Formulation Example 5 (Flowable Preparation) 20 parts of each of the compositions of the present disclosure, 3 parts of polyoxyethylene tristyrylphenyl ether phosphate ester triethanolamine, and 20 parts of water containing 0.2 parts of Rhodorsil 426R are mixed, the mixture is wet-pulverized using a Dynomill, and then mixed with 60 parts of water containing 8 parts of propylene glycol and 0.32 parts of xanthan gum to obtain a 20% suspension in water.

[0169] Formulation Example 6 (Liquid) 10 parts of each of the compositions of the present disclosure, 5 parts of polyoxyethylene sorbitan monostearate, 5 parts of propylene glycol and 70 parts of water are mixed with stirring to obtain a 10% solution of each.

[0170] The effectiveness of certain particularly preferred combinations of compositions has been confirmed through biological testing.

[0171] Biological Test Example 1: Preventive Effect A chemical solution containing the compounds (A) and (C) shown in Table 1 (Kumiten (registered trademark) added at a 5,000-fold dilution) was sprayed onto Chinese cabbage seedlings grown in 6.5 cm polypots, and the plants were air-dried. Approximately 24 hours after spraying, a suspension of Bacillus oryzae (containing 500 ppm Tween-20 aq.) was sprayed and inoculated, and the plants were kept in a moist chamber set at 25°C. After 6 days, the number of lesions was counted, and the control titer was calculated using the following formula. This test was carried out in one row with 5 plants per plot. Control titer = (1 - (average number of lesions in treated plots / average number of lesions in untreated plots)) x 100 The results are shown in Table 1.

[0172]

[0173] To show the degree of synergistic effect, the "expected control value" was calculated using the following formula based on the Colby method. When the control value is greater than each "expected control value," it is determined that a synergistic effect exists. Expected value = X + Y - XY / 100 X: Control value in the area where A is used alone Y: Control value in the area where C is used alone

[0174] Results As a result, the plant pest control composition containing compound (A) and compound (C) showed a synergistic effect against bacterial black spot of Chinese cabbage when applied to the target.

[0175] Biological Test Example 2: Curative Effect Chinese cabbage seedlings grown in 6.5 cm polypots were inoculated by spraying with a suspension of Bacillus oryzae (containing 500 ppm Tween-20 aq.) and then kept in a moist chamber set at 25°C for 1 day. Approximately 24 hours after inoculation, a chemical solution containing compounds (A) and (C) shown in Table 2 (containing Kumiten (registered trademark) at a 5,000-fold dilution) was sprayed on the plants, and the plants were returned to the moist chamber. After 6 days, the number of lesions was counted and the control titer was calculated using the following formula. This test was carried out in one row with 5 plants per group. Control titer = (1 - (average number of lesions in treated groups / average number of lesions in untreated groups)) x 100 The results are shown in Table 2.

[0176]

[0177] Results As a result, the plant pest control composition containing compound (A) and compound (C) showed a synergistic effect against bacterial black spot of Chinese cabbage when applied to the target.

[0178] Biological Test Example 3: Preventive Effect A chemical solution (containing 3,300 times the concentration of Kumiten (registered trademark)) containing the compounds (A) and (C) shown in Table 3 was sprayed onto cabbage seedlings grown in 6.5 cm polypots. Approximately 24 hours after spraying, flora disks were prepared from plate media on which vegetable sclerotium fungi had been previously cultured, and placed on leaves for inoculation, which was then maintained in a moist chamber set at 20°C. After 3 days, the lesion diameter was measured, and the control titer was calculated using the following formula. This test was carried out in one series of 5 plants per plot. Control titer = (1 - (lesion spot diameter in treated plot / lesion spot diameter in untreated plot)) x 100 The results are shown in Table 3.

[0179]

[0180] Results As a result, the plant pest control composition containing compound (A) and compound (C) showed a synergistic effect against cabbage stem rot when applied to a target. This application claims priority to Japanese Patent Application No. 2023-185781, filed October 30, 2023. Japanese Patent Application No. 2023-185781 is incorporated herein by reference.

Claims

1. An agricultural and horticultural pest control composition (excluding the pest control composition for paddy rice) containing (A) saccharin and / or its salt and at least one plant treatment composition selected from the group consisting of (B) an insecticidal active compound and (C) a bactericidal active compound.

