Synthesis method of bis (2, 2, 2-trifluoroethyl) carbonate
A synthesis method, trifluoroethyl technology, applied in the field of dicarbonate synthesis, can solve the problems of poor exchange reaction ability, complex reaction process, and reduced catalytic activity, achieving mild reaction, simple operation, and few by-products Effect
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Embodiment 1
[0020] The synthetic method of two (2,2,2-trifluoroethyl) carbonates, its synthetic steps are as follows:
[0021] Take 24g (0.24mol) of trifluoroethanol and add it to 100mL of dichloromethane, as a dichloromethane solution of trifluoroethanol for later use;
[0022] Under the protection of nitrogen, take 21.4g (0.1mol) of diphenyl carbonate and 40.95g (0.65mol) of imidazole and stir and mix, add 2.6g of aluminum chloride, heat to 80°C, keep stirring at 80°C for pre-reaction for 2h, and then lower to room temperature, add dropwise a dichloromethane solution containing trifluoroethanol, after the dropwise addition, reflux for 2 h for transesterification, after the reaction is complete, add hydrochloric acid dropwise to adjust the pH to 1, separate the phases, and concentrate the obtained dichloromethane phase , rectification, obtain 19.57g two (2,2,2-trifluoroethyl) carbonate, yield 86.59%, purity 99.97%, concrete chemical reaction formula is as follows:
[0023]
Embodiment 2
[0025] The synthetic method of two (2,2,2-trifluoroethyl) carbonates, its synthetic steps are as follows:
[0026] Take 23g (0.23mol) of trifluoroethanol and add it to 80mL of dichloromethane, as a dichloromethane solution of trifluoroethanol for later use;
[0027] Under nitrogen protection, take 21.4g (0.1mol) of diphenyl carbonate and 41.58g (0.66mol) of imidazole and stir and mix, add 2.14g of aluminum chloride, heat to 70°C, keep stirring at 70°C for pre-reaction for 3h, then drop to room temperature, dropwise add a dichloromethane solution containing trifluoroethanol, after the dropwise addition, reflux for 2.5 h for transesterification reaction, after the reaction is complete, add hydrochloric acid dropwise to adjust to pH = 1.5, separate the phases, and the obtained dichloromethane phase is After concentration and rectification, 19.14 g of bis(2,2,2-trifluoroethyl) carbonate was obtained, with a yield of 84.69% and a purity of 99.91%.
Embodiment 3
[0029] The synthetic method of two (2,2,2-trifluoroethyl) carbonates, its synthetic steps are as follows:
[0030] Take 24g (0.24mol) of trifluoroethanol and add it to 90mL of dichloromethane, as a dichloromethane solution of trifluoroethanol for later use;
[0031] Under the protection of nitrogen, take 21.4g (0.1mol) of diphenyl carbonate and 44.1g (0.7mol) of imidazole and stir and mix, add 3.21g of aluminum chloride, heat to 75°C, keep stirring at 75°C for pre-reaction for 2.5h, then Cool down to room temperature, add dropwise a dichloromethane solution containing trifluoroethanol, after the dropwise addition, reflux for 3 h for transesterification, after the reaction is complete, add hydrochloric acid dropwise to adjust to pH = 2, separate the phases, and the obtained dichloromethane phase is After concentration and rectification, 19.29 g of bis(2,2,2-trifluoroethyl) carbonate was obtained, with a yield of 85.35% and a purity of 99.93%.
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