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Triazole derivative and application thereof

A technology of triazole derivatives and compounds, applied in the field of chemistry, can solve the problems of phytotoxicity of next crops, deformed seedlings, low seedling emergence rate, etc., and achieve the effects of reducing phytotoxicity, preventing lodging activity, and reducing rice plant height

Active Publication Date: 2021-06-22
SHENYANG RES INST OF CHEM IND
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  • Summary
  • Abstract
  • Description
  • Claims
  • Application Information

AI Technical Summary

Problems solved by technology

However, due to its long residual period (pesticide electronic manual, the soil half-life is 0.5-1.0 years), it is easy to cause phytotoxicity to the next crops, resulting in no seedlings, late emergence, low emergence rate, deformed seedlings and other phytotoxicity

Method used

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  • Triazole derivative and application thereof
  • Triazole derivative and application thereof
  • Triazole derivative and application thereof

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Experimental program
Comparison scheme
Effect test

Embodiment 1

[0181] Embodiment 1: the synthesis of compound 6-55

[0182] Step A:

[0183]

[0184] Add 3.3 g of 1-(1,2,4-triazol-1-yl)-3,3-dimethyl-2-butanone, 50 mL of DMF, and 1.0 g of sodium hydride into a 100 mL flask, and stir at room temperature for 0.5 hours. 3-Chloromethyl-6-chloropyridine 3.3g, stirring and heating at 80°C for 4 hours, after the reaction was detected by TLC, add 150mL of water, extract with 50mL of ethyl acetate x 3, combine organic phases, dry over anhydrous sodium sulfate, column layer Analysis (eluent is ethyl acetate and petroleum ether (boiling range 60-90 ℃), volume ratio is 1:2) purification to obtain 2.53g compound 1-(6-chloropyridin-3-yl) 2-(1, 2,4-triazol-1-yl)-4,4-dimethyl-3-pentanone, white solid namely A6-55. 1 H NMR (600MHz, DMSO- d6 )δ8.63(s,1H),8.19(d,J=2.2Hz,1H),7.96(s,1H),7.65(dd,J=8.2,2.4Hz,1H),7.41(d,J=8.2 Hz,1H),6.08(t,J=7.7Hz,1H),3.31(d,J=7.7Hz,2H),1.06(s,9H).m / z(%):293.09[M+H] +

[0185] Step B:

[0186]

[0187] Add 1.5 g of 1...

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Abstract

The invention belongs to the field of chemistry, and particularly relates to a triazole derivative and application of the derivative in plant growth regulation and bactericide. The triazole derivative is a compound as shown in a general formula I defined in the description, a diastereoisomer, a chiral isomer or a salt thereof. The definition of each substituent group in the formula is shown in the description. The compound provided by the invention can be applied to plant growth regulation and bactericides.

Description

technical field [0001] The invention belongs to the field of chemistry, specifically a triazole derivative and the application of the derivative in plant growth regulation and fungicide. Background technique [0002] Paclobutrazol is a plant growth regulator, which has the effects of delaying plant growth, inhibiting stem elongation, shortening internodes, promoting plant tillering, increasing plant stress resistance, and increasing yield. However, due to its long residual period (pesticide electronic manual, the soil half-life is 0.5-1.0 years), it is easy to cause phytotoxicity to the next crops, resulting in no seedlings, late emergence, low emergence rate, deformed seedlings and other phytotoxicity. [0003] The development of plant growth regulators with fast metabolism and low residue is of great significance to agricultural production. Contents of the invention [0004] The object of the present invention is a triazole derivative and its application. [0005] In o...

Claims

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Application Information

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Patent Type & Authority Applications(China)
IPC IPC(8): C07D401/06A01N43/653A01P1/00A01P3/00A01P21/00
CPCC07D401/06A01N43/653C07D411/06C07D403/06Y02A40/10
Inventor 周繁冉兆晋孙朝辉毛志强王芳王志祥崔顺艳侯薪鑫王宇石凯强
Owner SHENYANG RES INST OF CHEM IND
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