2. The agricultural and horticultural pest control composition according to claim 1 (excluding the pest control composition for paddy rice), wherein the agricultural and horticultural pest control composition contains the (A) saccharin and / or its salt and the (C) bactericidal active compound.

3. The agricultural and horticultural pest control composition according to claim 2 (excluding the pest control composition for paddy rice), wherein the (C) bactericidal active compound is an antibiotic for agricultural pesticides.

4. The agricultural and horticultural pest control composition according to claim 3 (excluding the pest control composition for paddy rice), wherein the antibiotic for agricultural pesticides contains at least one antibiotic selected from the group consisting of a chitin synthase inhibitor, an enopyranuronic acid antibiotic, a hexopyranosyl antibiotic, a glucopyranosyl antibiotic, a tetracycline antibiotic, and an amphiphilic macrolide antifungal antibiotic.

5. The agricultural and horticultural pest control composition according to claim 4 (excluding the pest control composition for paddy rice), wherein the antibiotic for agricultural pesticides is at least one compound or its salt selected from the group consisting of polyoxin, kasugamycin, validamycin, streptomycin, and oxytetracycline.

6. The agricultural and horticultural pest control composition according to claim 5 (excluding the pest control composition for paddy rice), wherein the antibiotic for agricultural pesticides is polyoxin or its salt.

7. [Correction based on Rule 91, 25.04.2025] The said (B) insecticidal active compound is (b1) an acetylcholinesterase (AChE) inhibitor, (b2) a GABAergic chloride ion channel blocker, (b3) a sodium channel modulator, (b4) a nicotinic acetylcholine receptor (nAChR) competitive modulator, (b5) a nicotinic acetylcholine receptor (nAChR) allosteric modulator - Site I, (b6) a glutamate-gated chloride ion channel (GluCl) allosteric modulator, (b7) a juvenile hormone analogue, (b8) other non-specific (multi-site) inhibitors, (b9) a chordotonal organ TRPV channel modulator, (b10) a mite growth inhibitor acting on CHS1, (b11) a microbial-derived insect midgut intima disruptor, (b12) a mitochondrial ATP synthase inhibitor, (b13) an oxidative phosphorylation uncoupler that disturbs the proton gradient, (b14) a nicotinic acetylcholine receptor (nAChR) channel blocker, (b15) a chitin biosynthesis inhibitor acting on CHS1, (b16) a chitin biosynthesis inhibitor (Type 1), (b17) a molting inhibitor (for Diptera insects), (b18) a molting hormone (ecdysone) receptor agonist, (b19) an octopamine receptor agonist, (b20) a mitochondrial electron transport system complex III inhibitor - Qo site, (b21) a mitochondrial electron transport system complex I inhibitor (METI), (b22) a voltage-dependent sodium channel blocker, (b23) an acetyl-CoA carboxylase inhibitor, (b24) a mitochondrial electron transport system complex IV inhibitor, (b25) a mitochondrial electron transport system complex II inhibitor, (b26) a ryanodine receptor modulator, (b27) a chordotonal organ nicotinamidase inhibitor, (b28) a GABAergic chloride ion channel allosteric modulator, (b29) a baculovirus, (b30) a nicotinic acetylcholine receptor (nAChR) allosteric modulator - Site II, (b31) a calcium-activated potassium channel (KCa2) modulator, (b32) a mitochondrial electron transport system complex III inhibitor - Qi site, (b33) a target suppressor via RNA interference, (b34) a chordotonal organ modulator (target site unspecified),and at least one compound selected from the group consisting of agent A with unknown or uncertain mechanism of action, bacterial agent with unknown or uncertain mechanism of action (excluding BT agent), composition, extract or unrefined oil of plant origin with unknown or uncertain mechanism of action, fungal agent with unknown or uncertain mechanism of action, and physical disturbance with unknown or uncertain mechanism of action, wherein the (C) bactericidal active compound is (c1) an RNA polymerase I inhibitor, (c2) a DNA / RNA biosynthesis inhibitor, (c3) a DNA topoisomerase type II (gyrase) inhibitor, (c4) a dihydroorotate dehydrogenase inhibitor in de novo pyrimidine biosynthesis, (c5) a tubulin polymerization inhibitor, (c6) a cell division (unknown site of action) inhibitor, (c7) a delocalizer of spectrin-like protein, (c8) an inhibitor of actin / myosin / fimbrin function, (c9) a complex I (NADH oxidoreductase) inhibitor, (c10) a complex II (succinate dehydrogenase) inhibitor, (c11) a complex III (ubiquinol oxidase Qo site) inhibitor, (c12) a complex III (ubiquinone reductase Qi site) inhibitor, (c13) an uncoupler of oxidative phosphorylation, (c14) a complex III (ubiquinone reductase Qo site stigmatellin binding subsite) inhibitor, (c15) a methionine biosynthesis inhibitor, (c16) a protein biosynthesis (ribosome translation initiation stage) inhibitor, (c17) a protein biosynthesis (ribosome polypeptide elongation stage) inhibitor, (c18) a MAP histidine kinase (os-2, HOG1) inhibitor in osmotic signal transduction, (c19) a MAP histidine kinase (os-1, Daf1) inhibitor in osmotic signal transduction, (c20) a methyltransferase inhibitor of phospholipid biosynthesis, (c21) an inhibitor of cellular lipid peroxidation, (c22) a fatty acid inhibitor of cell membrane permeability, (c23) a lipid homeostasis and transport / storage inhibitor, (c24) a C14 demethylase inhibitor in sterol biosynthesis, (c25) a 3-keto reductase inhibitor in C4 demethylation of sterol biosynthesis, (c26) a squalene epoxidase inhibitor in sterol biosynthesis, (c27) a chitin synthase inhibitor, (c28) a cellulose synthase inhibitor, (c29) a reductase inhibitor of melanin biosynthesis, (c30) a dehydratase inhibitor of melanin biosynthesisThe agricultural and horticultural pest control composition according to claim 1 (excluding the pest control composition for paddy rice), which is at least one compound selected from the group consisting of (c31) a polyketamide synthase inhibitor for melanin synthesis, (c32) a resistance inducer for host plants (excluding saccharin or its salts), (c33) a compound with an unknown mechanism of action, (c34) a multi-site contact active compound, and (c35) an unclassified compound.

8. [Correction based on Rule 91, 25.04.2025] The said (B) insecticidal active compound is at least one compound selected from the group consisting of (b1) acetylcholinesterase (AChE) inhibitor, (b2) GABAergic chloride ion (chloride ion) channel blocker, (b3) sodium channel modulator, (b4) nicotinic acetylcholine receptor (nAChR) competitive modulator, (b5) nicotinic acetylcholine receptor (nAChR) allosteric modulator - Site I, (b9) chordotonal organ TRPV channel modulator, (b14) nicotinic acetylcholine receptor (nAChR) channel blocker, (b16) chitin biosynthesis inhibitor (Type 1), (b18) ecdysone receptor agonist, (b26) ryanodine receptor modulator, and (b33) oxathiazosulfyl, benzpyrioxan, and isocycloseram; the said (C) fungicidal active compound is at least one compound selected from the group consisting of (c1) RNA polymerase I inhibitor, (c2) DNA / RNA biosynthesis inhibitor, (c3) DNA topoisomerase Type II (gyrase) inhibitor, (c4) dihydroorotate dehydrogenase inhibitor in de novo pyrimidine biosynthesis, (c5) tubulin polymerization inhibitor, (c6) cell division (site of action unknown) inhibitor, (c10) complex II (succinate dehydrogenase) inhibitor, (c11) complex III (ubiquinol oxidase Qo site) inhibitor, (c12) complex III (ubiquinone reductase Qi site) inhibitor, (c16) protein biosynthesis (ribosome translation initiation stage) inhibitor, (c17) protein biosynthesis (ribosome polypeptide elongation stage) inhibitor, (c20) methyltransferase inhibitor of phospholipid biosynthesis, (c24) C14 demethylase inhibitor in sterol biosynthesis, (c27) chitin biosynthesis enzyme inhibitor, (c29) reductase inhibitor of melanin biosynthesis, (c31) polyketamide synthase inhibitor of melanin biosynthesis, (c32) host plant resistance inducer (excluding saccharin or its salts), (c33) compound with unknown mechanism of action, (c34) multi-site contact active compound, and (c35) quinofumelin. The agricultural and horticultural pest control composition according to claim 1 (excluding the pest control composition for paddy rice).

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